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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • Azaperone

    CAS:
    Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.
    Fórmula:C19H22FN3O
    Pureza:98.73%
    Cor e Forma:White Or Off-White Crystalline
    Peso molecular:327.4
  • Melanin Concentrating Hormone, salmon acetate


    <p>Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>
    Fórmula:C91H143N27O26S4
    Pureza:99.41%
    Cor e Forma:Solid
    Peso molecular:2157
  • Pizuglanstat

    CAS:
    <p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>
    Fórmula:C27H36N6O4
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:508.61
  • Betahistine EP Impurity C

    CAS:
    <p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>
    Fórmula:C15H19N3
    Pureza:≥95%
    Cor e Forma:Solid
    Peso molecular:241.33
  • Methiothepin mesylate

    CAS:
    <p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>
    Fórmula:C21H28N2O3S3
    Pureza:98% - 99.92%
    Cor e Forma:Solid
    Peso molecular:452.65
  • Praliciguat

    CAS:
    <p>Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.</p>
    Fórmula:C21H14F8N6O2
    Pureza:98.82%
    Cor e Forma:Solid
    Peso molecular:534.36
  • BMS 182874 hydrochloride

    CAS:
    <p>BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.</p>
    Fórmula:C17H20ClN3O3S
    Pureza:97.01%
    Cor e Forma:Solid
    Peso molecular:381.88
  • Landiolol hydrochloride

    CAS:
    <p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>
    Fórmula:C25H40ClN3O8
    Pureza:99.91%
    Cor e Forma:White Crystalline Powder
    Peso molecular:546.05
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Cor e Forma:Solid
    Peso molecular:538.64
  • A2B receptor antagonist 2

    CAS:
    <p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>
    Fórmula:C12H15N5
    Pureza:100%
    Cor e Forma:Solid
    Peso molecular:229.28
  • MF-766

    CAS:
    <p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>
    Fórmula:C27H21F3N2O3
    Pureza:99.54% - 99.59%
    Cor e Forma:Solid
    Peso molecular:478.46
  • Ciproxifan maleate

    CAS:
    <p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>
    Fórmula:C20H22N2O6
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:386.4
  • BWX 46 Acetate


    <p>BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.</p>
    Fórmula:C118H190N36O30S2
    Pureza:96.86%
    Cor e Forma:Solid
    Peso molecular:2657.12
  • AHN 1-055 hydrochloride

    CAS:
    <p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>
    Fórmula:C21H24ClF2NO
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:379.87
  • Raclopride

    CAS:
    <p>Raclopride is a selective antagonist of dopamine D2/D3 receptor.</p>
    Fórmula:C15H20Cl2N2O3
    Pureza:99.17%
    Cor e Forma:Solid
    Peso molecular:347.24
  • Piboserod

    CAS:
    <p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>
    Fórmula:C22H31N3O2
    Pureza:97.21% - 99.49%
    Cor e Forma:Solid
    Peso molecular:369.5
  • JNJ-7777120

    CAS:
    <p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits &gt;1000-fold selectivity over the other histamin receptors.</p>
    Fórmula:C14H16ClN3O
    Pureza:99.83% - 99.96%
    Cor e Forma:Solid
    Peso molecular:277.75
  • Bevantolol hydrochloride

    CAS:
    <p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>
    Fórmula:C20H28ClNO4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:381.9
  • Pimozide

    CAS:
    <p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>
    Fórmula:C28H29F2N3O
    Pureza:99.63% - >99.99%
    Cor e Forma:Solid
    Peso molecular:461.55
  • Clemizole

    CAS:
    <p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>
    Fórmula:C19H20ClN3
    Pureza:98% - 99.65%
    Cor e Forma:Solid
    Peso molecular:325.84
  • Taladegib

    CAS:
    <p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>
    Fórmula:C26H24F4N6O
    Pureza:98.75% - >99.99%
    Cor e Forma:Solid
    Peso molecular:512.5
  • CCG215022

    CAS:
    <p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>
    Fórmula:C26H22FN7O3
    Pureza:97.63% - 99.69%
    Cor e Forma:Solid
    Peso molecular:499.5
  • Clemizole hydrochloride

