
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Fórmula:C21H26D6Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:433.45Altanserin
CAS:<p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>Fórmula:C22H22FN3O2SCor e Forma:SolidPeso molecular:411.494-Hydroxypropranolol-d7 hydrochloride
CAS:<p>Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.</p>Fórmula:C16H22ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:318.85Doxepin D3 Hydrochloride
CAS:<p>Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and</p>Fórmula:C19H22ClNOPureza:98%Cor e Forma:SolidPeso molecular:318.86Substance P TFA
CAS:<p>Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.</p>Fórmula:C65H99F3N18O15SPureza:98%Cor e Forma:SolidPeso molecular:1461.67Diacetolol D7
CAS:<p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>Fórmula:C16H24N2O4Pureza:98%Cor e Forma:SolidPeso molecular:315.42Rebamipide-d4
CAS:<p>Rebamipide D4 is deuterium labeled Rebamipide.</p>Fórmula:C19H15ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:374.81R121919
CAS:<p>R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.</p>Fórmula:C22H32N6Pureza:99.75%Cor e Forma:SolidPeso molecular:380.53Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Fórmula:C19H23NOCor e Forma:SolidPeso molecular:281.39Flibanserin-d4
CAS:<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Fórmula:C20H21F3N4OPureza:98%Cor e Forma:SolidPeso molecular:394.43Clozapine-d8
CAS:<p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>Fórmula:C18H19ClN4Cor e Forma:SolidPeso molecular:334.87Dapagliflozin impurity
CAS:Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Fórmula:C21H25ClO7Cor e Forma:SolidPeso molecular:424.87Terlipressin
CAS:<p>Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.</p>Fórmula:C52H74N16O15S2Pureza:98%Cor e Forma:SolidPeso molecular:1227.37Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Fórmula:C20H22Cl2N2O4Cor e Forma:SolidPeso molecular:425.31Cefaclor
CAS:Cefaclor (Panoral) is a cephalosporin antibiotic.Fórmula:C15H14ClN3O4SPureza:99.03% - 99.98%Cor e Forma:SolidPeso molecular:367.81Antazoline phosphate
CAS:<p>Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.</p>Fórmula:C17H22N3O4PPureza:98%Cor e Forma:CoaPeso molecular:363.35NBI-27914
CAS:<p>NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.</p>Fórmula:C18H20Cl4N4Pureza:99.47% - 99.64%Cor e Forma:SolidPeso molecular:434.19Ramelteon-d5
CAS:<p>Ramelteon-d5 is a deuterated compound of Ramelteon.</p>Fórmula:C16H16D5NO2Cor e Forma:SolidPeso molecular:264.37SKF-82958 hydrobromide
CAS:<p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>Fórmula:C19H21BrClNO2Pureza:98%Cor e Forma:SolidPeso molecular:410.73Gizzerosine
CAS:<p>Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.</p>Fórmula:C11H20N4O2Cor e Forma:SolidPeso molecular:240.3Nadolol-d9
CAS:<p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>Fórmula:C17H27NO4Pureza:98%Cor e Forma:SolidPeso molecular:318.46(R)-Praziquantel-d11
CAS:<p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:323.47JNJ-10397049
CAS:<p>OX2 receptor antagonist</p>Fórmula:C19H20Br2N2O3Cor e Forma:SolidPeso molecular:484.18Clorprenaline
CAS:<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Fórmula:C11H16ClNOPureza:98.9%Cor e Forma:SolidPeso molecular:213.7SB-674042
CAS:<p>SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.</p>Fórmula:C24H21FN4O2SPureza:99.9%Cor e Forma:SolidPeso molecular:448.51LY223982
CAS:LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.Fórmula:C30H30O7Pureza:99.86%Cor e Forma:SolidPeso molecular:502.56Ozagrel Sodium
CAS:<p>Ozagrel Sodium is a thromboxane A2 synthase inhibitor. It is used to treat cerebrovascular diseases.</p>Fórmula:C13H12N2NaO2Pureza:98%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:251.245-HT3 antagonist 5
CAS:<p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>Fórmula:C16H13N3O2Pureza:99.84%Cor e Forma:SolidPeso molecular:279.29SLIGRL-NH2
CAS:<p>SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.</p>Fórmula:C29H56N10O7Pureza:98.29%Cor e Forma:SolidPeso molecular:656.82Dexloxiglumide
