GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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Jatrorrhizine chloride
CAS:<p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>Fórmula:C20H20ClNO4Pureza:99.79%Cor e Forma:SolidPeso molecular:373.8Trazpiroben
CAS:<p>Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.</p>Fórmula:C31H39N3O4Pureza:99.41% - >99.99%Cor e Forma:SolidPeso molecular:517.66Citalopram
CAS:<p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>Fórmula:C20H21FN2OPureza:99.78% - 99.89%Cor e Forma:SolidPeso molecular:324.39Syk Inhibitor II
CAS:<p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>Fórmula:C14H15F3N6OPureza:97.63%Cor e Forma:SolidPeso molecular:340.3Ropinirole
CAS:<p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>Fórmula:C16H24N2OPureza:99.68%Cor e Forma:SolidPeso molecular:260.38R 59-022
CAS:<p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>Fórmula:C27H26FN3OSPureza:98.55%Cor e Forma:SolidPeso molecular:459.58L-745870
CAS:<p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>Fórmula:C18H19ClN4Pureza:98%Cor e Forma:SolidPeso molecular:326.82SR59230A hydrochloride
CAS:<p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>Fórmula:C21H28ClNO2Pureza:99.49%Cor e Forma:SolidPeso molecular:361.91PACAP (1-38), human, ovine, rat
CAS:<p>PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.</p>Fórmula:C203H331N63O53SPureza:96.93% - 98.16%Cor e Forma:SolidPeso molecular:4534.26Travoprost
CAS:<p>Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.</p>Fórmula:C26H35F3O6Pureza:97.39% - 99.58%Cor e Forma:Colorless OilPeso molecular:500.55Cyproheptadine hydrochloride
CAS:<p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>Fórmula:C21H21N·HClPureza:99.88% - 99.97%Cor e Forma:SolidPeso molecular:323.86Arazasetron HCl
CAS:<p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>Fórmula:C17H20ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:349.81GPR183-IN-1
CAS:<p>GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.</p>Fórmula:C16H19BrN2O2Cor e Forma:SolidPeso molecular:351.24Metoxibutropate
CAS:<p>Metoxibutropate is a biochemical.</p>Fórmula:C20H24O3Cor e Forma:SolidPeso molecular:312.417-phenyl trinor Prostaglandin F2α isopropyl ester
CAS:<p>17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the Allergan</p>Fórmula:C26H38O5Cor e Forma:SolidPeso molecular:430.58Risperidone Mesylate
CAS:<p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>Fórmula:C24H31FN4O5SPureza:98%Cor e Forma:SolidPeso molecular:506.59Escitalopram
CAS:<p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>Fórmula:C20H21FN2OPureza:99.82%Cor e Forma:White Or White Crystalline PowderPeso molecular:324.39N-Methyl amisulpride
CAS:<p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>Fórmula:C18H29N3O4SCor e Forma:SolidPeso molecular:383.51Keto Ziprasidone
CAS:<p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>Fórmula:C21H19ClN4O2SPureza:98%Cor e Forma:SolidPeso molecular:426.92Fremanezumab
CAS:<p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>Pureza:95% - 95%Cor e Forma:LiquidCarlumab
CAS:<p>Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.</p>Pureza:95%Cor e Forma:LiquidUliledlimab
CAS:<p>Uliledlimab, a humanized monoclonal antibody against CD73, reduces extracellular adenosine production and modulates immunosuppressive pathways.</p>Pureza:95% - 95%Cor e Forma:LiquidMeticillin
CAS:<p>Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.</p>Fórmula:C17H20N2O6SCor e Forma:SolidPeso molecular:380.42Triflupromazine
CAS:<p>Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.</p>Fórmula:C18H19F3N2SCor e Forma:SolidPeso molecular:352.42PF-610355
CAS:<p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>Fórmula:C34H39N3O6SPureza:99.73%Cor e Forma:SolidPeso molecular:617.76Olopatadine
CAS:<p>Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.</p>Fórmula:C21H23NO3Pureza:98%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:337.41Tulobuterol
CAS:<p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>Fórmula:C12H18ClNOCor e Forma:Crystalline SolidPeso molecular:227.73Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Cor e Forma:LiquidMethaphenilene hydrochloride
CAS:<p>Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.</p>Fórmula:C15H21ClN2SPureza:99.84%Cor e Forma:SolidPeso molecular:296.86Mibavademab
CAS:<p>Mibavademab is a humanized anti-leptin receptor (LEPR) mAb under investigation for treating congenital leptin deficiency.</p>Pureza:95%Cor e Forma:LiquidP2Y14R antagonist 1
CAS:<p>P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.</p>Fórmula:C15H12BrN3O2Pureza:98.88%Cor e Forma:SolidPeso molecular:346.18DL-Phenylephrine HCl
CAS:<p>DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.</p>Fórmula:C9H14ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:203.67Eptinezumab
