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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5373 produtos de "GPCR/Proteína-G"

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  • Cariprazine D6

    CAS:
    <p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>
    Fórmula:C21H26D6Cl2N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.45
  • Altanserin

    CAS:
    <p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>
    Fórmula:C22H22FN3O2S
    Cor e Forma:Solid
    Peso molecular:411.49
  • 4-Hydroxypropranolol-d7 hydrochloride

    CAS:
    <p>Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.</p>
    Fórmula:C16H22ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.85
  • Doxepin D3 Hydrochloride

    CAS:
    <p>Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and</p>
    Fórmula:C19H22ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.86
  • Substance P TFA

    CAS:
    <p>Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.</p>
    Fórmula:C65H99F3N18O15S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1461.67
  • Diacetolol D7

    CAS:
    <p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>
    Fórmula:C16H24N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:315.42
  • Rebamipide-d4

    CAS:
    <p>Rebamipide D4 is deuterium labeled Rebamipide.</p>
    Fórmula:C19H15ClN2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:374.81
  • R121919

    CAS:
    <p>R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.</p>
    Fórmula:C22H32N6
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:380.53
  • Diphenylpyraline

    CAS:
    <p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>
    Fórmula:C19H23NO
    Cor e Forma:Solid
    Peso molecular:281.39
  • Flibanserin-d4

    CAS:
    <p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>
    Fórmula:C20H21F3N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:394.43
  • Clozapine-d8

    CAS:
    <p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>
    Fórmula:C18H19ClN4
    Cor e Forma:Solid
    Peso molecular:334.87
  • Dapagliflozin impurity

    CAS:
    Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.
    Fórmula:C21H25ClO7
    Cor e Forma:Solid
    Peso molecular:424.87
  • Terlipressin

    CAS:
    <p>Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.</p>
    Fórmula:C52H74N16O15S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1227.37
  • Fipexide hydrochloride

    CAS:
    Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.
    Fórmula:C20H22Cl2N2O4
    Cor e Forma:Solid
    Peso molecular:425.31
  • Cefaclor

    CAS:
    Cefaclor (Panoral) is a cephalosporin antibiotic.
    Fórmula:C15H14ClN3O4S
    Pureza:99.03% - 99.98%
    Cor e Forma:Solid
    Peso molecular:367.81
  • Antazoline phosphate

    CAS:
    <p>Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.</p>
    Fórmula:C17H22N3O4P
    Pureza:98%
    Cor e Forma:Coa
    Peso molecular:363.35
  • NBI-27914

    CAS:
    <p>NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.</p>
    Fórmula:C18H20Cl4N4
    Pureza:99.47% - 99.64%
    Cor e Forma:Solid
    Peso molecular:434.19
  • Ramelteon-d5

    CAS:
    <p>Ramelteon-d5 is a deuterated compound of Ramelteon.</p>
    Fórmula:C16H16D5NO2
    Cor e Forma:Solid
    Peso molecular:264.37
  • SKF-82958 hydrobromide

    CAS:
    <p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>
    Fórmula:C19H21BrClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:410.73
  • Gizzerosine

    CAS:
    <p>Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.</p>
    Fórmula:C11H20N4O2
    Cor e Forma:Solid
    Peso molecular:240.3
  • Nadolol-d9

    CAS:
    <p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>
    Fórmula:C17H27NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.46
  • (R)-Praziquantel-d11

    CAS:
    <p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>
    Fórmula:C19H24N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:323.47
  • JNJ-10397049

    CAS:
    <p>OX2 receptor antagonist</p>
    Fórmula:C19H20Br2N2O3
    Cor e Forma:Solid
    Peso molecular:484.18
  • Clorprenaline

    CAS:
    <p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>
    Fórmula:C11H16ClNO
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:213.7
  • SB-674042

    CAS:
    <p>SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.</p>
    Fórmula:C24H21FN4O2S
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:448.51
  • LY223982

    CAS:
    LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.
    Fórmula:C30H30O7
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:502.56
  • Ozagrel Sodium

