GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

Exibir 18 mais subcategorias

Foram encontrados 5696 produtos de "GPCR/Proteína-G"

Pureza (%)

100

produtos por página.

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Substance P, Free Acid
CAS:
- 71977-09-8
Substance P, Free Acid is a synthetic analog of native Substance P, however, it lacks the biological activity exhibited by Substance P.
Fórmula:C₆₃H₉₇N₁₇O₁₄S
Pureza:98%
Cor e Forma:Solid
Peso molecular:1348.61
Ref: TM-TP1788
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AL12180
CAS:
- 748816-43-5
AL12180 is a bioactive chemical.
Fórmula:C₂₁H₂₇ClO₆
Cor e Forma:Solid
Peso molecular:410.89
Ref: TM-T29810
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(±)12-HEPE
CAS:
- 81187-21-5
(±)12-HEPE is produced by non-enzymatic oxidation of EPA.
Fórmula:C₂₀H₃₀O₃
Cor e Forma:Solid
Peso molecular:318.457
Ref: TM-T35506
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BMS-196085
CAS:
- 170686-10-9
BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.
Fórmula:C₂₄H₂₆F₂N₂O₅S
Cor e Forma:Solid
Peso molecular:492.54
Ref: TM-T30504
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S1P2 antagonist 1
CAS:
- 2262402-83-3
S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.
Fórmula:C₂₃H₂₁ClN₄O₄
Cor e Forma:Solid
Peso molecular:452.9
Ref: TM-T39798
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Nemifitide diTFA
CAS:
- 204992-09-6
Nemifitide diTFA is a synthetic pentapeptide with antidepressant properties, resembling MIF, that crosses the blood-brain barrier.
Fórmula:C₃₇H₄₅F₇N₁₀O₁₀
Pureza:99.78% - 99.84%
Cor e Forma:Solid
Peso molecular:922.8
Ref: TM-TP1127
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[Tyr11]-Somatostatin
CAS:
- 59481-27-5
[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.
Fórmula:C₇₆H₁₀₄N₁₈O₂₀S₂
Peso molecular:1653.89
Ref: TM-T40680
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Levitide
CAS:
- 114281-19-5
Levitide is a neurohormone-like peptide which is from the skin of Xenopus laevis.
Fórmula:C₆₆H₁₁₉N₂₁O₁₉S
Pureza:98%
Cor e Forma:Solid
Peso molecular:1542.85
Ref: TM-T20704
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8-iso-15-keto Prostaglandin F2α
CAS:
- 191919-01-4
8-iso-15-keto Prostaglandin F2α (8-iso-15-keto PGF2α) is a metabolite of the isoprostane 8-iso PGF2α in rabbits, monkeys, and humans.
Fórmula:C₂₀H₃₂O₅
Cor e Forma:Solid
Peso molecular:352.471
Ref: TM-T36166
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AR ligand 40
AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.
Fórmula:C₂₁H₂₅N₅
Cor e Forma:Solid
Peso molecular:347.211
Ref: TM-T207383
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(R)-CJ 11974
CAS:
- 187281-35-2
(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.
Fórmula:C₃₁H₃₈N₂O
Pureza:97.15%
Cor e Forma:Soild
Peso molecular:454.65
Ref: TM-T68068L
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YFLLRNP
CAS:
- 149440-16-4
YFLLRNP is a biologically active peptide functioning as a partial agonist of PAR-1, selectively activating the G12/13 signaling pathway.
Fórmula:C₄₅H₆₇N₁₁O₁₀
Cor e Forma:Solid
Peso molecular:922.08
Ref: TM-T80235
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d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.
Fórmula:C₄₉H₇₁N₁₁O₁₃S₂
Pureza:98.86%
Cor e Forma:Solid
Peso molecular:1086.28
Ref: TM-TP1927L1
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PF-07062119
PF-07062119 is a humanized immunoglobulin G1 (IgG1) monoclonal antibody designed to target and inhibit GUCY2C.
Cor e Forma:Odour Liquid
Ref: TM-T9901A-899
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CH 275
CAS:
- 174688-78-9
Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.
Fórmula:C₇₄H₉₆N₁₄O₁₅S₂
Pureza:98%
Cor e Forma:Solid
Peso molecular:1485.8
Ref: TM-TP2045
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Hemokinin 1, human TFA
Hemokinin-1 is a human TFA and selective NK1 agonist; also activates NK2 & NK3 and induces opioid-independent analgesia.
Fórmula:C₅₆H₈₅F₃N₁₄O₁₆S
Cor e Forma:Solid
Peso molecular:1299.42
Ref: TM-T75840
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L-779976
CAS:
- 214770-19-1
L-779,976 is an agonist of somatostatin receptor.
Fórmula:C₃₃H₄₃N₇O₃
Cor e Forma:Solid
Peso molecular:585.74
Ref: TM-T27783
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M40
CAS:
- 143896-17-7
Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat
Fórmula:C₉₄H₁₄₅N₂₃O₂₄
Pureza:98%
Cor e Forma:Solid
Peso molecular:1981.33
Ref: TM-TP1992
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(D-Ala2)-GRF (1-29) amide (human)
CAS:
- 89453-59-8
(D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-
Fórmula:C₁₄₉H₂₄₆N₄₄O₄₂S
Peso molecular:3357.88
Ref: TM-T83549
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AL 34662
CAS:
- 210580-75-9
AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a
Fórmula:C₁₀H₁₃N₃O
Pureza:99.77%
Cor e Forma:Solid
Peso molecular:191.23
Ref: TM-T22029