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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • BN 50341

    CAS:
    <p>BN 50341 is an inhibitor of antithrombotic platelet activating factor.</p>
    Fórmula:C32H41ClN2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:553.13
  • Dacopafant

    CAS:
    <p>Dacopafant is an antagonist of platlet activationg factor receptor.</p>
    Fórmula:C12H11N3OS
    Cor e Forma:Solid
    Peso molecular:245.3
  • SNAP 5089

    CAS:
    α1A-adrenoceptor antagonist
    Fórmula:C36H40N4O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:608.73
  • CUMI-101

    CAS:
    <p>CUMI-101 is an agonist of 5-HT1A receptor.</p>
    Fórmula:C19H27N5O3
    Cor e Forma:Solid
    Peso molecular:373.45
  • Dihydroalprenolol, (S)-

    CAS:
    <p>Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.</p>
    Fórmula:C15H25NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:251.36
  • 2MeSAMP

    CAS:
    <p>2MeSAMP is a P2Y(12) antagonist that works by inhibiting platelet activation through a P2Y(12)/G(i)-dependent mechanism.</p>
    Fórmula:C11H16N5NaO7PS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:416.3
  • Gyki 32887

    CAS:
    <p>Gyki 32887 is a dopamine agonist.</p>
    Fórmula:C23H28N6O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:516.57
  • SMANT hydrochloride

    CAS:
    SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.
    Fórmula:C16H24BrClN2O
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:375.73
  • Carcainium chloride

    CAS:
    <p>Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.</p>
    Fórmula:C18H22ClN3O2
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:347.84
  • PGlu-3-methyl-His-Pro-NH2 TFA


    <p>PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding &amp; TSH release.</p>
    Fórmula:C19H25F3N6O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:490.43
  • RS 52367

    CAS:
    <p>RS 52367 is a beta-adrenergic antagonist.</p>
    Fórmula:C18H34ClN3O3S
    Cor e Forma:Solid
    Peso molecular:408
  • Lergotrile

    CAS:
    <p>Lergotrile is used as an enzyme Inhibitor (Prolactin).</p>
    Fórmula:C17H18ClN3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:299.8
  • FAUC-3019

    CAS:
    <p>FAUC-3019 is a partial agonist of the dopamine D(4) receptor.</p>
    Fórmula:C22H24N2O
    Cor e Forma:Solid
    Peso molecular:332.44
  • Butidrine

    CAS:
    <p>Butidrine has an Antiarrhythmic activities.</p>
    Fórmula:C16H25NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:247.38
  • WS 009B

    CAS:
    WS 009B is an antagonist of the endothelin receptor.
    Fórmula:C24H25NO11S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:535.52
  • SB 268262

    CAS:
    <p>CGRP1 antagonist</p>
    Fórmula:C18H15N3O4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:401.46
  • Losmiprofen

    CAS:
    <p>Losmiprofen is a nonsteroidal compound of antiinflammatory.</p>
    Fórmula:C17H15ClO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.75
  • Cafaminol

    CAS:
    <p>Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.</p>
    Fórmula:C11H17N5O3
    Cor e Forma:Solid
    Peso molecular:267.28
  • DAT 582

    CAS:
    <p>DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent</p>
    Fórmula:C22H28ClN5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:413.95
  • Daglutril

    CAS:
    <p>Daglutril is a NEP/ECE inhibitor for treating hypertension, heart failure, and pulmonary issues, blocking big endothelin-1 conversion.</p>
    Fórmula:C31H38N2O6
    Cor e Forma:Solid
    Peso molecular:534.64
  • JTH-601 free base

    CAS:
    <p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>
    Fórmula:C24H35NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:401.54
  • Iodophenpropit dihydrobromide

    CAS:
    <p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>
    Fórmula:C15H20BrIN4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:495.22
  • Asperlicin D

    CAS:
    <p>Asperlicin D is a cholecystokinin antagonist agent.</p>
    Fórmula:C25H18N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:406.44
  • LY 25648

    CAS:
    <p>LY 25648 is an antagonist of leukotriene B4.</p>
    Fórmula:C19H27NO2S
    Cor e Forma:Solid
    Peso molecular:333.49
  • VK-II-86

    CAS:
    VK-II-86 is a non-β-blocking carvedilol analog. It prevents ouabain-Induced cardiotoxicity
    Fórmula:C25H28N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:420.5
  • KLS-13019

