GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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Praliciguat
CAS:<p>Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.</p>Fórmula:C21H14F8N6O2Pureza:98.82%Cor e Forma:SolidPeso molecular:534.36Ataciguat
CAS:<p>Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.</p>Fórmula:C21H19Cl2N3O6S3Pureza:99.09%Cor e Forma:SolidPeso molecular:576.49Dimethocaine
CAS:<p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>Fórmula:C16H26N2O2Pureza:99.52%Cor e Forma:SolidPeso molecular:278.39N-Acetylhistamine acetate
<p>N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.</p>Fórmula:C9H15N3O3Pureza:98%Cor e Forma:SolidPeso molecular:213.23BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Cor e Forma:SolidPeso molecular:458.42FK962
CAS:<p>FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.</p>Fórmula:C14H17FN2O2Pureza:99.89%Cor e Forma:SolidPeso molecular:264.3AC 187 Acetate
<p>AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.</p>Fórmula:C129H209N37O42Pureza:99.71%Cor e Forma:SolidPeso molecular:2950.26Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Fórmula:C25H40ClN3O8Pureza:99.91%Cor e Forma:White Crystalline PowderPeso molecular:546.05WAY-100635 Monomaleate
CAS:<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Cor e Forma:SolidPeso molecular:538.64Detomidine hydrochloride
CAS:<p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>Fórmula:C12H14N2·HClPureza:99.97%Cor e Forma:SolidPeso molecular:222.71Indacaterol
CAS:<p>Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.</p>Fórmula:C24H28N2O3Pureza:99.96%Cor e Forma:SolidPeso molecular:392.49SAX-187
CAS:<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Fórmula:C15H13ClN4O2S2Pureza:97.82% - 98%Cor e Forma:SolidPeso molecular:380.87Calcitonin(salmon) Acetate(47931-85-1(free base))
<p>Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5</p>Fórmula:C145H240N44O48S2Pureza:99.29%Cor e Forma:SolidPeso molecular:3431.85GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Fórmula:C29H36F3N3O5Pureza:98.2% - 98.88%Cor e Forma:SolidPeso molecular:563.61Mequitazine
CAS:<p>Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.</p>Fórmula:C20H22N2SPureza:99.98%Cor e Forma:SolidPeso molecular:322.47MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Fórmula:C27H21F3N2O3Pureza:99.54% - 99.59%Cor e Forma:SolidPeso molecular:478.46Chlorcyclizine
CAS:<p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>Fórmula:C18H21ClN2Pureza:98.75%Cor e Forma:SolidPeso molecular:300.83Regadenoson
CAS:<p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>Fórmula:C15H18N8O5Pureza:99.57% - 99.81%Cor e Forma:Off-White SolidPeso molecular:390.35Ranitidine
CAS:<p>Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).</p>Fórmula:C13H22N4O3SPureza:99.52%Cor e Forma:Solid SolidPeso molecular:314.40S1RA hydrochloride
CAS:<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Fórmula:C20H24ClN3O2Pureza:98% - 99.84%Cor e Forma:SolidPeso molecular:373.87Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Fórmula:C20H22N2O6Pureza:99.39%Cor e Forma:SolidPeso molecular:386.4Epinastine hydrochloride
CAS:<p>Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.</p>Fórmula:C16H15N3·HClPureza:99.26% - 99.62%Cor e Forma:White SolidPeso molecular:285.77AM095
CAS:<p>AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.</p>Fórmula:C27H23N2NaO5Pureza:98.87%Cor e Forma:SolidPeso molecular:478.47AHN 1-055 hydrochloride
CAS:<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Fórmula:C21H24ClF2NOPureza:99.89%Cor e Forma:SolidPeso molecular:379.87SCH 58261
CAS:<p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>Fórmula:C18H15N7OPureza:99.07% - 99.75%Cor e Forma:SolidPeso molecular:345.36JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Fórmula:C14H16ClN3OPureza:99.83% - 99.96%Cor e Forma:SolidPeso molecular:277.75Neurokinin A(4-10) TFA(97559-35-8 free base)
<p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>Fórmula:C36H55F3N8O12SPureza:>99.99%Cor e Forma:SolidPeso molecular:880.93Bevantolol hydrochloride
CAS:<p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>Fórmula:C20H28ClNO4Pureza:99.49%Cor e Forma:SolidPeso molecular:381.9Pimozide
CAS:<p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>Fórmula:C28H29F2N3OPureza:99.63% - >99.99%Cor e Forma:SolidPeso molecular:461.55RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Fórmula:C25H27N3O3Pureza:98.64% - 99.62%Cor e Forma:SolidPeso molecular:417.5Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Cor e Forma:SolidPeso molecular:240.69HPI 1
CAS:<p>HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.</p>Fórmula:C27H29NO6Pureza:97.6%Cor e Forma:SolidPeso molecular:463.52C-021
CAS:<p>C 021 dihydrochloride is a potent CCR4 antagonist.</p>Fórmula:C27H41N5O2Pureza:99.74% - 99.90%Cor e Forma:SolidPeso molecular:467.65Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Cor e Forma:Appearance White Crystalline PowderPeso molecular:264.19LY334370
