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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • (±)12-HEPE
    Targetmol
    + Info

    (±)12-HEPE

    CAS:
    <p>(±)12-HEPE is produced by non-enzymatic oxidation of EPA.</p>
    Fórmula:C20H30O3
    Cor e Forma:Solid
    Peso molecular:318.457

    Ref: TM-T35506

  • 6α-Prostaglandin I1
    Targetmol
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    6α-Prostaglandin I1

    CAS:
    <p>6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.</p>
    Fórmula:C20H34O5
    Cor e Forma:Solid
    Peso molecular:354.487

    Ref: TM-T36238

  • Nocistatin(human)
    Targetmol
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    Nocistatin(human)

    CAS:
    <p>Blocker of nociceptin-induced allodynia and hyperalgesia</p>
    Fórmula:C149H238N42O53S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3561.93

    Ref: TM-TP2277

  • Logotipo do CymitQuimica
    Targetmol
    + Info

    Maridebart

    CAS:
    <p>Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].</p>
    Cor e Forma:Liquid

    Ref: TM-T81862

  • 5(S),6(R)-11-trans DiHETE
    Targetmol
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    5(S),6(R)-11-trans DiHETE

    CAS:
    <p>5(S),6(R)-11-trans DiHETE, a C-11 isomer of 5(S),6(R)-DiHETE, occurs in rat kidneys, formed enzymatically; not a soybean lipoxygenase substrate.</p>
    Fórmula:C20H32O4
    Cor e Forma:Solid
    Peso molecular:336.47

    Ref: TM-T37651

  • Tafluprost ethyl amide
    Targetmol
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    Tafluprost ethyl amide

    CAS:
    <p>Tafluprost ethyl amide is a prostaglandin derivative.</p>
    Fórmula:C24H33F2NO4
    Cor e Forma:Solid
    Peso molecular:437.52

    Ref: TM-T37956

  • Jmv 179
    Targetmol
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    Jmv 179

    CAS:
    <p>Jmv 179 is an antagonist of the cholecystokinin receptor.</p>
    Fórmula:C51H67N7O15S
    Cor e Forma:Solid
    Peso molecular:1050.19

    Ref: TM-T24204

  • [Tyr3]Octreotate
    Targetmol
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    [Tyr3]Octreotate

    CAS:
    <p>[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds.</p>
    Fórmula:C49H64N10O12S2
    Pureza:98.21%
    Cor e Forma:Soild
    Peso molecular:1049.22

    Ref: TM-T67931

  • D-Epinephrine
    Targetmol
    + Info

    D-Epinephrine

    CAS:
    <p>D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.</p>
    Fórmula:C9H13NO3
    Cor e Forma:Solid
    Peso molecular:183.2

    Ref: TM-T31383

  • CAY10597
    Targetmol
    + Info

    CAY10597

    CAS:
    <p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>
    Fórmula:C20H14ClFN2O5
    Cor e Forma:Solid
    Peso molecular:416.79

    Ref: TM-T38365

  • Halometasone
    Targetmol
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    Halometasone

    CAS:
    <p>Halometasone: synthetic corticosteroid for psoriasis and eczema treatment.</p>
    Fórmula:C22H27ClF2O5
    Cor e Forma:Solid
    Peso molecular:444.9

    Ref: TM-T36379

  • Logotipo do CymitQuimica
    Targetmol
    + Info

    TGR5 agonist 7

    <p>TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.</p>
    Fórmula:C37H59N2NaO9S
    Cor e Forma:Solid
    Peso molecular:730.93

    Ref: TM-T203565

  • Binospirone
    Targetmol
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    Binospirone

    CAS:
    <p>Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study of movement disorders associated with neurologic dysfunction.</p>
    Fórmula:C20H26N2O4
    Pureza:97.57% - 98.96%
    Cor e Forma:Soild
    Peso molecular:358.43

    Ref: TM-T71138L

  • Clotizolam
    Targetmol
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    Clotizolam

    CAS:
    <p>Clotizolam is a thienotriazolodiazepine derivative with PAF antagonistic properties, exhibiting sedative, anxiolytic, anticonvulsant, and muscle relaxant effects.</p>
    Fórmula:C15H10Cl2N4S
    Cor e Forma:Solid
    Peso molecular:349.24

    Ref: TM-T203541

  • Ro 25-1553
    Targetmol
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    Ro 25-1553

    CAS:
    <p>Ro 25-1553 is a 31-amino acid analog of vasoactive intestinal peptide (VIP) that functions as an agonist for the VIP2 receptor (VPAC2 receptor). In guinea pig models, Ro 25-1553 exhibits bronchodilator effects on tracheal smooth muscle contraction induced by neural stimuli or Carbachol.</p>
    Fórmula:C160H258N46O46
    Cor e Forma:Solid
    Peso molecular:3562.04

    Ref: TM-T203230

  • L-770644 dihydrochloride
    Targetmol
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    L-770644 dihydrochloride

    CAS:
    <p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>
    Fórmula:C30H38ClN7O4S
    Cor e Forma:Solid
    Peso molecular:628.19

    Ref: TM-T24377L

  • S1R agonist 1
    Targetmol
    + Info

    S1R agonist 1

    CAS:
    <p>Compound 6b: Selective S1R agonist, K i = 0.93 nM (S1R), 72 nM (S2R); neuroprotective against ROS, NMDA toxicity.</p>
    Fórmula:C20H25NO
    Cor e Forma:Solid
    Peso molecular:295.42

    Ref: TM-T74822

  • LRGILS-NH2
    Targetmol
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    LRGILS-NH2

    CAS:
    <p>LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.</p>
    Fórmula:C29H56N10O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:656.82

    Ref: TM-T22933

  • Apelin-12 acetate
    Targetmol
    + Info

    Apelin-12 acetate

    <p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>
    Fórmula:C66H107N21O16S
    Pureza:98.82%
    Cor e Forma:Solid
    Peso molecular:1482.75

    Ref: TM-T39823L

  • Khusimol
    Targetmol
    + Info

    Khusimol

    CAS:
    <p>Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.</p>
    Fórmula:C15H24O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:220.35

    Ref: TM-T25577