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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • (R)-Elagolix
    Targetmol
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    (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Fórmula:C32H30F5N3O5
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:631.59

    Ref: TM-T11174

  • Noradrenaline bitartrate
    Targetmol
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Fórmula:C12H19NO10
    Pureza:99.53% - >99.99%
    Cor e Forma:Solid
    Peso molecular:337.28

    Ref: TM-T0871

  • Olinciguat
    Targetmol
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    Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Fórmula:C21H16F5N7O3
    Pureza:99.33% - 99.71%
    Cor e Forma:Solid
    Peso molecular:509.39

    Ref: TM-T16383

  • Venlafaxine hydrochloride
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    Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Fórmula:C17H28ClNO2
    Pureza:97.32% - 99.86%
    Cor e Forma:White Crystalline Powder
    Peso molecular:313.86

    Ref: TM-T0472

  • YNT-185
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    YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:615.74

    Ref: TM-T39229

  • Urocortin (rat) acetate
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    Urocortin (rat) acetate

    <p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>
    Pureza:97.76%
    Cor e Forma:Soild

    Ref: TM-TP1020L

  • 2-Bromo-6-methoxynaphthalene
    Targetmol
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    2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Fórmula:C11H9BrO
    Pureza:98.51%
    Cor e Forma:White To Off-White Powder
    Peso molecular:237.09

    Ref: TM-T0663

  • Ketanserin
    Targetmol
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    Ketanserin

    CAS:
    <p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>
    Fórmula:C22H22FN3O3
    Pureza:99.19% - 99.73%
    Cor e Forma:Solid
    Peso molecular:395.43

    Ref: TM-T1066

  • Talastine
    Targetmol
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    Talastine

    CAS:
    <p>Talastine is an antihistamine compound that can induce an allergic rash.</p>
    Fórmula:C19H21N3O
    Pureza:98.50% - 99.44%
    Cor e Forma:Solid
    Peso molecular:307.39

    Ref: TM-T68150

  • CP-809101 hydrochloride
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    CP-809101 hydrochloride

    CAS:
    <p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Fórmula:C15H18Cl2N4O
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:341.24

    Ref: TM-T10871

  • Roxatidine Acetate hydrochloride
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    Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Fórmula:C19H29ClN2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:384.9

    Ref: TM-T0157

  • (3aR,9aR)-Fluparoxan
    Targetmol
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H10FNO2
    Pureza:97.82%
    Cor e Forma:Soild
    Peso molecular:195.19

    Ref: TM-T77566

  • Lafutidine
    Targetmol
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    Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Fórmula:C22H29N3O4S
    Pureza:98.55%
    Cor e Forma:Yellowish White Crystalline Powder
    Peso molecular:431.55

    Ref: TM-T0081

  • AH 6809
    Targetmol
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Fórmula:C17H14O5
    Pureza:97.59%
    Cor e Forma:Solid
    Peso molecular:298.29

    Ref: TM-T14148

  • Fluparoxan hydrochloride
    Targetmol
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:231.65

    Ref: TM-T77565

  • Levosulpiride
    Targetmol
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43

    Ref: TM-T1211

  • Moxisylyte hydrochloride
    Targetmol
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    Moxisylyte hydrochloride

    CAS:
    <p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>
    Fórmula:C16H26ClNO3
    Pureza:99.93% - ≥95%
    Cor e Forma:Solid
    Peso molecular:315.84

    Ref: TM-T0394

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79

    Ref: TM-T1519L

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Cor e Forma:Colourless Flake Crystalline Solid
    Peso molecular:448.39

    Ref: TM-T1566

  • Ondansetron hydrochloride dihydrate
    Targetmol
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    Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Fórmula:C18H19N3O·HCl·2H2O
    Pureza:99.92%
    Cor e Forma:White Crystal Powder
    Peso molecular:365.86

    Ref: TM-T1478