    CAS:
    <p>KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).</p>
    Fórmula:C22H29NO3
    Pureza:>99.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:355.47
  • GS 283

    CAS:
    <p>GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.</p>
    Fórmula:C17H17NO3
    Cor e Forma:Solid
    Peso molecular:283.32
  • Viprostol

    CAS:
    Viprostol is an agent of prostaglandin antihypertensive.
    Fórmula:C23H36O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:392.53
  • Garomefrine HCl

    CAS:
    <p>Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.</p>
    Fórmula:C9H14ClFN2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:284.73
  • Chloracyzine

    CAS:
    <p>Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.</p>
    Fórmula:C19H21ClN2OS
    Cor e Forma:Solid
    Peso molecular:360.9
  • Alclofenac sodium

    CAS:
    <p>Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.</p>
    Fórmula:C11H11ClNaO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:249.65
  • Tecalcet Hydrochloride

    CAS:
    <p>Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.</p>
    Fórmula:C18H23Cl2NO
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:340.29
  • SARS-CoV-2-IN-57

    CAS:
    <p>SARS-CoV-2-IN-57 (compound (+)-R-26) is a potent inhibitor of SARS-CoV-2 with an IC50 of 80 nM and demonstrates high affinity for the Sigma Receptor, exhibiting</p>
    Fórmula:C23H37N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:371.56
  • AMX12006

    CAS:
    <p>AMX12006, a potent and selective EP4 antagonist, exhibits cytotoxic and antitumor activity, demonstrating oral activity with an IC50 of 4.3 nM [1].</p>
    Fórmula:C26H22F3N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:481.47
  • Quinpirole Hydrochloride

    CAS:
    <p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>
    Fórmula:C13H22ClN3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:255.79
  • WAY 163909

    CAS:
    WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).
    Fórmula:C14H18N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:214.31
  • PF2562

    CAS:
    <p>PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).</p>
    Fórmula:C19H17N5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.37
  • Chlorazanil

    CAS:
    <p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>
    Fórmula:C9H8ClN5
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:221.65
  • Eplivanserin

    CAS:
    Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
    Fórmula:C19H21FN2O2
    Pureza:97.04%
    Cor e Forma:Solid
    Peso molecular:328.38
  • NRA-0160

    CAS:
    <p>NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)</p>
    Fórmula:C24H23F2N3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:439.52
  • BW 245C

    CAS:
    <p>BW 245C is a DP1 agonist with an inhibitory effect on the aggregation response of collagen and can be used to study diseases such as stroke.</p>
    Fórmula:C19H32N2O5
    Pureza:≥99%
    Cor e Forma:Solid
    Peso molecular:368.47
  • OMDM-6

    CAS:
    <p>OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.</p>
    Fórmula:C28H42N2O3
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:454.64
  • Mianserin

    CAS:
    <p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>
    Fórmula:C18H20N2
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:264.36
  • I942

    CAS:
    <p>I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to regulate inflammatory gene expression in human umbilical</p>
    Fórmula:C20H19NO4S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:369.43
  • Medroxalol

    CAS:
    <p>Medroxalol (RMI81968), an oral α- &amp; β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>
    Fórmula:C20H24N2O5
    Cor e Forma:Solid
    Peso molecular:372.42
  • Wy 49051

    CAS:
    <p>Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).</p>
    Fórmula:C28H33N5O3
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:487.59
  • PF-03654746

    CAS:
    <p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>
    Fórmula:C18H24F2N2O
    Pureza:98.85% - 99.57%
    Cor e Forma:Solid
    Peso molecular:322.39
  • ChemR23-IN-1

    CAS:
    <p>ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.</p>
    Fórmula:C28H29N7O2
    Cor e Forma:Solid
    Peso molecular:495.58
  • Edivoxetine

    CAS:
    <p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>
    Fórmula:C18H26FNO4
    Cor e Forma:Solid
    Peso molecular:339.4
  • PD 144418

    CAS:
    <p>PD 144418 displays potential antipsychotic activity.</p>
    Fórmula:C18H22N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:282.38
  • F13714 fumarate

    CAS:
    <p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>
    Fórmula:C25H29ClF2N4O5
    Pureza:98.86%
    Cor e Forma:Solid
    Peso molecular:538.97
  • Rec 15/2615 dihydrochloride

