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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • CE3F4
    Targetmol
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    CE3F4

    CAS:
    <p>CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).</p>
    Fórmula:C11H10Br2FNO
    Pureza:97.15% - 98.06%
    Cor e Forma:Solid
    Peso molecular:351.01

    Ref: TM-T12616L

  • Chlorpheniramine maleate
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    Chlorpheniramine maleate

    CAS:
    <p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>
    Fórmula:C20H23ClN2O4
    Pureza:99.64% - 99.98%
    Cor e Forma:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Peso molecular:390.87

    Ref: TM-T1553

  • RS 15385-198
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    RS 15385-198

    CAS:
    <p>RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.</p>
    Fórmula:C18H26N2O3S
    Pureza:>99.99%
    Cor e Forma:Soild
    Peso molecular:350.48

    Ref: TM-T68051L

  • Evatanepag
    Targetmol
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    Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Fórmula:C25H28N2O5S
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:468.57

    Ref: TM-T15259

  • Relenopride
    Targetmol
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    Relenopride

    CAS:
    <p>YKP 10811 (Relenopride) is a novel 5-HT4 receptor partial agonist, which can be used to study irritable bowel syndrome with constipation.</p>
    Fórmula:C24H30ClFN4O4
    Pureza:98.98% - 99.76%
    Cor e Forma:Soild
    Peso molecular:492.97

    Ref: TM-T83981

  • Nepafenac
    Targetmol
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    Nepafenac

    CAS:
    <p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>
    Fórmula:C15H14N2O2
    Pureza:98.94% - 99.43%
    Cor e Forma:Solid
    Peso molecular:254.28

    Ref: TM-T1280

  • Fluoxetine
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    Fluoxetine

    CAS:
    <p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>
    Fórmula:C17H18F3NO
    Pureza:99.07% - 99.28%
    Cor e Forma:Solid
    Peso molecular:309.33

    Ref: TM-T0450

  • Atomoxetine hydrochloride
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    Atomoxetine hydrochloride

    CAS:
    <p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>
    Fórmula:C17H22ClNO
    Pureza:99.86%
    Cor e Forma:White Solid
    Peso molecular:291.82

    Ref: TM-T0869

  • UCM-1306
    Targetmol
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    UCM-1306

    CAS:
    <p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>
    Fórmula:C14H14FNO2S
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:279.33

    Ref: TM-T67729

  • Pemirolast potassium
    Targetmol
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    Pemirolast potassium

    CAS:
    <p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>
    Fórmula:C10H7KN6O
    Pureza:98.91% - 99.63%
    Cor e Forma:Crystals From Dimethylformamide Crystalline Solid
    Peso molecular:266.31

    Ref: TM-T1425

  • PHM-27 (human) acetate
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    PHM-27 (human) acetate

    <p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>
    Fórmula:C137H215F3N34O42S
    Pureza:99.20%
    Cor e Forma:Soild
    Peso molecular:3099.44

    Ref: TM-TP1954L

  • PIT
    Targetmol
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    PIT

    CAS:
    <p>PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.</p>
    Fórmula:C20H16N2O5S
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:396.42

    Ref: TM-T23164

  • Ifenprodil
    Targetmol
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    Ifenprodil

    CAS:
    <p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 &amp; GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>
    Fórmula:C21H27NO2
    Pureza:99.58%
    Cor e Forma:White Crystalline Powder
    Peso molecular:325.44

    Ref: TM-T1186L

  • Quetiapine hemifumarate
    Targetmol
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    Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Fórmula:C46H54N6O8S2
    Pureza:99.32% - >99.99%
    Cor e Forma:White Crystalline Solid
    Peso molecular:883.09

    Ref: TM-T6241

  • Famotidine
    Targetmol
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    Famotidine

    CAS:
    Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.
    Fórmula:C8H15N7O2S3
    Pureza:98.93% - 99.91%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:337.45

    Ref: TM-T1627

  • DF-1012 FA
    Targetmol
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    DF-1012 FA

    <p>DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.</p>
    Fórmula:C17H22N4O3
    Pureza:99.15% - 99.97%
    Cor e Forma:Solid
    Peso molecular:330.382

    Ref: TM-T27158L

  • Azasetron hydrochloride
    Targetmol
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    Azasetron hydrochloride

    CAS:
    <p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>
    Fórmula:C17H20ClN3O3·HCl
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:386.27

    Ref: TM-T1528

  • Aripiprazole Lauroxil
    Targetmol
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    Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Fórmula:C36H51Cl2N3O4
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:660.71

    Ref: TM-T14319

  • Loratadine
    Targetmol
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    Loratadine

    CAS:
    <p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>
    Fórmula:C22H23ClN2O2
    Pureza:99.71% - 99.98%
    Cor e Forma:White Powder
    Peso molecular:382.88

    Ref: TM-T1097

  • Paroxetine hydrochloride
    Targetmol
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    Paroxetine hydrochloride

    CAS:
    <p>Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.</p>
    Fórmula:C19H21ClFNO3
    Pureza:98% - 99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:365.826

    Ref: TM-T1636