
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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BN 50341
CAS:<p>BN 50341 is an inhibitor of antithrombotic platelet activating factor.</p>Fórmula:C32H41ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:553.13Dacopafant
CAS:<p>Dacopafant is an antagonist of platlet activationg factor receptor.</p>Fórmula:C12H11N3OSCor e Forma:SolidPeso molecular:245.3SNAP 5089
CAS:α1A-adrenoceptor antagonistFórmula:C36H40N4O5Pureza:98%Cor e Forma:SolidPeso molecular:608.73CUMI-101
CAS:<p>CUMI-101 is an agonist of 5-HT1A receptor.</p>Fórmula:C19H27N5O3Cor e Forma:SolidPeso molecular:373.45Dihydroalprenolol, (S)-
CAS:<p>Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.</p>Fórmula:C15H25NO2Pureza:98%Cor e Forma:SolidPeso molecular:251.362MeSAMP
CAS:<p>2MeSAMP is a P2Y(12) antagonist that works by inhibiting platelet activation through a P2Y(12)/G(i)-dependent mechanism.</p>Fórmula:C11H16N5NaO7PSPureza:98%Cor e Forma:SolidPeso molecular:416.3Gyki 32887
CAS:<p>Gyki 32887 is a dopamine agonist.</p>Fórmula:C23H28N6O6SPureza:98%Cor e Forma:SolidPeso molecular:516.57SMANT hydrochloride
CAS:SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.Fórmula:C16H24BrClN2OPureza:99.81%Cor e Forma:SolidPeso molecular:375.73Carcainium chloride
CAS:<p>Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.</p>Fórmula:C18H22ClN3O2Pureza:99.89%Cor e Forma:SolidPeso molecular:347.84PGlu-3-methyl-His-Pro-NH2 TFA
<p>PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding & TSH release.</p>Fórmula:C19H25F3N6O6Pureza:98%Cor e Forma:SolidPeso molecular:490.43RS 52367
CAS:<p>RS 52367 is a beta-adrenergic antagonist.</p>Fórmula:C18H34ClN3O3SCor e Forma:SolidPeso molecular:408Lergotrile
CAS:<p>Lergotrile is used as an enzyme Inhibitor (Prolactin).</p>Fórmula:C17H18ClN3Pureza:98%Cor e Forma:SolidPeso molecular:299.8FAUC-3019
CAS:<p>FAUC-3019 is a partial agonist of the dopamine D(4) receptor.</p>Fórmula:C22H24N2OCor e Forma:SolidPeso molecular:332.44Butidrine
CAS:<p>Butidrine has an Antiarrhythmic activities.</p>Fórmula:C16H25NOPureza:98%Cor e Forma:SolidPeso molecular:247.38WS 009B
CAS:WS 009B is an antagonist of the endothelin receptor.Fórmula:C24H25NO11SPureza:98%Cor e Forma:SolidPeso molecular:535.52SB 268262
CAS:<p>CGRP1 antagonist</p>Fórmula:C18H15N3O4S2Pureza:98%Cor e Forma:SolidPeso molecular:401.46Losmiprofen
CAS:<p>Losmiprofen is a nonsteroidal compound of antiinflammatory.</p>Fórmula:C17H15ClO4Pureza:98%Cor e Forma:SolidPeso molecular:318.75Cafaminol
CAS:<p>Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.</p>Fórmula:C11H17N5O3Cor e Forma:SolidPeso molecular:267.28DAT 582
CAS:<p>DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent</p>Fórmula:C22H28ClN5OPureza:98%Cor e Forma:SolidPeso molecular:413.95Daglutril
CAS:<p>Daglutril is a NEP/ECE inhibitor for treating hypertension, heart failure, and pulmonary issues, blocking big endothelin-1 conversion.</p>Fórmula:C31H38N2O6Cor e Forma:SolidPeso molecular:534.64JTH-601 free base
CAS:<p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>Fórmula:C24H35NO4Pureza:98%Cor e Forma:SolidPeso molecular:401.54Iodophenpropit dihydrobromide
CAS:<p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>Fórmula:C15H20BrIN4SPureza:98%Cor e Forma:SolidPeso molecular:495.22Asperlicin D
CAS:<p>Asperlicin D is a cholecystokinin antagonist agent.</p>Fórmula:C25H18N4O2Pureza:98%Cor e Forma:SolidPeso molecular:406.44LY 25648
CAS:<p>LY 25648 is an antagonist of leukotriene B4.</p>Fórmula:C19H27NO2SCor e Forma:SolidPeso molecular:333.49VK-II-86
CAS:VK-II-86 is a non-β-blocking carvedilol analog. It prevents ouabain-Induced cardiotoxicityFórmula:C25H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:420.5KLS-13019
CAS:<p>KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).</p>Fórmula:C22H29NO3Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:355.47GS 283
CAS:<p>GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.</p>Fórmula:C17H17NO3Cor e Forma:SolidPeso molecular:283.32Viprostol
CAS:Viprostol is an agent of prostaglandin antihypertensive.Fórmula:C23H36O5Pureza:98%Cor e Forma:SolidPeso molecular:392.53Garomefrine HCl
CAS:<p>Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.</p>Fórmula:C9H14ClFN2O3SPureza:98%Cor e Forma:SolidPeso molecular:284.73Chloracyzine
CAS:<p>Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.</p>Fórmula:C19H21ClN2OSCor e Forma:SolidPeso molecular:360.9Alclofenac sodium
CAS:<p>Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.</p>Fórmula:C11H11ClNaO3Pureza:98%Cor e Forma:SolidPeso molecular:249.65Tecalcet Hydrochloride
