
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(993 produtos)
- Receptor de adenosina(246 produtos)
- Receptor adrenérgico(3.004 produtos)
- Receptor de Bombesina(33 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(153 produtos)
- CaSR(33 produtos)
- Receptor de Canabinóides(212 produtos)
- Receptor de Dopamina(433 produtos)
- Receptor Endotelina(79 produtos)
- Receptor GNRH(77 produtos)
- GPCR19(32 produtos)
- GRK(32 produtos)
- GTPase(22 produtos)
- Receptor Glucagon(182 produtos)
- Hedgehog/Smoothened(47 produtos)
- Receptor de Histamina(381 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(26 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(310 produtos)
- PAFR(12 produtos)
- PKA(51 produtos)
- Receptor S1P(18 produtos)
- SGLT(31 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5745 produtos de "GPCR/Proteína-G"
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SDZ NKT 343
CAS:<p>human tachykinin NK1 receptor antagonist</p>Fórmula:C33H33N5O5Pureza:98%Cor e Forma:SolidPeso molecular:579.65L 741671
CAS:L 741671 is an antagonist of the neurokinin-1 receptor.Fórmula:C23H22F6N4O2Cor e Forma:SolidPeso molecular:500.44CB1R Allosteric modulator 2
CAS:<p>Compound 18 is a potent CB1R allosteric modulator that acts as a negative modulator (NAM) for CB1R orthosteric ligands.</p>Fórmula:C19H15ClFN3OCor e Forma:SolidPeso molecular:355.79Isothipendyl
CAS:Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.Fórmula:C16H19N3SCor e Forma:SolidPeso molecular:285.41RB-005
CAS:RB-005 is a potent SK1 inhibitor with IC(50) of 3.6 μM, potentially treating proliferative diseases like hypertension and degrades SK1 in human cells.Fórmula:C21H35NOCor e Forma:SolidPeso molecular:317.51UCSF686
CAS:UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.Fórmula:C14H19N3O2SCor e Forma:SolidPeso molecular:293.38Neladenoson dalanate HCl
CAS:Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).Fórmula:C35H35Cl2N7O4S2Pureza:98%Cor e Forma:SolidPeso molecular:752.73Sortilin antagonist 1
CAS:Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.Fórmula:C20H24N2O4Cor e Forma:SolidPeso molecular:356.42Antiplatelet agent 1
CAS:Antiplatelet agent 1 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.Fórmula:C21H24F2N6O4SCor e Forma:SolidPeso molecular:494.51CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Fórmula:C21H22N8O3Cor e Forma:SolidPeso molecular:434.45SSTR4 agonist 3
CAS:SSTR4 agonist 3 activates SSTR4 in the hippocampus and neocortex, aiding memory and learning, and shows potent pain relief in rodents.Fórmula:C18H24N4OSCor e Forma:SolidPeso molecular:344.47ATC0065 HCl
CAS:ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.Fórmula:C25H31BrCl2F3N5OCor e Forma:SolidPeso molecular:625.35Clencyclohexerol
CAS:Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.Fórmula:C14H20Cl2N2O2Cor e Forma:SolidPeso molecular:319.23SGS518 oxalate
CAS:SGS518 oxalate is a 5-HT6 antagonist.Fórmula:C23H24F2N2O7SPureza:98%Cor e Forma:SolidPeso molecular:510.51GLP-1R agonist 1
CAS:GLP-1R agonist 1, an imidazole derivative and potent GLP-1R activator, may aid diabetes research.Fórmula:C32H29ClFN3O5Cor e Forma:SolidPeso molecular:590.04(Rac)-SEP-363856
CAS:(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a uniqueFórmula:C9H13NOSPureza:98%Cor e Forma:SolidPeso molecular:183.27COR 170
CAS:<p>inverse agonist of CB2 receptors</p>Fórmula:C31H36N2O2Pureza:98%Cor e Forma:SolidPeso molecular:468.63ML233
CAS:<p>"ML233: potent apelin receptor agonist, EC50=3.7 μM, 21-fold selective over AT1 receptor."</p>Fórmula:C19H21NO4SCor e Forma:SolidPeso molecular:359.44Ketotifen
CAS:Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.Fórmula:C19H19NOSCor e Forma:SolidPeso molecular:309.43CB1/2 agonist 2