    CAS:
    Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.
    Fórmula:C26H35Cl2N5O5
    Pureza:97.04% - 99.76%
    Cor e Forma:Solid
    Peso molecular:568.49
  • PGD2-IN-1

    CAS:
    <p>PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.</p>
    Fórmula:C23H23Cl2N3O3
    Pureza:98.21%
    Cor e Forma:Solid
    Peso molecular:460.35
  • INCB38579

    CAS:
    <p>INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.</p>
    Fórmula:C25H34N6O
    Cor e Forma:Solid
    Peso molecular:434.58
  • Org-13011 fumarate

    CAS:
    <p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>
    Fórmula:C22H29F3N4O5
    Pureza:98.92%
    Cor e Forma:Solid
    Peso molecular:486.48
  • CGP 35949

    CAS:
    <p>CGP 35949 is an LTD4 antagonist with phospholipase inhibitory activity.</p>
    Fórmula:C23H25ClN5NaO5
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:509.92
  • Povafonidine

    CAS:
    <p>Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.</p>
    Fórmula:C11H13N5
    Cor e Forma:Solid
    Peso molecular:215.25
  • CB2 modulator 1

    CAS:
    <p>CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.</p>
    Fórmula:C18H19F3N4O2
    Pureza:99.6%
    Cor e Forma:Solid
    Peso molecular:380.36
  • 5-HT7 agonist 2

    CAS:
    <p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>
    Fórmula:C23H29N3O
    Cor e Forma:Solid
    Peso molecular:363.5
  • Zenidolol

    CAS:
    <p>Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.</p>
    Fórmula:C17H27NO2
    Cor e Forma:Solid
    Peso molecular:277.4
  • (Rac)-HAMI 3379

    CAS:
    <p>HAMI 3379: potent CysLT2 receptor blocker; protects against acute/subacute brain injury; reduces microglia inflammation.</p>
    Fórmula:C34H45NO8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:595.72
  • BRL 37344 sodium

    CAS:
    <p>BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.</p>
    Fórmula:C19H22ClNNaO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.83
  • A-943931

    CAS:
    A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.
    Fórmula:C17H21N5
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:295.38
  • AL-3138

    CAS:
    <p>AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.</p>
    Fórmula:C20H33FO4
    Cor e Forma:Solid
    Peso molecular:356.47
  • ICI 192605

    CAS:
    <p>ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.</p>
    Fórmula:C22H23ClO5
    Cor e Forma:Solid
    Peso molecular:402.87
  • (S)-(-)-Propranolol hydrochloride

    CAS:
    <p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>
    Fórmula:C16H22ClNO2
    Pureza:99.02% - 99.91%
    Cor e Forma:Solid
    Peso molecular:295.8
  • Befetupitant

    CAS:
    <p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>
    Fórmula:C29H29F6N3O2
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:565.55
  • PD-156707

    CAS:
    <p>PD-156707 is a selective antagonist of endothelin A receptor.</p>
    Fórmula:C28H26NaO9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:529.497
  • Lidanserin

    CAS:
    <p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>
    Fórmula:C26H31FN2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.53
  • WAY208466 dihydrochloride

    CAS:
    <p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>
    Fórmula:C17H20Cl2FN3O2S
    Pureza:98.43%
    Cor e Forma:Solid
    Peso molecular:420.33
  • GAT228

    CAS:
    <p>GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].</p>
    Fórmula:C22H18N2O2
    Cor e Forma:Solid
    Peso molecular:342.39
  • PD 81723

    CAS:
    <p>Allosteric potentiator at the adenosine A1 receptor</p>
    Fórmula:C14H12F3NOS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:299.31
  • A-940894

    CAS:
    <p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>
    Fórmula:C17H21N5
    Cor e Forma:Solid
    Peso molecular:295.38
  • 5-HT7 receptor ligand 1

    CAS:
    <p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>
    Fórmula:C21H23N7
    Cor e Forma:Solid
    Peso molecular:373.45
  • LY 302148

    CAS:
    <p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>
    Fórmula:C19H23FN4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:326.41
  • SKF-104557

    CAS:
    <p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>
    Fórmula:C13H18N2O
    Cor e Forma:Solid
    Peso molecular:218.29
  • CP 135807

    CAS:
    <p>CP 135807 is a 5-HT1D receptor agonist.</p>
    Fórmula:C19H21N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:351.4
  • Enciprazine

