GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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Bag-1
CAS:<p>Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.</p>Fórmula:C22H27N3Cor e Forma:SolidPeso molecular:333.47JNJ-17156516
CAS:<p>JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.</p>Fórmula:C26H22Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:481.37Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Fórmula:C23H21FN8OCor e Forma:SolidPeso molecular:444.46ZK-90055 hydrochloride
CAS:ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.Fórmula:C16H23ClN2O4Pureza:99.26%Cor e Forma:SolidPeso molecular:342.82Aminaftone
CAS:<p>Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.</p>Fórmula:C18H15NO4Pureza:96.31% - 99.39%Cor e Forma:SolidPeso molecular:309.32GCGR antagonist 2
CAS:<p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>Fórmula:C28H26N4O2Cor e Forma:SolidPeso molecular:450.53Ko-3290
CAS:<p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>Fórmula:C19H25N3O3Pureza:98%Cor e Forma:SolidPeso molecular:343.42GB-110
CAS:<p>GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.</p>Fórmula:C33H48N6O5Pureza:98%Cor e Forma:SolidPeso molecular:608.77GSK334429
CAS:<p>GSK334429 is an antagonist of histamine H3 receptor.</p>Fórmula:C20H29F3N4OCor e Forma:SolidPeso molecular:398.47Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Fórmula:C22H26ClNPureza:98%Cor e Forma:SolidPeso molecular:339.9Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Fórmula:C20H25BrN4OCor e Forma:SolidPeso molecular:417.34S-5751
CAS:<p>S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.</p>Fórmula:C25H31NO4SCor e Forma:SolidPeso molecular:441.58Imiloxan hydrochloride
CAS:<p>Imiloxan hydrochloride is an α2-adrenoceptor antagonist.</p>Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75Abanoquil
CAS:Abanoquil is an antagonist of alpha-1 adrenoceptor.Fórmula:C22H25N3O4Cor e Forma:SolidPeso molecular:395.45Gastrazole disodium
CAS:<p>Gastrazole, a CCK2 receptor antagonist, is used potentially for the treatment of pancreatic cancer.</p>Fórmula:C34H34FN5Na2O7Cor e Forma:SolidPeso molecular:689.652Tiamenidine
CAS:<p>Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.</p>Fórmula:C8H10ClN3SPureza:98%Cor e Forma:SolidPeso molecular:215.7Methylcarbamyl PAF C-16
CAS:<p>Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.</p>Fórmula:C26H55N2O7PCor e Forma:SolidPeso molecular:538.7JMV3002
CAS:<p>JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.</p>Fórmula:C35H34N6O3Cor e Forma:SolidPeso molecular:586.68PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Fórmula:C17H21N3Pureza:98%Cor e Forma:SolidPeso molecular:267.37AK-IN-1
CAS:<p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>Fórmula:C22H21N3O4Cor e Forma:SolidPeso molecular:391.42IMTPPE
CAS:<p>IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.</p>Fórmula:C20H27N3O2SCor e Forma:SolidPeso molecular:373.51Sequifenadine
CAS:<p>Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].</p>Fórmula:C22H27NOCor e Forma:SolidPeso molecular:321.46NPC 17731
CAS:<p>NPC 17731 is a bradykinin receptor antagonist.</p>Fórmula:C59H95N19O14Cor e Forma:SolidPeso molecular:1294.5MK761
CAS:<p>MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.</p>Fórmula:C13H19N3O2Cor e Forma:SolidPeso molecular:249.31CCG-271423
CAS:<p>CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.</p>Fórmula:C28H26N4O3Cor e Forma:SolidPeso molecular:466.53LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.41DMP 696