    CAS:
    <p>Ozagrel Sodium is a thromboxane A2 synthase inhibitor. It is used to treat cerebrovascular diseases.</p>
    Fórmula:C13H12N2NaO2
    Pureza:98%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:251.24
  • 5-HT3 antagonist 5

    CAS:
    <p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>
    Fórmula:C16H13N3O2
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:279.29
  • SLIGRL-NH2

    CAS:
    <p>SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.</p>
    Fórmula:C29H56N10O7
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:656.82
  • Dexloxiglumide

    CAS:
    Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.
    Fórmula:C21H30Cl2N2O5
    Cor e Forma:Solid
    Peso molecular:461.38
  • GLP-1R modulator C5

    CAS:
    <p>GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.</p>
    Fórmula:C24H21NO3
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:371.43
  • Aripiprazole (D8)

    CAS:
    <p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:456.44
  • Alimemazine D6

    CAS:
    <p>Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.</p>
    Fórmula:C18H22N2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:304.48
  • GLP-1R modulator C16

    CAS:
    <p>GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.</p>
    Fórmula:C21H26ClFN2O3
    Pureza:99.6% - >99.99%
    Cor e Forma:Solid
    Peso molecular:408.89
  • Virodhamine

    CAS:
    <p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>
    Fórmula:C22H37NO2
    Pureza:98%
    Cor e Forma:Soild
    Peso molecular:347.53
  • ML224

    CAS:
    <p>ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism.</p>
    Fórmula:C31H31N3O5
    Pureza:99.14%
    Cor e Forma:Solid
    Peso molecular:525.59
  • GLP-1R modulator L7-028

    CAS:
    <p>GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.</p>
    Fórmula:C24H28N2O3
    Pureza:98.76% - >99.99%
    Cor e Forma:Solid
    Peso molecular:392.49
  • 4,4-Diphenylbutylamine hydrochloride

    CAS:
    <p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>
    Fórmula:C16H20ClN
    Cor e Forma:Solid
    Peso molecular:261.79
  • Ipragliflozin (L-Proline)

    CAS:
    Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.
    Fórmula:C26H30FNO7S
    Cor e Forma:Solid
    Peso molecular:519.58
  • 3-O-Methyldopa-d3

    CAS:
    3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.
    Fórmula:C10H10D3NO4
    Peso molecular:214.23
  • SB-269970 hydrochloride

    CAS:
    <p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits &gt;50-fold selectivity</p>
    Fórmula:C18H28N2O3S·HCl
    Pureza:98.45%
    Cor e Forma:Solid
    Peso molecular:388.95
  • SB-277011 hydrochloride

    CAS:
    <p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>
    Fórmula:C28H31ClN4O
    Pureza:98.54%
    Cor e Forma:Solid
    Peso molecular:475.03
  • Glucagon (1-29), bovine, human, porcine

    CAS:
    Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.
    Fórmula:C153H225N43O49S
    Pureza:99.56% - 99.56%
    Cor e Forma:Solid
    Peso molecular:3482.75
  • Agomelatine-d6

    CAS:
    Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.
    Fórmula:C15H17NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:249.34
  • Apraclonidine hydrochloride

    CAS:
    <p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>
    Fórmula:C9H11Cl3N4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:281.57
  • Pimozide-d4

    CAS:
    <p>Pimozide D4 is a deuterium labeled Pimozide.</p>
    Fórmula:C28H29F2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:465.57
  • Quetiapine-d4 hemifumarate

    CAS:
    <p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>
    Fórmula:C25H29N3O6S
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:503.61
  • Methyldopate

    CAS:
    <p>Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.</p>
    Fórmula:C12H17NO4
    Cor e Forma:Solid
    Peso molecular:239.27
  • Zagociguat

    CAS:
    <p>Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and can be used in the research of neurological diseases.</p>
    Fórmula:C16H10F4N6
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:362.28
  • WAY-100635

    CAS:
    <p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>
    Fórmula:C25H34N4O2
    Pureza:98.972%
    Cor e Forma:Solid
    Peso molecular:422.56
  • Telcagepant

