GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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Uroguanylin (human) TFA
<p>Uroguanylin (human) (TFA) is the natural ligand for the guanylate cyclase C (GCC) receptor expressed in metastatic colorectal cancer tumors. In animal models of human colon cancer, Uroguanylin (human) (TFA) demonstrates antitumor activity.</p>Cor e Forma:Odour SolidNeurokinin B (TFA)
CAS:<p>Neurokinin B TFA, a tachykinin, targets NK1R, NK2R, nk3r GPCRs, modulating effects.</p>Fórmula:C59H81F6N13O18S2Pureza:98%Cor e Forma:SolidPeso molecular:1438.47Tecastemizole
CAS:<p>Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.</p>Fórmula:C19H21FN4Pureza:99.70%Cor e Forma:SolidPeso molecular:324.4Nesiritide
CAS:<p>Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.</p>Fórmula:C143H244N50O42S4Pureza:98%Cor e Forma:SolidPeso molecular:3464.04Plecanatide acetate
CAS:Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Fórmula:C67H108N18O28S4Pureza:98%Cor e Forma:SolidPeso molecular:1741.9415(S)-HpEPE
CAS:<p>15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456(+)-5-trans Cloprostenol
CAS:<p>Cloprostenol, a synthetic PGF2α derivative, induces estrus and treats reproductive issues in livestock; its minor impurity, (+)-5-trans, is less effective.</p>Fórmula:C22H29ClO6Cor e Forma:SolidPeso molecular:424.92ACT-1016-0707
CAS:<p>ACT-1016-0707 is a selective, insurmountable LPA1 antagonist with antifibrotic and anti-inflammatory activity in lung fibrosis models</p>Fórmula:C19H23ClN4O4SPureza:99.905%Cor e Forma:SolidPeso molecular:438.93AL12180
CAS:<p>AL12180 is a bioactive chemical.</p>Fórmula:C21H27ClO6Cor e Forma:SolidPeso molecular:410.89d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Fórmula:C47H67N11O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1026.2PF-232798
CAS:<p>PF-232798 is a second generation oral CCR5 antagonist with potent broad-spectrum anti-HIV-1 activity.</p>Fórmula:C29H40FN5O2Cor e Forma:SolidPeso molecular:509.66Mirtazapine N-oxide
CAS:<p>Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.</p>Fórmula:C17H19N3OCor e Forma:SolidPeso molecular:281.359SRI-37330
CAS:<p>SRI-37330 inhibits glucagon secretion and function, reduces hepatic glucose production, and reverses hepatic steatosis.</p>Fórmula:C16H19F3N4O2SPureza:99.65%Cor e Forma:SolidPeso molecular:388.41CKLF1-C27 TFA
<p>CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.</p>Fórmula:C153H244F3N39O39Cor e Forma:SolidPeso molecular:3310.8Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:<p>CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.</p>Fórmula:C163H267N51O50S2Pureza:98%Cor e Forma:SolidPeso molecular:3805.31A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Fórmula:C23H25IN4Cor e Forma:SolidPeso molecular:484.38[D-Trp8]-γ-MSH
CAS:<p>[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).</p>Fórmula:C74H99N21O16SPureza:98%Cor e Forma:SolidPeso molecular:1570.795-hydroxy Propranolol
CAS:<p>5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.</p>Fórmula:C16H21NO3Cor e Forma:SolidPeso molecular:275.348Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Fórmula:C26H37N5O2Pureza:97.69% - 99.86%Cor e Forma:White Crystalline SolidPeso molecular:451.6[D-Trp8,Tyr11] Somatostatin
CAS:[D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,Fórmula:C76H104N18O20S2Peso molecular:1653.88(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Fórmula:C64H81N17O14Peso molecular:1312.43FSLLRY-NH2
CAS:<p>PAR2 antagonist; counters taxol effects, PKC in mice; inhibits ERK, collagen in fibroblasts; lessens dermatophyte itch in mice.</p>Fórmula:C39H60N10O8Pureza:98%Cor e Forma:SolidPeso molecular:796.97Alprostadil ethyl ester
CAS:<p>Alprostadil ethyl ester is a biochemical used in the treatment of scleroderma.</p>Fórmula:C22H38O5Cor e Forma:SolidPeso molecular:382.53Mapenterol hydrochloride
CAS:<p>Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.</p>Fórmula:C14H21Cl2F3N2OPureza:98.11% - 99.98%Cor e Forma:SolidPeso molecular:361.23Amylin (1-37), human acetate
<p>Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.</p>Pureza:96.21%Cor e Forma:Odour SolidsGnRH-A
