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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • 6-fluoro-DL-Tryptophan
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    6-fluoro-DL-Tryptophan

    CAS:
    <p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>
    Fórmula:C11H11FN2O2
    Pureza:99.25%
    Cor e Forma:Off-White Powder
    Peso molecular:222.22

    Ref: TM-T7694

  • HS 014 acetate(207678-81-7 free base)
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    HS 014 acetate(207678-81-7 free base)

    <p>HS 014 acetate is a potent MC4R antagonist with Ki: 3.16 nM (MC4), and boosts food intake and nociception in animals.</p>
    Fórmula:C73H98N20O19S2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1623.83

    Ref: TM-TP2015L

  • Sertindole
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    Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Cor e Forma:Off-White To Pale Yellow Solid
    Peso molecular:440.94

    Ref: TM-T5858

  • GLPG2938
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    GLPG2938

    CAS:
    <p>GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and</p>
    Fórmula:C20H19F6N7O2
    Pureza:98.25%
    Cor e Forma:Solid
    Peso molecular:503.4

    Ref: TM-T9199

  • Dioxopromethazine hydrochloride
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    Dioxopromethazine hydrochloride

    CAS:
    Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
    Fórmula:C17H20N2O2S·HCl
    Pureza:99.58%
    Cor e Forma:Solid
    Peso molecular:352.88

    Ref: TM-T3723

  • Nomifensine
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    Nomifensine

    CAS:
    <p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>
    Fórmula:C16H18N2
    Pureza:99.83% - ≥95%
    Cor e Forma:Solid
    Peso molecular:238.33

    Ref: TM-T7308

  • A-582941 dihydrochloride
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    A-582941 dihydrochloride

    CAS:
    <p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:353.29

    Ref: TM-T22016

  • Elagolix sodium
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    Elagolix sodium

    CAS:
    <p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>
    Fórmula:C32H29F5N3NaO5
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:653.57

    Ref: TM-T5031

  • Bimatoprost
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    Bimatoprost

    CAS:
    <p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>
    Fórmula:C25H37NO4
    Pureza:98% - >99.99%
    Cor e Forma:Crystalline Solid
    Peso molecular:415.57

    Ref: TM-T2538

  • Neuromedin N acetate(92169-45-4 free base)
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    Neuromedin N acetate(92169-45-4 free base)

    <p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>
    Fórmula:C40H67N7O10
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:805.9

    Ref: TM-TP1085L

  • Chlorphenoxamine
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    Chlorphenoxamine

    CAS:
    <p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>
    Fórmula:C18H22ClNO
    Pureza:99.44% - 99.85%
    Cor e Forma:Solid
    Peso molecular:303.83

    Ref: TM-T7564

  • UFP 803 acetate
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    UFP 803 acetate

    UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.
    Fórmula:C52H68N10O14S2
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:1121.29

    Ref: TM-TP2104L

  • Vorapaxar
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    Vorapaxar

    CAS:
    <p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>
    Fórmula:C29H33FN2O4
    Pureza:98.77% - 99.93%
    Cor e Forma:Solid
    Peso molecular:492.58

    Ref: TM-T7013

  • Octreotide Acetate
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    Octreotide Acetate

    CAS:
    <p>Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.</p>
    Fórmula:C51H70N10O12S2
    Pureza:99.03% - 99.87%
    Cor e Forma:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised Solid
    Peso molecular:1079.3

    Ref: TM-T4119

  • Betahistine
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    Betahistine

    CAS:
    <p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>
    Fórmula:C8H12N2
    Pureza:99.87% - 99.87%
    Cor e Forma:Yellowish Liquid Liquid Liquid
    Peso molecular:136.19

    Ref: TM-T4195

  • Sotagliflozin
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    Sotagliflozin

    CAS:
    <p>Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potential</p>
    Fórmula:C21H25ClO5S
    Pureza:99% - 99.86%
    Cor e Forma:Solid
    Peso molecular:424.94

    Ref: TM-T3547

  • M617 acetate
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    M617 acetate

    <p>M617 acetate is a selective agonist of galanin receptor 1 (GAL1).</p>
    Fórmula:C112H161N29O28
    Pureza:96.02%
    Cor e Forma:Solid
    Peso molecular:2361.65

    Ref: TM-TP1993L

  • HS024
    Targetmol
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    HS024

    CAS:
    <p>HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.</p>
    Fórmula:C58H79N19O10S2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1266.5

    Ref: TM-TP1898

  • SB-222200
    Targetmol
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    SB-222200

    CAS:
    <p>SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).</p>
    Fórmula:C26H24N2O
    Pureza:97.13%
    Cor e Forma:Solid
    Peso molecular:380.48

    Ref: TM-T16849

  • Guanabenz Acetate
    Targetmol
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    Guanabenz Acetate

    CAS:
    <p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>
    Fórmula:C8H8Cl2N4·C2H4O2
    Pureza:99% - 99.66%
    Cor e Forma:White Solid From Acetonitrile White Solid
    Peso molecular:291.13

    Ref: TM-T6522