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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5373 produtos de "GPCR/Proteína-G"

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  • Urocortin (rat) acetate
    Targetmol
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    Urocortin (rat) acetate

    Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
    Pureza:97.76%
    Cor e Forma:Soild

    Ref: TM-TP1020L

  • Indacaterol maleate
    Targetmol
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    Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Fórmula:C28H32N2O7
    Pureza:99.03% - 99.67%
    Cor e Forma:Solid
    Peso molecular:508.56

    Ref: TM-T1239

  • Lafutidine
    Targetmol
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    Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Fórmula:C22H29N3O4S
    Pureza:98.55%
    Cor e Forma:Yellowish White Crystalline Powder
    Peso molecular:431.55

    Ref: TM-T0081

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79

    Ref: TM-T1519L

  • 2-Bromo-6-methoxynaphthalene
    Targetmol
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    2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Fórmula:C11H9BrO
    Pureza:98.51%
    Cor e Forma:White To Off-White Powder
    Peso molecular:237.09

    Ref: TM-T0663

  • Amiselimod hydrochloride
    Targetmol
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    Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Fórmula:C19H31ClF3NO3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:413.9

    Ref: TM-T10305

  • Prucalopride
    Targetmol
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    Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Fórmula:C18H26ClN3O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:367.87

    Ref: TM-T2542

  • Clonidine hydrochloride
    Targetmol
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    Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55

    Ref: TM-T1247

  • Methyldopa
    Targetmol
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    Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21

    Ref: TM-T0505

  • CYM 50769
    Targetmol
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    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Fórmula:C24H17ClN2O3
    Pureza:98% - 99.08%
    Cor e Forma:Solid
    Peso molecular:416.86

    Ref: TM-T22702

  • Fluparoxan hydrochloride
    Targetmol
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:231.65

    Ref: TM-T77565

  • Fluvoxamine maleate
    Targetmol
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    Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:434.41

    Ref: TM-T1077

  • Levosulpiride
    Targetmol
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43

    Ref: TM-T1211

  • Alfuzosin hydrochloride
    Targetmol
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    Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Fórmula:C19H27N5O4·HCl
    Pureza:99.78%
    Cor e Forma:White To Off-White Solid
    Peso molecular:425.91

    Ref: TM-T0091

  • Roxatidine Acetate hydrochloride
    Targetmol
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    Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Fórmula:C19H29ClN2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:384.9

    Ref: TM-T0157

  • Urapidil hydrochloride
    Targetmol
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    Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94

    Ref: TM-T0088

  • Granisetron hydrochloride
    Targetmol
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    Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:348.87

    Ref: TM-T1042

  • Naftopidil
    Targetmol
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    Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49

    Ref: TM-T0696

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Cor e Forma:Colourless Flake Crystalline Solid
    Peso molecular:448.39

    Ref: TM-T1566

  • Fenspiride hydrochloride
    Targetmol
    + Info

    Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Fórmula:C15H20N2O2·HCl
    Pureza:99.64% - 99.92%
    Cor e Forma:Solid
    Peso molecular:296.79

    Ref: TM-T0383