    CAS:
    Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.
    Fórmula:C19H21Cl2N3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:362.3
  • BMS-813160

    CAS:
    <p>BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.</p>
    Fórmula:C25H40N8O2
    Pureza:99.66% - 99.79%
    Cor e Forma:Solid
    Peso molecular:484.64
  • RS102895

    CAS:
    <p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>
    Fórmula:C21H21F3N2O2
    Pureza:97.64% - 99.80%
    Cor e Forma:Solid
    Peso molecular:390.4
  • Vercirnon

    CAS:
    <p>Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.</p>
    Fórmula:C22H21ClN2O4S
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:444.93
  • Geissoschizine methyl ether

    CAS:
    <p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>
    Fórmula:C22H26N2O3
    Pureza:99.24% - 99.68%
    Cor e Forma:Solid
    Peso molecular:366.45
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Fórmula:C18H15BrF2N4O2
    Pureza:98.42% - 99.88%
    Cor e Forma:Solid
    Peso molecular:437.24
  • Neurokinin A

    CAS:
    <p>Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.</p>
    Fórmula:C50H80N14O14S
    Pureza:>99.99%
    Cor e Forma:White To Off-White Lyophilized Solid
    Peso molecular:1133.32
  • Gastrin I (human) acetate


    Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (
    Fórmula:C99H128N20O33S
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:2158.25
  • Lurasidone hydrochloride

    CAS:
    Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.
    Fórmula:C28H36N4O2S·HCl
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:529.14
  • 2-Pyridylethylamine dihydrochloride

    CAS:
    <p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>
    Fórmula:C7H12Cl2N2
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:195.09
  • Loxapine

    CAS:
    <p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>
    Fórmula:C18H18ClN3O
    Pureza:99.88%
    Cor e Forma:Pale Yellowish Crystals From Petroleum Ether Solid
    Peso molecular:327.81
  • Pergolide

    CAS:
    <p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>
    Fórmula:C19H26N2S
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:314.49
  • Decloxizine

    CAS:
    <p>Decloxizine is a H1 receptor antagonist</p>
    Fórmula:C21H28N2O2
    Pureza:99.53%
    Cor e Forma:White Or Similar To White Powder
    Peso molecular:340.46
  • PF-04418948

    CAS:
    <p>PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.</p>
    Fórmula:C23H20FNO5
    Pureza:98.67% - 99.45%
    Cor e Forma:Solid
    Peso molecular:409.41
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Cor e Forma:Solid
    Peso molecular:433.57
  • Scyliorhinin II acetate


    <p>Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.</p>
    Fórmula:C79H123N21O28S3
    Pureza:99.06%
    Cor e Forma:Solid
    Peso molecular:1911.14
  • IPSU

    CAS:
    <p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>
    Fórmula:C23H27N5O2
    Pureza:97.05%
    Cor e Forma:Solid
    Peso molecular:405.49
  • BD1063 dhydrochloride

    CAS:
    BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).
    Fórmula:C13H20Cl4N2
    Pureza:99.52% - ≥95%
    Cor e Forma:Solid
    Peso molecular:346.12
  • Conopressin S acetate(111317-90-9 free base)


    <p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>
    Fórmula:C43H77N17O12S2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:1088.32
  • HAEGTFT acetate(926018-95-3 free base)


    <p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>
    Fórmula:C35H51N9O14
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:821.84
  • Linzagolix

    CAS:
    <p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>
    Fórmula:C22H15F3N2O7S
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:508.42
  • ACH-000143

    CAS:
    <p>ACH-000143 是一种可口服的褪黑素受体激动剂,对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>
    Fórmula:C13H16ClN3O3
    Pureza:98.15%
    Cor e Forma:Solid
    Peso molecular:297.74
  • Betaxolol

    CAS:
    <p>Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.</p>
    Fórmula:C18H29NO3
    Pureza:99.01%
    Cor e Forma:White Crystalline Solid
    Peso molecular:307.43
  • Bradykinin (acetate)

