
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Fórmula:C18H23ClIN3O3SPureza:98%Cor e Forma:SolidPeso molecular:523.82Clothixamide
CAS:Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.Fórmula:C24H28ClN3OSPureza:95.51%Cor e Forma:SolidPeso molecular:442.02RS 52367
CAS:<p>RS 52367 is a beta-adrenergic antagonist.</p>Fórmula:C18H34ClN3O3SCor e Forma:SolidPeso molecular:408Lergotrile
CAS:<p>Lergotrile is used as an enzyme Inhibitor (Prolactin).</p>Fórmula:C17H18ClN3Pureza:98%Cor e Forma:SolidPeso molecular:299.8L 10503
CAS:L 10503 is an antifertility agent.Fórmula:C17H15N3OPureza:98%Cor e Forma:SolidPeso molecular:277.32FAUC-3019
CAS:<p>FAUC-3019 is a partial agonist of the dopamine D(4) receptor.</p>Fórmula:C22H24N2OCor e Forma:SolidPeso molecular:332.44ABT-299
CAS:<p>ABT-299 is a prodrug of A-85783.</p>Fórmula:C32H28ClFN4O4SCor e Forma:SolidPeso molecular:619.11Butidrine
CAS:<p>Butidrine has an Antiarrhythmic activities.</p>Fórmula:C16H25NOPureza:98%Cor e Forma:SolidPeso molecular:247.38A457
CAS:<p>A457 is an antagonist of the prokineticin receptor.</p>Fórmula:C26H33ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:457WS 009B
CAS:WS 009B is an antagonist of the endothelin receptor.Fórmula:C24H25NO11SPureza:98%Cor e Forma:SolidPeso molecular:535.52SB 268262
CAS:<p>CGRP1 antagonist</p>Fórmula:C18H15N3O4S2Pureza:98%Cor e Forma:SolidPeso molecular:401.46Losmiprofen
CAS:<p>Losmiprofen is a nonsteroidal compound of antiinflammatory.</p>Fórmula:C17H15ClO4Pureza:98%Cor e Forma:SolidPeso molecular:318.75Cafaminol
CAS:<p>Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.</p>Fórmula:C11H17N5O3Cor e Forma:SolidPeso molecular:267.28DAT 582
CAS:<p>DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent</p>Fórmula:C22H28ClN5OPureza:98%Cor e Forma:SolidPeso molecular:413.95Daglutril
CAS:<p>Daglutril is a NEP/ECE inhibitor for treating hypertension, heart failure, and pulmonary issues, blocking big endothelin-1 conversion.</p>Fórmula:C31H38N2O6Cor e Forma:SolidPeso molecular:534.64(-)-S-Timolol
CAS:<p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>Fórmula:C13H26N4O4SCor e Forma:SolidPeso molecular:334.44Opiranserin
CAS:<p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>Fórmula:C21H34N2O5Pureza:98%Cor e Forma:SolidPeso molecular:394.51Levoprotiline hydrochloride
CAS:<p>Levoprotiline hydrochloride is an antidepressant.</p>Fórmula:C20H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:329.86Tranterol hydrochloride
CAS:<p>Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.</p>Fórmula:C13H19Cl2F3N2OPureza:98%Cor e Forma:SolidPeso molecular:347.2LUF5831
CAS:<p>LUF5831 is an agonist of adenosine A1 receptor.</p>Fórmula:C15H12N4O2SCor e Forma:SolidPeso molecular:312.35BE 2254
CAS:<p>BE 2254 is an antagonist of central noradrenergic receptor.</p>Fórmula:C19H21NO2Cor e Forma:SolidPeso molecular:295.38Amitifadine free base
CAS:<p>Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.</p>Fórmula:C11H11Cl2NCor e Forma:SolidPeso molecular:228.12LG 82-4-00
CAS:<p>LG 82-4-00 is an inhibitor of thromboxane.</p>Fórmula:C10H11ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:274.72AHR-13268D
CAS:<p>AHR-13268D is a new agent of antiallergic/antihistaminic.</p>Fórmula:C28H29F2NNaO4Pureza:98%Cor e Forma:SolidPeso molecular:504.53NVP-QAV-680
CAS:<p>NVP-QAV-680: Powerful, selective CRTh2 antagonist with nM potency inhibiting eosinophil/Th2 activation.</p>Fórmula:C18H18N2O4SPureza:98%Cor e Forma:SolidPeso molecular:358.41S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Fórmula:C16H20ClN3OSCor e Forma:SolidPeso molecular:337.87A 69024
