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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • Navafenterol saccharinate
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    Navafenterol saccharinate

    CAS:
    <p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>
    Fórmula:C45H47N7O9S3
    Cor e Forma:Solid
    Peso molecular:926.09

    Ref: TM-T30265

  • Logotipo do CymitQuimica
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    Neuropeptide SF(mouse,rat) TFA

    <p>Neuropeptide SF TFA is a potent agonist for NPFF1 (Ki=48.4 nM) and NPFF2 (Ki=12.1 nM) and enhances ASIC3 current.</p>
    Fórmula:C42H66F3N13O12
    Cor e Forma:Solid
    Peso molecular:1002.05

    Ref: TM-T75865

  • Relamorelin TFA
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    Relamorelin TFA

    CAS:
    <p>Relamorelin (RM-131) TFA: ghrelin analog, GHSR agonist, 0.42 nM affinity, boosts growth hormone, enhances gastric emptying, potential in motility disorders.</p>
    Fórmula:C45H51F3N8O7S
    Cor e Forma:Solid
    Peso molecular:905

    Ref: TM-T75262

  • Lysophosphatidic acid
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    Lysophosphatidic acid

    CAS:
    <p>Lysophosphatidic acid is a bioactive chemical.</p>
    Fórmula:C21H41O7P
    Cor e Forma:Solid
    Peso molecular:436.52

    Ref: TM-T33076

  • Logotipo do CymitQuimica
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    PSB-1114 triethylamine

    <p>PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50</p>
    Fórmula:C10H15F2N3O13P3S·xC6H15N
    Pureza:98%
    Cor e Forma:Solid

    Ref: TM-T78080

  • FFN246
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    FFN246

    CAS:
    <p>FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and</p>
    Fórmula:C15H13FN2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:256.27

    Ref: TM-T78684

  • Emoghrelin
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    Emoghrelin

    CAS:
    <p>Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].</p>
    Fórmula:C24H22O13
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:518.42

    Ref: TM-T80006

  • Logotipo do CymitQuimica
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    Muscarinic toxin 3

    CAS:
    <p>Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57</p>
    Fórmula:C319H489N89O97S8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:7379.35

    Ref: TM-T80477

  • Gemeprost
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    Gemeprost

    CAS:
    <p>Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.</p>
    Fórmula:C23H38O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:394.54

    Ref: TM-T20855

  • Logotipo do CymitQuimica
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    TGR5 agonist 7

    <p>TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.</p>
    Fórmula:C37H59N2NaO9S
    Cor e Forma:Solid
    Peso molecular:730.93

    Ref: TM-T203565

  • SC-53116
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    SC-53116

    CAS:
    <p>SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.</p>
    Fórmula:C16H22ClN3O2
    Cor e Forma:Solid
    Peso molecular:323.82

    Ref: TM-T34559

  • DOTA-JR11
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    DOTA-JR11

    CAS:
    <p>DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.</p>
    Fórmula:C74H98ClN19O21S2
    Cor e Forma:Solid
    Peso molecular:1689.27

    Ref: TM-T80157

  • Logotipo do CymitQuimica
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    Kisspeptin-54(human) TFA

    <p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>
    Fórmula:C258H401N79O78·C2HF3O2
    Cor e Forma:Solid
    Peso molecular:5971.45

    Ref: TM-T75774

  • Logotipo do CymitQuimica
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    α-CGRP (mouse, rat) TFA

    <p>α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions and</p>
    Fórmula:C162H262N50O52S2·C2HF3O2
    Pureza:98%
    Cor e Forma:Solid

    Ref: TM-T78540

  • 4-Oxo-5-phenylpentanoic aci
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    4-Oxo-5-phenylpentanoic aci

    CAS:
    <p>4-Oxo-5-phenylpentanoic aci is a useful organic compound for research related to life sciences. The catalog number is T125056 and the CAS number is 3183-15-1.</p>
    Fórmula:C11H12O3
    Cor e Forma:Solid
    Peso molecular:192.214

    Ref: TM-T125056

  • 1,2,3-Trilinoelaidoyl-rac-glycerol
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    1,2,3-Trilinoelaidoyl-rac-glycerol

    CAS:
    <p>1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.</p>
    Fórmula:C57H98O6
    Cor e Forma:Solid
    Peso molecular:879.405

    Ref: TM-T37383

  • Logotipo do CymitQuimica
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    human GALP (3-32)

    <p>Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), as</p>
    Fórmula:C137H213N43O38S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3102.49

    Ref: TM-T80516

  • LMN-NKA acetate
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    LMN-NKA acetate

    <p>LMN-NKA acetate is a modified Neurokinin A (4-10) and selective NK2R (Neurokinin 2 receptor) agonist induces bladder contraction smooth muscle contraction.</p>
    Fórmula:C41H68N8O12
    Cor e Forma:Solid
    Peso molecular:865.03

    Ref: TM-T76426L

  • Nesiritide
    Targetmol
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    Nesiritide

    CAS:
    <p>Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.</p>
    Fórmula:C143H244N50O42S4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3464.04

    Ref: TM-TP1208

  • Velmupressin acetate
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    Velmupressin acetate

    CAS:
    <p>Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).</p>
    Fórmula:C44H64ClN11O10S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1006.63

    Ref: TM-TP1205