GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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BI-6901
CAS:<p>BI-6901 is a CCR10 antagonist. In a mouse model of DNFB exposure hypersensitivity, BI 6901 displays its anti-inflammatory response in a dose-dependent manner.</p>Fórmula:C23H27N5O3SPureza:99.83%Cor e Forma:SolidPeso molecular:453.56Trimopam
CAS:Trimopam is a dopamine receptor agonist of the benzazepine group.Fórmula:C19H23NO2Cor e Forma:SolidPeso molecular:297.39GS 283
CAS:<p>GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.</p>Fórmula:C17H17NO3Cor e Forma:SolidPeso molecular:283.32CCR2 antagonist 3
CAS:<p>CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.</p>Fórmula:C17H25FN2O2Pureza:99.87%Cor e Forma:SolidPeso molecular:308.39NPS-2143
CAS:NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.Fórmula:C24H25ClN2O2Pureza:99.56%Cor e Forma:SolidPeso molecular:408.92CCR1 antagonist 9
CAS:<p>CCR1 antagonist 9 (compound 19e) is a selective CCR1 antagonist based on aziridine. CCR1 inhibition in calcium flux assays.</p>Fórmula:C20H16FN5O3SPureza:99.13%Cor e Forma:SolidPeso molecular:425.44Amgen-23
CAS:<p>Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.</p>Fórmula:C23H25Cl2N3O2SPureza:97.31%Cor e Forma:SolidPeso molecular:478.44FR 121196
CAS:<p>FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.</p>Fórmula:C12H16FN3O3SCor e Forma:SolidPeso molecular:301.34A23887
CAS:<p>A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.</p>Fórmula:C22H24ClNPureza:98%Cor e Forma:SolidPeso molecular:337.89SUN 1334H
CAS:<p>SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).</p>Fórmula:C23H28Cl2F2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:489.38Org41841
CAS:Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.Fórmula:C19H22N4O2S2Pureza:99.46% - 99.92%Cor e Forma:SolidPeso molecular:402.53Dipiproverine hydrochloride
CAS:<p>Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.</p>Fórmula:C20H32Cl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:403.39PAF-AN-1
CAS:<p>PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of anaphylactic death.</p>Fórmula:C28H28N2O3Pureza:98.06%Cor e Forma:SolidPeso molecular:440.53Resomelagon
CAS:<p>Resomelagon (AP1189), an oral melanocortin receptor agonist, triggers Ca2+ and ERK1/2 activation; useful in obesity and inflammation studies.</p>Fórmula:C14H14N6O2Cor e Forma:SolidPeso molecular:298.3GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Cor e Forma:SolidPeso molecular:377.48Bamirastine
CAS:<p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>Fórmula:C31H37N5O3Pureza:96.68%Cor e Forma:SolidPeso molecular:527.66Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Cor e Forma:SolidPeso molecular:282.81GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93CGS 12066B dimaleate
CAS:<p>5-HT1B full agonist</p>Fórmula:C25H25F3N4O8Pureza:98%Cor e Forma:SolidPeso molecular:566.48KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Fórmula:C26H32N2O4Cor e Forma:SolidPeso molecular:436.54Cicloprolol hydrochloride
CAS:<p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>Fórmula:C18H30ClNO4Pureza:97.26%Cor e Forma:SolidPeso molecular:359.89MLN3126
CAS:<p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>Fórmula:C21H19ClN2O5SCor e Forma:SolidPeso molecular:446.9Pancopride
CAS:<p>Pancopride（LAS 30451） is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced</p>Fórmula:C18H24ClN3O2Pureza:93.64%Cor e Forma:SolidPeso molecular:349.86H3R-IN-1 Hydrochloride
CAS:<p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>Fórmula:C19H24ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:377.86Clonidine