CAS:CB1/2 agonist 2 binds tightly to cannabinoid receptors, acting fully on CB1 and inversely on CB2.Fórmula:C26H43NO3Cor e Forma:SolidPeso molecular:417.62Pitolisant oxalate
CAS:Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.Fórmula:C19H28ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:385.88WAY 161503 hydrochloride
CAS:WAY 161503 hydrochloride is a 5-HT2C receptor agonist.Fórmula:C11H12Cl3N3OPureza:98%Cor e Forma:SolidPeso molecular:308.59SKF-83822
CAS:SKF-83822 is an agonist of dopamine D1-like receptor.Fórmula:C20H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:343.85MRS 1523
CAS:MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.Fórmula:C23H29NO3SPureza:98%Cor e Forma:SolidPeso molecular:399.55JNJ-26070109
CAS:JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.Fórmula:C23H17BrF2N4O3SPureza:98%Cor e Forma:SolidPeso molecular:547.37SUN-C5174
CAS:<p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>Fórmula:C22H29FN4O2Pureza:98%Cor e Forma:SolidPeso molecular:400.49Tertatolol
CAS:Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.Fórmula:C16H25NO2SPureza:98%Cor e Forma:SolidPeso molecular:295.44Resomelagon
CAS:Resomelagon (AP1189), an oral melanocortin receptor agonist, triggers Ca2+ and ERK1/2 activation; useful in obesity and inflammation studies.Fórmula:C14H14N6O2Cor e Forma:SolidPeso molecular:298.3ONO-2952
CAS:ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.Fórmula:C22H20ClFN2O2Pureza:98%Cor e Forma:SolidPeso molecular:398.86S-3608
CAS:S-3608 is an atypical dopamine agonist.Fórmula:C16H20ClN3OSCor e Forma:SolidPeso molecular:337.87Panamesine
CAS:Panamesine (EMD 57445) is a high affinity receptor ligand for sigma (IC50: 6 nM) with potential for atypical antipsychotic studies.Fórmula:C23H26N2O6Cor e Forma:SolidPeso molecular:426.46PGN36
CAS:<p>PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).</p>Fórmula:C21H23N3O3Cor e Forma:SolidPeso molecular:365.43Methapyrilene
CAS:Methapyrilene is a histamine H1 antagonist with sedative action.Fórmula:C14H19N3SCor e Forma:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)Peso molecular:261.39Repirinast
CAS:<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Fórmula:C20H21NO5Cor e Forma:SolidPeso molecular:355.38R 121919 hydrochloride
CAS:CRF1 antagonist with Ki=3.5 nM, lowers stress-induced ACTH, has anxiolytic and antidepressant effects, orally bioavailable.Fórmula:C22H33ClN6Cor e Forma:SolidPeso molecular:417.0L 760735
CAS:<p>L 760735 is a NK1 receptor antagonist.</p>Fórmula:C26H29ClF7N5O2Pureza:98%Cor e Forma:SolidPeso molecular:611.98FR260010
CAS:FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.Fórmula:C22H19N5Cor e Forma:SolidPeso molecular:353.42Trimazosin
CAS:Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.Fórmula:C20H29N5O6Cor e Forma:SolidPeso molecular:435.47SMO-IN-3
CAS:SMO-IN-3: Strong SMO blocker, disrupts Hh pathway (IC50=34.09 nM), hinders Daoy cell growth, has anticancer properties.Fórmula:C27H25F4N3O2Cor e Forma:SolidPeso molecular:499.5L-902688
CAS:L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).Fórmula:C21H27F2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:419.47CM572
CAS:CM572 is a selective putative sigma-2 antagonist.Fórmula:C22H23FN4O2SCor e Forma:SolidPeso molecular:426.51Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Cor e Forma:SolidPeso molecular:255.74FR-194921
CAS:FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.Fórmula:C23H23N5OCor e Forma:SolidPeso molecular:385.46RP101442
CAS:RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).Fórmula:C23H22N4O3Cor e Forma:SolidPeso molecular:402.45ZM 169369
CAS:ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.Fórmula:C19H20N2SCor e Forma:SolidPeso molecular:308.44Immepip