CAS:Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.Fórmula:C21H30Cl2N2O5Cor e Forma:SolidPeso molecular:461.38GLP-1R modulator C5
CAS:<p>GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.</p>Fórmula:C24H21NO3Pureza:99.59%Cor e Forma:SolidPeso molecular:371.43Aripiprazole (D8)
CAS:<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Fórmula:C23H27Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:456.44Alimemazine D6
CAS:<p>Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.</p>Fórmula:C18H22N2SPureza:98%Cor e Forma:SolidPeso molecular:304.48GLP-1R modulator C16
CAS:<p>GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.</p>Fórmula:C21H26ClFN2O3Pureza:99.6% - >99.99%Cor e Forma:SolidPeso molecular:408.89Virodhamine
CAS:<p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>Fórmula:C22H37NO2Pureza:98%Cor e Forma:SoildPeso molecular:347.53ML224
CAS:<p>ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism.</p>Fórmula:C31H31N3O5Pureza:99.14%Cor e Forma:SolidPeso molecular:525.59GLP-1R modulator L7-028
CAS:<p>GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.</p>Fórmula:C24H28N2O3Pureza:98.76% - >99.99%Cor e Forma:SolidPeso molecular:392.494,4-Diphenylbutylamine hydrochloride
CAS:<p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>Fórmula:C16H20ClNCor e Forma:SolidPeso molecular:261.79Ipragliflozin (L-Proline)
CAS:Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.Fórmula:C26H30FNO7SCor e Forma:SolidPeso molecular:519.583-O-Methyldopa-d3
CAS:3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Fórmula:C10H10D3NO4Peso molecular:214.23SB-269970 hydrochloride
CAS:<p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity</p>Fórmula:C18H28N2O3S·HClPureza:98.45%Cor e Forma:SolidPeso molecular:388.95SB-277011 hydrochloride
CAS:<p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>Fórmula:C28H31ClN4OPureza:98.54%Cor e Forma:SolidPeso molecular:475.03Glucagon (1-29), bovine, human, porcine
CAS:Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.Fórmula:C153H225N43O49SPureza:99.56% - 99.56%Cor e Forma:SolidPeso molecular:3482.75Agomelatine-d6
CAS:Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Fórmula:C15H17NO2Pureza:98%Cor e Forma:SolidPeso molecular:249.34Apraclonidine hydrochloride
CAS:<p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>Fórmula:C9H11Cl3N4Pureza:99.74%Cor e Forma:SolidPeso molecular:281.57Pimozide-d4
CAS:<p>Pimozide D4 is a deuterium labeled Pimozide.</p>Fórmula:C28H29F2N3OPureza:98%Cor e Forma:SolidPeso molecular:465.57Quetiapine-d4 hemifumarate
CAS:<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Fórmula:C25H29N3O6SPureza:98%Cor e Forma:White SolidPeso molecular:503.61Methyldopate
CAS:<p>Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.</p>Fórmula:C12H17NO4Cor e Forma:SolidPeso molecular:239.27Zagociguat
CAS:<p>Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and can be used in the research of neurological diseases.</p>Fórmula:C16H10F4N6Pureza:99.37%Cor e Forma:SolidPeso molecular:362.28WAY-100635
CAS:<p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>Fórmula:C25H34N4O2Pureza:98.972%Cor e Forma:SolidPeso molecular:422.56Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Fórmula:C26H27F5N6O3Pureza:98.98% - 98.98%Cor e Forma:SolidPeso molecular:566.52Aramisulpride
CAS:<p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>Fórmula:C17H27N3O4SCor e Forma:SolidPeso molecular:369.48Ziprasidone amino acid
CAS:<p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>Fórmula:C21H23ClN4O2SCor e Forma:SolidPeso molecular:430.95PSB-0739
CAS:<p>PSB-0739 Selective platelet P2Y12 receptor antagonist characterized by competitive binding with antithrombotic and platelet aggregation modulating effects.</p>Fórmula:C26H17N3Na2O8S2Pureza:98%Cor e Forma:SolidPeso molecular:609.54Paliperidone Palmitate
CAS:<p>Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>Fórmula:C39H57FN4O4Pureza:98%Cor e Forma:SolidPeso molecular:664.89Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Fórmula:C22H25N3O3Pureza:99.94%Cor e Forma:SolidPeso molecular:379.45Eticlopride hydrochloride