CAS:<p>Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.</p>Fórmula:C9H9Cl2N3Pureza:99.42% - 99.44%Cor e Forma:Crystals SolidPeso molecular:230.09Trifluperidol HCl
CAS:Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Fórmula:C22H24ClF4NO2Cor e Forma:SolidPeso molecular:445.88QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Fórmula:C23H28N2O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:364.48AS1069562
CAS:<p>AS1069562 inhibits 5-HT/NE reuptake, boosts IGF-1, FGF2 mRNA in dorsal root ganglia, spinal cord.</p>Fórmula:C20H23NO5SPureza:98%Cor e Forma:SolidPeso molecular:389.46GPR183 antagonist-2
CAS:<p>GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].</p>Fórmula:C20H18F2N4O5Cor e Forma:SolidPeso molecular:432.38PRX-08066 Maleic acid
CAS:<p>PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.</p>Fórmula:C23H21ClFN5O4SPureza:97.59%Cor e Forma:SolidPeso molecular:517.96Dexnafenodone Hydrochloride
CAS:<p>Dexnafenodone Hydrochloride is an adrenergic receptor antagonist and serotonin uptake inhibitor.</p>Fórmula:C20H24ClNOCor e Forma:SolidPeso molecular:329.86Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Fórmula:C19H17NO7Pureza:95% - 97.34%Cor e Forma:SolidPeso molecular:371.34LY 87130
CAS:<p>LY 87130 is a phenylethanolamine-N-methyltransferase inhibitor.</p>Fórmula:C12H13NPureza:98%Cor e Forma:SolidPeso molecular:171.24A3AR antagonist 2
CAS:<p>A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.</p>Fórmula:C22H16N6O3Cor e Forma:SolidPeso molecular:412.4PNU-177864
CAS:<p>PNU-177864 is a selective dopamine D3 receptor antagonist.</p>Fórmula:C18H21F3N2O3SPureza:99.92%Cor e Forma:SolidPeso molecular:402.43Rocastine
CAS:<p>Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.</p>Fórmula:C13H19N3OSPureza:98.26%Cor e Forma:SolidPeso molecular:265.37FAUC-3019
CAS:<p>FAUC-3019 is a partial agonist of the dopamine D(4) receptor.</p>Fórmula:C22H24N2OCor e Forma:SolidPeso molecular:332.44Iodophenpropit dihydrobromide
CAS:<p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>Fórmula:C15H20BrIN4SPureza:98%Cor e Forma:SolidPeso molecular:495.22H3 receptor-MO-1
CAS:<p>H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.</p>Fórmula:C20H27N3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:341.45MK-0249
CAS:<p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>Fórmula:C23H24F3N3O2Pureza:99.90%Cor e Forma:SolidPeso molecular:431.45Bopindolol
CAS:<p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.48Lergotrile
CAS:<p>Lergotrile is used as an enzyme Inhibitor (Prolactin).</p>Fórmula:C17H18ClN3Pureza:98%Cor e Forma:SolidPeso molecular:299.8KLS-13019
CAS:<p>KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).</p>Fórmula:C22H29NO3Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:355.47WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Fórmula:C17H20Cl2FN3O2SPureza:98.43%Cor e Forma:SolidPeso molecular:420.33GW-876167
CAS:<p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>Fórmula:C16H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:315.37(S)-Terazosin
CAS:<p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>Fórmula:C19H25N5O4Cor e Forma:SolidPeso molecular:387.43SB-221284
CAS:5-HT2C/2B receptor antagonistFórmula:C16H14F3N3OSPureza:98%Cor e Forma:SolidPeso molecular:353.36Licogliflozin
CAS:<p>Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).</p>Fórmula:C23H28O7Pureza:98%Cor e Forma:SolidPeso molecular:416.46Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Cor e Forma:SolidPeso molecular:328.38Tecalcet Hydrochloride
CAS:<p>Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.</p>Fórmula:C18H23Cl2NOPureza:99.97%Cor e Forma:SolidPeso molecular:340.29RPT193
