GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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Rolapitant hydrochloride hydrate
CAS:<p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>Fórmula:C25H29ClF6N2O3Cor e Forma:SolidPeso molecular:554.95Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Fórmula:C17H25N3O2SPureza:99.08%Cor e Forma:SolidPeso molecular:335.47Melanin Concentrating Hormone, salmon acetate
<p>Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>Fórmula:C91H143N27O26S4Pureza:99.41%Cor e Forma:SolidPeso molecular:2157Procaterol hydrochloride hydrate
CAS:<p>Short-acting β2-adrenergic receptor agonist used to treat asthma.</p>Fórmula:C32H48Cl2N4O7Pureza:99.71% - 99.97%Cor e Forma:SolidPeso molecular:671.65ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS:<p>ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)</p>Fórmula:C14H15NO2SPureza:99.98%Cor e Forma:SolidPeso molecular:261.34Bosentan (hydrate)
CAS:<p>Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.</p>Fórmula:C27H29N5O6S·H2OPureza:99.31% - 99.86%Cor e Forma:White PowderPeso molecular:569.63Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Fórmula:C15H19N3Pureza:≥95%Cor e Forma:SolidPeso molecular:241.33Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Fórmula:C21H24ClN2NaO4SPureza:99.82%Cor e Forma:SolidPeso molecular:458.93GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Fórmula:C151H228N40O47Pureza:98.89%Cor e Forma:SolidPeso molecular:3355.67Ralinepag
CAS:<p>Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human and</p>Fórmula:C23H26ClNO5Pureza:99.79% - 99.85%Cor e Forma:SolidPeso molecular:431.91Etilevodopa hydrochloride
CAS:<p>Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.</p>Fórmula:C11H16ClNO4Pureza:95.00%Cor e Forma:SolidPeso molecular:261.7Eprazinone dihydrochloride
CAS:<p>Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.</p>Fórmula:C24H32N2O2·2HClPureza:99.25%Cor e Forma:A White Or Almost White CrysPeso molecular:453.44Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.444F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Cor e Forma:SolidPeso molecular:429.49Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Fórmula:C40H55N7O11SPureza:99.84% - >99.99%Cor e Forma:White PowderPeso molecular:841.97Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Cor e Forma:White Or Off-White CrystallinePeso molecular:327.4Hemokinin 1 (human) acetate(491851-53-7 free base)
<p>Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.</p>Fórmula:C56H88N14O16SPureza:97.82%Cor e Forma:SolidPeso molecular:1245.45Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Fórmula:C9H13NO2Pureza:99.5% - 99.89%Cor e Forma:SolidPeso molecular:167.21PAR-2-IN-1
CAS:<p>PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.</p>Fórmula:C12H14ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:267.71[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS:<p>[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.</p>Fórmula:C190H286N54O56Pureza:99.39%Cor e Forma:SolidPeso molecular:4223Enavogliflozin
CAS:<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Fórmula:C24H27ClO6Pureza:97.37%Cor e Forma:SolidPeso molecular:446.92MEN 10207 acetate
<p>MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.</p>Fórmula:C59H72N14O12Pureza:99.18%Cor e Forma:SolidPeso molecular:1169.29SKF 38393 hydrochloride
CAS:<p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>Fórmula:C16H17NO2·HClPureza:99.1% - 99.51%Cor e Forma:SolidPeso molecular:291.77idalopirdine
CAS:<p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>Fórmula:C20H19F5N2OPureza:99.73%Cor e Forma:SolidPeso molecular:398.37E7046
CAS:<p>E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.</p>Fórmula:C22H18F5N3O4Pureza:99.86%Cor e Forma:SolidPeso molecular:483.4Isocorynoxeine
CAS:<p>Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.</p>Fórmula:C22H26N2O4Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:382.45lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7Parmodulin 2
CAS:<p>ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).</p>Fórmula:C17H17BrN2O2Pureza:97.35% - 99.95%Cor e Forma:SolidPeso molecular:361.23Alcaftadine
CAS:<p>Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.</p>Fórmula:C19H21N3OPureza:98% - 98.65%Cor e Forma:SolidPeso molecular:307.397-Amino-4-(trifluoromethyl)coumarin
CAS:<p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16GR 125743
CAS:<p>GR 125743 is a novel antagonist of 5-HT1B/1D receptor.</p>Fórmula:C25H28N4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:416.52T-1095
CAS:<p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>Fórmula:C26H28O11Pureza:99.78%Cor e Forma:SolidPeso molecular:516.49Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Fórmula:C15H24ClNO2Pureza:99.79%Cor e Forma:SolidPeso molecular:285.81MK-571 sodium
