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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5373 produtos de "GPCR/Proteína-G"

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  • (3aR,9aR)-Fluparoxan
    Targetmol
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H10FNO2
    Pureza:97.82%
    Cor e Forma:Soild
    Peso molecular:195.19

    Ref: TM-T77566

  • Ro 10-5824 dihydrochloride
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    Ro 10-5824 dihydrochloride

    CAS:
    Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).
    Fórmula:C17H22Cl2N4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:353.29

    Ref: TM-T12761

  • AH 6809
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Fórmula:C17H14O5
    Pureza:97.59%
    Cor e Forma:Solid
    Peso molecular:298.29

    Ref: TM-T14148

  • Methyldopa
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    Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21

    Ref: TM-T0505

  • Fluvoxamine maleate
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    Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:434.41

    Ref: TM-T1077

  • Dimenhydrinate
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    Dimenhydrinate

    CAS:
    <p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>
    Fórmula:C24H28ClN5O3
    Pureza:99.57% - 99.77%
    Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Peso molecular:469.96

    Ref: TM-T0298

  • (R)-Elagolix
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    (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Fórmula:C32H30F5N3O5
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:631.59

    Ref: TM-T11174

  • Olinciguat
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    Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Fórmula:C21H16F5N7O3
    Pureza:99.33% - 99.71%
    Cor e Forma:Solid
    Peso molecular:509.39

    Ref: TM-T16383

  • Fosopamine(HCl)
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    Fosopamine(HCl)

    CAS:
    <p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>
    Fórmula:C9H15ClNO5P
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:283.65

    Ref: TM-T68076L

  • MP-A08
    Targetmol
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    MP-A08

    CAS:
    <p>MP-A08 selectively inhibits SPHK1; targets SphK1 &amp; SphK2 with Ki of 6.9 μM &amp; 27 μM, respectively.</p>
    Fórmula:C27H25N3O4S2
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:519.64

    Ref: TM-T16128

  • Moxisylyte hydrochloride
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    Moxisylyte hydrochloride

    CAS:
    Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
    Fórmula:C16H26ClNO3
    Pureza:99.94% - ≥95%
    Cor e Forma:Solid
    Peso molecular:315.84

    Ref: TM-T0394

  • YNT-185
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    YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:615.74

    Ref: TM-T39229

  • Phenothiazine
    Targetmol
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    Phenothiazine

    CAS:
    <p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>
    Fórmula:C12H9NS
    Pureza:99.95%
    Cor e Forma:Yellow Solid Pellets
    Peso molecular:199.27

    Ref: TM-T0776

  • NEO 376
    Targetmol
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    NEO 376

    CAS:
    <p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>
    Fórmula:C20H24ClN3O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:357.88

    Ref: TM-T12207

  • Clonidine hydrochloride
    Targetmol
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    Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55

    Ref: TM-T1247

  • Ketanserin
    Targetmol
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    Ketanserin

    CAS:
    <p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>
    Fórmula:C22H22FN3O3
    Pureza:99.19% - 99.73%
    Cor e Forma:Solid
    Peso molecular:395.43

    Ref: TM-T1066

  • Metaproterenol hemisulfate
    Targetmol
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    Metaproterenol hemisulfate

    CAS:
    <p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>
    Fórmula:C11H17NO3·5H2O4S
    Pureza:98.53% - 99.74%
    Cor e Forma:Solid
    Peso molecular:260.3

    Ref: TM-T0277

  • Cyproheptadine hydrochloride sesquihydrate
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    Cyproheptadine hydrochloride sesquihydrate

    CAS:
    <p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>
    Fórmula:C21H24ClNO
    Pureza:99.77% - >99.99%
    Cor e Forma:White To Slightly Yellowish Crystalline Solid
    Peso molecular:341.88

    Ref: TM-T0174

  • Roxatidine Acetate hydrochloride
    Targetmol
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    Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Fórmula:C19H29ClN2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:384.9

    Ref: TM-T0157

  • Ezlopitant
    Targetmol
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    Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Fórmula:C31H38N2O
    Pureza:97.49%
    Cor e Forma:Solid
    Peso molecular:454.65

    Ref: TM-T68068