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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5373 produtos de "GPCR/Proteína-G"

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  • Pizotifen
    Targetmol
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    Pizotifen

    CAS:
    <p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>
    Fórmula:C19H21NS
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:295.44

    Ref: TM-T1442

  • Silodosin
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    Silodosin

    CAS:
    Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
    Fórmula:C25H32F3N3O4
    Pureza:99.282% - 99.76%
    Cor e Forma:Colorless To Pink Solid
    Peso molecular:495.53

    Ref: TM-T1504

  • Rimonabant
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79

    Ref: TM-T1519L

  • ESI-05
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    ESI-05

    CAS:
    <p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>
    Fórmula:C16H18O2S
    Pureza:97.22%
    Cor e Forma:Solid
    Peso molecular:274.38

    Ref: TM-T15247

  • hGPR91 antagonist 1
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    hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:529.53

    Ref: TM-T11560

  • Duloxetine hydrochloride
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    Duloxetine hydrochloride

    CAS:
    <p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>
    Fórmula:C18H20ClNOS
    Pureza:99.93% - >99.99%
    Cor e Forma:White Or White Crystalline Powder
    Peso molecular:333.88

    Ref: TM-T1471

  • JNJ-18038683
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    JNJ-18038683

    CAS:
    <p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>
    Fórmula:C26H28ClN3O7
    Pureza:97.29%
    Cor e Forma:Solid
    Peso molecular:529.97

    Ref: TM-T11720

  • Asenapine Maleate
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    Asenapine Maleate

    CAS:
    Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.
    Fórmula:C21H20ClNO5
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:401.84

    Ref: TM-T1951

  • Urapidil hydrochloride
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    Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94

    Ref: TM-T0088

  • PF429242 dihydrochloride
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    PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Fórmula:C25H37Cl2N3O2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:482.49

    Ref: TM-T12437

  • Methyldopa
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    Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21

    Ref: TM-T0505

  • Nylidrin hydrochloride
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    Nylidrin hydrochloride

    CAS:
    <p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells &amp; human basophils.</p>
    Fórmula:C19H26ClNO2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:335.87

    Ref: TM-T0173

  • Naftopidil
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    Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49

    Ref: TM-T0696

  • Fluvoxamine maleate
    Targetmol
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    Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:434.41

    Ref: TM-T1077

  • Lafutidine
    Targetmol
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    Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Fórmula:C22H29N3O4S
    Pureza:98.55%
    Cor e Forma:Yellowish White Crystalline Powder
    Peso molecular:431.55

    Ref: TM-T0081

  • Prucalopride
    Targetmol
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    Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Fórmula:C18H26ClN3O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:367.87

    Ref: TM-T2542

  • Venlafaxine hydrochloride
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    Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Fórmula:C17H28ClNO2
    Pureza:97.32% - 99.86%
    Cor e Forma:White Crystalline Powder
    Peso molecular:313.86

    Ref: TM-T0472

  • Fluoxetine
    Targetmol
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    Fluoxetine

    CAS:
    <p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>
    Fórmula:C17H18F3NO
    Pureza:99.07% - 99.28%
    Cor e Forma:Solid
    Peso molecular:309.33

    Ref: TM-T0450

  • Talastine
    Targetmol
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    Talastine

    CAS:
    <p>Talastine is an antihistamine compound that can induce an allergic rash.</p>
    Fórmula:C19H21N3O
    Pureza:98.50% - 99.44%
    Cor e Forma:Solid
    Peso molecular:307.39

    Ref: TM-T68150

  • Imidazolidinyl urea
    Targetmol
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    Imidazolidinyl urea

    CAS:
    <p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>
    Fórmula:C11H16N8O8
    Pureza:98.6%
    Cor e Forma:White Fluid Powder With Slight Characteristic Odor
    Peso molecular:388.29

    Ref: TM-T0430