GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(1.025 produtos)
- Receptor de adenosina(249 produtos)
- Receptor adrenérgico(3.030 produtos)
- Receptor de Bombesina(35 produtos)
- Receptor de Bradicinina(61 produtos)
- CXCR(159 produtos)
- CaSR(34 produtos)
- Receptor de Canabinóides(217 produtos)
- Colecistocinina(1 produtos)
- Receptor de Dopamina(445 produtos)
- Receptor Endotelina(86 produtos)
- Receptor GNRH(84 produtos)
- GPCR19(33 produtos)
- GRK(33 produtos)
- GTPase(22 produtos)
- Receptor Glucagon(196 produtos)
- Hedgehog/Smoothened(49 produtos)
- Receptor de Histamina(385 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(26 produtos)
- Receptor OX(42 produtos)
- Receptor opioide(325 produtos)
- PAFR(14 produtos)
- PKA(58 produtos)
- Receptor S1P(17 produtos)
- SGLT(31 produtos)
- Receptor Sigma(46 produtos)
Exibir 19 mais subcategorias
Foram encontrados 5982 produtos de "GPCR/Proteína-G"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Alniditan dihydrochloride
CAS:Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.Fórmula:C17H28Cl2N4OCor e Forma:SolidPeso molecular:375.34GRK5-IN-3
CAS:GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5).GRK5-IN-3 significantly inhibits GRK5 (IC50: 0.22 μM) and GRK6 (IC50: 0.41 μM).Fórmula:C23H21N7O3Cor e Forma:SolidPeso molecular:443.46APC-3316 tosylate
CAS:APC-3316 tosylate is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.Fórmula:C39H46N4O7S2Cor e Forma:SolidPeso molecular:746.94ABT-546
CAS:ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.Fórmula:C30H48N2O6Pureza:98%Cor e Forma:SolidPeso molecular:532.71BGC201531
CAS:BGC201531 (AP-1531) is a EP4 antagonist for the treatment of acute migraine.
Fórmula:C26H28N2O6SPureza:98.51% - 99.33%Cor e Forma:SolidPeso molecular:496.58EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Fórmula:C15H22N2OPureza:97.66% - 99.78%Cor e Forma:SolidPeso molecular:246.35Ref: TM-T11183
1mg92,00€2mg125,00€5mg170,00€10mg213,00€25mg474,00€50mg688,00€100mg938,00€500mg1.882,00€1mL*10mM (DMSO)170,00€WIN 62,577
CAS:WIN 62,577 is a allosteric antagonist of mAChR.Fórmula:C29H31N3OPureza:98%Cor e Forma:SolidPeso molecular:437.58Esprolol hydrochloride
CAS:Esprolol is a β-adrenergic receptor antagonist.Fórmula:C17H28ClNO4Pureza:98%Cor e Forma:SolidPeso molecular:345.86T-0509
CAS:T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-
Fórmula:C18H23NO5Pureza:97.52% - 98.43%Cor e Forma:SolidPeso molecular:333.382-Methylthioadenosine diphosphate trisodium
CAS:2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.Fórmula:C11H14N5Na3O10P2SCor e Forma:SolidPeso molecular:539.24Chlorazanil
CAS:Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.Fórmula:C9H8ClN5Pureza:98.89%Cor e Forma:SolidPeso molecular:221.65Ulimorelin
CAS:Ulimorelin, ghrelin receptor agonist (EC50: 29 nM, Ki: 16 nM), is a prokinetic and vasorelaxant via α1-adrenoceptor antagonism.Fórmula:C30H39FN4O4Pureza:98%Cor e Forma:SolidPeso molecular:538.65Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Fórmula:C18H19NCor e Forma:SolidPeso molecular:249.35GCGR antagonist 2
CAS:Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.Fórmula:C28H26N4O2Cor e Forma:SolidPeso molecular:450.53Ko-3290
CAS:Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.Fórmula:C19H25N3O3Pureza:98%Cor e Forma:SolidPeso molecular:343.42Imiloxan hydrochloride
CAS:Imiloxan hydrochloride is an α2-adrenoceptor antagonist.Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75Dacemazine
CAS:Dacemazine is used to treat depression.Fórmula:C16H16N2OSCor e Forma:SolidPeso molecular:284.38Gastrazole disodium
CAS:Gastrazole, a CCK2 receptor antagonist, is used potentially for the treatment of pancreatic cancer.Fórmula:C34H34FN5Na2O7Cor e Forma:SolidPeso molecular:689.652Oxiperomide