CAS:<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Fórmula:C17H25ClN2O3·HClPureza:98%Cor e Forma:SolidPeso molecular:377.31Bromperidol hydrochloride
CAS:<p>Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.</p>Fórmula:C21H24BrClFNO2Cor e Forma:SolidPeso molecular:456.78ST-836 hydrochloride
CAS:ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .Fórmula:C23H35ClN4OSPureza:98%Cor e Forma:SolidPeso molecular:451.07Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Fórmula:C21H23ClFNO2Pureza:98%Cor e Forma:SolidPeso molecular:379.89Emedastine Difumarate
CAS:<p>Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.</p>Fórmula:C25H34N4O9Cor e Forma:SolidPeso molecular:534.56YNT-185 dihydrochloride
CAS:<p>Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.</p>Fórmula:C33H39Cl2N5O5SCor e Forma:SolidPeso molecular:688.67Tulobuterol-d9 HCl
CAS:Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.Fórmula:C12H10D9Cl2NOPeso molecular:273.25GLP-1 receptor agonist 7
CAS:<p>GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.</p>Fórmula:C31H30ClFN4O5Cor e Forma:SolidPeso molecular:593.05GSK682753A
CAS:GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).Fórmula:C23H21Cl3N2O3Cor e Forma:SolidPeso molecular:479.78Cetirizine D4
CAS:<p>Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:392.91Benoxathian hydrochloride
CAS:<p>Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.</p>Fórmula:C19H24ClNO4SCor e Forma:SolidPeso molecular:397.91Revdofilimab
CAS:<p>Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.</p>Pureza:98.80% - 98.80%Cor e Forma:LiquidNefazodone
CAS:<p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>Fórmula:C25H32ClN5O2Pureza:99.85%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:470.01Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Fórmula:C27H34N4O3Pureza:99.33%Cor e Forma:SolidPeso molecular:462.58Omidenepag
CAS:Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.Fórmula:C23H22N6O4SPureza:99.67% - 99.77%Cor e Forma:SolidPeso molecular:478.52MRGPRX4 modulator-2
CAS:MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value of less than 100 nM. Its notable applications include research on autoimmune diseases such as psoriasis, multiple sclerosis, Steven Johnson's Syndrome, and various chronic itch conditions [1].Fórmula:C15H9ClF4O3Pureza:99.24%Cor e Forma:SolidPeso molecular:348.68(S)-(+)-Dimethindene maleate
CAS:<p>(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors</p>Fórmula:C24H28N2O4Pureza:99.94%Cor e Forma:SolidPeso molecular:408.49Asenapine hydrochloride
CAS:<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Fórmula:C17H17Cl2NOCor e Forma:SolidPeso molecular:322.23V-0219
CAS:<p>V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.</p>Fórmula:C20H25F3N4O2Pureza:99.91%Cor e Forma:SoildPeso molecular:410.43LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Fórmula:C18H14FN5OPureza:99.03% - >99.99%Cor e Forma:SolidPeso molecular:335.34rac-Propranolol-d7
CAS:Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.Fórmula:C16H14D7NO2Cor e Forma:SolidPeso molecular:266.39Travoprost (Standard)
CAS:Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Fórmula:C26H35F3O6Peso molecular:500.55Agomelatine (L(+)-Tartaric acid)
CAS:<p>Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and</p>Fórmula:C19H23NO8Cor e Forma:SolidPeso molecular:393.39SYL-4
CAS:SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Fórmula:C20H15N3O5SPureza:95.76%Cor e Forma:SoildPeso molecular:409.42Tegaserod
CAS:<p>Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).</p>Fórmula:C16H23N5OPureza:99.20% - 99.89%Cor e Forma:SolidPeso molecular:301.39WZ4141
CAS:WZ4141 is an intermediate in compound synthesis.Fórmula:C16H13N3O2Pureza:98%Cor e Forma:SolidPeso molecular:279.29Eplivanserin (mixture)
CAS:<p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>Fórmula:C19H21FN2O2Cor e Forma:SolidPeso molecular:328.387Granisetron
CAS:<p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Fórmula:C10H18ClN3SPureza:98%Cor e Forma:White Crystalline PowderPeso molecular:247.79Sumatriptan
