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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5360 produtos de "GPCR/Proteína-G"

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  • L-796,778 acetate
    Targetmol
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    L-796,778 acetate

    <p>L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is &gt;1000nM.</p>
    Fórmula:C31H44N6O9
    Pureza:98%
    Cor e Forma:Soild
    Peso molecular:644.72

    Ref: TM-T32511L

  • 13,14-dihydro Prostaglandin F2α
    Targetmol
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    13,14-dihydro Prostaglandin F2α

    CAS:
    <p>13,14-dihydro Prostaglandin F2α (13,14-dihydro PGF2α) is the analog of PGF2α which has no unsaturation in the lower side chain.</p>
    Fórmula:C20H36O5
    Cor e Forma:Solid
    Peso molecular:356.503

    Ref: TM-T36146

  • Misoprostol
    Targetmol
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    Misoprostol

    CAS:
    <p>Misoprostol, a prostaglandin E1 derivative, has a strong inhibitory effect on gastric acid secretion, while having a contractile effect on pregnancy.</p>
    Fórmula:C22H38O5
    Pureza:99.78%
    Cor e Forma:Water-Soluble Viscous Liquid
    Peso molecular:382.53

    Ref: TM-T2573

  • ACTH (1-17)
    Targetmol
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    ACTH (1-17)

    CAS:
    <p>ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.</p>
    Fórmula:C95H145N29O23S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2093.41

    Ref: TM-TP1011

  • VU0453379
    Targetmol
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    VU0453379

    CAS:
    <p>VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).</p>
    Fórmula:C26H34N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.57

    Ref: TM-T17242

  • GLP-1 receptor agonist 8
    Targetmol
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    GLP-1 receptor agonist 8

    CAS:
    <p>GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.</p>
    Fórmula:C34H36ClFN6O4
    Cor e Forma:Solid
    Peso molecular:647.14

    Ref: TM-T74132

  • Logotipo do CymitQuimica
    Targetmol
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    Urocortin II, mouse

    CAS:
    <p>Mouse Urocortin II: Selective CRF2 agonist, Ki 0.66 nM for CRFR2, &gt;100 nM for CRFR1, affects central neural circuits.</p>
    Fórmula:C187H320N56O50
    Cor e Forma:Solid
    Peso molecular:4152.96

    Ref: TM-T76127

  • γ1-MSH
    Targetmol
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    γ1-MSH

    CAS:
    <p>Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4.</p>
    Fórmula:C72H97N21O14S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1512.76

    Ref: TM-TP1892

  • Dexchlorpheniramine free base
    Targetmol
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    Dexchlorpheniramine free base

    CAS:
    <p>Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.</p>
    Fórmula:C16H19ClN2
    Pureza:98%
    Cor e Forma:Oily Liquid Solid
    Peso molecular:274.79

    Ref: TM-T0785L

  • SB 258585
    Targetmol
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    SB 258585

    CAS:
    <p>SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.</p>
    Fórmula:C18H22IN3O3S
    Pureza:99.8%
    Cor e Forma:Soild
    Peso molecular:487.36

    Ref: TM-T23318L

  • (S)-Osanetant
    Targetmol
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    (S)-Osanetant

    CAS:
    <p>(S)-Osanetant, an S-enantiomer, is a selective NK3 antagonist with potential for treating schizophrenia and has anxiolytic and antidepressant effects.</p>
    Fórmula:C35H41Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:606.62

    Ref: TM-T74413

  • SFNGGP-NH2
    Targetmol
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    SFNGGP-NH2

    CAS:
    SFNGGP-NH2 is a biologically active peptide that interacts with Protease-Activated Receptor 3 (PAR-3), a high-affinity thrombin receptor.
    Fórmula:C25H36N8O8
    Cor e Forma:Solid
    Peso molecular:576.6

    Ref: TM-T80234

  • ARC 239 dihydrochloride
    Targetmol
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    ARC 239 dihydrochloride

    CAS:
    <p>ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).</p>
    Fórmula:C24H31Cl2N3O3
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:480.43

    Ref: TM-T22033

  • 4-Hydroxy MET
    Targetmol
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    4-Hydroxy MET

    CAS:
    4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.
    Fórmula:C13H18N2O
    Cor e Forma:Solid
    Peso molecular:218.3

    Ref: TM-T203151

  • RC-3095 TFA
    Targetmol
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    RC-3095 TFA

    CAS:
    <p>RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.</p>
    Fórmula:C58H80F3N15O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1220.34

    Ref: TM-TP1701

  • R 396
    Targetmol
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    R 396

    CAS:
    <p>R 396 (Acleu-asp-gln-trp-phe-glynh2) is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.</p>
    Fórmula:C39H51N9O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:805.88

    Ref: TM-T24697

  • M40
    Targetmol
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    M40

    CAS:
    <p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>
    Fórmula:C94H145N23O24
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1981.33

    Ref: TM-TP1992

  • Phoenixin-14 TFA
    Targetmol
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    Phoenixin-14 TFA

    <p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>
    Fórmula:C75H110N18O20·xC2HF3O2
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:1583.78 (free base)

    Ref: TM-T81485

  • ARL 15849XX
    Targetmol
    + Info

    ARL 15849XX

    CAS:
    <p>ARL 15849XX, a CCK-8 analog, is a novel anti-obesity agent.</p>
    Fórmula:C47H60N8O13S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:977.09

    Ref: TM-T25108

  • GS-2278
    Targetmol
    + Info

    GS-2278

    CAS:
    <p>GS-2278 is an antagonist of LPAR1 (lysophosphatidic acid receptor 1) with potential applications in the study of idiopathic pulmonary fibrosis (IPF).</p>
    Fórmula:C22H16F5N9O3
    Cor e Forma:Solid
    Peso molecular:549.41

    Ref: TM-T203480