CAS:Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.Fórmula:C20H23N3O2Pureza:98%Cor e Forma:SolidPeso molecular:337.42L-692429
CAS:L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can be used to study acromegaly and obesity.Fórmula:C29H31N7O2Pureza:98.64% - 99.90%Cor e Forma:SolidPeso molecular:509.614Ref: TM-T11798
1mg147,00€5mg356,00€10mg530,00€25mg848,00€50mg1.153,00€100mg1.549,00€1mL*10mM (DMSO)400,00€Dacopafant
CAS:Dacopafant is an antagonist of platlet activationg factor receptor.Fórmula:C12H11N3OSCor e Forma:SolidPeso molecular:245.3Methylcarbamyl PAF C-16
CAS:Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.Fórmula:C26H55N2O7PCor e Forma:SolidPeso molecular:538.7LUF5831
CAS:LUF5831 is an agonist of adenosine A1 receptor.Fórmula:C15H12N4O2SCor e Forma:SolidPeso molecular:312.35Aminaftone
CAS:Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.Fórmula:C18H15NO4Pureza:96.31% - 99.39%Cor e Forma:SolidPeso molecular:309.32Ambucetamide
CAS:Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Fórmula:C17H28N2O2Cor e Forma:SolidPeso molecular:292.42Licogliflozin
CAS:Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).Fórmula:C23H28O7Pureza:98%Cor e Forma:SolidPeso molecular:416.46SC 51089 free base
CAS:SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.Fórmula:C22H19ClN4O3Cor e Forma:SolidPeso molecular:422.86Metrenperone
CAS:Metrenperone is used as a S(2)-receptor blocker.Fórmula:C24H26FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:407.48KW-8232 free base
CAS:KW-8232 free base can reduces the biosynthesis of PGE2, is an anti-osteoporotic agent.Fórmula:C36H37ClN4O3Pureza:98%Cor e Forma:SolidPeso molecular:609.16CCG-271423
CAS:CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.Fórmula:C28H26N4O3Cor e Forma:SolidPeso molecular:466.53BAY-386
CAS:BAY-386 is a PAR1 receptor inhibitor which suppresses activation of thrombin and platelet activity.Fórmula:C22H25F3N4O5SCor e Forma:SolidPeso molecular:514.52PNU-177864
CAS:PNU-177864 is a selective dopamine D3 receptor antagonist.Fórmula:C18H21F3N2O3SPureza:99.92%Cor e Forma:SolidPeso molecular:402.43LY 302148
CAS:LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.41CAY10412
CAS:Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.Fórmula:C25H36O2SCor e Forma:SolidPeso molecular:400.62Ksg 504
CAS:Ksg 504 has superior selectivity and affinity to CCK-A receptors and derived from proglumide.Fórmula:C31H49N5O8SCor e Forma:SolidPeso molecular:651.81Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Fórmula:C70H92ClN17O14·xC2H4O2Pureza:97.96%Cor e Forma:SolidPeso molecular:1491.11CI-1015
CAS:CI-1015 is a CCK-B receptor antagonist with oral activity.Fórmula:C29H39N3O4Cor e Forma:SolidPeso molecular:493.64F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Fórmula:C26H29ClF2N4O4SCor e Forma:SolidPeso molecular:567.05BMS-193884
CAS:BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.Fórmula:C20H17N3O4SCor e Forma:SolidPeso molecular:395.43O-2093
CAS:anandamide uptake inhibitorFórmula:C34H43Cl2NO3Pureza:98%Cor e Forma:SolidPeso molecular:584.62MDL 73005EF hydrochloride
CAS:5-HT1A receptor antagonistFórmula:C20H27ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:394.89ATC0065
CAS:ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.Fórmula:C25H29BrF3N5OCor e Forma:SolidPeso molecular:552.43Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Fórmula:C19H17NO7Pureza:95% - 97.34%Cor e Forma:SolidPeso molecular:371.34Efpeglenatide
CAS:Efpeglenatide is a long-acting GLP-1 receptor agonist that improves insulin sensitivity, lowers blood glucose, delays weight gain, and supports metabolic disease research.Pureza:100% - 100%Cor e Forma:SolidAcetylaszonalenin
CAS:Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.Fórmula:C25H25N3O3Cor e Forma:SolidPeso molecular:415.48Tacitin
