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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • CYM50308
    Targetmol
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    CYM50308

    CAS:
    <p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>
    Fórmula:C20H21F2N3O2S
    Pureza:99.43% - 99.77%
    Cor e Forma:Solid
    Peso molecular:405.46

    Ref: TM-T15032

  • Ebalzotan
    Targetmol
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    Ebalzotan

    CAS:
    <p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>
    Fórmula:C19H30N2O2
    Pureza:98.09% - 99.41%
    Cor e Forma:Solid
    Peso molecular:318.45

    Ref: TM-T68059

  • Amp579 TFA
    Targetmol
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    Amp579 TFA

    <p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>
    Fórmula:C24H29ClF3N5O5S
    Pureza:96.56%
    Cor e Forma:Soild
    Peso molecular:592.03

    Ref: TM-T67972L

  • Carebastine
    Targetmol
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    Carebastine

    CAS:
    <p>Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.</p>
    Fórmula:C32H37NO4
    Pureza:99.16%
    Cor e Forma:Off-White Solid
    Peso molecular:499.64

    Ref: TM-T10680

  • Azelastine hydrochloride
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    Azelastine hydrochloride

    CAS:
    <p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>
    Fórmula:C22H24ClN3O·HCl
    Pureza:98% - >99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:418.36

    Ref: TM-T0211L

  • Imidazolidinyl urea
    Targetmol
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    Imidazolidinyl urea

    CAS:
    <p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>
    Fórmula:C11H16N8O8
    Pureza:98.6%
    Cor e Forma:White Fluid Powder With Slight Characteristic Odor
    Peso molecular:388.29

    Ref: TM-T0430

  • Evatanepag
    Targetmol
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    Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Fórmula:C25H28N2O5S
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:468.57

    Ref: TM-T15259

  • Naluzotan hydrochloride
    Targetmol
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    Naluzotan hydrochloride

    CAS:
    <p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>
    Fórmula:C23H39ClN4O3S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:487.1

    Ref: TM-T68113

  • Promethazine hydrochloride
    Targetmol
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    Promethazine hydrochloride

    CAS:
    Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.
    Fórmula:C17H20N2S·HCl
    Pureza:99.85%
    Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Peso molecular:320.88

    Ref: TM-T0445L

  • Nepafenac
    Targetmol
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    Nepafenac

    CAS:
    <p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>
    Fórmula:C15H14N2O2
    Pureza:98.94% - 99.43%
    Cor e Forma:Solid
    Peso molecular:254.28

    Ref: TM-T1280

  • (±) Clopidogrel hydrogen sulfate
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    (±) Clopidogrel hydrogen sulfate

    CAS:
    <p>(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots</p>
    Fórmula:C16H16ClNO2S·H2SO4
    Pureza:98.67% - 99.04%
    Cor e Forma:Colorless To Light Yellow Liquid
    Peso molecular:419.9

    Ref: TM-T0182L2

  • Quetiapine
    Targetmol
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    Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:383.51

    Ref: TM-T0162

  • Quetiapine hemifumarate
    Targetmol
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    Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Fórmula:C46H54N6O8S2
    Pureza:99.32% - >99.99%
    Cor e Forma:White Crystalline Solid
    Peso molecular:883.09

    Ref: TM-T6241

  • Lamotrigine
    Targetmol
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    Lamotrigine

    CAS:
    <p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>
    Fórmula:C9H7Cl2N5
    Pureza:99.76% - 99.95%
    Cor e Forma:White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
    Peso molecular:256.09

    Ref: TM-T0680

  • Metaraminol tartrate
    Targetmol
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    Metaraminol tartrate

    CAS:
    <p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>
    Fórmula:C13H19NO8
    Pureza:99.68%
    Cor e Forma:White Powder
    Peso molecular:317.29

    Ref: TM-T0279

  • Solabegron
    Targetmol
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    Solabegron

    CAS:
    <p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>
    Fórmula:C23H23ClN2O3
    Pureza:97.89%
    Cor e Forma:Solid
    Peso molecular:410.89

    Ref: TM-T12970

  • Relenopride
    Targetmol
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    Relenopride

    CAS:
    <p>YKP 10811 (Relenopride) is a novel 5-HT4 receptor partial agonist, which can be used to study irritable bowel syndrome with constipation.</p>
    Fórmula:C24H30ClFN4O4
    Pureza:98.98% - 99.76%
    Cor e Forma:Soild
    Peso molecular:492.97

    Ref: TM-T83981

  • JMV 2959 hydrochloride (925238-89-7 free base)
    Targetmol
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    JMV 2959 hydrochloride (925238-89-7 free base)

    CAS:
    <p>JMV 2959 hydrochloride (925238-89-7 free base) is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.</p>
    Fórmula:C30H33ClN6O2
    Pureza:98.09%
    Cor e Forma:Solid
    Peso molecular:545.08

    Ref: TM-T11719

  • Degarelix acetate(214766-78-6 free base)
    Targetmol
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    Degarelix acetate(214766-78-6 free base)

    CAS:
    <p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>
    Fórmula:C84H107ClN18O18
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:1692.34

    Ref: TM-T10988L

  • Alarelin Acetate
    Targetmol
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    Alarelin Acetate

    CAS:
    <p>Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.</p>
    Fórmula:C56H78N16O12
    Pureza:99.81% - >99.99%
    Cor e Forma:White Powder
    Peso molecular:1167.34

    Ref: TM-T1494