CAS:<p>MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.</p>Fórmula:C26H27ClN2O3S2·NaPureza:97.86% - 99.58%Cor e Forma:SolidPeso molecular:537.07Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Fórmula:C5H11Cl2N3Pureza:99.12%Cor e Forma:SolidPeso molecular:184.067N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Fórmula:C12H14N2OPureza:98.79%Cor e Forma:PowderPeso molecular:202.25ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Fórmula:C19H22N4O3Pureza:99.92%Cor e Forma:SolidPeso molecular:354.4Xamoterol
CAS:<p>Xamoterol is a cardiac stimulant.</p>Fórmula:C16H25N3O5Cor e Forma:SolidPeso molecular:339.39Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Fórmula:C15H20N8O6Pureza:98%Cor e Forma:SolidPeso molecular:408.37Dasotraline
CAS:<p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>Fórmula:C16H15Cl2NCor e Forma:SolidPeso molecular:292.2Amylin, amide, rat acetate(124447-81-0,free base)
<p>Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.</p>Fórmula:C169H276N52O55S2Pureza:98.93%Cor e Forma:SolidPeso molecular:3980.45BPTU
CAS:<p>BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).</p>Fórmula:C23H22F3N3O3Pureza:99.37% - 99.89%Cor e Forma:SolidPeso molecular:445.43PAR-4 Agonist Peptide, amide TFA
CAS:<p>PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.</p>Fórmula:C36H49F3N8O9Pureza:99.72%Cor e Forma:SolidPeso molecular:794.82PD 168568
CAS:<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Fórmula:C22H27N3OCor e Forma:SolidPeso molecular:349.47Protease-Activated Receptor-1, PAR-1 Agonist acetate
<p>PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.</p>Fórmula:C37H62N10O11Pureza:98.1800%Cor e Forma:SolidPeso molecular:822.95Secretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Fórmula:C129H216N42O42Pureza:98.12%Cor e Forma:SolidPeso molecular:3027.35GUANABENZ
CAS:<p>GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.</p>Fórmula:C8H8Cl2N4Pureza:98.31%Cor e Forma:White Solid From Acetonitrile SolidPeso molecular:231.08S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Cor e Forma:SolidPeso molecular:407.48Bradykinin (2-9)
CAS:<p>Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.</p>Fórmula:C44H61N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:904.02Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Fórmula:C19H21N5O4Pureza:99.86%Cor e Forma:White To Tan Powder SolidPeso molecular:383.4GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Fórmula:C22H21ClN4O4Pureza:99.04%Cor e Forma:SolidPeso molecular:440.88Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Fórmula:C23H29NO5SPureza:98%Cor e Forma:SolidPeso molecular:431.55Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Fórmula:C9H10Cl2N4Cor e Forma:SolidPeso molecular:245.11Substance P 1-9 aceate
<p>Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.</p>Fórmula:C54H81N15O14Pureza:99.01%Cor e Forma:SolidPeso molecular:1164.31Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Fórmula:C23H24FN3O2Pureza:99.2%Cor e Forma:SolidPeso molecular:393.45Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Fórmula:C21H20O9Pureza:98.90% - 99.21%Cor e Forma:Yellow Brown Fine PowderPeso molecular:416.38Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Fórmula:C18H24ClNO3Pureza:97.15% - 99.94%Cor e Forma:SolidPeso molecular:337.84CP 376395
CAS:<p>CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.</p>Fórmula:C21H30N2OPureza:99.86% - 99.94%Cor e Forma:SolidPeso molecular:326.48Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Fórmula:C19H16F2N8O2Pureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:426.38[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
<p>[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and</p>Fórmula:C76H103N21O18SPureza:99.75%Cor e Forma:SolidPeso molecular:1630.82Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Fórmula:C21H27ClN2O2Pureza:99.54% - ≥95%Cor e Forma:Oil SolidPeso molecular:374.9Peptide YY (PYY) (3-36), human
CAS:<p>Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.</p>Fórmula:C176H272N52O54Pureza:97.76%Cor e Forma:SolidPeso molecular:3980.42Derenofylline
CAS:<p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>Fórmula:C18H20N4OPureza:98.09%Cor e Forma:SolidPeso molecular:308.38CYM 50358 hydrochloride (1314212-39-9 free base)
CAS:<p>CYM50358 HCl is an S1P4 antagonist.</p>Fórmula:C20H19Cl3N2O2Pureza:99.57%Cor e Forma:SolidPeso molecular:425.73CJC-1295 acetate(863288-34-0 free base)
<p>CJC-1295 acetate is a synthetic GHRH analogue and GHS.</p>Fórmula:C154H256N44O44Pureza:97.29%Cor e Forma:SolidPeso molecular:3428.01Bindarit
CAS:<p>Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.</p>Fórmula:C19H20N2O3Pureza:98.35% - 98.55%Cor e Forma:SolidPeso molecular:324.37Laropiprant sodium
<p>Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.</p>Cor e Forma:SolidPEN (human) aceate