CAS:Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.Fórmula:C18H20ClNPureza:98%Cor e Forma:SolidPeso molecular:285.81VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Fórmula:C25H32N4O2Cor e Forma:SolidPeso molecular:420.55GRK5-IN-4
CAS:GRK5-IN-4: potent, selective covalent inhibitor of GRK5 (IC50=1.1 μM), 90x more specific than GRK2, useful for heart failure research.Fórmula:C26H25N7O3Cor e Forma:SolidPeso molecular:483.52TC-C 14G
CAS:CB1 receptor inverse agonistFórmula:C24H17Cl2F2NO4Pureza:98%Cor e Forma:SolidPeso molecular:492.3MRS2603
CAS:MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.Fórmula:C14H12ClN4O8PPureza:98%Cor e Forma:SolidPeso molecular:430.69SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Fórmula:C21H22ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:403.86CAY10498
CAS:A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.Fórmula:C18H20N6Cor e Forma:SolidPeso molecular:320.39Hexoprenaline
CAS:Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.Fórmula:C22H32N2O6Cor e Forma:SolidPeso molecular:420.5KW-8232
CAS:KW-8232, an orally active anti-osteoporotic agent, reduces the biosynthesis of PGE2[1].Fórmula:C37H41ClN4O6SCor e Forma:SolidPeso molecular:705.27VPC12249
CAS:VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity.Fórmula:C34H52NO6PCor e Forma:SolidPeso molecular:601.75CP-376395 HCl
CAS:CP 376395 hydrochloride is a potent and selective CRF-RI receptor antagonist.Fórmula:C21H31ClN2OCor e Forma:SolidPeso molecular:362.94PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFórmula:C14H12F3NOSPureza:98%Cor e Forma:SolidPeso molecular:299.31LEI-101
CAS:LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.Fórmula:C23H25FN4O4SPureza:98%Cor e Forma:SolidPeso molecular:472.53GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Fórmula:C22H18N2O2Cor e Forma:SolidPeso molecular:342.393-epi-Vitamin D3
CAS:3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM inFórmula:C27H44OCor e Forma:SolidPeso molecular:384.64Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Fórmula:C15H19N3O2Cor e Forma:SolidPeso molecular:273.33Fenmetozole Tosylate
CAS:Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,Fórmula:C17H18Cl2N2O4SPureza:98%Cor e Forma:SolidPeso molecular:417.31RUSKI-201
CAS:RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.Fórmula:C20H27N3OSCor e Forma:SolidPeso molecular:357.51SKF83959
CAS:SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.
Fórmula:C18H20ClNO2Pureza:98.68%Cor e Forma:SolidPeso molecular:317.81U-101958 Maleate
CAS:U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.Fórmula:C25H33N3O5Pureza:98%Cor e Forma:SolidPeso molecular:455.55Aceprometazine
CAS:Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].Fórmula:C19H22N2OSCor e Forma:SolidPeso molecular:326.46HSK0935
CAS:HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.Fórmula:C22H25ClO7Pureza:98%Cor e Forma:SolidPeso molecular:436.88MRS2768 tetrasodium salt
CAS:MRS2768 tetrasodium: a P2Y2 agonist; offers cardioprotection against ischemia.Fórmula:C15H16N2Na4O18P4Cor e Forma:SolidPeso molecular:728.14(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Fórmula:C23H32N6O3SPureza:99.54%Cor e Forma:SolidPeso molecular:472.6Ref: TM-T10000
1mg148,00€5mg284,00€10mg411,00€25mg645,00€50mg867,00€100mg1.121,00€1mL*10mM (DMSO)369,00€Linadryl hydrochloride
CAS:Linadryl hydrochloride may have antihistamine activity.Fórmula:C19H24ClNO2Cor e Forma:SolidPeso molecular:333.85Idremcinal
CAS:Idremcinal is a motilin receptor agonist.Fórmula:C39H69NO12Cor e Forma:SolidPeso molecular:743.96CCG-273463
CAS:CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.Fórmula:C26H25BrN4O3Cor e Forma:SolidPeso molecular:521.41SSTR5 antagonist 2
CAS:SSTR5 antagonist 2: potent, orally active, selective SSTR5 inhibitor, may treat Type 2 diabetes.Fórmula:C32H35FN2O5Pureza:98%Cor e Forma:SolidPeso molecular:546.63Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Fórmula:C26H31FN2O4Pureza:98%Cor e Forma:SolidPeso molecular:454.53RUSKI-201 dihydrochloride