CAS:RPT193 is an oral CCR4 inhibitor reducing Th2 cell migration in atopic dermatitis, asthma, and allergies.Fórmula:C27H34Cl3N5O2Cor e Forma:SolidPeso molecular:566.95MS-0022
CAS:<p>MS-0022: SMO antagonist, inhibits Hh signaling in nM-µM ranges, curbs tumor cell growth, and delays tumor progression in vivo.</p>Fórmula:C21H16BrN3OCor e Forma:SolidPeso molecular:406.28RS 52367
CAS:<p>RS 52367 is a beta-adrenergic antagonist.</p>Fórmula:C18H34ClN3O3SCor e Forma:SolidPeso molecular:408Fluphenazine Decanoate Dihydrochloride
CAS:<p>Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.</p>Fórmula:C32H46Cl2F3N3O2SPureza:98%Cor e Forma:SolidPeso molecular:664.69PGlu-3-methyl-His-Pro-NH2 TFA
<p>PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding & TSH release.</p>Fórmula:C19H25F3N6O6Pureza:98%Cor e Forma:SolidPeso molecular:490.43Etersalate
CAS:<p>Etersalate inhibits platelet function. It also reduces thromboxane A2 (TXA2) levels.</p>Fórmula:C19H19NO6Pureza:98%Cor e Forma:SolidPeso molecular:357.36RS 79948 hydrochloride
CAS:<p>α2-adrenoreceptor antagonist</p>Fórmula:C19H29ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:400.96Moprolol
CAS:<p>Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].</p>Fórmula:C13H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:239.31A-77636
CAS:<p>A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50</p>Fórmula:C20H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:329.43Trimazosin
CAS:<p>Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.</p>Fórmula:C20H29N5O6Cor e Forma:SolidPeso molecular:435.47Medroxalol
CAS:<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Fórmula:C20H24N2O5Cor e Forma:SolidPeso molecular:372.42ONO-2952
CAS:<p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>Fórmula:C22H20ClFN2O2Pureza:98%Cor e Forma:SolidPeso molecular:398.86Mrgx2 antagonist-1
CAS:Mrgx2 antagonist-1 is a potent antagonist of Mrgx2 (Mas-related Gene X2) and can be used to study Mrgx2-mediated diseases and disorders.Fórmula:C23H26F5N5O3Cor e Forma:SolidPeso molecular:515.48WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Fórmula:C14H18N2Pureza:98%Cor e Forma:SolidPeso molecular:214.31L 641953
CAS:<p>L 641953 is an antagonist of the thromboxane receptor.</p>Fórmula:C15H9FO3SCor e Forma:SolidPeso molecular:288.29Ifoxetine sulfate
CAS:<p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>Fórmula:C13H19NO2H2O4SPureza:98%Cor e Forma:SolidPeso molecular:270.34(R)-DOI hydrochloride
CAS:<p>(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.</p>Fórmula:C11H17ClINO2Pureza:99.88% - >99.99%Cor e Forma:SolidPeso molecular:357.62N-Methyldopamine hydrochloride
CAS:<p>N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.</p>Fórmula:C9H14ClNO2Cor e Forma:SolidPeso molecular:203.675-HT2A receptor agonist-2
CAS:<p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>Fórmula:C20H21ClN2O3Cor e Forma:SolidPeso molecular:372.85MAT2A-IN-3
CAS:<p>MAT2A-IN-3: potent MAT2A inhibitor, hinders MTAP-deficient cancer cell growth, potential for cancer research.</p>Fórmula:C24H16F5N5O3Cor e Forma:SolidPeso molecular:517.41Carcainium chloride
CAS:<p>Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.</p>Fórmula:C18H22ClN3O2Pureza:99.89%Cor e Forma:SolidPeso molecular:347.84Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Fórmula:C18H22BrNSPureza:99.65%Cor e Forma:SolidPeso molecular:364.34OMDM-6
CAS:<p>OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.</p>Fórmula:C28H42N2O3Pureza:99.66%Cor e Forma:SolidPeso molecular:454.64Napamezole
CAS:<p>Napamezole: α2 adrenergic receptor antagonist, blocks α1 in rat vas deferens (Kb 135 nM), reverses clonidine effects on twitch height.</p>Fórmula:C14H16N2Pureza:98%Cor e Forma:SolidPeso molecular:212.29L-692429