    CAS:
    <p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>
    Fórmula:C52H77N15O13
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1120.26
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Cor e Forma:Solid
    Peso molecular:463.87
  • 1-[(5-methylisoxazol-3-yl)methyl]piperazine

    CAS:
    <p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>
    Fórmula:C9H15N3O
    Pureza:95%
    Cor e Forma:Solid
    Peso molecular:181.23
  • VKGILS-NH2 Acetate


    <p>VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.</p>
    Fórmula:C30H58N8O9
    Pureza:98.83%
    Cor e Forma:Solid
    Peso molecular:674.83
  • DORA-22

    CAS:
    <p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>
    Fórmula:C23H22F2N4O2
    Pureza:97.67%
    Cor e Forma:Solid
    Peso molecular:424.44
  • Peptide YY (PYY) (3-36), human

    CAS:
    <p>Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.</p>
    Fórmula:C176H272N52O54
    Pureza:97.76%
    Cor e Forma:Solid
    Peso molecular:3980.42
  • Doxazosin

    CAS:
    <p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>
    Fórmula:C23H25N5O5
    Pureza:99.47% - 99.87%
    Cor e Forma:Solid
    Peso molecular:451.48
  • ZM241385

    CAS:
    <p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>
    Fórmula:C16H15N7O2
    Pureza:97.02% - 99.69%
    Cor e Forma:Solid
    Peso molecular:337.34
  • S 38093 HCl

    CAS:
    <p>S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.</p>
    Fórmula:C17H25ClN2O2
    Pureza:97.91%
    Cor e Forma:Solid
    Peso molecular:324.85
  • Cetirizine Impurity B dihydrochloride

    CAS:
    <p>Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.</p>
    Fórmula:C19H23Cl3N2O2
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:417.76
  • Antalarmin

    CAS:
    <p>Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.</p>
    Fórmula:C24H34N4
    Cor e Forma:Solid
    Peso molecular:378.55
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:417.89
  • Elinzanetant

    CAS:
    <p>Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.</p>
    Fórmula:C33H35F7N4O3
    Pureza:98% - 99.13%
    Cor e Forma:Solid
    Peso molecular:668.64
  • Galanin Receptor Ligand M35 TFA


    <p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>
    Fórmula:C109H154N27F3O28
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:2347.62
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Fórmula:C35H47FN10O8
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:754.85
  • Carazolol

    CAS:
    <p>Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.</p>
    Fórmula:C18H22N2O2
    Pureza:99% - 99.53%
    Cor e Forma:Yellowish Solid
    Peso molecular:298.38
  • Pancreatic Polypeptide, rat acetate


    Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.
    Pureza:97.53%
    Cor e Forma:Solid
    Peso molecular:N/A
  • ML382

    CAS:
    <p>ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).</p>
    Fórmula:C18H20N2O4S
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:360.43
  • CGP 20712 A

    CAS:
    <p>CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.</p>
    Fórmula:C24H29F3N4O8S
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:590.57
  • BMS-986278

    CAS:
    <p>BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,</p>
    Fórmula:C22H31N5O5
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:445.51
  • Tandospirone

    CAS:
    <p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>
    Fórmula:C21H29N5O2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:383.49
  • Maropitant citrate

    CAS:
    <p>Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.</p>
    Fórmula:C38H50N2O9
    Pureza:98.91%
    Cor e Forma:Solid
    Peso molecular:678.81
  • Rotigotine

    CAS:
    Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.
    Fórmula:C19H25NOS
    Pureza:99.04% - 99.88%
    Cor e Forma:Solid
    Peso molecular:315.47
  • CB1/2 agonist 3

    CAS:
    <p>CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.</p>
    Fórmula:C25H41NO2
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:387.6
  • Clopidogrel thiolactone

    CAS:
    Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.
    Fórmula:C16H16ClNO3S
    Pureza:98.79%
    Cor e Forma:Solid
    Peso molecular:337.82
  • L-368,899 hydrochloride

    CAS:
    <p>L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.</p>
    Fórmula:C26H43ClN4O5S2
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:591.23
  • Medetomidine