CAS:<p>A 69024 is a highly selective antagonist of dopamine D-1 receptor.</p>Fórmula:C20H24BrNO4Pureza:98%Cor e Forma:SolidPeso molecular:422.31SB 272183
CAS:<p>SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.</p>Fórmula:C29H28ClN5OPureza:98%Cor e Forma:SolidPeso molecular:498.02Sch 24518
CAS:<p>Sc h24518 is an antagonist of D1 receptor.</p>Fórmula:C16H17BrClNOPureza:98%Cor e Forma:SolidPeso molecular:354.67SKF-83822
CAS:<p>SKF-83822 is an agonist of dopamine D1-like receptor.</p>Fórmula:C20H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:343.85Iprindole
CAS:<p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>Fórmula:C19H28N2Pureza:99.54%Cor e Forma:SolidPeso molecular:284.44WAY 161503 hydrochloride
CAS:<p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>Fórmula:C11H12Cl3N3OPureza:98%Cor e Forma:SolidPeso molecular:308.59Cicloprolol hydrochloride
CAS:<p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>Fórmula:C18H30ClNO4Pureza:97.26%Cor e Forma:SolidPeso molecular:359.89Bamirastine
CAS:<p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>Fórmula:C31H37N5O3Pureza:96.68%Cor e Forma:SolidPeso molecular:527.66PAF-AN-1
CAS:<p>PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of anaphylactic death.</p>Fórmula:C28H28N2O3Pureza:98.06%Cor e Forma:SolidPeso molecular:440.53TD-5471 hydrochloride
CAS:<p>TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (</p>Fórmula:C32H32ClN3O4Pureza:99.57%Cor e Forma:SolidPeso molecular:558.07Pitolisant oxalate
CAS:<p>Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Fórmula:C19H28ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:385.88Quinpirole Hydrochloride
CAS:<p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>Fórmula:C13H22ClN3Pureza:98%Cor e Forma:SolidPeso molecular:255.79PF-03654764
CAS:<p>PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.</p>Fórmula:C20H28F2N2OPureza:>99.99%Cor e Forma:SolidPeso molecular:350.45Methdilazine Hydrochloride
CAS:<p>Methdilazine Hydrochloride (Bristaline) is a histamine H1 receptor antagonist for dermatologic conditions and relief of itching by allergies or rhinitis.</p>Fórmula:C18H21ClN2SCor e Forma:Light-Tan Crystalline Powder 4 8-6 (Ntp 1992)Peso molecular:332.89COR 170
CAS:<p>inverse agonist of CB2 receptors</p>Fórmula:C31H36N2O2Pureza:98%Cor e Forma:SolidPeso molecular:468.63GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Cor e Forma:SolidPeso molecular:377.48Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Fórmula:C17H20N4O2Pureza:99.97%Cor e Forma:SolidPeso molecular:312.37Niperotidine
CAS:<p>Niperotidine is an antagonist of histamine H2-receptor.</p>Fórmula:C20H26N4O5SPureza:98%Cor e Forma:SolidPeso molecular:434.51FR-194921
CAS:<p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>Fórmula:C23H23N5OCor e Forma:SolidPeso molecular:385.46RP101442
CAS:<p>RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).</p>Fórmula:C23H22N4O3Cor e Forma:SolidPeso molecular:402.45SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Fórmula:C18H20ClNO2Pureza:98.68%Cor e Forma:SolidPeso molecular:317.81EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Fórmula:C24H31N3O2Pureza:95.64% - 99.39%Cor e Forma:SolidPeso molecular:393.522mPGES-1 Inhibitor-1
CAS:<p>mPGES-1 Inhibitor-1 is an mPGES-1 inhibitor with anti-inflammatory and analgesic activity, which can be used to study acute liver injury.</p>Fórmula:C16H19ClN4O2Pureza:96.84% - 98.75%Cor e Forma:SolidPeso molecular:334.8(S)-(-)-Propranolol hydrochloride
