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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5696 produtos de "GPCR/Proteína-G"

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  • ML-180
    Targetmol
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    ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Fórmula:C20H25ClN4O2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:388.89

    Ref: TM-T12075

  • Citalopram hydrobromide
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    Citalopram hydrobromide

    CAS:
    <p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>
    Fórmula:C20H22BrFN2O
    Pureza:99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:405.304

    Ref: TM-T1483

  • Anamorelin
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    Anamorelin

    CAS:
    <p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>
    Fórmula:C31H42N6O3
    Pureza:99.35% - 99.94%
    Cor e Forma:Solid
    Peso molecular:546.7

    Ref: TM-T10319

  • Quetiapine
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    Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:383.51

    Ref: TM-T0162

  • Tripelennamine hydrochloride
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    Tripelennamine hydrochloride

    CAS:
    Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
    Fórmula:C16H21N3·HCl
    Pureza:99.54% - 99.81%
    Cor e Forma:White Solid
    Peso molecular:291.82

    Ref: TM-T1269

  • SEP-363856 hydrochloride
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    SEP-363856 hydrochloride

    CAS:
    <p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>
    Fórmula:C9H14ClNOS
    Pureza:99.86% - 99.99%
    Cor e Forma:Solid
    Peso molecular:219.73

    Ref: TM-T12899L

  • Lofepramine
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    Lofepramine

    CAS:
    <p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>
    Fórmula:C26H27ClN2O
    Pureza:98.38%
    Cor e Forma:Crystals From Methanol Or Acetone Solid
    Peso molecular:418.96

    Ref: TM-T15773

  • Flopropione
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    Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Fórmula:C9H10O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:182.17

    Ref: TM-T0525

  • Quetiapine hemifumarate
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    Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Fórmula:C46H54N6O8S2
    Pureza:99.32% - >99.99%
    Cor e Forma:White Crystalline Solid
    Peso molecular:883.09

    Ref: TM-T6241

  • Mizolastine
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    Mizolastine

    CAS:
    Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.
    Fórmula:C24H25FN6O
    Pureza:98% - 99.75%
    Cor e Forma:Solid
    Peso molecular:432.49

    Ref: TM-T0118

  • Doxylamine succinate
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    Doxylamine succinate

    CAS:
    <p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>
    Fórmula:C21H28N2O5
    Pureza:99.61%
    Cor e Forma:5 1 (Ntp 1992)
    Peso molecular:388.46

    Ref: TM-T1115

  • Carteolol hydrochloride
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    Carteolol hydrochloride

    CAS:
    Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.
    Fórmula:C16H24N2O3·HCl
    Pureza:99.84% - 99.91%
    Cor e Forma:Solid
    Peso molecular:328.83

    Ref: TM-T1282

  • Xylometazoline hydrochloride
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    Xylometazoline hydrochloride

    CAS:
    <p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>
    Fórmula:C16H24N2·HCl
    Pureza:99.77% - 99.87%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:280.84

    Ref: TM-T0042

  • (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carbo…
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    (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid

    CAS:
    (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.
    Fórmula:C20H29N3O8
    Pureza:99.72%
    Cor e Forma:Soild
    Peso molecular:439.46

    Ref: TM-T77670

  • Adenosine A1 receptor activator T62
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    Adenosine A1 receptor activator T62

    CAS:
    <p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>
    Fórmula:C15H14ClNOS
    Pureza:97.83%
    Cor e Forma:Solid
    Peso molecular:291.8

    Ref: TM-T14127

  • Bromperidol
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    Bromperidol

    CAS:
    Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.
    Fórmula:C21H23BrFNO2
    Pureza:99.89%
    Cor e Forma:Tan Solid
    Peso molecular:420.32

    Ref: TM-T14830

  • Pamabrom
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    Pamabrom

    CAS:
    Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.
    Fórmula:C11H18BrN5O3
    Pureza:99.84% - >99.99%
    Cor e Forma:Coa
    Peso molecular:348.2

    Ref: TM-T1230

  • p-MPPI hydrochloride
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    p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Fórmula:C25H28ClIN4O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:578.87

    Ref: TM-T16421

  • PIT
    Targetmol
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    PIT

    CAS:
    PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.
    Fórmula:C20H16N2O5S
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:396.42

    Ref: TM-T23164

  • Rebamipide
    Targetmol
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    Rebamipide

    CAS:
    <p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>
    Fórmula:C19H15ClN2O4
    Pureza:99.48% - 99.61%
    Cor e Forma:White Powder
    Peso molecular:370.79

    Ref: TM-T1562