CAS:<p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>Fórmula:C14H21N3O2SPureza:99.93%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:295.4Cimbuterol-d9
CAS:<p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>Fórmula:C13H10D9N3OPureza:99.22%Cor e Forma:SolidPeso molecular:242.37UCSF924
CAS:<p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>Fórmula:C20H22N2O2Pureza:98%Cor e Forma:SolidPeso molecular:322.4GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Fórmula:C15H21N5O5Cor e Forma:SolidPeso molecular:351.36Asenapine
CAS:<p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>Fórmula:C17H16ClNOPureza:99.64%Cor e Forma:CoaPeso molecular:285.77PD176252
CAS:<p>PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.</p>Fórmula:C32H36N6O5Pureza:99.18%Cor e Forma:SolidPeso molecular:584.67Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Fórmula:C15H21D3N2O4SCor e Forma:SolidPeso molecular:331.45Taranabant racemate
CAS:<p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>Fórmula:C27H25ClF3N3O2Pureza:98%Cor e Forma:SolidPeso molecular:515.95TP-16
CAS:<p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>Fórmula:C24H22FNO4SPureza:98.53% - 99.15%Cor e Forma:SolidPeso molecular:439.5Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Fórmula:C18H18ClN3SPureza:99.93%Cor e Forma:SolidPeso molecular:343.87Zilpaterol-d7
CAS:<p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>Fórmula:C14H12D7N3O2Cor e Forma:SolidPeso molecular:268.36Argipressin
CAS:<p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>Fórmula:C46H65N15O12S2Pureza:98%Cor e Forma:White PowderPeso molecular:1084.23Thiethylperazine
CAS:<p>Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.</p>Fórmula:C22H29N3S2Pureza:98.72%Cor e Forma:SolidPeso molecular:399.62L-798106
CAS:L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Fórmula:C27H22BrNO4SPureza:98.97%Cor e Forma:SolidPeso molecular:536.44MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Fórmula:C17H19N5OC2H2O4Pureza:97.10%Cor e Forma:SolidPeso molecular:354.39Clencyclohexerol-d10
CAS:<p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>Fórmula:C14H20Cl2N2O2Cor e Forma:SolidPeso molecular:329.29Furprofen
CAS:Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Fórmula:C14H12O4Pureza:98.62% - 99.25%Cor e Forma:SolidPeso molecular:244.24Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Fórmula:C19H24N2OSPureza:99.15%Cor e Forma:SolidPeso molecular:328.47BMS-986224
CAS:<p>BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.</p>Fórmula:C24H23ClN4O6Pureza:98.61% - 99.67%Cor e Forma:SolidPeso molecular:498.923-Hydroxy agomelatine
CAS:<p>3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.</p>Fórmula:C15H17NO3Cor e Forma:SolidPeso molecular:259.3Docosahexaenoic acid ethyl ester
CAS:<p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>Fórmula:C24H36O2Cor e Forma:SolidPeso molecular:356.54SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Fórmula:C15H15ClN4OPureza:98%Cor e Forma:SolidPeso molecular:302.76Sumanirole maleate
CAS:<p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>Fórmula:C15H17N3O5Pureza:98%Cor e Forma:SolidPeso molecular:319.31cis-(Z)-Flupentixol dihydrochloride
CAS:<p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>Fórmula:C23H27Cl2F3N2OSPureza:98.07%Cor e Forma:SolidPeso molecular:507.44Calcitonin (salmon)
CAS:<p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>Fórmula:C145H240N44O48S2Pureza:99.41% - 99.80%Cor e Forma:PowderPeso molecular:3431.85Scopine hydrochloride
CAS:<p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>Fórmula:C8H13NO2·HClPureza:98%Cor e Forma:White PowderPeso molecular:191.66SANT 2
CAS:<p>SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.</p>Fórmula:C26H26ClN3O4Pureza:99.23%Cor e Forma:SolidPeso molecular:479.96Neurotensin(8-13)
CAS:<p>Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>Fórmula:C38H64N12O8Pureza:99.95%Cor e Forma:SolidPeso molecular:816.99EST64454 Maleic acid salt
CAS:<p>EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.</p>Fórmula:C22H26F2N4O6Pureza:97.54%Cor e Forma:SolidPeso molecular:480.46Asapiprant
