GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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RU 24969 succinate
CAS:<p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>Fórmula:C18H22N2O5Cor e Forma:SolidPeso molecular:346.38Midaglizole
CAS:<p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>Fórmula:C16H17N3Cor e Forma:SolidPeso molecular:251.33DAPTA
CAS:DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Fórmula:C35H56N10O15Pureza:>99.99%Cor e Forma:SolidPeso molecular:856.88Cangrelor free acid
CAS:<p>Cangrelor, a reversible P2Y12 inhibitor for IV use, was approved in June 2015; it rapidly blocks ADP-induced platelet aggregation.</p>Fórmula:C17H25Cl2F3N5O12P3S2Cor e Forma:SolidPeso molecular:776.36GLPG2938
CAS:<p>GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and</p>Fórmula:C20H19F6N7O2Pureza:98.25%Cor e Forma:SolidPeso molecular:503.4AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Fórmula:C27H23N2NaO5Pureza:98.87%Cor e Forma:SolidPeso molecular:478.47Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Cor e Forma:Off-White To Pale Yellow SolidPeso molecular:440.94Ataciguat
CAS:Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Fórmula:C21H19Cl2N3O6S3Pureza:99.09%Cor e Forma:SolidPeso molecular:576.49BCTC
CAS:<p>BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)</p>Fórmula:C20H25ClN4OPureza:99.21%Cor e Forma:SolidPeso molecular:372.89Prasugrel Hydrochloride
CAS:<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Fórmula:C20H20FNO3S·HClPureza:99.39% - 99.79%Cor e Forma:SolidPeso molecular:409.9Thozalinone
CAS:<p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>Fórmula:C11H12N2O2Pureza:99.68%Cor e Forma:SolidPeso molecular:204.239-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Fórmula:C7H9N5Pureza:99.35% - 99.41%Cor e Forma:SolidPeso molecular:163.18Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Fórmula:C23H30N4O2SPureza:99.23%Cor e Forma:White PowderPeso molecular:426.57Ibutamoren
CAS:<p>Ibutamoren (MK-677) is a drug which acts as a potent, orally active growth hormone secretagogue, mimicking the GH stimulating action of the endogenous hormone ghrelin. It also alters the metabolism of body fat and so may have an application in the treatment of obesity.</p>Fórmula:C27H36N4O5SPureza:97.59%Cor e Forma:SolidPeso molecular:528.66Neuropeptide S (Rat) acetate
<p>Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor.</p>Fórmula:C97H164N34O29Pureza:95.36%Cor e Forma:SolidPeso molecular:2270.592-ATHBI
CAS:<p>2-ATHBI is a S1P lyase inhibitor.</p>Fórmula:C9H14N2O5Pureza:95.00%Cor e Forma:SolidPeso molecular:230.22Fosaprepitant dimeglumine
CAS:<p>Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.</p>Fórmula:C37H56F7N6O16PPureza:98% - 99.03%Cor e Forma:SolidPeso molecular:1004.83GBR 12935
CAS:<p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>Fórmula:C28H34N2OCor e Forma:SolidPeso molecular:414.58M 1145 acetate
<p>M1145 acetate: chimeric peptide, selective GAL2 agonist, Ki=6.55 nM; >90x affinity vs GAL1, 76x vs GalR3. Enhances galanin signal.</p>Fórmula:C130H209N37O34Pureza:99.1%Cor e Forma:SolidPeso molecular:2834.28HS 014 acetate(207678-81-7 free base)
<p>HS 014 acetate is a potent MC4R antagonist with Ki: 3.16 nM (MC4), and boosts food intake and nociception in animals.</p>Fórmula:C73H98N20O19S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:1623.83BRL-15572 dihydrochloride
CAS:<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Fórmula:C25H27ClN2O·2HClPureza:99.74%Cor e Forma:SolidPeso molecular:479.87Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Fórmula:C25H25Cl2N7OPureza:99.43%Cor e Forma:SolidPeso molecular:510.42Loxapine hydrochloride
CAS:<p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>Fórmula:C18H19Cl2N3OCor e Forma:SolidPeso molecular:364.27CGP71683 hydrochloride
CAS:<p>CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).</p>Fórmula:C26H30ClN5O2SPureza:99.92%Cor e Forma:SolidPeso molecular:512.07GSK 789472 hydrochloride
CAS:GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Fórmula:C15H22ClN3OPureza:99.89%Cor e Forma:SolidPeso molecular:295.816-fluoro-DL-Tryptophan