CAS:RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.Fórmula:C20H29Cl2N3OSCor e Forma:SolidPeso molecular:430.43Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Fórmula:C22H25NO6Pureza:98%Cor e Forma:SolidPeso molecular:399.44(E)-Guanabenz
CAS:(E)-Guanabenz is an oral α2-adrenoceptor agonist, antihypertensive, GADD34 inhibitor, and has neuroprotective properties.Fórmula:C8H8Cl2N4Cor e Forma:SolidPeso molecular:231.08Quinpirole Hydrochloride
CAS:Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and miceFórmula:C13H22ClN3Pureza:98%Cor e Forma:SolidPeso molecular:255.79LY 171859
CAS:LY 171859 is an agonist of D2-receptor.Fórmula:C17H14O5Pureza:98%Cor e Forma:SolidPeso molecular:298.29Midodrine (hydrochloride)
CAS:Midodrine hydrochloride ((±)-Midodrine hydrochloride) is an α1-receptor agonist used in the treatment of dysautonomia and orthostatic hypotension.Fórmula:C12H19ClN2O4Peso molecular:290.74Alprenolol hydrochloride, (S)-
CAS:Alprenolol hydrochloride, (S)- is a nonselective β-blocker. It is also a serotonin 5HT1A receptor antagonist.Fórmula:C15H24ClNO2Cor e Forma:SolidPeso molecular:285.81Atigliflozin
CAS:Atigliflozin is an antihyperglycaemic drug candidate.Fórmula:C18H22O7SCor e Forma:SolidPeso molecular:382.43Ro 363 hydrochloride
CAS:Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.Fórmula:C19H26ClNO6Cor e Forma:SolidPeso molecular:399.87GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Fórmula:C32H38N2O5Cor e Forma:SolidPeso molecular:530.665FG-5893
CAS:FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.Fórmula:C27H29F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:465.53ASP7657
CAS:ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.Fórmula:C28H26F3N3O3Cor e Forma:SolidPeso molecular:509.52MAT2A-IN-2
CAS:MAT2A-IN-2 is a potent inhibitor of MAT2A. MAT2A-IN-2 has potential for cancer disease research.Fórmula:C23H17F3N6O2Cor e Forma:SolidPeso molecular:466.42Flerobuterol
CAS:Flerobuterol is a potential antidepressant agent related to beta-adrenergic agonists.Fórmula:C12H18FNOPureza:98%Cor e Forma:SolidPeso molecular:211.28Fosnetupitant
CAS:Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.Fórmula:C31H35F6N4O5PPureza:98%Cor e Forma:SolidPeso molecular:688.6Proglumide sodium
CAS:Non-selective cholecystokinin (CCK) antagonistFórmula:C18H26N2NaO4Pureza:98%Cor e Forma:SolidPeso molecular:357.4Befetupitant
CAS:Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.Fórmula:C29H29F6N3O2Pureza:98.72%Cor e Forma:SolidPeso molecular:565.55RTI 336
CAS:RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.Fórmula:C24H26Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:429.38L-826266
CAS:L-826266 is an antagonist of EP(1) receptor.Fórmula:C27H21BrClNO4SCor e Forma:SolidPeso molecular:570.88GSK3004774
CAS:GSK3004774 is a nonabsorbable agonist of CaSR (pEC50: 7.3, 6.6, and 6.5 for human, mouse, and rat CaSR). GSK3004774 shows an EC50 of 50 nM for human CaSR.Fórmula:C32H40N4O3Pureza:98%Cor e Forma:SolidPeso molecular:528.68LY314228
CAS:LY314228 is an antagonist of 5-HT2A receptor.Fórmula:C20H24N4O3Cor e Forma:SolidPeso molecular:368.43Epanolol
CAS:Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.Fórmula:C20H23N3O4Pureza:98%Cor e Forma:SolidPeso molecular:369.41PQ-69
CAS:PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.Fórmula:C20H19FN4OCor e Forma:SolidPeso molecular:350.39Autotaxin-IN-6
CAS:Autotaxin-IN-6 is a strong ATX inhibitor with a 30 nM IC50, potentially aiding anticancer research by hindering cell migration.Fórmula:C35H54BNO6Cor e Forma:SolidPeso molecular:595.62Izuforant
CAS:Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).Fórmula:C12H12BrN7Cor e Forma:SolidPeso molecular:334.17