CAS:<p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>Fórmula:C16H22ClNO2Pureza:99.02% - 99.91%Cor e Forma:SolidPeso molecular:295.8Befetupitant
CAS:<p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>Fórmula:C29H29F6N3O2Pureza:98.72%Cor e Forma:SolidPeso molecular:565.55Aminaftone
CAS:<p>Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.</p>Fórmula:C18H15NO4Pureza:96.31% - 99.39%Cor e Forma:SolidPeso molecular:309.32ABT-546
CAS:<p>ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.</p>Fórmula:C30H48N2O6Pureza:98%Cor e Forma:SolidPeso molecular:532.71CYM-5478
CAS:<p>CYM-5478, a strong S1P2 agonist, boosts C6 cell survival over 100nM under serum-starvation.</p>Fórmula:C21H19F3N2O2Pureza:98%Cor e Forma:SolidPeso molecular:388.38MK-4256
CAS:MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively).Fórmula:C27H23FN8OCor e Forma:SolidPeso molecular:494.52PG 01037 dihydrochloride
CAS:<p>PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.</p>Fórmula:C26H28Cl4N4OPureza:99.89%Cor e Forma:SolidPeso molecular:554.34CH 141
CAS:<p>CH 141 is a new type of peripheral vasodilator.</p>Fórmula:C19H21N3OCor e Forma:SolidPeso molecular:307.39Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Fórmula:C24H27Cl2FN6OPureza:98%Cor e Forma:SolidPeso molecular:505.42ZM 169369
CAS:<p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>Fórmula:C19H20N2SCor e Forma:SolidPeso molecular:308.44(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFórmula:C25H31FN4O3Pureza:97.79%Cor e Forma:SolidPeso molecular:454.54GPR183 antagonist-2
CAS:<p>GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].</p>Fórmula:C20H18F2N4O5Cor e Forma:SolidPeso molecular:432.38CP94253 hydrochloride
CAS:<p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>Fórmula:C15H20ClN3OPureza:99.78%Cor e Forma:SolidPeso molecular:293.79PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Fórmula:C20H22N4O3Pureza:98%Cor e Forma:SolidPeso molecular:366.41RS 15385-197
CAS:<p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>Fórmula:C18H26N2O3SCor e Forma:SolidPeso molecular:350.485-Carboxamidotryptamine maleate
CAS:<p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>Fórmula:C15H17N3O5Pureza:99.88%Cor e Forma:SolidPeso molecular:319.31DuP 734
CAS:<p>DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].</p>Fórmula:C17H23BrFNOCor e Forma:SolidPeso molecular:356.279QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Fórmula:C23H28N2O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:364.48Rocastine
CAS:<p>Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.</p>Fórmula:C13H19N3OSPureza:98.26%Cor e Forma:SolidPeso molecular:265.37RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Fórmula:C16H24Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:363.28H3 receptor-MO-1
CAS:<p>H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.</p>Fórmula:C20H27N3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:341.45Adenosine receptor inhibitor 2
CAS:<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Fórmula:C17H20BrN5O2Cor e Forma:SolidPeso molecular:406.28LBP-1
CAS:<p>LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.</p>Fórmula:C23H29ClN6O3Cor e Forma:SolidPeso molecular:472.97Seproxetine HCl
CAS:<p>Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.</p>Fórmula:C16H17ClF3NOPureza:98%Cor e Forma:SolidPeso molecular:331.76ER819762
CAS:<p>ER819762, an antagonist of the prostaglandin E2 EP4 receptor, inhibits Th1 differentiation and Th17 expansion.</p>Fórmula:C30H39N3O3Cor e Forma:SolidPeso molecular:489.65Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Fórmula:C26H32N2O7Cor e Forma:SolidPeso molecular:484.549Phenindamine