CAS:<p>Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.</p>Fórmula:C18H23Cl2NOPureza:99.97%Cor e Forma:SolidPeso molecular:340.29SARS-CoV-2-IN-57
CAS:<p>SARS-CoV-2-IN-57 (compound (+)-R-26) is a potent inhibitor of SARS-CoV-2 with an IC50 of 80 nM and demonstrates high affinity for the Sigma Receptor, exhibiting</p>Fórmula:C23H37N3OPureza:98%Cor e Forma:SolidPeso molecular:371.56AMX12006
CAS:<p>AMX12006, a potent and selective EP4 antagonist, exhibits cytotoxic and antitumor activity, demonstrating oral activity with an IC50 of 4.3 nM [1].</p>Fórmula:C26H22F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:481.47Quinpirole Hydrochloride
CAS:<p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>Fórmula:C13H22ClN3Pureza:98%Cor e Forma:SolidPeso molecular:255.79WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Fórmula:C14H18N2Pureza:98%Cor e Forma:SolidPeso molecular:214.31PF2562
CAS:<p>PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).</p>Fórmula:C19H17N5OPureza:98%Cor e Forma:SolidPeso molecular:331.37Chlorazanil
CAS:<p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>Fórmula:C9H8ClN5Pureza:98.89%Cor e Forma:SolidPeso molecular:221.65Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Cor e Forma:SolidPeso molecular:328.38NRA-0160
CAS:<p>NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)</p>Fórmula:C24H23F2N3OSPureza:98%Cor e Forma:SolidPeso molecular:439.52BW 245C
CAS:<p>BW 245C is a DP1 agonist with an inhibitory effect on the aggregation response of collagen and can be used to study diseases such as stroke.</p>Fórmula:C19H32N2O5Pureza:≥99%Cor e Forma:SolidPeso molecular:368.47OMDM-6
CAS:<p>OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.</p>Fórmula:C28H42N2O3Pureza:99.66%Cor e Forma:SolidPeso molecular:454.64Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Fórmula:C18H20N2Pureza:99.85%Cor e Forma:SolidPeso molecular:264.36I942
CAS:<p>I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to regulate inflammatory gene expression in human umbilical</p>Fórmula:C20H19NO4SPureza:99.75%Cor e Forma:SolidPeso molecular:369.43Medroxalol
CAS:<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Fórmula:C20H24N2O5Cor e Forma:SolidPeso molecular:372.42Wy 49051
CAS:<p>Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).</p>Fórmula:C28H33N5O3Pureza:99.89%Cor e Forma:SolidPeso molecular:487.59PF-03654746
CAS:<p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>Fórmula:C18H24F2N2OPureza:98.85% - 99.57%Cor e Forma:SolidPeso molecular:322.39ChemR23-IN-1
CAS:<p>ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.</p>Fórmula:C28H29N7O2Cor e Forma:SolidPeso molecular:495.58Edivoxetine
CAS:<p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>Fórmula:C18H26FNO4Cor e Forma:SolidPeso molecular:339.4PD 144418
CAS:<p>PD 144418 displays potential antipsychotic activity.</p>Fórmula:C18H22N2OPureza:98%Cor e Forma:SolidPeso molecular:282.38F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Fórmula:C25H29ClF2N4O5Pureza:98.86%Cor e Forma:SolidPeso molecular:538.97Rec 15/2615 dihydrochloride
CAS:Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.Fórmula:C26H35Cl2N5O5Pureza:97.04% - 99.76%Cor e Forma:SolidPeso molecular:568.49PGD2-IN-1
CAS:<p>PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.</p>Fórmula:C23H23Cl2N3O3Pureza:98.21%Cor e Forma:SolidPeso molecular:460.35INCB38579
CAS:<p>INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.</p>Fórmula:C25H34N6OCor e Forma:SolidPeso molecular:434.58Org-13011 fumarate
CAS:<p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>Fórmula:C22H29F3N4O5Pureza:98.92%Cor e Forma:SolidPeso molecular:486.48CGP 35949
CAS:<p>CGP 35949 is an LTD4 antagonist with phospholipase inhibitory activity.</p>Fórmula:C23H25ClN5NaO5Pureza:99.62%Cor e Forma:SolidPeso molecular:509.92Povafonidine
CAS:<p>Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.</p>Fórmula:C11H13N5Cor e Forma:SolidPeso molecular:215.25CB2 modulator 1
CAS:<p>CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.</p>Fórmula:C18H19F3N4O2Pureza:99.6%Cor e Forma:SolidPeso molecular:380.365-HT7 agonist 2
CAS:<p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>Fórmula:C23H29N3OCor e Forma:SolidPeso molecular:363.5Zenidolol
CAS:<p>Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.</p>Fórmula:C17H27NO2Cor e Forma:SolidPeso molecular:277.4(Rac)-HAMI 3379
CAS:<p>HAMI 3379: potent CysLT2 receptor blocker; protects against acute/subacute brain injury; reduces microglia inflammation.</p>Fórmula:C34H45NO8Pureza:98%Cor e Forma:SolidPeso molecular:595.72BRL 37344 sodium