CAS:<p>Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.</p>Fórmula:C24H27N3O7SPureza:99.64%Cor e Forma:SolidPeso molecular:501.55[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Fórmula:C69H108N22O16SPureza:99.71%Cor e Forma:SolidPeso molecular:1533.8Lecirelin acetate(61012-19-9 free base)
<p>Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts</p>Fórmula:C61H88N16O14Pureza:98.1%Cor e Forma:SolidPeso molecular:1269.45Nelociguat
CAS:<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Fórmula:C19H17FN8O2Pureza:99.19%Cor e Forma:SolidPeso molecular:408.39Neurokinin A
CAS:<p>Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.</p>Fórmula:C50H80N14O14SPureza:>99.99%Cor e Forma:White To Off-White Lyophilized SolidPeso molecular:1133.32Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Fórmula:C19H21N5O4Pureza:99.86%Cor e Forma:White To Tan Powder SolidPeso molecular:383.4Phenylbiguanide
CAS:<p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>Fórmula:C8H11N5Pureza:99.54%Cor e Forma:SolidPeso molecular:177.21WAY-100635 Monomaleate
CAS:<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Cor e Forma:SolidPeso molecular:538.645-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Fórmula:C18H20N2OPureza:99.13%Cor e Forma:SolidPeso molecular:280.36Lys-[Des-Arg9]Bradykinin acetate
<p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and</p>Fórmula:C52H77N13O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1092.27Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Fórmula:C23H30N2O10Pureza:99.98%Cor e Forma:SolidPeso molecular:494.49I-191
CAS:<p>I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.</p>Fórmula:C23H26FN5O2Pureza:99.8%Cor e Forma:SolidPeso molecular:423.48M40 acetate(143896-17-7 free base)
<p>M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29)</p>Fórmula:C96H149N23O26Pureza:99.88%Cor e Forma:SolidPeso molecular:2041.38Zatebradine
CAS:<p>Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).</p>Fórmula:C26H36N2O5Pureza:98%Cor e Forma:SolidPeso molecular:456.57Grapiprant
CAS:<p>Grapiprant (AAT-007) is a selective EP4 receptor antagonist.</p>Fórmula:C26H29N5O3SPureza:99.49% - 99.843%Cor e Forma:SolidPeso molecular:491.61Ursodeoxycholic acid sodium
CAS:<p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>Fórmula:C24H40NaO4Pureza:99.66% - 99.96%Cor e Forma:SolidPeso molecular:415.56Dimethocaine
CAS:<p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>Fórmula:C16H26N2O2Pureza:99.52%Cor e Forma:SolidPeso molecular:278.39ML-184
CAS:<p>ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.</p>Fórmula:C25H34N4O3SPureza:99.45%Cor e Forma:SolidPeso molecular:470.63Hemokinin 1 (human) acetate(491851-53-7 free base)
<p>Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.</p>Fórmula:C56H88N14O16SPureza:97.82%Cor e Forma:SolidPeso molecular:1245.45Ataciguat
CAS:<p>Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.</p>Fórmula:C21H19Cl2N3O6S3Pureza:99.09%Cor e Forma:SolidPeso molecular:576.49Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38M871 acetate
<p>M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptive</p>Fórmula:C110H167N27O30Pureza:99.84%Cor e Forma:SolidPeso molecular:2347.67GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Cor e Forma:SolidPeso molecular:415.53Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Fórmula:C15H19N3Pureza:≥95%Cor e Forma:SolidPeso molecular:241.33Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Fórmula:C12H17ClN2O2Pureza:99.35%Cor e Forma:SolidPeso molecular:256.73Guanfacine hydrochloride
CAS:<p>Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.</p>Fórmula:C9H10Cl3N3OPureza:99.89% - 99.91%Cor e Forma:SolidPeso molecular:282.55Pizuglanstat
CAS:<p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>Fórmula:C27H36N6O4Pureza:99.62%Cor e Forma:SolidPeso molecular:508.61Plecanatide
CAS:<p>Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.</p>Fórmula:C65H104N18O26S4Pureza:97.51%Cor e Forma:SolidPeso molecular:1681.89Melanin Concentrating Hormone, salmon acetate