    CAS:
    Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.
    Fórmula:C26H27F5N6O3
    Pureza:98.98% - 98.98%
    Cor e Forma:Solid
    Peso molecular:566.52
  • Aramisulpride

    CAS:
    <p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>
    Fórmula:C17H27N3O4S
    Cor e Forma:Solid
    Peso molecular:369.48
  • Ziprasidone amino acid

    CAS:
    <p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>
    Fórmula:C21H23ClN4O2S
    Cor e Forma:Solid
    Peso molecular:430.95
  • PSB-0739

    CAS:
    <p>PSB-0739 Selective platelet P2Y12 receptor antagonist characterized by competitive binding with antithrombotic and platelet aggregation modulating effects.</p>
    Fórmula:C26H17N3Na2O8S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:609.54
  • Paliperidone Palmitate

    CAS:
    <p>Paliperidone: atypical antipsychotic, dopamine &amp; serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>
    Fórmula:C39H57FN4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:664.89
  • Spiroxatrine

    CAS:
    <p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>
    Fórmula:C22H25N3O3
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:379.45
  • Eticlopride hydrochloride

    CAS:
    <p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>
    Fórmula:C17H25ClN2O3·HCl
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:377.31
  • Bromperidol hydrochloride

    CAS:
    <p>Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.</p>
    Fórmula:C21H24BrClFNO2
    Cor e Forma:Solid
    Peso molecular:456.78
  • ST-836 hydrochloride

    CAS:
    ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .
    Fórmula:C23H35ClN4OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:451.07
  • Haloperidol (D4')

    CAS:
    Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.
    Fórmula:C21H23ClFNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:379.89
  • Emedastine Difumarate

    CAS:
    <p>Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.</p>
    Fórmula:C25H34N4O9
    Cor e Forma:Solid
    Peso molecular:534.56
  • YNT-185 dihydrochloride

    CAS:
    <p>Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.</p>
    Fórmula:C33H39Cl2N5O5S
    Cor e Forma:Solid
    Peso molecular:688.67
  • Tulobuterol-d9 HCl

    CAS:
    Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.
    Fórmula:C12H10D9Cl2NO
    Peso molecular:273.25
  • GLP-1 receptor agonist 7

    CAS:
    <p>GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.</p>
    Fórmula:C31H30ClFN4O5
    Cor e Forma:Solid
    Peso molecular:593.05
  • GSK682753A

    CAS:
    GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).
    Fórmula:C23H21Cl3N2O3
    Cor e Forma:Solid
    Peso molecular:479.78
  • Cetirizine D4

    CAS:
    <p>Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>
    Fórmula:C21H25ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:392.91
  • Benoxathian hydrochloride

    CAS:
    <p>Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.</p>
    Fórmula:C19H24ClNO4S
    Cor e Forma:Solid
    Peso molecular:397.91
  • Revdofilimab

    CAS:
    <p>Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.</p>
    Pureza:98.80% - 98.80%
    Cor e Forma:Liquid
  • Nefazodone

    CAS:
    <p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>
    Fórmula:C25H32ClN5O2
    Pureza:99.85%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:470.01
  • Fedovapagon

    CAS:
    <p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>
    Fórmula:C27H34N4O3
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:462.58
  • Omidenepag

    CAS:
    Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.
    Fórmula:C23H22N6O4S
    Pureza:99.67% - 99.77%
    Cor e Forma:Solid
    Peso molecular:478.52
  • MRGPRX4 modulator-2

    CAS:
    MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value of less than 100 nM. Its notable applications include research on autoimmune diseases such as psoriasis, multiple sclerosis, Steven Johnson's Syndrome, and various chronic itch conditions [1].
    Fórmula:C15H9ClF4O3
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:348.68
  • (S)-(+)-Dimethindene maleate

    CAS:
    <p>(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors</p>
    Fórmula:C24H28N2O4
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:408.49
  • Asenapine hydrochloride

    CAS:
    <p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>
    Fórmula:C17H17Cl2NO
    Cor e Forma:Solid
    Peso molecular:322.23
  • V-0219

    CAS:
    <p>V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.</p>
    Fórmula:C20H25F3N4O2
    Pureza:99.91%
    Cor e Forma:Soild
    Peso molecular:410.43
  • LAS101057