CAS:<p>sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.</p>Fórmula:C64H83N17O12Cor e Forma:SolidPeso molecular:1282.45Prepro VIP (81-122), human
CAS:Prepro VIP (81-122), human is a prepro-vasoactive intestinal polypeptide (VIP) derived peptide, corresponding to residues 81-122.Fórmula:C202H325N53O64SPureza:98%Cor e Forma:SolidPeso molecular:4552.13γ-2-MSH (41-58), amide
CAS:Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.Fórmula:C74H100N22O15SPureza:98%Cor e Forma:SolidPeso molecular:1569.79INCB3344 R-isomer
<p>INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.</p>Fórmula:C29H34F3N3O6Pureza:98%Cor e Forma:SolidPeso molecular:577.5919(R)-hydroxy Prostaglandin E1
CAS:<p>19(R)-hydroxy Prostaglandin E1 is an agonist of EP1 and EP3 receptor subtypes and exhibits contractile activity on smooth muscle and is the major prostaglandin</p>Fórmula:C20H34O6Cor e Forma:SolidPeso molecular:370.4865-HT6R antagonist 6
<p>5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.</p>Fórmula:C24H26N4O2SCor e Forma:SolidPeso molecular:434.55Sufotidine
CAS:<p>Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.</p>Fórmula:C20H31N5O3SPureza:99.03% - 99.92%Cor e Forma:SolidPeso molecular:421.56ONO-0300302
CAS:ONO-0300302: LPA1 antagonist, treats Benign Prostatic Hyperplasia, IC50 = 0.16 nM, reduces IUP in rats and dogs for 12h.Fórmula:C29H35NO5Pureza:98%Cor e Forma:SolidPeso molecular:477.59D-Epinephrine
CAS:<p>D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.</p>Fórmula:C9H13NO3Cor e Forma:SolidPeso molecular:183.2Vatinoxan
CAS:<p>Vatinoxan is a peripheral α2 adrenoreceptor antagonist.</p>Fórmula:C20H26N4O4SPureza:98%Cor e Forma:SolidPeso molecular:418.51BAM(8-22) TFA
<p>BAM(8-22) TFA activates Mrgprs, induces mouse scratching, and is a proenkephalin A derivative.</p>Fórmula:C93H128F3N25O25SCor e Forma:SolidPeso molecular:2085.2217-phenoxy trinor Prostaglandin F2α ethyl amide
CAS:<p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>Fórmula:C25H37NO5Cor e Forma:SolidPeso molecular:431.573TRAP-6 amide TFA
CAS:<p>TRAP-6 amide TFA is a PAR-1 thrombin receptor agonist peptide.</p>Fórmula:C36H58F3N11O10Cor e Forma:SolidPeso molecular:861.922BMS-604992 free base
CAS:<p>BMS-604992 (EX-1314), a selective GHSR agonist, binds strongly (ki=2.3 nM), is orally active, and increases rodent food intake.</p>Fórmula:C24H31N7O5Cor e Forma:SolidPeso molecular:497.556Dolcanatide
CAS:Dolcanatide: oral GC-C agonist with laxative, pain-relief, and anti-inflammatory properties for IBD research.Fórmula:C65H104N18O26S4Cor e Forma:SolidPeso molecular:1681.89MM 07
CAS:<p>Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.</p>Fórmula:C67H106N22O14S3Pureza:98%Cor e Forma:SolidPeso molecular:1539.9Ici 216140
CAS:<p>ICI 216140: GRP/bombesin receptor 2 blocker, potent at 2 nM. Reduces amylase at 2 mg/kg and lowers bombesin-induced blood pressure at 1 mM in rats.</p>Fórmula:C45H65N13O8Cor e Forma:SolidPeso molecular:916.08Jmv 167
CAS:<p>Jmv 167 is an antagonist of the Cholecystokinin receptor.</p>Fórmula:C51H68N8O14SPureza:98%Cor e Forma:SolidPeso molecular:1049.2116-phenoxy tetranor Prostaglandin F2α methyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Fórmula:C23H32O6Cor e Forma:SolidPeso molecular:404.503Benzomalvin B
CAS:<p>Benzomalvin B, a metabolite from Penicillium, blocks 24% NK1 receptor binding at 100 μg/ml.</p>Fórmula:C24H17N3O2Cor e Forma:SolidPeso molecular:379.419Vapreotide diacetate
CAS:<p>Vapreotide diacetate, a synthetic somatostatin analog, blocks NK1R to provide analgesic effects.</p>Fórmula:C61H78N12O13S2Pureza:98%Cor e Forma:SolidPeso molecular:1251.47Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Fórmula:C10H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:233.69Neuropeptide Y 13-36 (porcine)
CAS:<p>Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.</p>Fórmula:C135H209N41O36Cor e Forma:SolidPeso molecular:2982.408Azaline B
CAS:<p>Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.</p>Fórmula:C80H102ClN23O12Cor e Forma:SolidPeso molecular:1613.27ZL-1101