<p>Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>Fórmula:C91H143N27O26S4Pureza:99.41%Cor e Forma:SolidPeso molecular:2157Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Cor e Forma:White Or Off-White CrystallinePeso molecular:327.4Metoclopramide hydrochloride hydrate
CAS:<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Fórmula:C14H25Cl2N3O3Pureza:99.33%Cor e Forma:SolidPeso molecular:354.27Galanin Receptor Ligand M35 TFA
<p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>Fórmula:C109H154N27F3O28Pureza:99.45%Cor e Forma:SolidPeso molecular:2347.62Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Fórmula:C68H90N18O14Pureza:99.92%Cor e Forma:SolidPeso molecular:1383.55TY-52156
CAS:<p>TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).</p>Fórmula:C18H19Cl2N3OPureza:99.91% - 99.91%Cor e Forma:SolidPeso molecular:364.27[D-Phe12,Leu14]-Bombesin acetate
<p>[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Fórmula:C77H118N22O20Pureza:98.41% - 99.14%Cor e Forma:SolidPeso molecular:1671.9RS102895
CAS:<p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>Fórmula:C21H21F3N2O2Pureza:97.64% - 99.80%Cor e Forma:SolidPeso molecular:390.4SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Fórmula:C28H28ClN3OSPureza:97.37% - 98.88%Cor e Forma:SolidPeso molecular:490.06Ciliobrevin A
CAS:<p>Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.</p>Fórmula:C17H9Cl2N3O2Pureza:98.54% - 99.57%Cor e Forma:SolidPeso molecular:358.18Taprenepag
CAS:<p>Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).</p>Fórmula:C24H22N4O5SPureza:98.89% - 99.15%Cor e Forma:SolidPeso molecular:478.52MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Fórmula:C27H21F3N2O3Pureza:99.54% - 99.59%Cor e Forma:SolidPeso molecular:478.46SKF 38393 hydrochloride
CAS:<p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>Fórmula:C16H17NO2·HClPureza:99.1% - 99.51%Cor e Forma:SolidPeso molecular:291.77SANT-1
CAS:<p>SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).</p>Fórmula:C23H27N5Pureza:99.98% - >99.99%Cor e Forma:SolidPeso molecular:373.49MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Fórmula:C24H23N3O5SPureza:99.73%Cor e Forma:SolidPeso molecular:465.52F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Fórmula:C19H21ClF2N4OPureza:98.72%Cor e Forma:SolidPeso molecular:394.85Ondansetron
CAS:<p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>Fórmula:C18H19N3OPureza:99.92%Cor e Forma:White To Yellow CrystalsPeso molecular:293.36ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Fórmula:C19H22N4O3Pureza:99.92%Cor e Forma:SolidPeso molecular:354.4RE-640
CAS:<p>NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.</p>Fórmula:C20H16Cl2N4Pureza:99.60% - 99.87%Cor e Forma:SolidPeso molecular:383.27Vercirnon
CAS:<p>Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.</p>Fórmula:C22H21ClN2O4SPureza:99.23%Cor e Forma:SolidPeso molecular:444.93Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Fórmula:C215H347N61O65S·6C2H4O2Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:5218.88SAG hydrochloride (912545-86-9(free base))
CAS:<p>SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.</p>Fórmula:C28H29Cl2N3OSPureza:99.19% - 99.77%Cor e Forma:SolidPeso molecular:526.52R243
CAS:<p>R243 is CCR8 signaling and chemotaxis inhibitor.</p>Fórmula:C21H27NO4Pureza:99.03%Cor e Forma:SolidPeso molecular:357.44A2B receptor antagonist 2
CAS:<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Fórmula:C12H15N5Pureza:100%Cor e Forma:SolidPeso molecular:229.28Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Fórmula:C20H22N2SPureza:99.98%Cor e Forma:SolidPeso molecular:322.47Sonidegib
CAS:<p>Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.</p>Fórmula:C26H26F3N3O3Pureza:98% - 99.97%Cor e Forma:SolidPeso molecular:485.5Salmeterol Xinafoate
CAS:<p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>Fórmula:C36H45NO7Pureza:98% - 98.24%Cor e Forma:White SolidPeso molecular:603.75MRT-81
CAS:<p>MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.</p>Fórmula:C31H29N3O5SPureza:99.72%Cor e Forma:SolidPeso molecular:555.64SB297006