CAS:<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Fórmula:C21H22FN3OPureza:99.32%Cor e Forma:SolidPeso molecular:351.42Ozagrel hydrochloride
CAS:<p>Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contraction</p>Fórmula:C13H12N2O2·HClPureza:99.80%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:264.71Aprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Fórmula:C23H21F7N4O3Pureza:98% - 99.68%Cor e Forma:Off-White To Light Yellow Cyrstalline SolidPeso molecular:534.43CCG215022
CAS:<p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>Fórmula:C26H22FN7O3Pureza:97.63% - 99.69%Cor e Forma:SolidPeso molecular:499.5Clemizole hydrochloride
CAS:<p>Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.</p>Fórmula:C19H21Cl2N3Pureza:>99.99%Cor e Forma:SolidPeso molecular:362.3Vicriviroc maleate
CAS:<p>Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.</p>Fórmula:C32H42F3N5O6Pureza:98.16% - 98.37%Cor e Forma:SolidPeso molecular:649.7JK184
CAS:<p>JK184 is a potent Hedgehog (Hh) pathway inhibitor.</p>Fórmula:C19H18N4OSPureza:98.93% - 99.89%Cor e Forma:SolidPeso molecular:350.44AZD-4818
CAS:<p>AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Fórmula:C27H32Cl2N2O7Pureza:99.01%Cor e Forma:SolidPeso molecular:567.46BX471
CAS:<p>BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.</p>Fórmula:C21H24ClFN4O3Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:434.89Glasdegib
CAS:<p>Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.</p>Fórmula:C21H22N6OPureza:98.72%Cor e Forma:SolidPeso molecular:374.44RS102895
CAS:<p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>Fórmula:C21H21F3N2O2Pureza:97.64% - 99.80%Cor e Forma:SolidPeso molecular:390.4MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Fórmula:C24H23N3O5SPureza:99.73%Cor e Forma:SolidPeso molecular:465.52RE-640
CAS:<p>NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.</p>Fórmula:C20H16Cl2N4Pureza:99.60% - 99.87%Cor e Forma:SolidPeso molecular:383.27SAG hydrochloride (912545-86-9(free base))
CAS:<p>SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.</p>Fórmula:C28H29Cl2N3OSPureza:99.19% - 99.77%Cor e Forma:SolidPeso molecular:526.52R243
CAS:<p>R243 is CCR8 signaling and chemotaxis inhibitor.</p>Fórmula:C21H27NO4Pureza:99.03%Cor e Forma:SolidPeso molecular:357.44Sonidegib
CAS:<p>Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.</p>Fórmula:C26H26F3N3O3Pureza:98% - 99.97%Cor e Forma:SolidPeso molecular:485.5Salmeterol Xinafoate
CAS:<p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>Fórmula:C36H45NO7Pureza:98% - 98.24%Cor e Forma:White SolidPeso molecular:603.75MRT-81
CAS:<p>MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.</p>Fórmula:C31H29N3O5SPureza:99.72%Cor e Forma:SolidPeso molecular:555.64Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Fórmula:C46H65N13O11S2Pureza:99.65%Cor e Forma:SolidPeso molecular:1040.22Geissoschizine methyl ether
CAS:<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Fórmula:C22H26N2O3Pureza:99.24% - 99.68%Cor e Forma:SolidPeso molecular:366.45Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Fórmula:C59H80N14O13Pureza:95.3%Cor e Forma:SolidPeso molecular:1193.35Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Fórmula:C18H15BrF2N4O2Pureza:98.42% - 99.88%Cor e Forma:SolidPeso molecular:437.24Lecirelin acetate(61012-19-9 free base)
<p>Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts</p>Fórmula:C61H88N16O14Pureza:98.1%Cor e Forma:SolidPeso molecular:1269.45M40 acetate(143896-17-7 free base)
<p>M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29)</p>Fórmula:C96H149N23O26Pureza:99.88%Cor e Forma:SolidPeso molecular:2041.38Gastrin I (human) acetate
<p>Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (</p>Fórmula:C99H128N20O33SPureza:98.84%Cor e Forma:SolidPeso molecular:2158.25ML-184
CAS:<p>ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.</p>Fórmula:C25H34N4O3SPureza:99.45%Cor e Forma:SolidPeso molecular:470.63AM966
CAS:<p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>Fórmula:C27H23ClN2O5Pureza:98.06% - 99.79%Cor e Forma:SolidPeso molecular:490.932-Pyridylethylamine dihydrochloride
CAS:<p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>Fórmula:C7H12Cl2N2Pureza:99.42%Cor e Forma:SolidPeso molecular:195.09GBR 12935 dihydrochloride
CAS:<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Fórmula:C28H36Cl2N2OPureza:99.09% - ≥95%Cor e Forma:SolidPeso molecular:487.5Loxapine
CAS:<p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>Fórmula:C18H18ClN3OPureza:99.88%Cor e Forma:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.81ACTH (1-17) acetate
<p>ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).</p>Fórmula:C97H149N29O25SPureza:98.53%Cor e Forma:SolidPeso molecular:2153.47Pergolide