    CAS:
    LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
    Fórmula:C18H14FN5O
    Pureza:99.03% - >99.99%
    Cor e Forma:Solid
    Peso molecular:335.34
  • rac-Propranolol-d7

    CAS:
    Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.
    Fórmula:C16H14D7NO2
    Cor e Forma:Solid
    Peso molecular:266.39
  • Travoprost (Standard)

    CAS:
    Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.
    Fórmula:C26H35F3O6
    Peso molecular:500.55
  • Agomelatine (L(+)-Tartaric acid)

    CAS:
    <p>Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and</p>
    Fórmula:C19H23NO8
    Cor e Forma:Solid
    Peso molecular:393.39
  • SYL-4

    CAS:
    SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.
    Fórmula:C20H15N3O5S
    Pureza:95.76%
    Cor e Forma:Soild
    Peso molecular:409.42
  • Tegaserod

    CAS:
    <p>Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).</p>
    Fórmula:C16H23N5O
    Pureza:99.20% - 99.89%
    Cor e Forma:Solid
    Peso molecular:301.39
  • WZ4141

    CAS:
    WZ4141 is an intermediate in compound synthesis.
    Fórmula:C16H13N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:279.29
  • Eplivanserin (mixture)

    CAS:
    <p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>
    Fórmula:C19H21FN2O2
    Cor e Forma:Solid
    Peso molecular:328.387
  • Granisetron

    CAS:
    <p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>
    Fórmula:C18H24N4O
    Cor e Forma:Solid
    Peso molecular:312.41
  • Pramipexole dihydrochloride

    CAS:
    Pramipexole dihydrochloride could be used to treat Parkinson disease.
    Fórmula:C10H18ClN3S
    Pureza:98%
    Cor e Forma:White Crystalline Powder
    Peso molecular:247.79
  • Sumatriptan

    CAS:
    <p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>
    Fórmula:C14H21N3O2S
    Pureza:99.93%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:295.4
  • Cimbuterol-d9

    CAS:
    <p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>
    Fórmula:C13H10D9N3O
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:242.37
  • UCSF924

    CAS:
    <p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>
    Fórmula:C20H22N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:322.4
  • GR79236

    CAS:
    GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
    Fórmula:C15H21N5O5
    Cor e Forma:Solid
    Peso molecular:351.36
  • Asenapine

    CAS:
    <p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>
    Fórmula:C17H16ClNO
    Pureza:99.64%
    Cor e Forma:Coa
    Peso molecular:285.77
  • PD176252

    CAS:
    <p>PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.</p>
    Fórmula:C32H36N6O5
    Pureza:99.18%
    Cor e Forma:Solid
    Peso molecular:584.67
  • Tiapride-d3


    Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.
    Fórmula:C15H21D3N2O4S
    Cor e Forma:Solid
    Peso molecular:331.45
  • Taranabant racemate

    CAS:
    <p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>
    Fórmula:C27H25ClF3N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:515.95
  • TP-16

    CAS:
    <p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>
    Fórmula:C24H22FNO4S
    Pureza:98.53% - 99.15%
    Cor e Forma:Solid
    Peso molecular:439.5
  • Clothiapine

    CAS:
    Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
    Fórmula:C18H18ClN3S
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:343.87
  • Zilpaterol-d7

    CAS:
    <p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>
    Fórmula:C14H12D7N3O2
    Cor e Forma:Solid
    Peso molecular:268.36
  • Argipressin

    CAS:
    <p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>
    Fórmula:C46H65N15O12S2
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:1084.23
  • Thiethylperazine

    CAS:
    <p>Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.</p>
    Fórmula:C22H29N3S2
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:399.62
  • L-798106

    CAS:
    L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.
    Fórmula:C27H22BrNO4S
    Pureza:98.97%
    Cor e Forma:Solid
    Peso molecular:536.44
  • MRS-3777 hemioxalate

    CAS:
    <p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>
    Fórmula:C17H19N5OC2H2O4
    Pureza:97.10%
    Cor e Forma:Solid
    Peso molecular:354.39
  • Clencyclohexerol-d10