CAS:<p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>Fórmula:C11H11FN2O2Pureza:99.25%Cor e Forma:Off-White PowderPeso molecular:222.22Tafluprost
CAS:<p>Tafluprost, a prostaglandin analog, is the selective agonist of fluoroprostaglandin (FP) receptor PGF2α.</p>Fórmula:C25H34F2O5Pureza:97.7% - 99.67%Cor e Forma:LiquidPeso molecular:452.53Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Cor e Forma:SolidPeso molecular:379.36MK-1064
CAS:<p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>Fórmula:C24H20ClN5O3Pureza:99.19% - 99.82%Cor e Forma:SolidPeso molecular:461.9Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Cor e Forma:SolidPeso molecular:301.81HT-2157
CAS:<p>HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target.</p>Fórmula:C21H13F3N2OPureza:98.33%Cor e Forma:SolidPeso molecular:366.343-CPMT
CAS:<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Fórmula:C21H25Cl2NOPureza:99.03%Cor e Forma:SolidPeso molecular:378.33Epinastine
CAS:<p>Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.</p>Fórmula:C16H15N3Pureza:99.94%Cor e Forma:SolidPeso molecular:249.31TCS 1102
CAS:TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Fórmula:C27H26N4O2SPureza:99.35% - 99.52%Cor e Forma:SolidPeso molecular:470.59Metoclopramide hydrochloride hydrate
CAS:<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Fórmula:C14H25Cl2N3O3Pureza:99.33%Cor e Forma:SolidPeso molecular:354.27GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Fórmula:C25H28N4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:416.52Praliciguat
CAS:<p>Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.</p>Fórmula:C21H14F8N6O2Pureza:98.82%Cor e Forma:SolidPeso molecular:534.36GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFórmula:C23H24Cl2N2O3Pureza:99.82% - 99.93%Cor e Forma:SolidPeso molecular:447.35Bexagliflozin
CAS:<p>Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 2 nM for human SGLT2.</p>Fórmula:C24H29ClO7Pureza:98.99% - 99.89%Cor e Forma:SolidPeso molecular:464.94Enavogliflozin
CAS:<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Fórmula:C24H27ClO6Pureza:97.37%Cor e Forma:SolidPeso molecular:446.92Bosentan (hydrate)
CAS:Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.Fórmula:C27H29N5O6S·H2OPureza:99.31% - 99.86%Cor e Forma:White PowderPeso molecular:569.63Plecanatide
CAS:<p>Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.</p>Fórmula:C65H104N18O26S4Pureza:97.51%Cor e Forma:SolidPeso molecular:1681.89JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Fórmula:C14H16ClN3OPureza:99.83% - 99.96%Cor e Forma:SolidPeso molecular:277.75Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Fórmula:C14H23BrClN3O2Cor e Forma:SolidPeso molecular:380.71PSB-SB-487
CAS:<p>PSB-SB-487 is antagonist of GPR55.</p>Fórmula:C26H32O4Pureza:98.53%Cor e Forma:SolidPeso molecular:408.53Glasdegib
CAS:<p>Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.</p>Fórmula:C21H22N6OPureza:98.72%Cor e Forma:SolidPeso molecular:374.44Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Fórmula:C29H34O6Pureza:≥98%Cor e Forma:LiquidPeso molecular:478.58PAR-2-IN-1
CAS:<p>PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.</p>Fórmula:C12H14ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:267.71[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
<p>[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and</p>Fórmula:C76H103N21O18SPureza:99.75%Cor e Forma:SolidPeso molecular:1630.82BX471
CAS:<p>BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.</p>Fórmula:C21H24ClFN4O3Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:434.89TS-011
CAS:<p>N-(3-Chloro-4-morpholinophenyl)-N'-hydroxyformimidamide (TS-011) is a selective 20-Hydroxyeicosatetraenoic acid synthesis inhibitor.</p>Fórmula:C11H14ClN3O2Pureza:99.48%Cor e Forma:SolidPeso molecular:255.7Bay 59-3074
CAS:<p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>Fórmula:C18H13F6NO4SPureza:97.68% - 99.69%Cor e Forma:SolidPeso molecular:453.36RFRP3(human) acetate(311309-27-0 free base)
<p>RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.</p>Fórmula:C47H76N14O12Pureza:97.09%Cor e Forma:SolidPeso molecular:1029.19ML221
