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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5373 produtos de "GPCR/Proteína-G"

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  • ML-180
    Targetmol
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    ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Fórmula:C20H25ClN4O2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:388.89

    Ref: TM-T12075

  • PF-06882961
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    PF-06882961

    CAS:
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Fórmula:C31H30FN5O4
    Pureza:97.19% - 99.56%
    Cor e Forma:Solid
    Peso molecular:555.6

    Ref: TM-T12431

  • Fluparoxan hydrochloride
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:231.65

    Ref: TM-T77565

  • Phenothiazine
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    Phenothiazine

    CAS:
    <p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>
    Fórmula:C12H9NS
    Pureza:99.95%
    Cor e Forma:Yellow Solid Pellets
    Peso molecular:199.27

    Ref: TM-T0776

  • JNJ-18038683
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    JNJ-18038683

    CAS:
    <p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>
    Fórmula:C26H28ClN3O7
    Pureza:97.29%
    Cor e Forma:Solid
    Peso molecular:529.97

    Ref: TM-T11720

  • Desipramine hydrochloride
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    Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Fórmula:C18H23ClN2
    Pureza:99.58% - 99.94%
    Cor e Forma:White To Off-White Powder
    Peso molecular:302.842

    Ref: TM-T0991

  • Levosulpiride
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43

    Ref: TM-T1211

  • Zolmitriptan
    Targetmol
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Fórmula:C16H21N3O2
    Pureza:99.69% - 99.91%
    Cor e Forma:White Or Kind Of White Powder
    Peso molecular:287.36

    Ref: TM-T1092

  • PF429242 dihydrochloride
    Targetmol
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    PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Fórmula:C25H37Cl2N3O2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:482.49

    Ref: TM-T12437

  • Urapidil hydrochloride
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    Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94

    Ref: TM-T0088

  • Cetirizine dihydrochloride
    Targetmol
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    Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Fórmula:C21H27Cl3N2O3
    Pureza:99.4% - 99.97%
    Cor e Forma:Solid
    Peso molecular:461.81

    Ref: TM-T0089

  • Ezlopitant
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    Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Fórmula:C31H38N2O
    Pureza:97.49%
    Cor e Forma:Solid
    Peso molecular:454.65

    Ref: TM-T68068

  • PF-610355 HCl
    Targetmol
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    PF-610355 HCl

    <p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>
    Fórmula:C19H22ClN7O6
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:479.87

    Ref: TM-T16509L

  • Granisetron hydrochloride
    Targetmol
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    Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:348.87

    Ref: TM-T1042

  • Olinciguat
    Targetmol
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    Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Fórmula:C21H16F5N7O3
    Pureza:99.33% - 99.71%
    Cor e Forma:Solid
    Peso molecular:509.39

    Ref: TM-T16383

  • NF-56-EJ40 hydrochloride
    Targetmol
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    NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Fórmula:C27H31Cl2N3O3
    Pureza:99.33%
    Cor e Forma:Soild
    Peso molecular:516.46

    Ref: TM-T12216L

  • Quetiapine
    Targetmol
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    Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:383.51

    Ref: TM-T0162

  • Naftopidil
    Targetmol
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    Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49

    Ref: TM-T0696

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Cor e Forma:Colourless Flake Crystalline Solid
    Peso molecular:448.39

    Ref: TM-T1566

  • Ornidazole
    Targetmol
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    Ornidazole

    CAS:
    <p>Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.</p>
    Fórmula:C7H10ClN3O3
    Pureza:99.47%
    Cor e Forma:Crystalline Solid
    Peso molecular:219.63

    Ref: TM-T1556