CAS:<p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>Fórmula:C19H26N2SPureza:99.95%Cor e Forma:SolidPeso molecular:314.49Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Cor e Forma:SolidPeso molecular:433.57Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Fórmula:C12H17NO9Pureza:97.32% - 99.97%Cor e Forma:SolidPeso molecular:319.27LRGILS-NH2 acetate
<p>LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.</p>Fórmula:C29H56N10O7Pureza:96.65%Cor e Forma:SolidPeso molecular:656.82Hemopressin (human, mouse) acetate
<p>Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.</p>Fórmula:C52H83N13O14Pureza:99.86%Cor e Forma:SolidPeso molecular:1114.29Brimonidine Tartrate
CAS:<p>Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).</p>Fórmula:C15H16BrN5O6Pureza:99.95%Cor e Forma:Off-White Crystalline SolidPeso molecular:442.22Ki16425
CAS:<p>Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.</p>Fórmula:C23H23ClN2O5SPureza:97.6% - 97.78%Cor e Forma:SolidPeso molecular:474.96Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Cor e Forma:White SolidPeso molecular:463Serotonin
CAS:<p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>Fórmula:C10H12N2OPureza:97.47% - 99.92%Cor e Forma:SolidPeso molecular:176.22Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Cor e Forma:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28Verucerfont
CAS:<p>Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .</p>Fórmula:C22H26N6O2Pureza:99.90%Cor e Forma:SolidPeso molecular:406.48tcY-NH2 TFA(327177-34-4 free base)
<p>tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.</p>Fórmula:C42H50F3N7O9Pureza:>99.99%Cor e Forma:SolidPeso molecular:853.9IPSU
CAS:<p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>Fórmula:C23H27N5O2Pureza:97.05%Cor e Forma:SolidPeso molecular:405.498-Cyclopentyl-1,3-dimethylxanthine
CAS:<p>8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.</p>Fórmula:C12H16N4O2Pureza:98.58% - >99.99%Cor e Forma:SolidPeso molecular:248.283-AQC
CAS:<p>3-AQC is a competitive antagonist of 5-HT3.</p>Fórmula:C20H21N5O4Pureza:99.45%Cor e Forma:SolidPeso molecular:395.41CHEMBL241987
CAS:<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Fórmula:C16H11N3OPureza:99.81%Cor e Forma:SolidPeso molecular:261.28BD1063 dhydrochloride
CAS:<p>BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).</p>Fórmula:C13H20Cl4N2Pureza:99.52% - ≥95%Cor e Forma:SolidPeso molecular:346.12Tiprenolol
CAS:<p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>Fórmula:C13H21NO2SPureza:99.43%Cor e Forma:SolidPeso molecular:255.38BAR 501 impurity
CAS:<p>BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。</p>Fórmula:C26H46O3Pureza:98.78%Cor e Forma:SolidPeso molecular:406.64AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C21H25ClN2Pureza:99.61%Cor e Forma:SolidPeso molecular:340.89ONO-7300243
CAS:<p>ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).</p>Fórmula:C28H31NO5Pureza:99.66%Cor e Forma:SolidPeso molecular:461.55Thrombin Receptor Activator for Peptide
<p>Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.</p>Fórmula:C32H51F3N8O9Pureza:99.88%Cor e Forma:SolidPeso molecular:748.79Ablukast
CAS:<p>Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.</p>Fórmula:C28H34O8Pureza:98.58%Cor e Forma:SolidPeso molecular:498.56GW842166X
CAS:<p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>Fórmula:C18H17Cl2F3N4O2Pureza:99.47%Cor e Forma:SolidPeso molecular:449.25Ibutamoren Mesylate
CAS:<p>Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.</p>Fórmula:C28H40N4O8S2Pureza:97.98% - ≥98%Cor e Forma:SolidPeso molecular:624.77SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Fórmula:C17H13N5O2Pureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:319.322-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
<p>2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.</p>Fórmula:C38H64F3N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:891.98Ditolylguanidine
CAS:<p>Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).</p>Fórmula:C15H17N3Pureza:98.42%Cor e Forma:White To Pinkish Solid PowderPeso molecular:239.321-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:<p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>Fórmula:C9H15N3OPureza:95%Cor e Forma:SolidPeso molecular:181.23VKGILS-NH2 Acetate
<p>VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.</p>Fórmula:C30H58N8O9Pureza:98.83%Cor e Forma:SolidPeso molecular:674.83DORA-22
CAS:<p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>Fórmula:C23H22F2N4O2Pureza:97.67%Cor e Forma:SolidPeso molecular:424.44Pridopidine
CAS:<p>Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.</p>Fórmula:C15H23NO2SPureza:95.2% - 99.89%Cor e Forma:SolidPeso molecular:281.41AZ3451
CAS:<p>AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).</p>Fórmula:C30H27BrN4O3Pureza:98.12%Cor e Forma:SolidPeso molecular:571.46lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7
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