CAS:Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.Fórmula:C9H15N3Cor e Forma:SolidPeso molecular:165.24Phenyltoloxamine
CAS:Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).Fórmula:C17H21NOCor e Forma:SolidPeso molecular:255.35Prucalopride hydrochloride
CAS:Prucalopride hydrochloride is a selective agonist of the 5-HT4.Fórmula:C18H27Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:404.33(S)-SLV 319
CAS:Ibipinabant (SLV319), a potent CB1 antagonist, K i = 7.8 nM, >1000x selective over CB2, for obesity and diabetic research.Fórmula:C23H20Cl2N4O2SCor e Forma:SolidPeso molecular:487.4Primidolol
CAS:Primidolol is a beta adrenergic receptor antagonist and antihypertensive agent.Fórmula:C17H23N3O4Pureza:98%Cor e Forma:SolidPeso molecular:333.38COR167
CAS:<p>COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.</p>Fórmula:C28H38N2O2Cor e Forma:SolidPeso molecular:434.61MRS2395
CAS:MRS2395, a dipivaloyl P2Y12 receptor blocker, inhibits ADP-induced platelet activation with a Ki of 3.6 μM and boosts TRAP-6-triggered dense granule release.Fórmula:C20H30ClN5O4Cor e Forma:SolidPeso molecular:439.94PNU-177864 hydrochloride
CAS:<p>PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor.</p>Fórmula:C18H22ClF3N2O3SPureza:99.95%Cor e Forma:SolidPeso molecular:438.89Mizolastine dihydrochloride
CAS:Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).Fórmula:C24H27Cl2FN6OPureza:98%Cor e Forma:SolidPeso molecular:505.42CH 141
CAS:CH 141 is a new type of peripheral vasodilator.Fórmula:C19H21N3OCor e Forma:SolidPeso molecular:307.39CID1172084
CAS:CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Fórmula:C23H18FN5O2S2Cor e Forma:SolidPeso molecular:479.55MS012
CAS:MS012 is a Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase (Kd = 46 ± 15 nM).Fórmula:C22H35N5O2Cor e Forma:SolidPeso molecular:401.55GRK5-IN-3
CAS:GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5).GRK5-IN-3 significantly inhibits GRK5 (IC50: 0.22 μM) and GRK6 (IC50: 0.41 μM).Fórmula:C23H21N7O3Cor e Forma:SolidPeso molecular:443.46SSTR4 agonist 2
CAS:<p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41ASP-4058 hydrochloride
CAS:<p>ASP-4058 hydrochloride: selective oral S1P1/S1P5 agonist, safe, mitigates mouse autoimmune encephalomyelitis.</p>Fórmula:C19H13ClF6N4O2Cor e Forma:SolidPeso molecular:478.78GB-110
CAS:GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.Fórmula:C33H48N6O5Pureza:98%Cor e Forma:SolidPeso molecular:608.77GSK334429
CAS:GSK334429 is an antagonist of histamine H3 receptor.Fórmula:C20H29F3N4OCor e Forma:SolidPeso molecular:398.47Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Fórmula:C22H26ClNPureza:98%Cor e Forma:SolidPeso molecular:339.9Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Fórmula:C20H25BrN4OCor e Forma:SolidPeso molecular:417.34SKF-104557
CAS:<p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>Fórmula:C13H18N2OCor e Forma:SolidPeso molecular:218.29S-5751
CAS:S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.Fórmula:C25H31NO4SCor e Forma:SolidPeso molecular:441.58Methylcarbamyl PAF C-16
CAS:Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.Fórmula:C26H55N2O7PCor e Forma:SolidPeso molecular:538.7PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Fórmula:C17H21N3Pureza:98%Cor e Forma:SolidPeso molecular:267.37AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Fórmula:C22H21N3O4Cor e Forma:SolidPeso molecular:391.42SC 51089 free base
CAS:<p>SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.</p>Fórmula:C22H19ClN4O3Cor e Forma:SolidPeso molecular:422.86Metrenperone
CAS:Metrenperone is used as a S(2)-receptor blocker.Fórmula:C24H26FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:407.48Sequifenadine