CAS:<p>DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.</p>Fórmula:C18H21Cl2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:410.3Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Fórmula:C18H29NO2Pureza:98%Cor e Forma:SolidPeso molecular:291.43Foscarbidopa
CAS:<p>Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.</p>Fórmula:C10H15N2O7PPureza:96.17% - 97.27%Cor e Forma:SolidPeso molecular:306.21Zinterol hydrochloride
CAS:<p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>Fórmula:C19H27ClN2O4SCor e Forma:SolidPeso molecular:414.952-ThioUTP tetrasodium salt
CAS:<p>2-ThioUTP tetrasodium salt is a P2Y2 agonist.</p>Fórmula:C9H15N2O14P3SPureza:98%Cor e Forma:SolidPeso molecular:500.21Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Fórmula:C25H27N3O5SPureza:98%Cor e Forma:SolidPeso molecular:481.56BI-L 239
CAS:BI-L 239 is an inhibition of 5-lipoxygenase products that cause bronchoconstriction.Fórmula:C16H15FOCor e Forma:SolidPeso molecular:242.29CCG-224406
CAS:<p>CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.</p>Fórmula:C29H27FN6O5Cor e Forma:SolidPeso molecular:558.565-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45PD 119819
CAS:PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.Fórmula:C21H25Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:438.35A-940894
CAS:<p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>Fórmula:C17H21N5Cor e Forma:SolidPeso molecular:295.38Guanoxabenz hydrochloride
CAS:<p>Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.</p>Fórmula:C8H9Cl3N4OCor e Forma:SolidPeso molecular:283.54Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.53Alprenolol tartrate, (S)-
CAS:<p>Alprenolol tartrate, (S)- is an 5-HT1A antagonist.</p>Fórmula:C19H29NO8Pureza:98%Cor e Forma:SolidPeso molecular:399.44Sultopride
CAS:<p>Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.</p>Fórmula:C17H26N2O4SCor e Forma:SolidPeso molecular:354.46GRK5-IN-4
CAS:<p>GRK5-IN-4: potent, selective covalent inhibitor of GRK5 (IC50=1.1 μM), 90x more specific than GRK2, useful for heart failure research.</p>Fórmula:C26H25N7O3Cor e Forma:SolidPeso molecular:483.52SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Cor e Forma:SolidPeso molecular:376.29(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Fórmula:C16H26BrNOPureza:98%Cor e Forma:SolidPeso molecular:328.29(Rac)-WAY-161503
CAS:<p>(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.</p>Fórmula:C11H11Cl2N3OPureza:99.51%Cor e Forma:SolidPeso molecular:272.13VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Fórmula:C21H15N3OCor e Forma:SolidPeso molecular:325.36Bufetolol
CAS:Bufetolol is an antagonist of beta-adrenoceptor.Fórmula:C18H29NO4Pureza:98%Cor e Forma:SolidPeso molecular:323.43AZD-1678
CAS:<p>AZD-1678 is a potent CCR4 receptor antagonist.</p>Fórmula:C11H8Cl2FN3O3SCor e Forma:SolidPeso molecular:352.17Kadsurenone
CAS:<p>Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.</p>Fórmula:C21H24O5Cor e Forma:SolidPeso molecular:356.41CP 96345
CAS:<p>CP 96345 is a NK1 receptor antagonist.</p>Fórmula:C28H32N2OPureza:98%Cor e Forma:SolidPeso molecular:412.573-epi-Vitamin D3
CAS:<p>3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM in</p>Fórmula:C27H44OCor e Forma:SolidPeso molecular:384.64Mosapramine
CAS:<p>Mosapramine is a dopamine D2-receptor antagonist.</p>Fórmula:C28H35ClN4OPureza:98%Cor e Forma:SolidPeso molecular:479.06Fenmetozole Tosylate
CAS:<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Fórmula:C17H18Cl2N2O4SPureza:98%Cor e Forma:SolidPeso molecular:417.31S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Fórmula:C22H29Cl2N3O2SCor e Forma:SolidPeso molecular:470.45GSK-345931A