CAS:<p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>Pureza:95% - 95%Cor e Forma:LiquidBuflomedil
CAS:<p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>Fórmula:C17H25NO4Pureza:98%Cor e Forma:SolidPeso molecular:307.38Cinnarizine D8
CAS:<p>Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.</p>Fórmula:C26H28N2Pureza:98%Cor e Forma:SolidPeso molecular:376.573Brexpiprazole-d8
CAS:<p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>Fórmula:C25H27N3O2SPureza:98%Cor e Forma:SolidPeso molecular:441.6215-keto Prostaglandin F2α
CAS:<p>15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.</p>Fórmula:C20H32O5Pureza:98%Cor e Forma:SolidPeso molecular:352.47Mirtazapine D3
CAS:<p>Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .</p>Fórmula:C17H19N3Pureza:98%Cor e Forma:SolidPeso molecular:268.37Dapagliflozin-d5
CAS:Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Fórmula:C21H25ClO6Pureza:98%Cor e Forma:SolidPeso molecular:413.9Amitriptyline-d6 Hydrochloride
CAS:<p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>Fórmula:C20H18D6ClNCor e Forma:SolidPeso molecular:319.90Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Fórmula:C18H29NO2H2O4SPureza:98.55%Cor e Forma:SolidPeso molecular:340.47Amthamine
CAS:<p>Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.</p>Fórmula:C6H11N3SCor e Forma:SoildPeso molecular:157.24Diclofensine
CAS:<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Fórmula:C17H17Cl2NOPureza:97.01% - 98.13%Cor e Forma:SolidPeso molecular:322.237-Desmethyl-3-hydroxyagomelatine
CAS:<p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>Fórmula:C14H15NO3Pureza:98%Cor e Forma:SolidPeso molecular:245.275-Methyltryptamine hydrochloride
CAS:<p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>Fórmula:C11H15ClN2Pureza:99.45%Cor e Forma:SolidPeso molecular:210.703Amidephrine hydrochloride
CAS:<p>Amidephrine hydrochloride is a biochemical.</p>Fórmula:C10H17ClN2O3SCor e Forma:SolidPeso molecular:280.77Ketanserinol
CAS:<p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>Fórmula:C22H24FN3O3Cor e Forma:SolidPeso molecular:397.44(RS)-ICI-118551 Hydrochloride
CAS:<p>ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3</p>Fórmula:C17H27NO2·HClPureza:98.02%Cor e Forma:SolidPeso molecular:313.86Roxatidine acetate
CAS:<p>Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.</p>Fórmula:C19H28N2O4Pureza:98%Cor e Forma:White Or Off-White PowderPeso molecular:348.44Litorin
CAS:<p>Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.</p>Fórmula:C51H68N14O11SCor e Forma:White PowderPeso molecular:1085.24Vanoxerine
CAS:<p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>Fórmula:C28H32F2N2OPureza:98%Cor e Forma:SolidPeso molecular:450.56Isoproterenol sulfate anhydrous
CAS:<p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>Fórmula:C22H36N2O10SPureza:98%Cor e Forma:CoaPeso molecular:520.59Tivumecirnon
CAS:<p>Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumour</p>Fórmula:C24H27Cl2F3N6OPureza:99.88%Cor e Forma:SolidPeso molecular:543.41Ciproxifan
CAS:<p>Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).</p>Fórmula:C16H18N2O2Pureza:98.00%Cor e Forma:SolidPeso molecular:270.33Dehydroabiethylamine
CAS:<p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.</p>Fórmula:C20H31NPureza:98.79%Cor e Forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecular:285.47R-138727
CAS:<p>R-138727 is a novel P2Y12 receptor inhibitor.</p>Fórmula:C18H20FNO3SPureza:98%Cor e Forma:SolidPeso molecular:349.42Hydroxy ziprasidone
CAS:<p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>Fórmula:C21H21ClN4O2SPureza:98%Cor e Forma:SolidPeso molecular:428.94MK-447
CAS:<p>MK-447 is a nonsteroidal antiinflammatory agent.</p>Fórmula:C11H16INOPureza:98%Cor e Forma:SolidPeso molecular:305.16S 25585
CAS:<p>S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Fórmula:C22H23F3N4O6SPureza:98%Cor e Forma:SolidPeso molecular:528.5Amidephrine
CAS:<p>Amidephrine is an adrenergic agent.</p>Fórmula:C10H16N2O3SCor e Forma:SolidPeso molecular:244.31Atenolol Hydrochloride
CAS:<p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>Fórmula:C14H23ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:302.80Norreticuline
CAS:<p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>Fórmula:C18H21NO4Cor e Forma:SolidPeso molecular:315.36Ticlopidine
CAS:<p>Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.</p>Fórmula:C14H14ClNSPureza:99.67%Cor e Forma:SolidPeso molecular:263.79Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Fórmula:C12H15N3O2Pureza:98%Cor e Forma:SolidPeso molecular:233.27Caerulein, desulfated
CAS:<p>Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.</p>Fórmula:C58H73N13O18SPureza:99.46%Cor e Forma:SolidPeso molecular:1272.34Ridazolol HCl
CAS:<p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>Fórmula:C15H19Cl3N4O3Pureza:99.48%Cor e Forma:SoildPeso molecular:409.7SB 271046 hydrochloride