CAS:Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].Fórmula:C22H27NOCor e Forma:SolidPeso molecular:321.46CCG-271423
CAS:CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.Fórmula:C28H26N4O3Cor e Forma:SolidPeso molecular:466.53LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.412-Thio-UTP
CAS:2-ThioUTP tetrasodium salt is a P2Y2 agonist.Fórmula:C9H15N2O14P3SPureza:98%Cor e Forma:SolidPeso molecular:500.21BMS-193884
CAS:BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.Fórmula:C20H17N3O4SCor e Forma:SolidPeso molecular:395.43O-2093
CAS:<p>anandamide uptake inhibitor</p>Fórmula:C34H43Cl2NO3Pureza:98%Cor e Forma:SolidPeso molecular:584.625-HT7 receptor ligand 1
CAS:Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45A-940894
CAS:A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.Fórmula:C17H21N5Cor e Forma:SolidPeso molecular:295.38Usmarapride
CAS:Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.53GRK5-IN-4
CAS:GRK5-IN-4: potent, selective covalent inhibitor of GRK5 (IC50=1.1 μM), 90x more specific than GRK2, useful for heart failure research.Fórmula:C26H25N7O3Cor e Forma:SolidPeso molecular:483.52MRS2603
CAS:MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.Fórmula:C14H12ClN4O8PPureza:98%Cor e Forma:SolidPeso molecular:430.69CAY10498
CAS:A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.Fórmula:C18H20N6Cor e Forma:SolidPeso molecular:320.39Hexoprenaline
CAS:Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.Fórmula:C22H32N2O6Cor e Forma:SolidPeso molecular:420.5KW-8232
CAS:<p>KW-8232, an orally active anti-osteoporotic agent, reduces the biosynthesis of PGE2[1].</p>Fórmula:C37H41ClN4O6SCor e Forma:SolidPeso molecular:705.27SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Fórmula:C19H22BrNO2Pureza:98%Cor e Forma:SolidPeso molecular:376.29AZD-1678
CAS:<p>AZD-1678 is a potent CCR4 receptor antagonist.</p>Fórmula:C11H8Cl2FN3O3SCor e Forma:SolidPeso molecular:352.17CP 96345
CAS:<p>CP 96345 is a NK1 receptor antagonist.</p>Fórmula:C28H32N2OPureza:98%Cor e Forma:SolidPeso molecular:412.573-epi-Vitamin D3
CAS:3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM inFórmula:C27H44OCor e Forma:SolidPeso molecular:384.64Fenmetozole Tosylate
CAS:<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Fórmula:C17H18Cl2N2O4SPureza:98%Cor e Forma:SolidPeso molecular:417.31S 14063
CAS:S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.Fórmula:C22H29Cl2N3O2SCor e Forma:SolidPeso molecular:470.45GSK-345931A
CAS:GSK-345931A is an EP(1) antagonist with CNS uptake in mice/rats, offering strong pain relief in acute and prolonged inflammation.Fórmula:C22H20ClNNaO3Cor e Forma:SolidPeso molecular:404.85Agroclavine
CAS:Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.Fórmula:C16H18N2Cor e Forma:SolidPeso molecular:238.33RUSKI-201
CAS:RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.Fórmula:C20H27N3OSCor e Forma:SolidPeso molecular:357.51ADRA1D receptor antagonist 1 free base
CAS:ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.Fórmula:C15H13ClN4OCor e Forma:SolidPeso molecular:300.74Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Fórmula:C19H25N3O2S2Cor e Forma:SolidPeso molecular:391.55Idremcinal
CAS:<p>Idremcinal is a motilin receptor agonist.</p>Fórmula:C39H69NO12Cor e Forma:SolidPeso molecular:743.96CCG-273463
CAS:<p>CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.</p>Fórmula:C26H25BrN4O3Cor e Forma:SolidPeso molecular:521.41Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Fórmula:C26H31FN2O4Pureza:98%Cor e Forma:SolidPeso molecular:454.53PD-156707
CAS:PD-156707 is a selective antagonist of endothelin A receptor.Fórmula:C28H26NaO9Pureza:98%Cor e Forma:SolidPeso molecular:529.497