CAS:<p>GSK-345931A is an EP(1) antagonist with CNS uptake in mice/rats, offering strong pain relief in acute and prolonged inflammation.</p>Fórmula:C22H20ClNNaO3Cor e Forma:SolidPeso molecular:404.85Agroclavine
CAS:<p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>Fórmula:C16H18N2Cor e Forma:SolidPeso molecular:238.33RUSKI-201
CAS:<p>RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.</p>Fórmula:C20H27N3OSCor e Forma:SolidPeso molecular:357.51SNT-207858 free base
CAS:<p>SNT-207858: selective MC-4 receptor antagonist, passes blood-brain barrier, orally active, IC50: 22 nM (binding), 11 nM (function).</p>Fórmula:C32H43Cl2N5O3Pureza:98%Cor e Forma:SolidPeso molecular:616.62ADRA1D receptor antagonist 1 free base
CAS:<p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>Fórmula:C15H13ClN4OCor e Forma:SolidPeso molecular:300.74MRS2179
CAS:<p>MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.</p>Fórmula:C11H17N5O9P2Cor e Forma:SolidPeso molecular:425.23CI 1020
CAS:<p>endothelin-A receptor (ETA) antagonist</p>Fórmula:C28H26O9Pureza:98%Cor e Forma:SolidPeso molecular:506.5Fonazine
CAS:<p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>Fórmula:C19H25N3O2S2Cor e Forma:SolidPeso molecular:391.55BMS-665053
CAS:<p>BMS-665053: CRF1 receptor antagonist, IC50 = 1.0 nM; inhibits cAMP in Y-79 cells, IC50 = 4.9 nM; anti-anxiety in rats, Cl = 17 mL/min/kg, t½ = 7.8 h.</p>Fórmula:C16H14Cl3F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:424.66Levobunolol
CAS:<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Fórmula:C17H25NO3Cor e Forma:White To Pink PowderPeso molecular:291.39B-HT 933 dihydrochloride
CAS:<p>Azepexole (B-HT 933) dihydrochloride is an α2-adrenoceptor agonist, pKi: 8.3/α2A, 7.6/α2B, 7.5/α2C; IC50: 78.72 nM for peristalsis inhibition.</p>Fórmula:C9H17Cl2N3OCor e Forma:SolidPeso molecular:254.16Broxaterol
CAS:<p>Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.</p>Fórmula:C9H15BrN2O2Pureza:98%Cor e Forma:SolidPeso molecular:263.13L 651142
CAS:<p>L 651142 is a weak inhibitor of the platelet-activating factor receptor. It is also binding to polymorphonuclear leukocytes.</p>Fórmula:C21H23NO4SCor e Forma:SolidPeso molecular:385.48CFM 1571 hydrochloride
CAS:<p>CFM 1571 hydrochloride stimulates sGC with EC50 of 5.49 μM; potential for cardiovascular research.</p>Fórmula:C23H29ClN4O3Cor e Forma:SolidPeso molecular:444.96Repinotan HCl
CAS:<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Fórmula:C21H25ClN2O4SPureza:99.57%Cor e Forma:SolidPeso molecular:436.95Atigliflozin
CAS:<p>Atigliflozin is an antihyperglycaemic drug candidate.</p>Fórmula:C18H22O7SCor e Forma:SolidPeso molecular:382.43Ro 363 hydrochloride
CAS:<p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>Fórmula:C19H26ClNO6Cor e Forma:SolidPeso molecular:399.87JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Fórmula:C20H28N2OPureza:98%Cor e Forma:SolidPeso molecular:312.45FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Fórmula:C27H29F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:465.53Pargolol hydrochloride
CAS:<p>Pargolol hydrochloride is an antagonist of β adrenergic receptor.</p>Fórmula:C16H24ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:313.82Octoclothepin maleate salt
CAS:<p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>Fórmula:C23H25ClN2O4SCor e Forma:SolidPeso molecular:460.97Substance P Receptor Antagonist 1
CAS:<p>Substance P Receptor Antagonist 1 may aid in treating GI, inflammatory, respiratory, and CNS disorders.</p>Fórmula:C24H29F3N2O2Pureza:98%Cor e Forma:SolidPeso molecular:434.49ICI 192605