CAS:<p>ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in</p>Fórmula:C17H11N3O6SPureza:97.74%Cor e Forma:SolidPeso molecular:385.35Vorapaxar sulfate
CAS:<p>Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.</p>Fórmula:C29H35FN2O8SPureza:99.9% - >99.99%Cor e Forma:SolidPeso molecular:590.66Droxidopa
CAS:Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Fórmula:C9H11NO5Pureza:97.27% - 99.88%Cor e Forma:SolidPeso molecular:213.19Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Fórmula:C32H44F3N3O2SPureza:98.14%Cor e Forma:SolidPeso molecular:591.77Eptapirone
CAS:<p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>Fórmula:C16H23N7O2Pureza:99.39% - 99.65%Cor e Forma:SolidPeso molecular:345.4Opaganib
CAS:<p>Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).</p>Fórmula:C23H25ClN2OPureza:98.86% - 99.85%Cor e Forma:SolidPeso molecular:380.91Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFórmula:C49H70N12O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1035.15AM1241
CAS:<p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>Fórmula:C22H22IN3O3Pureza:98.937% - 99.1%Cor e Forma:SolidPeso molecular:503.33Ibrolipim
CAS:<p>Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.</p>Fórmula:C19H20BrN2O4PPureza:98.04%Cor e Forma:SolidPeso molecular:451.25FAUC 346
CAS:<p>FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.</p>Fórmula:C24H29N3O2SPureza:99.46%Cor e Forma:SolidPeso molecular:423.57ML417
CAS:<p>ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).</p>Fórmula:C22H25N3O3Pureza:98.4% - 99.42%Cor e Forma:SolidPeso molecular:379.45Istradefylline
CAS:<p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>Fórmula:C20H24N4O4Pureza:98.18% - 99.95%Cor e Forma:SolidPeso molecular:384.43Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Cor e Forma:SolidPeso molecular:331.86Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Cor e Forma:SolidPeso molecular:434.83TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Cor e Forma:SolidPeso molecular:448.43Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Fórmula:C68H87N17O15Pureza:99.98%Cor e Forma:SolidPeso molecular:1382.55Poloxamer 407
CAS:<p>Poloxamer 407 is a nonionic surfactant.</p>Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:7700(Average)Aripiprazole monohydrate
CAS:<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Fórmula:C23H29Cl2N3O3Cor e Forma:SolidPeso molecular:466.4Bavisant dihydrochloride hydrate
CAS:Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.Fórmula:C19H31Cl2N3O3Cor e Forma:SolidPeso molecular:420.38Quipazine
CAS:<p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>Fórmula:C13H15N3Cor e Forma:SolidPeso molecular:213.28Brefonalol
CAS:<p>Brefonalol is a vasodilating beta-adrenergic receptor blocker.</p>Fórmula:C22H28N2O2Cor e Forma:SolidPeso molecular:352.47Raclopride tartrate
CAS:<p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>Fórmula:C19H26Cl2N2O9Cor e Forma:SolidPeso molecular:497.32Eltoprazine dihydrochloride
CAS:<p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>Fórmula:C12H18Cl2N2O2Pureza:99.64%Cor e Forma:SolidPeso molecular:293.19Brompheniramine
CAS:<p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>Fórmula:C16H19BrN2Cor e Forma:SolidPeso molecular:319.24Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Fórmula:C65H102N16O25Pureza:95.55%Cor e Forma:SolidPeso molecular:1507.6Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.44Olodaterol hydrochloride
CAS:<p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>Fórmula:C21H27ClN2O5Pureza:99.11%Cor e Forma:SolidPeso molecular:422.9Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Fórmula:C20H22N2O4Pureza:98.46%Cor e Forma:SolidPeso molecular:354.4Mecamylamine hydrochloride
CAS:<p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>Fórmula:C11H22ClNPureza:99.76% - >99.99%Cor e Forma:White SolidPeso molecular:203.75Buserelin Acetate (57982-77-1 free base)