    CAS:
    <p>Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.</p>
    Fórmula:C13H16N2
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:200.28
  • UCM 608

    CAS:
    <p>UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.</p>
    Fórmula:C19H20N2O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:308.37
  • Nebentan potassium

    CAS:
    <p>Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.</p>
    Fórmula:C24H20KN5O5S
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:529.61
  • Trabodenoson

    CAS:
    <p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>
    Fórmula:C15H20N6O6
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:380.36
  • S1RA

    CAS:
    <p>S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2</p>
    Fórmula:C20H23N3O2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:337.42
  • Fenoterol hydrobromide

    CAS:
    Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.
    Fórmula:C17H22BrNO4
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:384.27
  • S-Methoprene

    CAS:
    <p>S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.</p>
    Fórmula:C19H34O3
    Pureza:97.05% - 98.55%
    Cor e Forma:Solid
    Peso molecular:310.47
  • GRK6-IN-2

    CAS:
    <p>GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.</p>
    Fórmula:C21H21FN6
    Pureza:98.94%
    Cor e Forma:Solid
    Peso molecular:376.43
  • Jatrorrhizine chloride

    CAS:
    <p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>
    Fórmula:C20H20ClNO4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:373.8
  • Citalopram

    CAS:
    <p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>
    Fórmula:C20H21FN2O
    Pureza:99.78% - 99.89%
    Cor e Forma:Solid
    Peso molecular:324.39
  • Opipramol

    CAS:
    <p>Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.</p>
    Fórmula:C23H29N3O
    Pureza:99.84% - 99.98%
    Cor e Forma:Solid
    Peso molecular:363.5
  • A2ti-1

    CAS:
    A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.
    Fórmula:C20H22N4O2S
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:382.48
  • Rizatriptan

    CAS:
    <p>Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.</p>
    Fórmula:C15H19N5
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:269.35
  • Fenoprofen

    CAS:
    Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.
    Fórmula:C15H14O3
    Pureza:98.4%
    Cor e Forma:Solid
    Peso molecular:242.27
  • Ketanserin tartrate

    CAS:
    Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.
    Fórmula:C26H28FN3O9
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:545.51
  • WIN 51,708

    CAS:
    WIN 51,708 is an antagonist of neurokinin-1 receptor.
    Fórmula:C29H33N3O
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:439.59
  • Bucindolol

    CAS:
    <p>Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.</p>
    Fórmula:C22H25N3O2
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:363.45
  • AF-710B

    CAS:
    <p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>
    Fórmula:C20H27N3OS
    Pureza:98.62% - 99.89%
    Cor e Forma:Solid
    Peso molecular:357.51
  • Atipamezole

    CAS:
    Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
    Fórmula:C14H16N2
    Pureza:99.88%
    Cor e Forma:Off-White To Light Yellow Crystal Powder
    Peso molecular:212.29
  • SB 243213

    CAS:
    <p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>
    Fórmula:C22H19F3N4O2
    Pureza:98.78% - 99.86%
    Cor e Forma:Solid
    Peso molecular:428.41
  • Setiptiline

    CAS:
    Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.
    Fórmula:C19H19N
    Pureza:98.05% - 98.07%
    Cor e Forma:Solid
    Peso molecular:261.36
  • Atogepant

    CAS:
    <p>Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.</p>
    Fórmula:C29H23F6N5O3
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:603.52
  • Pentoxyverine

    CAS:
    Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.
    Fórmula:C20H31NO3
    Pureza:97.11%
    Cor e Forma:Solid
    Peso molecular:333.47
  • Protein deglycase DJ-1 against-1

    CAS:
    <p>Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.</p>
    Fórmula:C24H23N3O4
    Pureza:97.23%
    Cor e Forma:Solid
    Peso molecular:417.46
  • Canagliflozin hemihydrate

    CAS:
    <p>Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.</p>
    Fórmula:C48H52F2O11S2
    Pureza:99.42% - 99.96%
    Cor e Forma:Solid
    Peso molecular:907.05
  • ACT-462206

    CAS:
    ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.
    Fórmula:C20H24N2O4S
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:388.48
  • Levocetirizine Dihydrochloride