    CAS:
    <p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>
    Fórmula:C14H20Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:329.29
  • Furprofen

    CAS:
    Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.
    Fórmula:C14H12O4
    Pureza:98.62% - 99.25%
    Cor e Forma:Solid
    Peso molecular:244.24
  • Levomepromazine

    CAS:
    Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.
    Fórmula:C19H24N2OS
    Pureza:99.15%
    Cor e Forma:Solid
    Peso molecular:328.47
  • BMS-986224

    CAS:
    <p>BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.</p>
    Fórmula:C24H23ClN4O6
    Pureza:98.61% - 99.67%
    Cor e Forma:Solid
    Peso molecular:498.92
  • 3-Hydroxy agomelatine

    CAS:
    <p>3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.</p>
    Fórmula:C15H17NO3
    Cor e Forma:Solid
    Peso molecular:259.3
  • Docosahexaenoic acid ethyl ester

    CAS:
    <p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>
    Fórmula:C24H36O2
    Cor e Forma:Solid
    Peso molecular:356.54
  • SB-200646A

    CAS:
    SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.
    Fórmula:C15H15ClN4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:302.76
  • Sumanirole maleate

    CAS:
    <p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>
    Fórmula:C15H17N3O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:319.31
  • cis-(Z)-Flupentixol dihydrochloride

    CAS:
    <p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:507.44
  • Calcitonin (salmon)

    CAS:
    <p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>
    Fórmula:C145H240N44O48S2
    Pureza:99.41% - 99.80%
    Cor e Forma:Powder
    Peso molecular:3431.85
  • Scopine hydrochloride

    CAS:
    <p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>
    Fórmula:C8H13NO2·HCl
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:191.66
  • SANT 2

    CAS:
    <p>SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.</p>
    Fórmula:C26H26ClN3O4
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:479.96
  • Neurotensin(8-13)

    CAS:
    <p>Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>
    Fórmula:C38H64N12O8
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:816.99
  • EST64454 Maleic acid salt

    CAS:
    <p>EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.</p>
    Fórmula:C22H26F2N4O6
    Pureza:97.54%
    Cor e Forma:Solid
    Peso molecular:480.46
  • Asapiprant

    CAS:
    <p>Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.</p>
    Fórmula:C24H27N3O7S
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:501.55
  • [Pyr1]-Apelin-13

    CAS:
    [Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.
    Fórmula:C69H108N22O16S
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:1533.8
  • Lecirelin acetate(61012-19-9 free base)


    <p>Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts</p>
    Fórmula:C61H88N16O14
    Pureza:98.1%
    Cor e Forma:Solid
    Peso molecular:1269.45
  • Nelociguat

    CAS:
    <p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>
    Fórmula:C19H17FN8O2
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:408.39
  • Neurokinin A

    CAS:
    <p>Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.</p>
    Fórmula:C50H80N14O14S
    Pureza:>99.99%
    Cor e Forma:White To Off-White Lyophilized Solid
    Peso molecular:1133.32
  • Prazosin

    CAS:
    <p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>
    Fórmula:C19H21N5O4
    Pureza:99.86%
    Cor e Forma:White To Tan Powder Solid
    Peso molecular:383.4
  • Phenylbiguanide

    CAS:
    <p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>
    Fórmula:C8H11N5
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:177.21
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Cor e Forma:Solid
    Peso molecular:538.64
  • 5-Benzyloxygramine

    CAS:
    5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
    Fórmula:C18H20N2O
    Pureza:99.13%
    Cor e Forma:Solid
    Peso molecular:280.36
  • Lys-[Des-Arg9]Bradykinin acetate


    <p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and &gt; 30000 nM at human B1 and</p>
    Fórmula:C52H77N13O13
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:1092.27
  • Arformoterol Tartrate

    CAS:
    <p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>
    Fórmula:C23H30N2O10
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:494.49
  • I-191

    CAS:
    <p>I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.</p>
    Fórmula:C23H26FN5O2
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:423.48
  • M40 acetate(143896-17-7 free base)