CAS:<p>Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).</p>Fórmula:C62H90N16O15Pureza:99.31% - 99.78%Cor e Forma:SolidPeso molecular:1299.481-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Cor e Forma:SolidPeso molecular:248.75Alimemazine hemitartrate
CAS:<p>Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.</p>Fórmula:C18H22N2SC4H6O6Pureza:98.16% - 99.69%Cor e Forma:SolidPeso molecular:448.53CRT0273750
CAS:<p>CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.</p>Fórmula:C25H22ClF3N4O2Pureza:99.91%Cor e Forma:SolidPeso molecular:502.92Bevantolol
CAS:<p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>Fórmula:C20H27NO4Cor e Forma:SolidPeso molecular:345.43Sigma-LIGAND-1 hydrochloride
CAS:<p>Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.</p>Fórmula:C27H34ClNO4Cor e Forma:SolidPeso molecular:472.02Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Cor e Forma:SolidPeso molecular:356.44Tavapadon
CAS:<p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>Fórmula:C19H16F3N3O3Pureza:99.33% - 99.8%Cor e Forma:SolidPeso molecular:391.34Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Cor e Forma:SolidPeso molecular:336.38Dolasetron Mesylate hydrate
CAS:<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Fórmula:C20H26N2O7SPureza:99.86% - 99.9%Cor e Forma:SolidPeso molecular:438.49BMY-25368
CAS:<p>BMY-25368 is a long-acting antagonist of the H2-receptor.</p>Fórmula:C19H25N3O3Cor e Forma:SolidPeso molecular:343.42Mecamylamine
CAS:<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Fórmula:C11H21NCor e Forma:SolidPeso molecular:167.29Syk Inhibitor II dihydrochloride
CAS:<p>Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.</p>Fórmula:C14H17Cl2F3N6OPureza:98.53%Cor e Forma:SolidPeso molecular:413.22ACTH 1-14 acetate(25696-21-3 free base)
<p>ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.</p>Fórmula:C79H113N21O22SPureza:>99.99%Cor e Forma:SolidPeso molecular:1740.96LM11A-31 dihydrochloride
CAS:<p>LM11A-31 dihydrochloride is a water-soluble, BBB-penetrating p75NTR ligand and proNGF antagonist.</p>Fórmula:C12H27Cl2N3O2Pureza:99.9%Cor e Forma:SolidPeso molecular:316.27SCH-37370
CAS:<p>SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.</p>Fórmula:C21H21ClN2OPureza:99.07%Cor e Forma:SolidPeso molecular:352.86Emedastine
CAS:<p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>Fórmula:C17H26N4OPureza:97.1% - 97.76%Cor e Forma:OilPeso molecular:302.41Eltoprazine
CAS:<p>Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.</p>Fórmula:C12H16N2O2Cor e Forma:SolidPeso molecular:220.27REV 5901
CAS:<p>REV 5901: oral leukotriene receptor antagonist and 5-lipoxygenase inhibitor with Ki of 0.7 μM, researched for asthma.</p>Fórmula:C22H25NO2Cor e Forma:SolidPeso molecular:335.44ML-18
CAS:<p>ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.</p>Fórmula:C32H35N5O5Pureza:98.62% - >99.99%Cor e Forma:SolidPeso molecular:569.65Men 10376 TFA(135306-85-3,free)
<p>Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4</p>Fórmula:C59H69F3N12O12Pureza:99.22%Cor e Forma:SolidPeso molecular:1195.25Temanogrel
CAS:<p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>Fórmula:C24H28N4O4Pureza:99.24%Cor e Forma:SolidPeso molecular:436.5Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Fórmula:C22H25ClN4O4S2Cor e Forma:SolidPeso molecular:509.04ENMD-1068 HBr
CAS:<p>ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.</p>Fórmula:C15H30BrN3O2Cor e Forma:SolidPeso molecular:364.32Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Fórmula:C11H16N2O3Pureza:98%Cor e Forma:SolidPeso molecular:224.26Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Fórmula:C21H21FO5SPureza:99.38% - 99.70%Cor e Forma:SolidPeso molecular:404.45Laropiprant sodium
<p>Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.</p>Cor e Forma:SolidGSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Fórmula:C22H21ClN4O4Pureza:99.04%Cor e Forma:SolidPeso molecular:440.88Tiapride
CAS:<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Fórmula:C15H24N2O4SCor e Forma:SolidPeso molecular:328.43Tripelennamine citrate
CAS:<p>Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.</p>Fórmula:C22H29N3O7Cor e Forma:SolidPeso molecular:447.488Ajmalicine hydrochloride