CAS:<p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.</p>Fórmula:C20H22ClN3O3S2·HClPureza:99.77%Cor e Forma:SolidPeso molecular:488.45Itopride free base
CAS:<p>Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.</p>Fórmula:C20H26N2O4Cor e Forma:WhitePeso molecular:358.437-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene
CAS:<p>7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).</p>Fórmula:C42H44N2O6SPureza:98%Cor e Forma:SolidPeso molecular:704.87Paroxetine hydrochloride hemihydrate
CAS:<p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>Fórmula:C38H44Cl2F2N2O7Pureza:99.949%Cor e Forma:SolidPeso molecular:749.67Dolasetron Mesylate
CAS:<p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>Fórmula:C20H24N2O6SPureza:99.05%Cor e Forma:White PowderPeso molecular:420.48LY 344864
CAS:<p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>Fórmula:C21H22FN3OPureza:98%Cor e Forma:SolidPeso molecular:351.42MK-5046
CAS:<p>MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).</p>Fórmula:C20H18F6N4OPureza:98.56%Cor e Forma:SolidPeso molecular:444.37Lodoxamide tromethamine
CAS:<p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>Fórmula:C19H28ClN5O12Pureza:98.8%Cor e Forma:SolidPeso molecular:553.91Guacetisal
CAS:<p>Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.</p>Fórmula:C16H14O5Pureza:99.18%Cor e Forma:SolidPeso molecular:286.282-Iodomelatonin
CAS:<p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.</p>Fórmula:C13H15IN2O2Pureza:99.7%Cor e Forma:SolidPeso molecular:358.17Chlorazanil
CAS:<p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>Fórmula:C9H8ClN5Pureza:98.89%Cor e Forma:SolidPeso molecular:221.65RUSKI-201
CAS:<p>RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.</p>Fórmula:C20H27N3OSCor e Forma:SolidPeso molecular:357.51GAT228
CAS:<p>GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].</p>Fórmula:C22H18N2O2Cor e Forma:SolidPeso molecular:342.39Quinpirole Hydrochloride
CAS:<p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>Fórmula:C13H22ClN3Pureza:98%Cor e Forma:SolidPeso molecular:255.79H3R-IN-1 Hydrochloride
CAS:<p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>Fórmula:C19H24ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:377.86PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Fórmula:C14H12F3NOSPureza:98%Cor e Forma:SolidPeso molecular:299.31KW-8232
CAS:<p>KW-8232, an orally active anti-osteoporotic agent, reduces the biosynthesis of PGE2[1].</p>Fórmula:C37H41ClN4O6SCor e Forma:SolidPeso molecular:705.27Hexoprenaline
CAS:<p>Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.</p>Fórmula:C22H32N2O6Cor e Forma:SolidPeso molecular:420.5CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Fórmula:C18H20N6Cor e Forma:SolidPeso molecular:320.39MRS2603
CAS:<p>MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.</p>Fórmula:C14H12ClN4O8PPureza:98%Cor e Forma:SolidPeso molecular:430.69Org-12962
CAS:<p>Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).</p>Fórmula:C10H11ClF3N3Pureza:98.34%Cor e Forma:SolidPeso molecular:265.66Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.535-Carboxamidotryptamine maleate
CAS:<p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>Fórmula:C15H17N3O5Pureza:99.88%Cor e Forma:SolidPeso molecular:319.31Mirisetron
CAS:<p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>Fórmula:C24H31N3O2Pureza:99.88%Cor e Forma:SolidPeso molecular:393.52O-2093
CAS:<p>anandamide uptake inhibitor</p>Fórmula:C34H43Cl2NO3Pureza:98%Cor e Forma:SolidPeso molecular:584.622-ThioUTP tetrasodium salt
CAS:<p>2-ThioUTP tetrasodium salt is a P2Y2 agonist.</p>Fórmula:C9H15N2O14P3SPureza:98%Cor e Forma:SolidPeso molecular:500.21ICI 162,846
CAS:<p>ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.</p>Fórmula:C11H17F3N6OPureza:97.45%Cor e Forma:SolidPeso molecular:306.29MK761
CAS:<p>MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.</p>Fórmula:C13H19N3O2Cor e Forma:SolidPeso molecular:249.31NPC 17731
CAS:<p>NPC 17731 is a bradykinin receptor antagonist.</p>Fórmula:C59H95N19O14Cor e Forma:SolidPeso molecular:1294.5PRX-08066 Maleic acid
CAS:<p>PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.</p>Fórmula:C23H21ClFN5O4SPureza:97.59%Cor e Forma:SolidPeso molecular:517.96Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Fórmula:C20H25BrN4OCor e Forma:SolidPeso molecular:417.34Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Fórmula:C22H26ClNPureza:98%Cor e Forma:SolidPeso molecular:339.9GSK334429
CAS:<p>GSK334429 is an antagonist of histamine H3 receptor.</p>Fórmula:C20H29F3N4OCor e Forma:SolidPeso molecular:398.47GB-110
CAS:<p>GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.</p>Fórmula:C33H48N6O5Pureza:98%Cor e Forma:SolidPeso molecular:608.77
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