    <p>M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29)</p>
    Fórmula:C96H149N23O26
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:2041.38
  • Zatebradine

    CAS:
    <p>Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).</p>
    Fórmula:C26H36N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:456.57
  • Grapiprant

    CAS:
    <p>Grapiprant (AAT-007) is a selective EP4 receptor antagonist.</p>
    Fórmula:C26H29N5O3S
    Pureza:99.49% - 99.843%
    Cor e Forma:Solid
    Peso molecular:491.61
  • Ursodeoxycholic acid sodium

    CAS:
    <p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>
    Fórmula:C24H40NaO4
    Pureza:99.66% - 99.96%
    Cor e Forma:Solid
    Peso molecular:415.56
  • Dimethocaine

    CAS:
    <p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>
    Fórmula:C16H26N2O2
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:278.39
  • ML-184

    CAS:
    <p>ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.</p>
    Fórmula:C25H34N4O3S
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:470.63
  • Hemokinin 1 (human) acetate(491851-53-7 free base)


    <p>Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.</p>
    Fórmula:C56H88N14O16S
    Pureza:97.82%
    Cor e Forma:Solid
    Peso molecular:1245.45
  • Ataciguat

    CAS:
    <p>Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.</p>
    Fórmula:C21H19Cl2N3O6S3
    Pureza:99.09%
    Cor e Forma:Solid
    Peso molecular:576.49
  • Lerisetron

    CAS:
    <p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>
    Fórmula:C18H20N4
    Pureza:99.15% - 99.82%
    Cor e Forma:Solid
    Peso molecular:292.38
  • M871 acetate


    <p>M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptive</p>
    Fórmula:C110H167N27O30
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:2347.67
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Fórmula:C25H29N5O
    Pureza:99.2%
    Cor e Forma:Solid
    Peso molecular:415.53
  • Betahistine EP Impurity C

    CAS:
    <p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>
    Fórmula:C15H19N3
    Pureza:≥95%
    Cor e Forma:Solid
    Peso molecular:241.33
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Fórmula:C12H17ClN2O2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:256.73
  • Guanfacine hydrochloride

    CAS:
    <p>Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.</p>
    Fórmula:C9H10Cl3N3O
    Pureza:99.89% - 99.91%
    Cor e Forma:Solid
    Peso molecular:282.55
  • Pizuglanstat

    CAS:
    <p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>
    Fórmula:C27H36N6O4
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:508.61
  • Plecanatide

    CAS:
    <p>Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.</p>
    Fórmula:C65H104N18O26S4
    Pureza:97.51%
    Cor e Forma:Solid
    Peso molecular:1681.89
  • Melanin Concentrating Hormone, salmon acetate


    <p>Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>
    Fórmula:C91H143N27O26S4
    Pureza:99.41%
    Cor e Forma:Solid
    Peso molecular:2157
  • Azaperone

    CAS:
    <p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>
    Fórmula:C19H22FN3O
    Pureza:98.73%
    Cor e Forma:White Or Off-White Crystalline
    Peso molecular:327.4
  • Metoclopramide hydrochloride hydrate

    CAS:
    <p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>
    Fórmula:C14H25Cl2N3O3
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:354.27
  • Galanin Receptor Ligand M35 TFA


    <p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>
    Fórmula:C109H154N27F3O28
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:2347.62
  • Histrelin acetate

    CAS:
    <p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>
    Fórmula:C68H90N18O14
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:1383.55
  • TY-52156

    CAS:
    <p>TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).</p>
    Fórmula:C18H19Cl2N3O
    Pureza:99.91% - 99.91%
    Cor e Forma:Solid
    Peso molecular:364.27
  • [D-Phe12,Leu14]-Bombesin acetate


    <p>[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>
    Fórmula:C77H118N22O20
    Pureza:98.41% - 99.14%
    Cor e Forma:Solid
    Peso molecular:1671.9
  • RS102895

    CAS:
    <p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>
    Fórmula:C21H21F3N2O2
    Pureza:97.64% - 99.80%
    Cor e Forma:Solid
    Peso molecular:390.4
  • SAG