CAS:<p>Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.</p>Fórmula:C21H25ClN2O3Cor e Forma:SolidPeso molecular:388.89Betazole
CAS:<p>Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.</p>Fórmula:C5H9N3Cor e Forma:SolidPeso molecular:111.15Talnetant
CAS:<p>Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.</p>Fórmula:C25H22N2O2Pureza:97.88%Cor e Forma:SolidPeso molecular:382.45Secretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Fórmula:C129H216N42O42Pureza:98.12%Cor e Forma:SolidPeso molecular:3027.35L-765314
CAS:<p>L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.</p>Fórmula:C27H34N6O5Pureza:99.73%Cor e Forma:SolidPeso molecular:522.6ESI-09
CAS:ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.Fórmula:C16H15ClN4O2Pureza:97.24% - 99.57%Cor e Forma:SolidPeso molecular:330.77β-CGRP, human acetate
<p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>Fórmula:C164H271N51O50S3Pureza:99.35%Cor e Forma:SolidPeso molecular:3853.46Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Fórmula:C40H42ClN5O7Pureza:97.94% - 98.4%Cor e Forma:SolidPeso molecular:740.24RG7713
CAS:<p>RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.</p>Fórmula:C25H28ClN3O2Pureza:99.74%Cor e Forma:SolidPeso molecular:437.96SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Fórmula:C21H19ClN4O2Pureza:99.75% - ≥98%Cor e Forma:SolidPeso molecular:394.85CS 2100
CAS:<p>CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.</p>Fórmula:C25H23N3O4SPureza:99.19%Cor e Forma:SolidPeso molecular:461.531-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Fórmula:C6H9N3O2Pureza:99.29%Cor e Forma:SolidPeso molecular:155.15Gadolinium chloride
CAS:<p>Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist</p>Fórmula:Cl3GdPureza:98%Cor e Forma:White Crystalline SolidPeso molecular:263.61Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Cor e Forma:SolidPeso molecular:427.41Paltusotine
CAS:<p>Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.</p>Fórmula:C27H22F2N4OPureza:99.91%Cor e Forma:SolidPeso molecular:456.49Desvenlafaxine succinate hydrate
CAS:<p>Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).</p>Fórmula:C20H33NO7Pureza:99.26%Cor e Forma:White Crystalline PowdePeso molecular:399.48Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Fórmula:C16H16Cl3NPureza:98.92% - 99.6%Cor e Forma:SolidPeso molecular:328.66SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Fórmula:C18H21Cl2N3O4SPureza:98.94%Cor e Forma:SolidPeso molecular:446.35ABT-724
CAS:<p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>Fórmula:C17H19N5Pureza:99.73%Cor e Forma:SolidPeso molecular:293.37LGnRH-III, lamprey acetate(147859-97-0 free base)
<p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>Fórmula:C61H78N18O16Pureza:99.66%Cor e Forma:SolidPeso molecular:1319.38Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Fórmula:C10H8BrN7Pureza:99.11%Cor e Forma:SolidPeso molecular:306.12Etrasimod
CAS:<p>Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).</p>Fórmula:C26H26F3NO3Pureza:98.52% - 99.73%Cor e Forma:SolidPeso molecular:457.48CYN 154806 TFA
CAS:<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Fórmula:C58H69F3N12O16S2Pureza:99.7%Cor e Forma:SolidPeso molecular:1311.36Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Fórmula:C25H34FN3O2Pureza:97.84% - 99.69%Cor e Forma:Pale Yellow To Pale Orange SolidPeso molecular:427.55β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Fórmula:C120H178N34O37SPureza:99.64%Cor e Forma:SolidPeso molecular:2720.97L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Fórmula:C18H20Cl2N4Pureza:97.36%Cor e Forma:SolidPeso molecular:363.28Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Cor e Forma:Almost White To White Crystalline PowderPeso molecular:351.93PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Fórmula:C21H29Cl2N3O4SPureza:98.5%Cor e Forma:SolidPeso molecular:490.44Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Fórmula:C21H30N4O4Pureza:99.52%Cor e Forma:SolidPeso molecular:402.49DPCPX
CAS:<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Fórmula:C16H24N4O2Pureza:99.23% - 99.93%Cor e Forma:White SolidPeso molecular:304.39RBC8