CAS:<p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>Fórmula:C19H19NCor e Forma:SolidPeso molecular:261.36Eplivanserin hemifumarate
CAS:<p>Eplivanserin is an inverse agonist of 5-HT2A.</p>Fórmula:C23H25FN2O6Cor e Forma:SolidPeso molecular:444.45KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Fórmula:C26H32N2O4Cor e Forma:SolidPeso molecular:436.54Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Fórmula:C15H23Cl3N6Pureza:98%Cor e Forma:SolidPeso molecular:393.74Tilisolol HCl
CAS:<p>Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.</p>Fórmula:C17H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:340.85GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93LP 20 hydrochloride
CAS:<p>ligand of the 5-HT7 receptor</p>Fórmula:C17H21ClN2OPureza:98%Cor e Forma:SolidPeso molecular:304.81Usmarapride free base
CAS:<p>Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.</p>Fórmula:C21H29N5O2Pureza:99.91% - 99.91%Cor e Forma:SolidPeso molecular:383.49LY 25648
CAS:<p>LY 25648 is an antagonist of leukotriene B4.</p>Fórmula:C19H27NO2SCor e Forma:SolidPeso molecular:333.49GW-876167
CAS:<p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>Fórmula:C16H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:315.37Asperlicin D
CAS:<p>Asperlicin D is a cholecystokinin antagonist agent.</p>Fórmula:C25H18N4O2Pureza:98%Cor e Forma:SolidPeso molecular:406.44Org-12962
CAS:<p>Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).</p>Fórmula:C10H11ClF3N3Pureza:98.34%Cor e Forma:SolidPeso molecular:265.66Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Fórmula:C22H24ClN3OPureza:99.35%Cor e Forma:White Crystal PowderPeso molecular:381.90JTH-601 free base
CAS:<p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>Fórmula:C24H35NO4Pureza:98%Cor e Forma:SolidPeso molecular:401.54Ro 04-6790 dihydrochloride
CAS:<p>Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.</p>Fórmula:C12H18Cl2N6O2SPureza:98%Cor e Forma:SolidPeso molecular:381.28HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Fórmula:C21H21FN2O3Pureza:98%Cor e Forma:SolidPeso molecular:368.4CB1R Allosteric modulator 1
CAS:<p>CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.</p>Fórmula:C24H24ClN3OCor e Forma:SolidPeso molecular:405.92ICI 162,846
CAS:<p>ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.</p>Fórmula:C11H17F3N6OPureza:97.45%Cor e Forma:SolidPeso molecular:306.29TAS 205
CAS:<p>TAS 205 blocks H-PGDS (IC50= 55.8 nM), beats L-PGDS at 100 μM. Reduces PGD2 in human/rat basophils, dampens allergy in guinea pigs (30 mg/kg).</p>Fórmula:C27H38N6O5Cor e Forma:SolidPeso molecular:526.638Octahydroisoindole
CAS:<p>Octahydroisoindole is a natural product and a reference standard.</p>Fórmula:C8H15NPureza:≥98%Cor e Forma:SolidPeso molecular:125.21CB1R Allosteric modulator 3
CAS:<p>CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.</p>Fórmula:C22H17ClN2O2Pureza:98.18%Cor e Forma:SolidPeso molecular:376.84(S)-Viloxazine Hydrochloride
CAS:<p>(S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.</p>Fórmula:C13H20ClNO3Pureza:99.95%Cor e Forma:SolidPeso molecular:273.76MG 1
CAS:<p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>Fórmula:C17H25N3O2Pureza:98.98% - >99.99%Cor e Forma:SolidPeso molecular:303.4Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Fórmula:C20H25ClN2OSCor e Forma:SolidPeso molecular:376.94OSU 6162 hydrochloride
CAS:Dopamine stabilizerFórmula:C15H24ClNO2SPureza:98%Cor e Forma:SolidPeso molecular:317.88