<p>ZL-1101 is a human monoclonal antibody (mAb) targeting TNFRSF4/OX40/CD134.</p>Cor e Forma:Odour LiquidSenktide TFA
<p>Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.</p>Cor e Forma:Odour SolidSLB1122168 formic
<p>SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of 94 nM [1].</p>Fórmula:C23H37N3O3Pureza:98%Cor e Forma:SolidPeso molecular:403.56MCL0129
CAS:<p>MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.</p>Fórmula:C34H47FN4OPureza:98%Cor e Forma:SolidPeso molecular:546.76[Sar4] Substance P (4-11)
<p>'[Sar4] Substance P (4-11) is a C-terminus fragment and agonist of Substance P.'</p>Fórmula:C44H65N11O10SCor e Forma:SolidPeso molecular:940.12Substance P(1-7)
CAS:<p>Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.</p>Fórmula:C41H65N13O10Pureza:98%Cor e Forma:SolidPeso molecular:900.04ELA-32(human)
CAS:<p>Potent apelin receptor agonist with IC50 = 0.27 nM; does not bind GPR15/GPR25. Boosts hESC self-renewal and angiogenesis.</p>Fórmula:C170H289N63O39S4Pureza:98%Cor e Forma:SolidPeso molecular:3967.8Linaclotide acetate
CAS:<p>Linaclotide acetate, an oral guanylate cyclase C agonist with 14 amino acids, treats constipation-predominant IBS and chronic constipation.</p>Fórmula:C61H83N15O23S6Pureza:98%Cor e Forma:SolidPeso molecular:1586.79Detomidine carboxylic acid
CAS:<p>Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.</p>Fórmula:C12H12N2O2Pureza:98%Cor e Forma:SolidPeso molecular:216.24Phoenixin-14 TFA
<p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>Fórmula:C75H110N18O20·xC2HF3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:1583.78 (free base)SAR441255
SAR441255 is a potent unimolecular peptide that acts as a GLP-1/GIP/GCG receptor triagonist, demonstrating balanced activation across all three target receptorsCor e Forma:Odour SolidNafetolol
CAS:<p>Nafetolol (K 5407) is a biochemical reagent that can be used to synthesize other compounds.</p>Fórmula:C19H29NO3Pureza:98.91%Cor e Forma:SolidPeso molecular:319.44Fenoldopam
CAS:<p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>Fórmula:C16H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:305.76CART(55-102)(rat) TFA
<p>Rat CART(55-102) TFA suppresses appetite, links to leptin/neuropeptide Y, and may induce anxiety/stress.</p>Fórmula:C228H368F3N65O67S7Cor e Forma:SolidPeso molecular:5373.2Substance P (alligator)
CAS:<p>Substance P from alligator: a neuropeptide with structure Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2.</p>Fórmula:C63H98N20O13SCor e Forma:SolidPeso molecular:1375.64PACAP (1-38) free acid
CAS:<p>PACAP (1-38) free acid, an endogenous neuropeptide, potently modulates gastrointestinal and neuroendocrine functions.</p>Cor e Forma:Solid(Phe2,Orn8)-Oxytocin acetate
<p>(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.</p>Fórmula:C44H69N13O13S2Cor e Forma:SolidPeso molecular:1052.23SB234551
CAS:<p>SB234551 is a selective antagonist of endothelin ETA receptor.</p>Fórmula:C34H34N2O9Cor e Forma:SolidPeso molecular:614.64S1R agonist 2 hydrochloride
<p>Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 nM for S1R and 88 nM for S2R.</p>Fórmula:C21H28ClNOPureza:98%Cor e Forma:SolidPeso molecular:345.91Secretin (28-54), human
CAS:Secretin (28-54), human, is a 27-amino acid residue peptide with a C-terminal amidation, acting on human secretin receptors.Fórmula:C130H220N44O40Pureza:98%Cor e Forma:PowderPeso molecular:3039.46Oxmetidine
CAS:<p>Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.</p>Fórmula:C19H21N5O3SPureza:99.67%Cor e Forma:SolidPeso molecular:399.47CB2R/FAAH modulator-3
CAS:<p>CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.</p>Fórmula:C22H31NO2Pureza:99.81%Cor e Forma:SoildPeso molecular:341.49(±)5(6)-EET
CAS:<p>5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.</p>Fórmula:C20H32O3Cor e Forma:SolidPeso molecular:320.473Pramlintide
CAS:<p>Pramlintide, a polypeptide analog of human amylin, is an antidiabetic agent with antineoplastic properties in colorectal cancer.</p>Cor e Forma:SolidApelin-12 acetate
<p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>Fórmula:C66H107N21O16SPureza:98.82%Cor e Forma:SolidPeso molecular:1482.75Fabesetron