    CAS:
    <p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>
    Fórmula:C28H28ClN3OS
    Pureza:97.37% - 98.88%
    Cor e Forma:Solid
    Peso molecular:490.06
  • Ciliobrevin A

    CAS:
    <p>Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 &lt;10 μM.</p>
    Fórmula:C17H9Cl2N3O2
    Pureza:98.54% - 99.57%
    Cor e Forma:Solid
    Peso molecular:358.18
  • Taprenepag

    CAS:
    <p>Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).</p>
    Fórmula:C24H22N4O5S
    Pureza:98.89% - 99.15%
    Cor e Forma:Solid
    Peso molecular:478.52
  • MF-766

    CAS:
    <p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>
    Fórmula:C27H21F3N2O3
    Pureza:99.54% - 99.59%
    Cor e Forma:Solid
    Peso molecular:478.46
  • SKF 38393 hydrochloride

    CAS:
    <p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>
    Fórmula:C16H17NO2·HCl
    Pureza:99.1% - 99.51%
    Cor e Forma:Solid
    Peso molecular:291.77
  • SANT-1

    CAS:
    <p>SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).</p>
    Fórmula:C23H27N5
    Pureza:99.98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:373.49
  • MRT-10

    CAS:
    <p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>
    Fórmula:C24H23N3O5S
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:465.52
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Fórmula:C19H21ClF2N4O
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:394.85
  • Ondansetron

    CAS:
    <p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>
    Fórmula:C18H19N3O
    Pureza:99.92%
    Cor e Forma:White To Yellow Crystals
    Peso molecular:293.36
  • ICI 89406

    CAS:
    <p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>
    Fórmula:C19H22N4O3
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:354.4
  • RE-640

    CAS:
    <p>NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.</p>
    Fórmula:C20H16Cl2N4
    Pureza:99.60% - 99.87%
    Cor e Forma:Solid
    Peso molecular:383.27
  • Vercirnon

    CAS:
    <p>Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.</p>
    Fórmula:C22H21ClN2O4S
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:444.93
  • Lixisenatide acetate (320367-13-3 free base)

    CAS:
    <p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>
    Fórmula:C215H347N61O65S·6C2H4O2
    Pureza:98% - 99.9%
    Cor e Forma:Solid
    Peso molecular:5218.88
  • SAG hydrochloride (912545-86-9(free base))

    CAS:
    <p>SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.</p>
    Fórmula:C28H29Cl2N3OS
    Pureza:99.19% - 99.77%
    Cor e Forma:Solid
    Peso molecular:526.52
  • R243

    CAS:
    <p>R243 is CCR8 signaling and chemotaxis inhibitor.</p>
    Fórmula:C21H27NO4
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:357.44
  • A2B receptor antagonist 2

    CAS:
    <p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>
    Fórmula:C12H15N5
    Pureza:100%
    Cor e Forma:Solid
    Peso molecular:229.28
  • Mequitazine

    CAS:
    Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
    Fórmula:C20H22N2S
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:322.47
  • Sonidegib

    CAS:
    <p>Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.</p>
    Fórmula:C26H26F3N3O3
    Pureza:98% - 99.97%
    Cor e Forma:Solid
    Peso molecular:485.5
  • Salmeterol Xinafoate

    CAS:
    <p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>
    Fórmula:C36H45NO7
    Pureza:98% - 98.24%
    Cor e Forma:White Solid
    Peso molecular:603.75
  • MRT-81

    CAS:
    <p>MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.</p>
    Fórmula:C31H29N3O5S
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:555.64
  • SB297006

    CAS:
    <p>SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.</p>
    Fórmula:C18H18N2O5
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:342.35
  • Emorfazone

    CAS:
    Emorfazone (PH011085) has an anti-nociceptive effect.
    Fórmula:C11H17N3O3
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:239.27
  • BAY-545

    CAS:
    <p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>
    Fórmula:C18H22F3N3O4S
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:433.45
  • Felypressin

    CAS:
    <p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>
    Fórmula:C46H65N13O11S2
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:1040.22
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Fórmula:C19H29ClN2O2
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:352.9
  • Tolnapersine