CAS:<p>RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.</p>Fórmula:C25H20N4O3Pureza:98.44% - 99.81%Cor e Forma:SolidPeso molecular:424.45Pranlukast hemihydrate
CAS:<p>Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.</p>Fórmula:C27H23N5O40·5H2OPureza:99.28%Cor e Forma:SolidPeso molecular:490.52AP1189 acetate
CAS:<p>AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.</p>Fórmula:C16H18N6O4Pureza:99.95%Cor e Forma:SolidPeso molecular:358.35Bucindolol hydrochloride
CAS:<p>Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.</p>Fórmula:C22H26ClN3O2Cor e Forma:SolidPeso molecular:399.91Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Fórmula:C20H20NO4Pureza:97.18% - 99.06%Cor e Forma:SolidPeso molecular:338.38Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Fórmula:C19H22ClN3OPureza:98%Cor e Forma:SolidPeso molecular:343.86LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Cor e Forma:SolidPeso molecular:226.53Fabomotizole
CAS:<p>Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.</p>Fórmula:C15H21N3O2SPureza:99.4%Cor e Forma:SolidPeso molecular:307.41ACTH (1-39) human
CAS:<p>Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor.</p>Fórmula:C207H308N56O58SPureza:99.6%Cor e Forma:White Lyophilised SolidPeso molecular:4541.14ARN272
CAS:<p>ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).</p>Fórmula:C27H20N4O2Pureza:98.23%Cor e Forma:SolidPeso molecular:432.47Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Fórmula:C15H19Cl2N3O3SPureza:98.48%Cor e Forma:SolidPeso molecular:392.3Phosphorylcholine chloride
CAS:<p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>Fórmula:C5H15ClNO4PPureza:99.481% - 99.85%Cor e Forma:SolidPeso molecular:219.6Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Fórmula:C11H17N3O3Pureza:99.89%Cor e Forma:SolidPeso molecular:239.27Opromazine hydrochloride
CAS:<p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>Fórmula:C17H20Cl2N2OSPureza:98.03%Cor e Forma:SolidPeso molecular:371.32ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Fórmula:C29H29ClN4O2Pureza:99.88%Cor e Forma:SolidPeso molecular:501.02Cloprostenol sodium salt
CAS:<p>Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.</p>Fórmula:C22H28ClNaO6Pureza:97.17% - 98.47%Cor e Forma:White To Almost White Hygroscopic PowderPeso molecular:446.9Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Fórmula:C68H90N18O14Pureza:99.92%Cor e Forma:SolidPeso molecular:1383.55Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95PRX-08066
CAS:<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Fórmula:C19H17ClFN5SPureza:97.79% - 98.07%Cor e Forma:SolidPeso molecular:401.89Zacopride hydrochloride
CAS:<p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>Fórmula:C15H20ClN3O2·HClPureza:98.32%Cor e Forma:SolidPeso molecular:346.26SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Fórmula:C16H20N2O2·HClPureza:99.64%Cor e Forma:SolidPeso molecular:308.81CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Fórmula:C20H21N7O3Pureza:98.78%Cor e Forma:SolidPeso molecular:407.43BPTU
CAS:<p>BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).</p>Fórmula:C23H22F3N3O3Pureza:99.37% - 99.89%Cor e Forma:SolidPeso molecular:445.43Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Fórmula:C15H24ClNO2Pureza:99.79%Cor e Forma:SolidPeso molecular:285.81idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Fórmula:C20H19F5N2OPureza:99.73%Cor e Forma:SolidPeso molecular:398.37Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Fórmula:C18H24ClNO3Pureza:97.15% - 99.94%Cor e Forma:SolidPeso molecular:337.84GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Fórmula:C151H228N40O47Pureza:98.89%Cor e Forma:SolidPeso molecular:3355.67Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFórmula:C23H26ClNO5Pureza:99.79% - 99.85%Cor e Forma:SolidPeso molecular:431.91Mini Gastrin I, human acetate
<p>Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.</p>Fórmula:C76H103N15O28SPureza:99.35% - 99.82%Cor e Forma:SolidPeso molecular:1706.78Selexipag