    CAS:
    Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.
    Fórmula:C23H32N2O6
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:432.51
  • CID1172084

    CAS:
    CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.
    Fórmula:C23H18FN5O2S2
    Cor e Forma:Solid
    Peso molecular:479.55
  • PNU-177864 hydrochloride

    CAS:
    <p>PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor.</p>
    Fórmula:C18H22ClF3N2O3S
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:438.89
  • PF-184298

    CAS:
    <p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>
    Fórmula:C15H20Cl2N2O
    Pureza:98.67%
    Cor e Forma:Solid
    Peso molecular:315.24
  • Tedatioxetine hydrobromide

    CAS:
    Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.
    Fórmula:C18H22BrNS
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:364.34
  • Licogliflozin

    CAS:
    <p>Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).</p>
    Fórmula:C23H28O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:416.46
  • CCG-2046

    CAS:
    <p>CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.</p>
    Fórmula:C11H10N4
    Cor e Forma:Solid
    Peso molecular:198.22
  • L-692429

    CAS:
    L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can be used to study acromegaly and obesity.
    Fórmula:C29H31N7O2
    Pureza:98.64% - 99.90%
    Cor e Forma:Solid
    Peso molecular:509.614
  • CP 93129 dihydrochloride

    CAS:
    <p>5-HT1B agonist, potent and highly selective</p>
    Fórmula:C12H14ClN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:251.71
  • Cyclazosin HCl

    CAS:
    <p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>
    Fórmula:C23H28ClN5O4
    Pureza:99.10%
    Cor e Forma:Solid
    Peso molecular:473.95
  • 6-Chloromelatonin

    CAS:
    <p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>
    Fórmula:C13H15ClN2O2
    Pureza:98.01% - 99.25%
    Cor e Forma:Solid
    Peso molecular:266.72
  • Prucalopride hydrochloride

    CAS:
    <p>Prucalopride hydrochloride is a selective agonist of the 5-HT4.</p>
    Fórmula:C18H27Cl2N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:404.33
  • Alaproclate

    CAS:
    <p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>
    Fórmula:C13H18ClNO2
    Pureza:98.29% - 98.64%
    Cor e Forma:Solid
    Peso molecular:255.74
  • FR 64822

    CAS:
    <p>FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.</p>
    Fórmula:C11H14N4O
    Cor e Forma:Solid
    Peso molecular:218.26
  • TC-2153

    CAS:
    <p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>
    Fórmula:C7H5ClF3NS5
    Cor e Forma:Solid
    Peso molecular:355.89
  • Panamesine

    CAS:
    <p>Panamesine (EMD 57445) is a high affinity receptor ligand for sigma (IC50: 6 nM) with potential for atypical antipsychotic studies.</p>
    Fórmula:C23H26N2O6
    Cor e Forma:Solid
    Peso molecular:426.46
  • CB1/2 agonist 2

    CAS:
    <p>CB1/2 agonist 2 binds tightly to cannabinoid receptors, acting fully on CB1 and inversely on CB2.</p>
    Fórmula:C26H43NO3
    Cor e Forma:Solid
    Peso molecular:417.62
  • Dapiprazole

    CAS:
    <p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>
    Fórmula:C19H27N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:325.45
  • A-65186

    CAS:
    <p>A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.</p>
    Fórmula:C25H35N3O4
    Pureza:98.85% - 99.94%
    Cor e Forma:Solid
    Peso molecular:441.56
  • SKF83959

    CAS:
    <p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>
    Fórmula:C18H20ClNO2
    Pureza:98.68%
    Cor e Forma:Solid
    Peso molecular:317.81
  • Isothipendyl

    CAS:
    Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.
    Fórmula:C16H19N3S
    Cor e Forma:Solid
    Peso molecular:285.41
  • S-15535

    CAS:
    <p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>
    Fórmula:C21H24N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:336.43
  • ER819762

    CAS:
    <p>ER819762, an antagonist of the prostaglandin E2 EP4 receptor, inhibits Th1 differentiation and Th17 expansion.</p>
    Fórmula:C30H39N3O3
    Cor e Forma:Solid
    Peso molecular:489.65
  • OSU 6162 hydrochloride

    CAS:
    Dopamine stabilizer
    Fórmula:C15H24ClNO2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:317.88
  • SCH-202676 HBr

    CAS:
    <p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>
    Fórmula:C15H13N3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.35
  • JNJ-40255293