    CAS:
    <p>Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.</p>
    Fórmula:C21H26N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:322.44
  • Geissoschizine methyl ether

    CAS:
    <p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>
    Fórmula:C22H26N2O3
    Pureza:99.24% - 99.68%
    Cor e Forma:Solid
    Peso molecular:366.45
  • GRA Ex-25

    CAS:
    <p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>
    Fórmula:C29H36F3N3O5
    Pureza:98.2% - 98.88%
    Cor e Forma:Solid
    Peso molecular:563.61
  • Calcitonin(salmon) Acetate(47931-85-1(free base))


    <p>Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5</p>
    Fórmula:C145H240N44O48S2
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:3431.85
  • MK-1064

    CAS:
    <p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>
    Fórmula:C24H20ClN5O3
    Pureza:99.19% - 99.82%
    Cor e Forma:Solid
    Peso molecular:461.9
  • VUF10460

    CAS:
    <p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>
    Fórmula:C15H19N5
    Pureza:99.44% - 99.57%
    Cor e Forma:Solid
    Peso molecular:269.34
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Cor e Forma:Solid
    Peso molecular:379.36
  • SAX-187

    CAS:
    <p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>
    Fórmula:C15H13ClN4O2S2
    Pureza:97.82% - 98%
    Cor e Forma:Solid
    Peso molecular:380.87
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Cor e Forma:Solid
    Peso molecular:417.97
  • Treprostinil

    CAS:
    <p>Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).</p>
    Fórmula:C23H34O5
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:390.51
  • BA 1 acetate(183241-31-8 free base)


    <p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>
    Fórmula:C59H80N14O13
    Pureza:95.3%
    Cor e Forma:Solid
    Peso molecular:1193.35
  • Desmopressin acetate (16679-58-6 free base)

    CAS:
    <p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>
    Fórmula:C48H68N14O14S2
    Pureza:98.84% - >99.99%
    Cor e Forma:Solid
    Peso molecular:1129.26
  • VPC171

    CAS:
    <p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>
    Fórmula:C18H12F3NOS
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:347.35
  • Binodenoson

    CAS:
    <p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>
    Fórmula:C17H25N7O4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:391.42
  • Opromazine hydrochloride

    CAS:
    <p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>
    Fórmula:C17H20Cl2N2OS
    Pureza:98.03%
    Cor e Forma:Solid
    Peso molecular:371.32
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Fórmula:C18H15BrF2N4O2
    Pureza:98.42% - 99.88%
    Cor e Forma:Solid
    Peso molecular:437.24
  • Human growth hormone-releasing factor acetate


    Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on
    Pureza:99.26%
    Cor e Forma:Liquid
    Peso molecular:N/A
  • Aprepitant

    CAS:
    <p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>
    Fórmula:C23H21F7N4O3
    Pureza:98% - 99.68%
    Cor e Forma:Off-White To Light Yellow Cyrstalline Solid
    Peso molecular:534.43
  • AM095

    CAS:
    <p>AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.</p>
    Fórmula:C27H23N2NaO5
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:478.47
  • Urotensin I acetate (83930-33-0 Free base)


    Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.
    Pureza:95.44% - 99.73%
    Cor e Forma:Solid
    Peso molecular:N/A
  • Sevoflurane

    CAS:
    <p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>
    Fórmula:C4H3F7O
    Pureza:98%
    Cor e Forma:Less Oil Colorless Oil
    Peso molecular:200.05
  • ML-SI3

    CAS:
    <p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>
    Fórmula:C23H31N3O3S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:429.58
  • CCG215022

    CAS:
    <p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>
    Fórmula:C26H22FN7O3
    Pureza:97.63% - 99.69%
    Cor e Forma:Solid
    Peso molecular:499.5
  • Clemizole hydrochloride

    CAS:
    Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.
    Fórmula:C19H21Cl2N3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:362.3
  • Pancreatic Polypeptide (human) acetate


    Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.
    Pureza:97.26%
    Cor e Forma:Liquid
    Peso molecular:N/A