CAS:<p>Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.</p>Fórmula:C18H19N3OCor e Forma:SolidPeso molecular:293.3720-Carboxy-Leukotriene B4
CAS:<p>20-COOH LTB4, a metabolite of LTB4, binds BLT1 receptor and inhibits LTB4-induced neutrophil responses.</p>Fórmula:C20H30O6Cor e Forma:SolidPeso molecular:366.45Leukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Fórmula:C22H37NO4Cor e Forma:SolidPeso molecular:379.541ABT 724 trihydrochloride
CAS:<p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>Fórmula:C17H22Cl3N5Pureza:99.91%Cor e Forma:SolidPeso molecular:402.75Adrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Fórmula:C194H304N58O59S4Pureza:98%Cor e Forma:SolidPeso molecular:4521.17CCZ01048 TFA
CCZ01048 TFA, α-MSH analog, binds MC1R with 0.31 nM affinity, internalizes in melanoma cells, and is stable for melanoma PET imaging.Fórmula:C73H106F3N21O18Cor e Forma:SolidPeso molecular:1622.75Amylin, amide, human TFA
<p>Amylin, a 37-amino acid human hormone, moderates glucose regulation by reducing glucagon, delaying digestion, and increasing satiety.</p>Fórmula:C167H262F3N51O57S2Cor e Forma:SolidPeso molecular:4017.3Oxaprotiline hydrochloride
CAS:Oxaprotiline hydrochloride is an antidepressant.Fórmula:C20H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:329.86LRGILS-NH2
CAS:<p>LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.</p>Fórmula:C29H56N10O7Pureza:98%Cor e Forma:SolidPeso molecular:656.82Elabela(19-32)
CAS:<p>APJ receptor agonist with Ki of 0.93 nM, derived from ELA-32, activates Gαi1, β-arrestin-2, lowers rat heart arterial pressure, effective in vivo.</p>Fórmula:C75H119N25O17S2Pureza:98%Cor e Forma:SolidPeso molecular:1707.03[D-Phe12]-Bombesin
CAS:<p>Bombesin receptor antagonist</p>Fórmula:C74H112N22O18SPureza:98%Cor e Forma:SolidPeso molecular:1629.88Neurokinin B acetate(86933-75-7 free base)
<p>Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological effects.</p>Fórmula:C57H83N13O16S2Pureza:98.53%Cor e Forma:SolidPeso molecular:1270.48TT-OAD2
CAS:<p>TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.</p>Fórmula:C50H49Cl4N3O6Pureza:98%Cor e Forma:SolidPeso molecular:929.75PF-03382792
CAS:<p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>Fórmula:C23H32FN3O4Pureza:99.64%Cor e Forma:SolidPeso molecular:433.52Imnopitant dihydrochloride
CAS:<p>Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .</p>Fórmula:C28H30Cl2F6N4OCor e Forma:SolidPeso molecular:623.46NI-0701
<p>NI-0701 is a humanized antibody targeting CCL5/RANTES.</p>Pureza:95.4% (SDS-PAGE); 99.4% (SEC-HPLC) - 95.4% (SDS-PAGE); 99.4% (SEC-HPLC)Cor e Forma:LiquidPeso molecular:145.5kDaL-770644 dihydrochloride
CAS:<p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>Fórmula:C30H38ClN7O4SCor e Forma:SolidPeso molecular:628.19Lys-Bradykinin
CAS:<p>Endogenous bradykinin receptor agonist</p>Fórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Fórmula:C50H73N13O11Pureza:98%Cor e Forma:SolidPeso molecular:1032.21β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Fórmula:C162H267N51O48S3Pureza:98%Cor e Forma:SolidPeso molecular:3793.41Calcitonin (8-32), salmon
CAS:Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.Fórmula:C119H198N36O37Pureza:98%Cor e Forma:SolidPeso molecular:2725.06Anthramycin
CAS:<p>Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.</p>Fórmula:C16H17N3O4Cor e Forma:SolidPeso molecular:315.32Fluphenazine free base
CAS:<p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>Fórmula:C22H26F3N3OSCor e Forma:SolidPeso molecular:437.52Efranarelaxin alfa
CAS:<p>Efranarelaxin alfa is an agonist of the relaxin receptor. It shows potential for research in cardiovascular diseases and tissue repair.</p>Cor e Forma:LiquidRubraxanthone
CAS:<p>Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.</p>Fórmula:C24H26O6Cor e Forma:SolidPeso molecular:410.466Orexin B, rat, mouse TFA
<p>Orexin B, rat/mouse TFA, activates OX1-R & OX2-R receptors, influencing food intake, energy, and sleep regulation.</p>Fórmula:C128H216F3N45O36SCor e Forma:SolidPeso molecular:3050.42
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