CAS:<p>SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.</p>Fórmula:C18H18N2O5Pureza:99.59%Cor e Forma:SolidPeso molecular:342.35Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Fórmula:C11H17N3O3Pureza:99.89%Cor e Forma:SolidPeso molecular:239.27BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Fórmula:C18H22F3N3O4SPureza:98.05%Cor e Forma:SolidPeso molecular:433.45Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Fórmula:C46H65N13O11S2Pureza:99.65%Cor e Forma:SolidPeso molecular:1040.22RS-67333
CAS:<p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>Fórmula:C19H29ClN2O2Pureza:99.24%Cor e Forma:SolidPeso molecular:352.9Tolnapersine
CAS:<p>Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.</p>Fórmula:C21H26N2OPureza:98%Cor e Forma:SolidPeso molecular:322.44Geissoschizine methyl ether
CAS:<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Fórmula:C22H26N2O3Pureza:99.24% - 99.68%Cor e Forma:SolidPeso molecular:366.45GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Fórmula:C29H36F3N3O5Pureza:98.2% - 98.88%Cor e Forma:SolidPeso molecular:563.61Calcitonin(salmon) Acetate(47931-85-1(free base))
<p>Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5</p>Fórmula:C145H240N44O48S2Pureza:99.29%Cor e Forma:SolidPeso molecular:3431.85MK-1064
CAS:<p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>Fórmula:C24H20ClN5O3Pureza:99.19% - 99.82%Cor e Forma:SolidPeso molecular:461.9VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Fórmula:C15H19N5Pureza:99.44% - 99.57%Cor e Forma:SolidPeso molecular:269.34Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Cor e Forma:SolidPeso molecular:379.36SAX-187
CAS:<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Fórmula:C15H13ClN4O2S2Pureza:97.82% - 98%Cor e Forma:SolidPeso molecular:380.87Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97Treprostinil
CAS:<p>Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).</p>Fórmula:C23H34O5Pureza:99.29%Cor e Forma:SolidPeso molecular:390.51BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Fórmula:C59H80N14O13Pureza:95.3%Cor e Forma:SolidPeso molecular:1193.35Desmopressin acetate (16679-58-6 free base)
CAS:<p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>Fórmula:C48H68N14O14S2Pureza:98.84% - >99.99%Cor e Forma:SolidPeso molecular:1129.26VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Fórmula:C18H12F3NOSPureza:99.78%Cor e Forma:SolidPeso molecular:347.35Binodenoson
CAS:<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Fórmula:C17H25N7O4Pureza:99.74%Cor e Forma:SolidPeso molecular:391.42Opromazine hydrochloride
CAS:<p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>Fórmula:C17H20Cl2N2OSPureza:98.03%Cor e Forma:SolidPeso molecular:371.32Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Fórmula:C18H15BrF2N4O2Pureza:98.42% - 99.88%Cor e Forma:SolidPeso molecular:437.24Human growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) onPureza:99.26%Cor e Forma:LiquidPeso molecular:N/AAprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Fórmula:C23H21F7N4O3Pureza:98% - 99.68%Cor e Forma:Off-White To Light Yellow Cyrstalline SolidPeso molecular:534.43AM095
CAS:<p>AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.</p>Fórmula:C27H23N2NaO5Pureza:98.87%Cor e Forma:SolidPeso molecular:478.47Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.Pureza:95.44% - 99.73%Cor e Forma:SolidPeso molecular:N/ASevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Fórmula:C4H3F7OPureza:98%Cor e Forma:Less Oil Colorless OilPeso molecular:200.05ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Fórmula:C23H31N3O3SPureza:99.75%Cor e Forma:SolidPeso molecular:429.58CCG215022
CAS:<p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>Fórmula:C26H22FN7O3Pureza:97.63% - 99.69%Cor e Forma:SolidPeso molecular:499.5Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Fórmula:C19H21Cl2N3Pureza:>99.99%Cor e Forma:SolidPeso molecular:362.3Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Pureza:97.26%Cor e Forma:LiquidPeso molecular:N/A