    CAS:
    <p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>
    Fórmula:C21H27Cl3N2O3
    Pureza:99.89%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:461.81
  • LP-533401 hydrochloride

    CAS:
    LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.
    Fórmula:C27H23ClF4N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:562.94
  • Poly-D-lysine hydrobromide (MW 30000-70000)

    CAS:
    Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.
    Fórmula:(C6H14N2O2)x·xHBr
    Cor e Forma:Solid
    Peso molecular:227.102
  • SID 7969543

    CAS:
    <p>SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.</p>
    Fórmula:C24H24N2O7
    Pureza:98.94%
    Cor e Forma:Solid
    Peso molecular:452.46
  • Ozanimod hydrochloride

    CAS:
    Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.
    Fórmula:C23H25ClN4O3
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:440.92
  • CP-105696

    CAS:
    <p>CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.</p>
    Fórmula:C28H28O4
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:428.52
  • Rolofylline

    CAS:
    <p>Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.</p>
    Fórmula:C20H28N4O2
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:356.46
  • Dexpramipexole

    CAS:
    Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.
    Fórmula:C10H17N3S
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:211.33
  • GAT211

    CAS:
    <p>GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.</p>
    Fórmula:C22H18N2O2
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:342.39
  • WAY-100635 maleate

    CAS:
    <p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>
    Fórmula:C25H34N4O2·xC4H4O4
    Pureza:>99.99%
    Cor e Forma:White Solid
    Peso molecular:538.645
  • INCB 3284

    CAS:
    INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.
    Fórmula:C26H31F3N4O4
    Pureza:97.81% - 99.42%
    Cor e Forma:Solid
    Peso molecular:520.54
  • Alfuzosin

    CAS:
    <p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>
    Fórmula:C19H27N5O4
    Pureza:99.64%
    Cor e Forma:White Crystaline Powder
    Peso molecular:389.45
  • KB-5492 free base

    CAS:
    <p>KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.</p>
    Fórmula:C23H30N2O6
    Pureza:97.10% - 97.94%
    Cor e Forma:Solid
    Peso molecular:430.49
  • Latrepirdine dihydrochloride

    CAS:
    Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.
    Fórmula:C21H25N3·2HCl
    Pureza:98.45%
    Cor e Forma:Solid
    Peso molecular:392.37
  • (R)-Mirtazapine

    CAS:
    <p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>
    Fórmula:C17H19N3
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Trazpiroben

    CAS:
    Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.
    Fórmula:C31H39N3O4
    Pureza:99.41% - >99.99%
    Cor e Forma:Solid
    Peso molecular:517.66
  • Renzapride

    CAS:
    Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.
    Fórmula:C16H22ClN3O2
    Pureza:98.97% - 99.09%
    Cor e Forma:Solid
    Peso molecular:323.82
  • (S)-Mirtazapine

    CAS:
    (S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.
    Fórmula:C17H19N3
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Syk Inhibitor II

    CAS:
    <p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>
    Fórmula:C14H15F3N6O
    Pureza:97.63%
    Cor e Forma:Solid
    Peso molecular:340.3
  • R 59-022

    CAS:
    <p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>
    Fórmula:C27H26FN3OS
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:459.58
  • L-745870

    CAS:
    <p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>
    Fórmula:C18H19ClN4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:326.82
  • Ropinirole

    CAS:
    <p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>
    Fórmula:C16H24N2O
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:260.38
  • SR59230A hydrochloride

    CAS:
    <p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>
    Fórmula:C21H28ClNO2
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:361.91
  • Travoprost

    CAS:
    <p>Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.</p>
    Fórmula:C26H35F3O6
    Pureza:97.39% - 99.58%
    Cor e Forma:Colorless Oil
    Peso molecular:500.55
  • PACAP (1-38), human, ovine, rat

    CAS:
    PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.
    Fórmula:C203H331N63O53S
    Pureza:96.93% - 98.16%
    Cor e Forma:Solid
    Peso molecular:4534.26
  • Cyproheptadine hydrochloride

