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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5360 produtos de "GPCR/Proteína-G"

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  • Logotipo do CymitQuimica
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    Petrelintide acetate

    <p>Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.</p>
    Fórmula:C185H305N49O61·xC2H4O2
    Cor e Forma:Solid
    Peso molecular:4191.69 (free base)

    Ref: TM-TP3039

  • Logotipo do CymitQuimica
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    5-HT5AR/5-HT6R ligand-1

    <p>5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.</p>
    Fórmula:C25H30N4O2S
    Cor e Forma:Solid
    Peso molecular:450.6

    Ref: TM-T205096

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    Amylin (1-37), human acetate

    <p>Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.</p>
    Pureza:96.21%
    Cor e Forma:Odour Solid

    Ref: TM-T76480L

  • Xanthine amine congener dihydrochloride
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    Xanthine amine congener dihydrochloride

    CAS:
    <p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>
    Fórmula:C21H30Cl2N6O4
    Cor e Forma:Solid
    Peso molecular:501.41

    Ref: TM-T39387

  • DSP-1053
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    DSP-1053

    CAS:
    <p>Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.</p>
    Fórmula:C26H32BrNO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:502.44

    Ref: TM-T11107

  • [Des-His1,Glu9]-Glucagon amide
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    [Des-His1,Glu9]-Glucagon amide

    CAS:
    <p>Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.</p>
    Fórmula:C148H221N41O47S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3358.68

    Ref: TM-TP2033

  • GLP-1(7-37)
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    GLP-1(7-37)

    CAS:
    <p>GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.</p>
    Fórmula:C151H228N40O47
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3355.67

    Ref: TM-TP1306

  • Apelin-36(rat, mouse)
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    Apelin-36(rat, mouse)

    CAS:
    <p>Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.</p>
    Fórmula:C185H304N68O43S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4200.93

    Ref: TM-TP2094

  • (S)-Osanetant
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    (S)-Osanetant

    CAS:
    <p>(S)-Osanetant, an S-enantiomer, is a selective NK3 antagonist with potential for treating schizophrenia and has anxiolytic and antidepressant effects.</p>
    Fórmula:C35H41Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:606.62

    Ref: TM-T74413

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    Human growth hormone-releasing factor TFA

    <p>Human growth hormone-releasing factor TFA is a hypothalamic peptide that promotes GH secretion by targeting pituitary GHRHR.</p>
    Fórmula:C217H359F3N72O68S
    Cor e Forma:Solid
    Peso molecular:5153.67

    Ref: TM-T75713

  • [D-Trp34]-Neuropeptide Y
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    [D-Trp34]-Neuropeptide Y

    CAS:
    <p>Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.</p>
    Fórmula:C196H289N55O56
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4311.77

    Ref: TM-TP1984

  • Kadsurenin B
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    Kadsurenin B

    CAS:
    <p>Kadsurenin B, a platelet-activating factor (PAF) antagonist, exhibits neuroprotective properties and has a broad spectrum of pharmacological research</p>
    Fórmula:C20H22O5
    Cor e Forma:Solid
    Peso molecular:342.39

    Ref: TM-T79948

  • ARC 239 dihydrochloride
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    ARC 239 dihydrochloride

    CAS:
    <p>ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).</p>
    Fórmula:C24H31Cl2N3O3
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:480.43

    Ref: TM-T22033

  • PY-60
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    PY-60

    CAS:
    <p>PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.</p>
    Fórmula:C16H15N3O2S
    Pureza:99.5% - 99.67%
    Cor e Forma:Solid
    Peso molecular:313.37

    Ref: TM-T9566

  • Prostaglandin H1
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    Prostaglandin H1

    CAS:
    <p>Prostaglandin H1 is the cyclooxygenase metabolite of DGLA, a CRTh2 agonist and a precursor of a family of 1 anti-inflammatory prostaglandins.</p>
    Fórmula:C20H34O5
    Cor e Forma:Solid
    Peso molecular:354.487

    Ref: TM-T37328

  • SC 31391
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    SC 31391

    CAS:
    <p>SC 31391 is a PGE1 analog.</p>
    Fórmula:C24H32O6
    Cor e Forma:Solid
    Peso molecular:416.51

    Ref: TM-T34550

  • Benzomalvin A
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    Benzomalvin A

    CAS:
    <p>Benzomalvin A is a filamentous fungal secondary metabolite.</p>
    Fórmula:C24H19N3O2
    Cor e Forma:Solid
    Peso molecular:381.43

    Ref: TM-T30407

  • 4-P-PDOT
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    4-P-PDOT

    CAS:
    <p>4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.</p>
    Fórmula:C19H21NO
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:279.38

    Ref: TM-T14042

  • Logotipo do CymitQuimica
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    CCR6 antagonist 2

    <p>CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.</p>
    Fórmula:C19H24N4O4
    Cor e Forma:Solid
    Peso molecular:372.42

    Ref: TM-T205072

  • EP4-IN-1
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    EP4-IN-1

    CAS:
    <p>EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.</p>
    Fórmula:C27H24N2O4
    Pureza:99.94%
    Cor e Forma:Soild
    Peso molecular:440.49

    Ref: TM-T77699