    CAS:
    <p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>
    Fórmula:C23H22N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:402.45
  • 5-HT6/5-HT2A receptor ligand-2

    CAS:
    <p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>
    Fórmula:C20H18FN3O2
    Cor e Forma:Solid
    Peso molecular:351.37
  • Hedgehog IN-3

    CAS:
    <p>Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].</p>
    Fórmula:C18H13ClF3N5O
    Cor e Forma:Solid
    Peso molecular:407.78
  • RS 23597-190 hydrochloride

    CAS:
    <p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>
    Fórmula:C16H24Cl2N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:363.28
  • NSC12404

    CAS:
    <p>NSC-12404 is a selective non-lipid LPA2/3 agonist.</p>
    Fórmula:C21H13NO4
    Cor e Forma:Solid
    Peso molecular:343.33
  • VUF-10497

    CAS:
    <p>VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).</p>
    Fórmula:C18H20ClN5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.9
  • (R)-V-0219


    <p>(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.</p>
    Fórmula:C20H25F3N4O2
    Cor e Forma:Solid
    Peso molecular:410.43
  • SC-41930

    CAS:
    <p>SC-41930 is a potent and selective antagonist of leukotriene B4 receptor.</p>
    Fórmula:C28H36O7
    Cor e Forma:Solid
    Peso molecular:484.58
  • MJ 15

    CAS:
    <p>MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.</p>
    Fórmula:C23H17Cl3N4O
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:471.77
  • OPC-14523 hydrochloride

    CAS:
    <p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>
    Fórmula:C23H29Cl2N3O2
    Pureza:99.60%
    Cor e Forma:Solid
    Peso molecular:450.4
  • ADRA1D receptor antagonist 1 HCl

    CAS:
    <p>ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.</p>
    Fórmula:C15H14Cl2N4O
    Pureza:98.13%
    Cor e Forma:Solid
    Peso molecular:337.2
  • Hedgehog Antagonist VIII

    CAS:
    <p>Hh antagonist VIII is a quinazolinyl-urea that inhibits Gli transcription in the Hh pathway, linked to cancer, with an IC50 of 70 nM.</p>
    Fórmula:C23H15ClF4N4O2
    Cor e Forma:Solid
    Peso molecular:490.84
  • RS 79948 hydrochloride

    CAS:
    <p>α2-adrenoreceptor antagonist</p>
    Fórmula:C19H29ClN2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:400.96
  • Romifidine

    CAS:
    Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.
    Fórmula:C9H9BrFN3
    Cor e Forma:Solid
    Peso molecular:258.09
  • (Iso)-FK-480

    CAS:
    (Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.
    Fórmula:C26H19FN4O2
    Pureza:98.36% - 99.41%
    Cor e Forma:Solid
    Peso molecular:438.45
  • L-749372

    CAS:
    L-749372 is the beta 3 adrenergic receptor 3-Pyridyloxypropanolamine agonist.
    Fórmula:C22H24IN3O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:553.41
  • SB-221284

    CAS:
    5-HT2C/2B receptor antagonist
    Fórmula:C16H14F3N3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:353.36
  • BAY-27-9955

    CAS:
    <p>BAY-27-9955 is a glucagon receptor antagonist.</p>
    Fórmula:C23H31FO
    Cor e Forma:Solid
    Peso molecular:342.49
  • mPGES-1 Inhibitor-1

    CAS:
    <p>mPGES-1 Inhibitor-1 is an mPGES-1 inhibitor with anti-inflammatory and analgesic activity, which can be used to study acute liver injury.</p>
    Fórmula:C16H19ClN4O2
    Pureza:96.84% - 98.75%
    Cor e Forma:Solid
    Peso molecular:334.8
  • 2-Acetylbenzoic acid

    CAS:
    <p>2-Acetylbenzoic acid outperforms 2-propionyloxybenzoic in hindering platelet function and PG synthesis; both similar in blocking PGI2 creation.</p>
    Fórmula:C9H8O3
    Pureza:99.62%
    Cor e Forma:Off-White Solid
    Peso molecular:164.16
  • 5-HT4 antagonist 1

    CAS:
    <p>5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).</p>
    Fórmula:C23H36N4O5S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:480.62
  • Mabuterol, (S)-

    CAS:
    Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.
    Fórmula:C13H18ClF3N2O
    Cor e Forma:Solid
    Peso molecular:310.74
  • VL-0395