<p>PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.</p>Fórmula:C99H163N27O34Pureza:99.25%Cor e Forma:SolidPeso molecular:2275.51Tafluprost
CAS:<p>Tafluprost, a prostaglandin analog, is the selective agonist of fluoroprostaglandin (FP) receptor PGF2α.</p>Fórmula:C25H34F2O5Pureza:97.7% - 99.67%Cor e Forma:LiquidPeso molecular:452.53ACTH 11-24 acetate(4237-93-8 free base)
CAS:<p>ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.</p>Fórmula:C79H138N24O18Pureza:>99.99%Cor e Forma:SolidPeso molecular:1712.12AM281
CAS:<p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>Fórmula:C21H19Cl2IN4O2Pureza:98.6% - >99.99%Cor e Forma:White To Off-White SolidPeso molecular:557.21Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Fórmula:C17H18ClN4OCor e Forma:SolidPeso molecular:329.11691ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Fórmula:C129H207N45O41S3Pureza:98.24%Cor e Forma:SolidPeso molecular:3140.5PNU 22394 hydrochloride
CAS:<p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>Fórmula:C13H17ClN2Pureza:97.83%Cor e Forma:SolidPeso molecular:236.74BAR501
CAS:<p>BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。</p>Fórmula:C26H46O3Pureza:99.29% - 99.68%Cor e Forma:SolidPeso molecular:406.64PF-06882961 Tris
CAS:<p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Fórmula:C35H41FN6O7Pureza:98.74% - 99.79%Cor e Forma:SolidPeso molecular:676.7TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Cor e Forma:SolidPeso molecular:448.43CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Fórmula:C20H21N7O3Pureza:98.78%Cor e Forma:SolidPeso molecular:407.43SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Fórmula:C16H20N2O2·HClPureza:99.64%Cor e Forma:SolidPeso molecular:308.81Vortioxetine
CAS:<p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>Fórmula:C18H22N2SPureza:99.34% - 99.34%Cor e Forma:SolidPeso molecular:298.45Adrenocorticotropic Hormone (ACTH) (4-10) TFA
<p>Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .</p>Fórmula:C46H60F3N13O12SPureza:98.49%Cor e Forma:SolidPeso molecular:1076.12CID 16020046
CAS:<p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>Fórmula:C25H19N3O4Pureza:99.03%Cor e Forma:SolidPeso molecular:425.44Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Fórmula:C14H16N2·HClPureza:99.74%Cor e Forma:SolidPeso molecular:248.75BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Fórmula:C25H28Cl2N2OCor e Forma:SolidPeso molecular:443.41Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Fórmula:C20H24N2OSCor e Forma:SolidPeso molecular:340.48Mini Gastrin I, human acetate
<p>Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.</p>Fórmula:C76H103N15O28SPureza:99.35% - 99.82%Cor e Forma:SolidPeso molecular:1706.78Dimemorfan phosphate
CAS:<p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>Fórmula:C18H25N·H3O4PPureza:99.65%Cor e Forma:SolidPeso molecular:353.4Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Fórmula:C38H73N21O10S2HClPureza:>99.99%Cor e Forma:SolidPeso molecular:1353.33Diclofensine hydrochloride
CAS:<p>Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。</p>Fórmula:C17H18Cl3NOPureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:358.69Pizuglanstat
CAS:<p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>Fórmula:C27H36N6O4Pureza:99.62%Cor e Forma:SolidPeso molecular:508.61Neuropeptide SF(mouse,rat) acetate
<p>Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.</p>Fórmula:C42H69N13O12Pureza:98.37%Cor e Forma:SolidPeso molecular:948.08Neuropeptide EI, rat acetate
<p>Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.</p>Fórmula:C65H102N16O25Pureza:95.55%Cor e Forma:SolidPeso molecular:1507.6NIBR189
CAS:<p>NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively)</p>Fórmula:C21H21BrN2O3Pureza:97%Cor e Forma:ColourlessPeso molecular:429.31[Lys8, Lys9]-Neurotensin (8-13) acetate
<p>[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2</p>Fórmula:C40H68N8O10Pureza:99.31%Cor e Forma:SolidPeso molecular:821.02Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Fórmula:C21H21FO5SPureza:99.38% - 99.70%Cor e Forma:SolidPeso molecular:404.45Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Cor e Forma:SolidPeso molecular:434.83Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Cor e Forma:SolidPeso molecular:446.95RS-127445 hydrochloride
CAS:<p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>Fórmula:C17H17ClFN3Pureza:99.48%Cor e Forma:SolidPeso molecular:317.79Fexofenadine
CAS:<p>Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.</p>Fórmula:C32H39NO4Pureza:99.35%Cor e Forma:White To Off-White SolidPeso molecular:501.66PRX-08066
CAS:<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Fórmula:C19H17ClFN5SPureza:97.79% - 98.07%Cor e Forma:SolidPeso molecular:401.89
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