    CAS:
    <p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>
    Fórmula:C21H21N·HCl
    Pureza:99.88% - 99.97%
    Cor e Forma:Solid
    Peso molecular:323.86
  • Methaphenilene hydrochloride

    CAS:
    <p>Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.</p>
    Fórmula:C15H21ClN2S
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:296.86
  • GPR183-IN-1

    CAS:
    <p>GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.</p>
    Fórmula:C16H19BrN2O2
    Cor e Forma:Solid
    Peso molecular:351.24
  • Buflomedil

    CAS:
    <p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>
    Fórmula:C17H25NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:307.38
  • Eptinezumab

    CAS:
    <p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>
    Pureza:95% - 95%
    Cor e Forma:Liquid
  • Olopatadine

    CAS:
    <p>Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.</p>
    Fórmula:C21H23NO3
    Pureza:98%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:337.41
  • Carlumab

    CAS:
    <p>Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.</p>
    Pureza:95%
    Cor e Forma:Liquid
  • Mibavademab

    CAS:
    <p>Mibavademab is a humanized anti-leptin receptor (LEPR) mAb under investigation for treating congenital leptin deficiency.</p>
    Pureza:95%
    Cor e Forma:Liquid
  • 17-phenyl trinor Prostaglandin F2α isopropyl ester

    CAS:
    <p>17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the Allergan</p>
    Fórmula:C26H38O5
    Cor e Forma:Solid
    Peso molecular:430.58
  • PF-610355

    CAS:
    <p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>
    Fórmula:C34H39N3O6S
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:617.76
  • DL-Phenylephrine HCl

    CAS:
    DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.
    Fórmula:C9H14ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:203.67
  • Fremanezumab

    CAS:
    <p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>
    Pureza:95% - 95%
    Cor e Forma:Liquid
  • Risperidone Mesylate

    CAS:
    <p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>
    Fórmula:C24H31FN4O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:506.59
  • Keto Ziprasidone

    CAS:
    <p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>
    Fórmula:C21H19ClN4O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:426.92
  • N-Methyl amisulpride

    CAS:
    <p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>
    Fórmula:C18H29N3O4S
    Cor e Forma:Solid
    Peso molecular:383.51
  • Blontuvetmab

    CAS:
    <p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>
    Cor e Forma:Liquid
  • Metoxibutropate

    CAS:
    <p>Metoxibutropate is a biochemical.</p>
    Fórmula:C20H24O3
    Cor e Forma:Solid
    Peso molecular:312.4
  • Arazasetron HCl

    CAS:
    <p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>
    Fórmula:C17H20ClN3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:349.81
  • P2Y14R antagonist 1

    CAS:
    <p>P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.</p>
    Fórmula:C15H12BrN3O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:346.18
  • Meticillin

    CAS:
    <p>Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.</p>
    Fórmula:C17H20N2O6S
    Cor e Forma:Solid
    Peso molecular:380.42
  • Tulobuterol

    CAS:
    <p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>
    Fórmula:C12H18ClNO
    Cor e Forma:Crystalline Solid
    Peso molecular:227.73
  • Triflupromazine

    CAS:
    <p>Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.</p>
    Fórmula:C18H19F3N2S
    Cor e Forma:Solid
    Peso molecular:352.42
  • Uliledlimab

    CAS:
    <p>Uliledlimab, a humanized monoclonal antibody against CD73, reduces extracellular adenosine production and modulates immunosuppressive pathways.</p>
    Pureza:95% - 95%
    Cor e Forma:Liquid
  • Escitalopram

    CAS:
    <p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>
    Fórmula:C20H21FN2O
    Pureza:99.82%
    Cor e Forma:White Or White Crystalline Powder
    Peso molecular:324.39
  • 15-keto Prostaglandin F2α

    CAS:
    <p>15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.</p>
    Fórmula:C20H32O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.47
  • Brexpiprazole-d8

    CAS:
    <p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>
    Fórmula:C25H27N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:441.62
  • Mirtazapine D3

    CAS:
    Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .
    Fórmula:C17H19N3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:268.37
  • Dapagliflozin-d5

    CAS:
    Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.
    Fórmula:C21H25ClO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:413.9
  • Cinnarizine D8