    CAS:
    VL-0395 is an antagonist of CCK1 receptor.
    Fórmula:C25H21N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:427.45
  • Bamirastine

    CAS:
    <p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>
    Fórmula:C31H37N5O3
    Pureza:96.68%
    Cor e Forma:Solid
    Peso molecular:527.66
  • Cicloprolol hydrochloride

    CAS:
    <p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>
    Fórmula:C18H30ClNO4
    Pureza:97.26%
    Cor e Forma:Solid
    Peso molecular:359.89
  • NVP-QAV-680

    CAS:
    <p>NVP-QAV-680: Powerful, selective CRTh2 antagonist with nM potency inhibiting eosinophil/Th2 activation.</p>
    Fórmula:C18H18N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.41
  • Levoprotiline hydrochloride

    CAS:
    <p>Levoprotiline hydrochloride is an antidepressant.</p>
    Fórmula:C20H24ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.86
  • Butaclamol free base

    CAS:
    <p>Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.</p>
    Fórmula:C25H31NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:361.52
  • Argiprestocin

    CAS:
    Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.
    Fórmula:C43H67N15O12S2
    Pureza:99.34%
    Cor e Forma:Solid
    Peso molecular:1050.22
  • Quininib

    CAS:
    <p>Quininib inhibits ocular angiogenesis, blocks HMEC-1 tubules, aortic sprouts, and retinal revascularization in OIR mice.</p>
    Fórmula:C17H13NO
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:247.29
  • (+/-)-PPCC oxalate

    CAS:
    <p>Sigma receptor ligand with high sigma-1 affinity; binds sigma-2 as well (Ki = 1.5 &amp; 50.8 nM). Selective over dopaminergic, muscarinic receptors, DAT, SERT.</p>
    Fórmula:C50H60N2O10
    Cor e Forma:Solid
    Peso molecular:849.034
  • Sipagladenant

    CAS:
    <p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>
    Fórmula:C20H19N3O4S
    Cor e Forma:Solid
    Peso molecular:397.45
  • AZ-GHS-22

    CAS:
    <p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>
    Fórmula:C27H33ClN6O5S2
    Cor e Forma:Solid
    Peso molecular:621.17
  • MLN3126

    CAS:
    <p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>
    Fórmula:C21H19ClN2O5S
    Cor e Forma:Solid
    Peso molecular:446.9
  • KSCM-1

    CAS:
    <p>KSCM-1 is a selective sigma-1 receptor ligand.</p>
    Fórmula:C26H32N2O4
    Cor e Forma:Solid
    Peso molecular:436.54
  • GR-55562 dihydrobromide

    CAS:
    <p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>
    Fórmula:C23H26ClN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:411.93
  • Quinelorane dihydrochloride

    CAS:
    <p>Dopamine D2 and D3 receptor agonist</p>
    Fórmula:C14H23ClN4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:282.81
  • (Rac)-SEP-363856

    CAS:
    <p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>
    Fórmula:C9H13NOS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:183.27
  • Ro 19-1400

    CAS:
    <p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>
    Fórmula:C31H56N2O8S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:616.85
  • L-902688

    CAS:
    <p>L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).</p>
    Fórmula:C21H27F2N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:419.47
  • ALK4290

    CAS:
    <p>ALK4290 (AKST4290), a potent oral CCR3 inhibitor with a Ki of 3.2 nM, may treat macular degeneration and Parkinsonism.</p>
    Fórmula:C27H34ClN5O3
    Cor e Forma:Solid
    Peso molecular:512.04
  • SV-156

    CAS:
    <p>SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).</p>
    Fórmula:C21H23BrN2O2
    Cor e Forma:Solid
    Peso molecular:415.32
  • RPT193

    CAS:
    RPT193 is an oral CCR4 inhibitor reducing Th2 cell migration in atopic dermatitis, asthma, and allergies.
    Fórmula:C27H34Cl3N5O2
    Cor e Forma:Solid
    Peso molecular:566.95
  • SSTR4 agonist 2

    CAS:
    <p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>
    Fórmula:C18H24N4O
    Cor e Forma:Solid
    Peso molecular:312.41
  • GCGR antagonist 2

    CAS:
    <p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>
    Fórmula:C28H26N4O2
    Cor e Forma:Solid
    Peso molecular:450.53
  • Ko-3290