CAS:<p>Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.</p>Fórmula:C26H32N4O4SPureza:99.98% - >99.99%Cor e Forma:SolidPeso molecular:496.62Methiothepin mesylate
CAS:<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Fórmula:C21H28N2O3S3Pureza:98% - 99.92%Cor e Forma:SolidPeso molecular:452.65Ursodeoxycholic acid sodium
CAS:<p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>Fórmula:C24H40NaO4Pureza:99.66% - 99.96%Cor e Forma:SolidPeso molecular:415.56FK962
CAS:<p>FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.</p>Fórmula:C14H17FN2O2Pureza:99.89%Cor e Forma:SolidPeso molecular:264.3Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Fórmula:C25H40ClN3O8Pureza:99.91%Cor e Forma:White Crystalline PowderPeso molecular:546.05Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Fórmula:C12H14N2·HClPureza:99.97%Cor e Forma:SolidPeso molecular:222.71A2B receptor antagonist 2
CAS:<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Fórmula:C12H15N5Pureza:100%Cor e Forma:SolidPeso molecular:229.28Ondansetron
CAS:<p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>Fórmula:C18H19N3OPureza:99.92%Cor e Forma:White To Yellow CrystalsPeso molecular:293.36F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Fórmula:C19H21ClF2N4OPureza:98.72%Cor e Forma:SolidPeso molecular:394.85S1RA hydrochloride
CAS:<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Fórmula:C20H24ClN3O2Pureza:98% - 99.84%Cor e Forma:SolidPeso molecular:373.87BWX 46 Acetate
<p>BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.</p>Fórmula:C118H190N36O30S2Pureza:96.86%Cor e Forma:SolidPeso molecular:2657.12Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:<p>Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>Fórmula:C40H65F3N12O10Pureza:98.31%Cor e Forma:SolidPeso molecular:931.03Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Cor e Forma:SolidPeso molecular:369.54i
CAS:<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Fórmula:C16H12ClN3OPureza:99.49%Cor e Forma:SolidPeso molecular:297.74Neurokinin A(4-10) TFA(97559-35-8 free base)
<p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>Fórmula:C36H55F3N8O12SPureza:>99.99%Cor e Forma:SolidPeso molecular:880.93RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Fórmula:C25H27N3O3Pureza:98.64% - 99.62%Cor e Forma:SolidPeso molecular:417.5Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Cor e Forma:SolidPeso molecular:240.69HPI 1
CAS:<p>HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.</p>Fórmula:C27H29NO6Pureza:97.6%Cor e Forma:SolidPeso molecular:463.52ZK 756326
CAS:<p>ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.</p>Fórmula:C21H28N2O3Pureza:99.43%Cor e Forma:SolidPeso molecular:356.46Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Fórmula:C19H20ClN3Pureza:98% - 99.65%Cor e Forma:SolidPeso molecular:325.84Taladegib
CAS:<p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>Fórmula:C26H24F4N6OPureza:98.75% - >99.99%Cor e Forma:SolidPeso molecular:512.5LY334370
CAS:<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Fórmula:C21H22FN3OPureza:99.32%Cor e Forma:SolidPeso molecular:351.42Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Fórmula:C4H3F7OPureza:98%Cor e Forma:Less Oil Colorless OilPeso molecular:200.05ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Fórmula:C23H31N3O3SPureza:99.75%Cor e Forma:SolidPeso molecular:429.58PGS-IN-1
CAS:<p>PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).</p>Fórmula:C19H26O3Pureza:99.39%Cor e Forma:SolidPeso molecular:302.41HhAntag
CAS:<p>HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity</p>Fórmula:C24H23ClN4O3Pureza:95.73%Cor e Forma:SolidPeso molecular:450.92SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Fórmula:C28H28ClN3OSPureza:97.37% - 98.88%Cor e Forma:SolidPeso molecular:490.06Ciliobrevin A
CAS:<p>Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.</p>Fórmula:C17H9Cl2N3O2Pureza:98.54% - 99.57%Cor e Forma:SolidPeso molecular:358.18SANT-1
CAS:<p>SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).</p>Fórmula:C23H27N5Pureza:99.98% - >99.99%Cor e Forma:SolidPeso molecular:373.49
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