    CAS:
    <p>Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.</p>
    Fórmula:C26H28N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:376.573
  • Amitriptyline-d6 Hydrochloride

    CAS:
    <p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>
    Fórmula:C20H18D6ClN
    Cor e Forma:Solid
    Peso molecular:319.90
  • 5-Methyltryptamine hydrochloride

    CAS:
    <p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>
    Fórmula:C11H15ClN2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:210.703
  • 7-Desmethyl-3-hydroxyagomelatine

    CAS:
    <p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>
    Fórmula:C14H15NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:245.27
  • Tivumecirnon

    CAS:
    <p>Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumour</p>
    Fórmula:C24H27Cl2F3N6O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:543.41
  • (RS)-ICI-118551 Hydrochloride

    CAS:
    ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3
    Fórmula:C17H27NO2·HCl
    Pureza:98.02%
    Cor e Forma:Solid
    Peso molecular:313.86
  • Ketanserinol

    CAS:
    <p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>
    Fórmula:C22H24FN3O3
    Cor e Forma:Solid
    Peso molecular:397.44
  • Amthamine

    CAS:
    <p>Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.</p>
    Fórmula:C6H11N3S
    Cor e Forma:Soild
    Peso molecular:157.24
  • MK-447

    CAS:
    <p>MK-447 is a nonsteroidal antiinflammatory agent.</p>
    Fórmula:C11H16INO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:305.16
  • Roxatidine acetate

    CAS:
    <p>Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.</p>
    Fórmula:C19H28N2O4
    Pureza:98%
    Cor e Forma:White Or Off-White Powder
    Peso molecular:348.44
  • Diclofensine

    CAS:
    <p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>
    Fórmula:C17H17Cl2NO
    Pureza:97.01% - 98.13%
    Cor e Forma:Solid
    Peso molecular:322.23
  • Dehydroabiethylamine

    CAS:
    <p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs &amp; cholesterol transport, and has anti-tumor effects.</p>
    Fórmula:C20H31N
    Pureza:98.79%
    Cor e Forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber Liquid
    Peso molecular:285.47
  • Amidephrine hydrochloride

    CAS:
    <p>Amidephrine hydrochloride is a biochemical.</p>
    Fórmula:C10H17ClN2O3S
    Cor e Forma:Solid
    Peso molecular:280.77
  • 7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene

    CAS:
    <p>7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).</p>
    Fórmula:C42H44N2O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:704.87
  • Isoproterenol sulfate anhydrous

    CAS:
    <p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>
    Fórmula:C22H36N2O10S
    Pureza:98%
    Cor e Forma:Coa
    Peso molecular:520.59
  • Ticlopidine

    CAS:
    <p>Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.</p>
    Fórmula:C14H14ClNS
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:263.79
  • Atenolol Hydrochloride

    CAS:
    <p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>
    Fórmula:C14H23ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:302.80
  • Vanoxerine

    CAS:
    <p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>
    Fórmula:C28H32F2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:450.56
  • Hydroxy ziprasidone

    CAS:
    <p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>
    Fórmula:C21H21ClN4O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:428.94
  • Itopride free base

    CAS:
    <p>Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.</p>
    Fórmula:C20H26N2O4
    Cor e Forma:White
    Peso molecular:358.43
  • S 25585

    CAS:
    <p>S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>
    Fórmula:C22H23F3N4O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:528.5
  • Norreticuline

    CAS:
    <p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>
    Fórmula:C18H21NO4
    Cor e Forma:Solid
    Peso molecular:315.36
  • Pardoprunox

    CAS:
    <p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>
    Fórmula:C12H15N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:233.27
  • R-138727

    CAS:
    <p>R-138727 is a novel P2Y12 receptor inhibitor.</p>
    Fórmula:C18H20FNO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:349.42
  • Litorin

    CAS:
    <p>Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.</p>
    Fórmula:C51H68N14O11S
    Cor e Forma:White Powder
    Peso molecular:1085.24
  • Penbutolol sulfate

    CAS:
    <p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>
    Fórmula:C18H29NO2H2O4S
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:340.47
  • Ciproxifan