    CAS:
    <p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>
    Fórmula:C19H25N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.42
  • SC 51089 free base

    CAS:
    <p>SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.</p>
    Fórmula:C22H19ClN4O3
    Cor e Forma:Solid
    Peso molecular:422.86
  • Metrenperone

    CAS:
    <p>Metrenperone is used as a S(2)-receptor blocker.</p>
    Fórmula:C24H26FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:407.48
  • O-2093

    CAS:
    <p>anandamide uptake inhibitor</p>
    Fórmula:C34H43Cl2NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:584.62
  • Usmarapride

    CAS:
    <p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>
    Fórmula:C23H31N5O6
    Cor e Forma:Solid
    Peso molecular:473.53
  • TH-162

    CAS:
    <p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>
    Fórmula:C19H23N5O4
    Cor e Forma:Solid
    Peso molecular:385.42
  • Idremcinal

    CAS:
    <p>Idremcinal is a motilin receptor agonist.</p>
    Fórmula:C39H69NO12
    Cor e Forma:Solid
    Peso molecular:743.96
  • CCG-273463

    CAS:
    <p>CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.</p>
    Fórmula:C26H25BrN4O3
    Cor e Forma:Solid
    Peso molecular:521.41
  • ASP7657

    CAS:
    <p>ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.</p>
    Fórmula:C28H26F3N3O3
    Cor e Forma:Solid
    Peso molecular:509.52
  • RTI 336

    CAS:
    <p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>
    Fórmula:C24H26Cl2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:429.38
  • L-826266

    CAS:
    <p>L-826266 is an antagonist of EP(1) receptor.</p>
    Fórmula:C27H21BrClNO4S
    Cor e Forma:Solid
    Peso molecular:570.88
  • LY314228

    CAS:
    <p>LY314228 is an antagonist of 5-HT2A receptor.</p>
    Fórmula:C20H24N4O3
    Cor e Forma:Solid
    Peso molecular:368.43
  • CP-195543

    CAS:
    <p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>
    Fórmula:C24H19F3O4
    Cor e Forma:Solid
    Peso molecular:428.4
  • SKF-75670 Hydrobromide

    CAS:
    <p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>
    Fórmula:C17H20BrNO2
    Cor e Forma:Solid
    Peso molecular:350.25
  • Zicronapine

    CAS:
    <p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>
    Fórmula:C22H27ClN2
    Cor e Forma:Solid
    Peso molecular:354.92
  • NAEPA

    CAS:
    <p>NAEPA, an LPA mimetic, is a selective agonist of the lysophosphatidic acid-1 (LPA1) receptor.</p>
    Fórmula:C20H40NO5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:405.51
  • EP2 receptor antagonist-1

    CAS:
    <p>EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.</p>
    Fórmula:C24H22N4O5
    Cor e Forma:Solid
    Peso molecular:446.46
  • S-777469

    CAS:
    <p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>
    Fórmula:C23H27FN2O4
    Cor e Forma:Solid
    Peso molecular:414.47
  • CB2 receptor agonist 3

    CAS:
    <p>GP 2A is a selective agonist of CB2 receptor.</p>
    Fórmula:C24H23Cl2N3O
    Cor e Forma:Solid
    Peso molecular:440.36
  • DuP 734

    CAS:
    <p>DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].</p>
    Fórmula:C17H23BrFNO
    Cor e Forma:Solid
    Peso molecular:356.279
  • GPR183 antagonist-2

    CAS:
    <p>GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].</p>
    Fórmula:C20H18F2N4O5
    Cor e Forma:Solid
    Peso molecular:432.38
  • CJ 033466

    CAS:
    <p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>
    Fórmula:C19H28ClN5O
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:377.91
  • Nedocromil

    CAS:
    <p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>
    Fórmula:C19H17NO7
    Pureza:95% - 97.34%
    Cor e Forma:Solid
    Peso molecular:371.34
  • H3R-IN-1 Hydrochloride

    CAS:
    <p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>
    Fórmula:C19H24ClN3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:377.86
  • 5-Carboxamidotryptamine maleate

    CAS:
    <p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>
    Fórmula:C15H17N3O5
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:319.31
  • Mirisetron

    CAS:
    <p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>
    Fórmula:C24H31N3O2
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:393.52
  • Iprindole

