CymitQuimica logo
GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

Exibir 18 mais subcategorias

Foram encontrados 5378 produtos de "GPCR/Proteína-G"

Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
produtos por página.
  • Gemeprost
    Targetmol
    + Info

    Gemeprost

    CAS:
    <p>Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.</p>
    Fórmula:C23H38O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:394.54

    Ref: TM-T20855

  • Adrogolide HCl
    Targetmol
    + Info

    Adrogolide HCl

    CAS:
    Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.
    Fórmula:C22H26ClNO4S
    Cor e Forma:Solid
    Peso molecular:435.96

    Ref: TM-T29674

  • Danshenol B
    Targetmol
    + Info

    Danshenol B

    <p>Danshenol B is a natural product that can be used as a reference standard.</p>
    Fórmula:C22H26O4
    Cor e Forma:Solid
    Peso molecular:354.446

    Ref: TM-T125490

  • MMC(TMZ)-TOC TFA
    Targetmol
    + Info

    MMC(TMZ)-TOC TFA

    <p>MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.</p>
    Fórmula:C74H99F3N20O21S2
    Cor e Forma:Solid
    Peso molecular:1725.82

    Ref: TM-T204151

  • SGLT1/2-IN-2
    Targetmol
    + Info

    SGLT1/2-IN-2

    CAS:
    <p>SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).</p>
    Fórmula:C23H26F2O7
    Cor e Forma:Solid
    Peso molecular:452.451

    Ref: TM-T39966

  • Agaridoxin
    Targetmol
    + Info

    Agaridoxin

    CAS:
    <p>Agaridoxin is a mushroom metabolite.</p>
    Fórmula:C11H14N2O5
    Cor e Forma:Solid
    Peso molecular:254.242

    Ref: TM-T29709

  • Guanylate cyclase-IN-1
    Targetmol
    + Info

    Guanylate cyclase-IN-1

    CAS:
    <p>Guanylate cyclase-IN-1 (Example 46) is a specific inhibitor of guanylate cyclase, employed in research related to cardiovascular diseases.</p>
    Fórmula:C20H17FN8O
    Cor e Forma:Solid
    Peso molecular:404.409

    Ref: TM-T38770

  • O-Desmethyl Mebeverine alcohol hydrochloride
    Targetmol
    + Info

    O-Desmethyl Mebeverine alcohol hydrochloride

    CAS:
    <p>O-Desmethyl Mebeverine alcohol HCl, a metabolite of Mebeverine, is a strong α1 inhibitor, relaxing the GI tract.</p>
    Fórmula:C15H26ClNO2
    Cor e Forma:Solid
    Peso molecular:287.83

    Ref: TM-T75423

  • 17-trifluoromethylphenyl trinor Prostaglandin F2α ethyl amide
    Targetmol
    + Info

    17-trifluoromethylphenyl trinor Prostaglandin F2α ethyl amide

    CAS:
    <p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>
    Fórmula:C26H36F3NO4
    Cor e Forma:Solid
    Peso molecular:483.572

    Ref: TM-T37777

  • Tafluprost ethyl amide
    Targetmol
    + Info

    Tafluprost ethyl amide

    CAS:
    <p>Tafluprost ethyl amide is a prostaglandin derivative.</p>
    Fórmula:C24H33F2NO4
    Cor e Forma:Solid
    Peso molecular:437.52

    Ref: TM-T37956

  • 5-HT7R antagonist 1 free base
    Targetmol
    + Info

    5-HT7R antagonist 1 free base

    CAS:
    <p>5-HT7R antagonist 1 (free base) is a G protein-biased antagonist for the 5-HT 7 R receptor, with a dissociation constant (K i) of 6.5 nM.</p>
    Fórmula:C14H17ClN4
    Cor e Forma:Solid
    Peso molecular:276.77

    Ref: TM-T39870

  • YM 09538
    Targetmol
    + Info

    YM 09538

    CAS:
    <p>YM 09538 is a biochemical.</p>
    Fórmula:C18H25ClN2O5S
    Cor e Forma:Solid
    Peso molecular:416.92

    Ref: TM-T35252

  • HAEGT
    Targetmol
    + Info

    HAEGT

    CAS:
    <p>HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.</p>
    Fórmula:C20H31N7O9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:513.5

    Ref: TM-TP1381

  • Logotipo do CymitQuimica
    Targetmol
    + Info

    HDAC6-IN-49

    <p>HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.</p>
    Cor e Forma:Odour Solid

    Ref: TM-T200554

  • 2-Methyl-N,N-dimethyltryptamine
    Targetmol
    + Info

    2-Methyl-N,N-dimethyltryptamine

    CAS:
    <p>2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.</p>
    Fórmula:C13H18N2
    Cor e Forma:Solid
    Peso molecular:202.3

    Ref: TM-T203691

  • Pentagastrin meglumine
    Targetmol
    + Info

    Pentagastrin meglumine

    CAS:
    <p>Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.</p>
    Fórmula:C44H66N8O14S
    Cor e Forma:Solid
    Peso molecular:963.11

    Ref: TM-T33916

  • RF9 acetate
    Targetmol
    + Info

    RF9 acetate

    <p>RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.</p>
    Fórmula:C28H42N6O5
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:542.67

    Ref: TM-T16738L

  • Lys-[Des-Arg9]Bradykinin
    Targetmol
    + Info

    Lys-[Des-Arg9]Bradykinin

    CAS:
    Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.
    Fórmula:C50H73N13O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1032.21

    Ref: TM-TP1918

  • Logotipo do CymitQuimica
    Targetmol
    + Info

    GLP-1R agonist 29

    <p>GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.</p>
    Cor e Forma:Odour Solid

    Ref: TM-T206400

  • Logotipo do CymitQuimica
    Targetmol
    + Info

    Spns2-IN-2

    <p>Spns2-IN-2 (compound 3a) is an inhibitor of SPNS2.</p>
    Fórmula:C22H30ClN3O2
    Cor e Forma:Solid
    Peso molecular:403.95

    Ref: TM-T200979