GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

Exibir 18 mais subcategorias

Foram encontrados 5378 produtos de "GPCR/Proteína-G"

Pureza (%)

100

produtos por página.

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Tripelennamine hydrochloride
CAS:
- 154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
Fórmula:C₁₆H₂₁N₃·HCl
Pureza:99.54% - 99.81%
Cor e Forma:White Solid
Peso molecular:291.82
Ref: TM-T1269
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Anamorelin
CAS:
- 249921-19-5
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
Fórmula:C₃₁H₄₂N₆O₃
Pureza:99.35% - 99.94%
Cor e Forma:Solid
Peso molecular:546.7
Ref: TM-T10319
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Cisapride
CAS:
- 81098-60-4
Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.
Fórmula:C₂₃H₂₉ClFN₃O₄
Pureza:99.77%
Cor e Forma:White To Slightly Biege Powder Solid
Peso molecular:465.95
Ref: TM-T1291
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PF-06882961
CAS:
- 2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Fórmula:C₃₁H₃₀FN₅O₄
Pureza:97.19% - 99.56%
Cor e Forma:Solid
Peso molecular:555.6
Ref: TM-T12431
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YNT-185
CAS:
- 1804978-81-1
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
Fórmula:C₃₃H₃₇N₅O₅S
Pureza:99.67%
Cor e Forma:Solid
Peso molecular:615.74
Ref: TM-T39229
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Protriptyline hydrochloride
CAS:
- 1225-55-4
Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.
Fórmula:C₁₉H₂₁N·HCl
Pureza:98.54% - 99.98%
Cor e Forma:Solid
Peso molecular:299.84
Ref: TM-T0204
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Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
Pureza:97.76%
Cor e Forma:Soild
Ref: TM-TP1020L
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Terlipressin Acetate
CAS:
- 1884420-36-3
Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).
Fórmula:C₅₆H₈₂N₁₆O₁₉S₂
Pureza:98.50% - 99.69%
Cor e Forma:Solid
Peso molecular:1347.5
Ref: TM-T13920L
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ML604086
CAS:
- 850330-18-6
ML604086 suppresses CCL1 mediated chemotaxis and enhances intracellular Ca2 concentrations.
Fórmula:C₂₇H₃₂N₄O₄S
Pureza:99.91%
Cor e Forma:Solid
Peso molecular:508.63
Ref: TM-T16111
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Sonepcizumab
CAS:
- 1031360-18-5
Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.
Pureza:SDS-PAGE:95% SEC-HPLC:98.90%
Cor e Forma:Liquid
Peso molecular:146.43 kDa
Ref: TM-T76828
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Benztropine mesylate
CAS:
- 132-17-2
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON
Fórmula:C₂₁H₂₅NO·CH₄SO₃
Pureza:98.41% - 99.96%
Cor e Forma:White Crystalline Powder; Odourless Or Almost Odourless
Peso molecular:403.53
Ref: TM-T1336
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Erenumab
CAS:
- 1582205-90-0
Erenumab: human antibody blocking CGRP receptors to prevent migraines.
Pureza:99.43% (SEC-HPLC) - > 95%
Cor e Forma:Liquid
Peso molecular:146.2 kDa
Ref: TM-T76874
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Azacyclonol
CAS:
- 115-46-8
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
Fórmula:C₁₈H₂₁NO
Pureza:99.46%
Cor e Forma:Solid Powder
Peso molecular:267.37
Ref: TM-T0318
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Balovaptan
CAS:
- 1228088-30-9
Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.
Fórmula:C₂₂H₂₄ClN₅O
Pureza:99.88%
Cor e Forma:Solid
Peso molecular:409.91
Ref: TM-T14494
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Desipramine hydrochloride
CAS:
- 58-28-6
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
Fórmula:C₁₈H₂₃ClN₂
Pureza:99.58% - 99.94%
Cor e Forma:White To Off-White Powder
Peso molecular:302.842
Ref: TM-T0991
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Sergliflozin A
CAS:
- 360775-96-8
Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.
Fórmula:C₂₀H₂₄O₇
Pureza:99.43%
Cor e Forma:Solid
Peso molecular:376.4
Ref: TM-T68174
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hGPR91 antagonist 1
CAS:
- 1314796-00-3
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
Fórmula:C₃₁H₂₃F₄N₃O
Pureza:98.89%
Cor e Forma:Solid
Peso molecular:529.53
Ref: TM-T11560
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Fluoxetine hydrochloride
CAS:
- 56296-78-7
Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.
Fórmula:C₁₇H₁₉ClF₃NO
Pureza:99.6% - 99.98%
Cor e Forma:White To Off-White Crystalline Solid White To Off-White Powder
Peso molecular:345.787
Ref: TM-T0450L
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Gevotroline
CAS:
- 107266-06-8
Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.
Fórmula:C₁₉H₂₀FN₃
Pureza:98.65%
Cor e Forma:Solid
Peso molecular:309.38
Ref: TM-T68080
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RS 15385-198
CAS:
- 121961-55-5
RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.
Fórmula:C₁₈H₂₆N₂O₃S
Pureza:>99.99%
Cor e Forma:Soild
Peso molecular:350.48
Ref: TM-T68051L