CAS:L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can be used to study acromegaly and obesity.Fórmula:C29H31N7O2Pureza:98.64% - 99.90%Cor e Forma:SolidPeso molecular:509.614(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Fórmula:C23H32N6O3SPureza:99.54%Cor e Forma:SolidPeso molecular:472.6Latanoprost ethyl amide
CAS:<p>Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.</p>Fórmula:C25H39NO4Cor e Forma:SolidPeso molecular:417.58Adatanserin
CAS:<p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>Fórmula:C21H31N5OPureza:99.33%Cor e Forma:SolidPeso molecular:369.5MM-22
CAS:<p>biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide</p>Fórmula:C36H60N4O5SPureza:98%Cor e Forma:SolidPeso molecular:660.95Hedgehog IN-3
CAS:<p>Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].</p>Fórmula:C18H13ClF3N5OCor e Forma:SolidPeso molecular:407.78Etoperidone hydrochloride
CAS:<p>Etoperidone hydrochloride is an antidepressant agent.</p>Fórmula:C19H29Cl2N5OCor e Forma:SolidPeso molecular:414.37CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Fórmula:C19H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:351.4Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Fórmula:C16H24Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:363.28Adenosine receptor inhibitor 2
CAS:<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Fórmula:C17H20BrN5O2Cor e Forma:SolidPeso molecular:406.28p-MPPF dihydrochloride
CAS:<p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>Fórmula:C25H29Cl2FN4O2Pureza:99.55%Cor e Forma:SolidPeso molecular:507.43E55888
CAS:<p>E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.</p>Fórmula:C16H23N3Cor e Forma:SolidPeso molecular:257.37Antiplatelet agent 2
CAS:<p>Antiplatelet agent 2 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.</p>Fórmula:C21H24F2N6O4SCor e Forma:SolidPeso molecular:494.51ST1936
CAS:<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Fórmula:C13H17ClN2Pureza:98%Cor e Forma:SolidPeso molecular:236.74Gyki 32887
CAS:<p>Gyki 32887 is a dopamine agonist.</p>Fórmula:C23H28N6O6SPureza:98%Cor e Forma:SolidPeso molecular:516.57PD 144418
CAS:<p>PD 144418 displays potential antipsychotic activity.</p>Fórmula:C18H22N2OPureza:98%Cor e Forma:SolidPeso molecular:282.38Povafonidine
CAS:<p>Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.</p>Fórmula:C11H13N5Cor e Forma:SolidPeso molecular:215.25SMO-IN-3
CAS:<p>SMO-IN-3: Strong SMO blocker, disrupts Hh pathway (IC50=34.09 nM), hinders Daoy cell growth, has anticancer properties.</p>Fórmula:C27H25F4N3O2Cor e Forma:SolidPeso molecular:499.5CB2 receptor agonist 3
CAS:<p>GP 2A is a selective agonist of CB2 receptor.</p>Fórmula:C24H23Cl2N3OCor e Forma:SolidPeso molecular:440.36S-777469
CAS:<p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>Fórmula:C23H27FN2O4Cor e Forma:SolidPeso molecular:414.47L748337
CAS:<p>L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.</p>Fórmula:C26H31N3O5SPureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:497.61(RS)-Minesapride
CAS:<p>Minesapride is a serotonin receptor agonist.</p>Fórmula:C21H31ClN4O5Pureza:98%Cor e Forma:SolidPeso molecular:454.95UCM-05194
CAS:<p>UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD 19.6 nM, inactive at LPA2-6/autotaxin).</p>Fórmula:C19H30BrO6PPureza:90% - 91.22%Cor e Forma:SolidPeso molecular:465.32EP2 receptor antagonist-1
CAS:<p>EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.</p>Fórmula:C24H22N4O5Cor e Forma:SolidPeso molecular:446.46PGN-9856
CAS:PGN-9856 is an EP2 receptor ligand and EP2 receptor agonist with anti-inflammatory and intraocular pressure-lowering properties, useful for glaucoma research.Fórmula:C21H15F2NO4Pureza:99.27%Cor e Forma:SolidPeso molecular:383.35