CAS:<p>ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.</p>Fórmula:C22H23ClO5Cor e Forma:SolidPeso molecular:402.87AL-3138
CAS:<p>AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.</p>Fórmula:C20H33FO4Cor e Forma:SolidPeso molecular:356.47DW-1350
CAS:DW-1350 is an antagonist of LTB4 receptor.Fórmula:C25H31N3O3SPureza:98%Cor e Forma:SolidPeso molecular:453.6CCR8 antagonist 2
CAS:<p>CCR8 antagonist 2 blocks CCR8 activity, mainly on Treg and Th2 cells, for treating related diseases. See WO2022000443A1, compound 220.</p>Fórmula:C23H30ClN3O3SCor e Forma:SolidPeso molecular:464.02PQ-69
CAS:<p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>Fórmula:C20H19FN4OCor e Forma:SolidPeso molecular:350.39Autotaxin-IN-6
CAS:<p>Autotaxin-IN-6 is a strong ATX inhibitor with a 30 nM IC50, potentially aiding anticancer research by hindering cell migration.</p>Fórmula:C35H54BNO6Cor e Forma:SolidPeso molecular:595.62Izuforant
CAS:<p>Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).</p>Fórmula:C12H12BrN7Cor e Forma:SolidPeso molecular:334.17MK-8133
CAS:<p>MK-8133 is an antagonist of orexin-2 selective receptor with favorable development properties.</p>Fórmula:C23H21N5O2Cor e Forma:SolidPeso molecular:399.45A-943931
CAS:A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.Fórmula:C17H21N5Pureza:99.79%Cor e Forma:SolidPeso molecular:295.38BRL 37344 sodium
CAS:<p>BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.</p>Fórmula:C19H22ClNNaO4Pureza:98%Cor e Forma:SolidPeso molecular:386.83(Rac)-HAMI 3379
CAS:<p>HAMI 3379: potent CysLT2 receptor blocker; protects against acute/subacute brain injury; reduces microglia inflammation.</p>Fórmula:C34H45NO8Pureza:98%Cor e Forma:SolidPeso molecular:595.72QCC-374
CAS:<p>QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.</p>Fórmula:C28H33N3O2Pureza:98%Cor e Forma:SolidPeso molecular:443.58UK 1745
CAS:<p>UK 1745 is a novel drug of cardiotonic.</p>Fórmula:C16H23ClN2O2Cor e Forma:SolidPeso molecular:310.82Zenidolol
CAS:<p>Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.</p>Fórmula:C17H27NO2Cor e Forma:SolidPeso molecular:277.4CP-195543
CAS:<p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>Fórmula:C24H19F3O4Cor e Forma:SolidPeso molecular:428.4Guanethidine
CAS:<p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>Fórmula:C10H22N4Cor e Forma:SolidPeso molecular:198.31EP4 receptor antagonist 4
CAS:<p>EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].</p>Fórmula:C19H14N2OSCor e Forma:SolidPeso molecular:318.39SM-130686
CAS:<p>SM-130,686: orally-active GHSR agonist, 50% as potent as ghrelin in stimulating growth hormone.</p>Fórmula:C22H24Cl2F3N3O3Cor e Forma:SolidPeso molecular:506.355'-(N-Cyclopropyl)carboxamidoadenosine
CAS:<p>adenosine A2 receptor agonist</p>Fórmula:C13H16N6O4Pureza:98%Cor e Forma:SolidPeso molecular:320.35-HT7 agonist 2
CAS:<p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>Fórmula:C23H29N3OCor e Forma:SolidPeso molecular:363.5ROS 234
CAS:<p>ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.</p>Fórmula:C13H15N5Cor e Forma:SolidPeso molecular:241.29SDZ 21009
CAS:β-adrenoceptor and 5-HT1A/1B receptor antagonistFórmula:C19H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:348.44A 55453
CAS:<p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>Fórmula:C25H32N6O3Cor e Forma:SolidPeso molecular:464.56Adrenaline sulfate
CAS:<p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>Fórmula:C9H15NO7SCor e Forma:SolidPeso molecular:281.279
