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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • Methyldopa
    Targetmol
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    Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21

    Ref: TM-T0505

  • Clopidogrel
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    Clopidogrel

    CAS:
    <p>Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.</p>
    Fórmula:C16H16ClNO2S
    Pureza:98.23% - 98.83%
    Cor e Forma:White Powder
    Peso molecular:321.82

    Ref: TM-T0182

  • Terfenadine
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    Terfenadine

    CAS:
    Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
    Fórmula:C32H41NO2
    Pureza:98.76% - 99.75%
    Cor e Forma:Solid
    Peso molecular:471.67

    Ref: TM-T1266

  • Amiselimod hydrochloride
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    Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Fórmula:C19H31ClF3NO3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:413.9

    Ref: TM-T10305

  • Alverine citrate
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    Alverine citrate

    CAS:
    <p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>
    Fórmula:C26H35NO7
    Pureza:98.53% - 99.43%
    Cor e Forma:Coa
    Peso molecular:473.57

    Ref: TM-T0428

  • Cefaclor monohydrate
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    Cefaclor monohydrate

    CAS:
    <p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>
    Fórmula:C15H16ClN3O5S
    Pureza:97.36% - 99.9%
    Cor e Forma:White Crystaling Powder
    Peso molecular:385.82

    Ref: TM-T1495

  • Filorexant
    Targetmol
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    Filorexant

    CAS:
    <p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki &lt;3 nM).</p>
    Fórmula:C24H25FN4O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:420.48

    Ref: TM-T16096

  • RS 15385-198
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    RS 15385-198

    CAS:
    <p>RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.</p>
    Fórmula:C18H26N2O3S
    Pureza:>99.99%
    Cor e Forma:Soild
    Peso molecular:350.48

    Ref: TM-T68051L

  • Clonidine hydrochloride
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    Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55

    Ref: TM-T1247

  • Triflupromazine hydrochloride
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    Triflupromazine hydrochloride

    CAS:
    Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
    Fórmula:C18H20ClF3N2S
    Pureza:99.76% - 99.82%
    Cor e Forma:Crystals
    Peso molecular:388.88

    Ref: TM-T0302

  • CYM 50769
    Targetmol
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    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Fórmula:C24H17ClN2O3
    Pureza:98% - 99.08%
    Cor e Forma:Solid
    Peso molecular:416.86

    Ref: TM-T22702

  • Naluzotan hydrochloride
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    Naluzotan hydrochloride

    CAS:
    <p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>
    Fórmula:C23H39ClN4O3S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:487.1

    Ref: TM-T68113

  • Ondansetron hydrochloride dihydrate
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    Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Fórmula:C18H19N3O·HCl·2H2O
    Pureza:99.92%
    Cor e Forma:White Crystal Powder
    Peso molecular:365.86

    Ref: TM-T1478

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79

    Ref: TM-T1519L

  • Urapidil hydrochloride
    Targetmol
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    Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94

    Ref: TM-T0088

  • Antazoline hydrochloride
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    Antazoline hydrochloride

    CAS:
    <p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>
    Fórmula:C17H19N3·HCl
    Pureza:98% - 99.53%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:301.82

    Ref: TM-T0092

  • Palonosetron hydrochloride
    Targetmol
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    Palonosetron hydrochloride

    CAS:
    <p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>
    Fórmula:C19H24N2O·HCl
    Pureza:99.84% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:332.87

    Ref: TM-T1156

  • Proglumide
    Targetmol
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    Proglumide

    CAS:
    <p>Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.</p>
    Fórmula:C18H26N2O4
    Pureza:99.4% - 99.45%
    Cor e Forma:White Crystalline Powder
    Peso molecular:334.41

    Ref: TM-T1052

  • Trazodone hydrochloride
    Targetmol
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    Trazodone hydrochloride

    CAS:
    <p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>
    Fórmula:C19H23Cl2N5O
    Pureza:99.5% - 99.52%
    Cor e Forma:Solid
    Peso molecular:408.33

    Ref: TM-T1619

  • Bisoprolol hemifumarate
    Targetmol
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    Bisoprolol hemifumarate

    CAS:
    Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,
    Fórmula:C20H33NO6
    Pureza:98.69% - 99.84%
    Cor e Forma:White To Offf-White Powder
    Peso molecular:383.49

    Ref: TM-T0143