    CAS:
    <p>Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).</p>
    Fórmula:C16H18N2O2
    Pureza:98.00%
    Cor e Forma:Solid
    Peso molecular:270.33
  • Caerulein, desulfated

    CAS:
    Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.
    Fórmula:C58H73N13O18S
    Pureza:99.46%
    Cor e Forma:Solid
    Peso molecular:1272.34
  • SB 271046 hydrochloride

    CAS:
    <p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is &gt; 200-fold selective over 55 other receptors, enzymes and ion channels.</p>
    Fórmula:C20H22ClN3O3S2·HCl
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:488.45
  • Ridazolol HCl

    CAS:
    <p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>
    Fórmula:C15H19Cl3N4O3
    Pureza:99.48%
    Cor e Forma:Soild
    Peso molecular:409.7
  • Amidephrine

    CAS:
    <p>Amidephrine is an adrenergic agent.</p>
    Fórmula:C10H16N2O3S
    Cor e Forma:Solid
    Peso molecular:244.31
  • Guacetisal

    CAS:
    <p>Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.</p>
    Fórmula:C16H14O5
    Pureza:99.18%
    Cor e Forma:Solid
    Peso molecular:286.28
  • MK-5046

    CAS:
    MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
    Fórmula:C20H18F6N4O
    Pureza:98.56%
    Cor e Forma:Solid
    Peso molecular:444.37
  • Paroxetine hydrochloride hemihydrate

    CAS:
    <p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>
    Fórmula:C38H44Cl2F2N2O7
    Pureza:99.949%
    Cor e Forma:Solid
    Peso molecular:749.67
  • LY 344864

    CAS:
    <p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>
    Fórmula:C21H22FN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:351.42
  • Dolasetron Mesylate

    CAS:
    <p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>
    Fórmula:C20H24N2O6S
    Pureza:99.05%
    Cor e Forma:White Powder
    Peso molecular:420.48
  • Lodoxamide tromethamine

    CAS:
    <p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>
    Fórmula:C19H28ClN5O12
    Pureza:98.8%
    Cor e Forma:Solid
    Peso molecular:553.91
  • Ketotifen

    CAS:
    <p>Ketotifen: Oral H1 blocker &amp; mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE &amp; asthma prevention research.</p>
    Fórmula:C19H19NOS
    Cor e Forma:Solid
    Peso molecular:309.43
  • CB1/2 agonist 2

    CAS:
    <p>CB1/2 agonist 2 binds tightly to cannabinoid receptors, acting fully on CB1 and inversely on CB2.</p>
    Fórmula:C26H43NO3
    Cor e Forma:Solid
    Peso molecular:417.62
  • (Rac)-WAY-161503

    CAS:
    <p>(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.</p>
    Fórmula:C11H11Cl2N3O
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:272.13
  • Pitolisant oxalate

    CAS:
    <p>Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>
    Fórmula:C19H28ClNO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:385.88
  • WAY 161503 hydrochloride

    CAS:
    <p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>
    Fórmula:C11H12Cl3N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:308.59
  • SKF-83822

    CAS:
    <p>SKF-83822 is an agonist of dopamine D1-like receptor.</p>
    Fórmula:C20H22ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.85
  • Ro 19-1400

    CAS:
    <p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>
    Fórmula:C31H56N2O8S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:616.85
  • (Rac)-E1R

    CAS:
    <p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>
    Fórmula:C13H16N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:232.28
  • Bufetolol

    CAS:
    Bufetolol is an antagonist of beta-adrenoceptor.
    Fórmula:C18H29NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:323.43
  • GSK 189254 HCl

    CAS:
    <p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>
    Fórmula:C21H26ClN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:387.9
  • Kadsurenone

    CAS:
    <p>Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.</p>
    Fórmula:C21H24O5
    Cor e Forma:Solid
    Peso molecular:356.41
  • SUN-C5174

    CAS:
    <p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>
    Fórmula:C22H29FN4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:400.49
  • Tertatolol

    CAS:
    <p>Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.</p>
    Fórmula:C16H25NO2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:295.44