    CAS:
    <p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>
    Fórmula:C19H28N2
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:284.44
  • LPA2 antagonist 2

    CAS:
    LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.
    Fórmula:C20H16N2O6
    Pureza:96.13%
    Cor e Forma:Solid
    Peso molecular:380.35
  • SDZ 205-557 hydrochloride

    CAS:
    <p>5-HT3/5-HT4 receptor antagonist</p>
    Fórmula:C14H22Cl2N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:337.24
  • RS 15385-197

    CAS:
    <p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>
    Fórmula:C18H26N2O3S
    Cor e Forma:Solid
    Peso molecular:350.48
  • LBP-1

    CAS:
    <p>LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.</p>
    Fórmula:C23H29ClN6O3
    Cor e Forma:Solid
    Peso molecular:472.97
  • Seproxetine HCl

    CAS:
    <p>Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.</p>
    Fórmula:C16H17ClF3NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.76
  • Amitifadine free base

    CAS:
    <p>Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.</p>
    Fórmula:C11H11Cl2N
    Cor e Forma:Solid
    Peso molecular:228.12
  • BE 2254

    CAS:
    <p>BE 2254 is an antagonist of central noradrenergic receptor.</p>
    Fórmula:C19H21NO2
    Cor e Forma:Solid
    Peso molecular:295.38
  • LUF5831

    CAS:
    <p>LUF5831 is an agonist of adenosine A1 receptor.</p>
    Fórmula:C15H12N4O2S
    Cor e Forma:Solid
    Peso molecular:312.35
  • Opiranserin

    CAS:
    <p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>
    Fórmula:C21H34N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:394.51
  • Ro 04-6790 dihydrochloride

    CAS:
    <p>Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.</p>
    Fórmula:C12H18Cl2N6O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:381.28
  • HSR-609

    CAS:
    <p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>
    Fórmula:C21H21FN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:368.4
  • (E)-Alprenoxime

    CAS:
    (E)-Alprenoxime is the isomer of the Alprenoxime which is a site-activated ocular β-blocker.
    Fórmula:C15H22N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:262.35
  • Caprospinol

    CAS:
    Caprospinol inhibits β-Amyloid (Aβ) protein neurotoxicity.
    Fórmula:C33H52O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:512.76
  • Draflazine

    CAS:
    <p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>
    Fórmula:C30H33Cl2F2N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:604.52
  • Lergotrile mesylate

    CAS:
    Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.
    Fórmula:C18H22ClN3O3S
    Cor e Forma:Solid
    Peso molecular:395.9
  • RGH 1756

    CAS:
    <p>RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.</p>
    Fórmula:C26H30N4O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:462.61
  • S 12024-2

    CAS:
    <p>S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.</p>
    Fórmula:C16H26N2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.45
  • ML 10375

    CAS:
    <p>ML 10375 is an antagonist of 5-HT4 receptor.</p>
    Fórmula:C17H25ClN2O3
    Cor e Forma:Solid
    Peso molecular:340.85
  • L 659,877

    CAS:
    <p>L 659,877 is an antagonist of the Tachykinin and neurokinin-2 receptor.</p>
    Fórmula:C38H50N8O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:762.92
  • KSCM-11

    CAS:
    <p>KSCM-11 is a sigma receptor ligand.</p>
    Fórmula:C25H30N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:406.52
  • YM 114

    CAS:
    <p>YM 114 is an anatagonist of 5-HT(3) receptor.</p>
    Fórmula:C16H18ClN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:303.79
  • Mequitamium iodide

    CAS:
    <p>Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.</p>
    Fórmula:C21H25IN2S
    Cor e Forma:Solid
    Peso molecular:464.41
  • Virodhamine trifluoroacetate

    CAS:
    <p>Virodhamine trifluoroacetate: full GPR55 &amp; CB2 agonist, partial CB1 antagonist, cannabinoid receptor mixed antagonist.</p>
    Fórmula:C24H38F3NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:461.56
  • ADX-10061

    CAS:
    <p>ADX-10061 is a dopamine D1 receptor antagonist.</p>
    Fórmula:C19H20N2O4
    Cor e Forma:Solid
    Peso molecular:340.37
  • Mepixanox

    CAS:
    Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.
    Fórmula:C20H21NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:323.39
  • Diftalone

    CAS:
    <p>Diftalone is an anti-Inflammatory agent.</p>
    Fórmula:C16H12N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:264.28