CAS:<p>BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.</p>Fórmula:C19H22ClNNaO4Pureza:98%Cor e Forma:SolidPeso molecular:386.83A-943931
CAS:A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.Fórmula:C17H21N5Pureza:99.79%Cor e Forma:SolidPeso molecular:295.38AL-3138
CAS:<p>AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.</p>Fórmula:C20H33FO4Cor e Forma:SolidPeso molecular:356.47ICI 192605
CAS:<p>ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.</p>Fórmula:C22H23ClO5Cor e Forma:SolidPeso molecular:402.87(S)-(-)-Propranolol hydrochloride
CAS:<p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>Fórmula:C16H22ClNO2Pureza:99.02% - 99.91%Cor e Forma:SolidPeso molecular:295.8Befetupitant
CAS:<p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>Fórmula:C29H29F6N3O2Pureza:98.72%Cor e Forma:SolidPeso molecular:565.55PD-156707
CAS:<p>PD-156707 is a selective antagonist of endothelin A receptor.</p>Fórmula:C28H26NaO9Pureza:98%Cor e Forma:SolidPeso molecular:529.497Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Fórmula:C26H31FN2O4Pureza:98%Cor e Forma:SolidPeso molecular:454.53WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Fórmula:C17H20Cl2FN3O2SPureza:98.43%Cor e Forma:SolidPeso molecular:420.33GAT228
CAS:<p>GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].</p>Fórmula:C22H18N2O2Cor e Forma:SolidPeso molecular:342.39PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Fórmula:C14H12F3NOSPureza:98%Cor e Forma:SolidPeso molecular:299.31A-940894
CAS:<p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>Fórmula:C17H21N5Cor e Forma:SolidPeso molecular:295.385-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.41SKF-104557
CAS:<p>N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.</p>Fórmula:C13H18N2OCor e Forma:SolidPeso molecular:218.29CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Fórmula:C19H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:351.4Enciprazine
CAS:Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.Fórmula:C23H32N2O6Pureza:98.63%Cor e Forma:SolidPeso molecular:432.51CID1172084
CAS:CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Fórmula:C23H18FN5O2S2Cor e Forma:SolidPeso molecular:479.55PNU-177864 hydrochloride
CAS:<p>PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor.</p>Fórmula:C18H22ClF3N2O3SPureza:99.95%Cor e Forma:SolidPeso molecular:438.89PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Fórmula:C15H20Cl2N2OPureza:98.67%Cor e Forma:SolidPeso molecular:315.24Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Fórmula:C18H22BrNSPureza:99.65%Cor e Forma:SolidPeso molecular:364.34Licogliflozin
CAS:<p>Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).</p>Fórmula:C23H28O7Pureza:98%Cor e Forma:SolidPeso molecular:416.46CCG-2046
CAS:<p>CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.</p>Fórmula:C11H10N4Cor e Forma:SolidPeso molecular:198.22L-692429
CAS:L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can be used to study acromegaly and obesity.Fórmula:C29H31N7O2Pureza:98.64% - 99.90%Cor e Forma:SolidPeso molecular:509.614CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Fórmula:C12H14ClN3OPureza:98%Cor e Forma:SolidPeso molecular:251.71Cyclazosin HCl
CAS:<p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>Fórmula:C23H28ClN5O4Pureza:99.10%Cor e Forma:SolidPeso molecular:473.956-Chloromelatonin
CAS:<p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>Fórmula:C13H15ClN2O2Pureza:98.01% - 99.25%Cor e Forma:SolidPeso molecular:266.72Prucalopride hydrochloride
CAS:<p>Prucalopride hydrochloride is a selective agonist of the 5-HT4.</p>Fórmula:C18H27Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:404.33Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Cor e Forma:SolidPeso molecular:255.74FR 64822
CAS:<p>FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.</p>Fórmula:C11H14N4OCor e Forma:SolidPeso molecular:218.26TC-2153
CAS:<p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>Fórmula:C7H5ClF3NS5Cor e Forma:SolidPeso molecular:355.89Panamesine
CAS:<p>Panamesine (EMD 57445) is a high affinity receptor ligand for sigma (IC50: 6 nM) with potential for atypical antipsychotic studies.</p>Fórmula:C23H26N2O6Cor e Forma:SolidPeso molecular:426.46CB1/2 agonist 2
CAS:<p>CB1/2 agonist 2 binds tightly to cannabinoid receptors, acting fully on CB1 and inversely on CB2.</p>Fórmula:C26H43NO3Cor e Forma:SolidPeso molecular:417.62Dapiprazole
CAS:<p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>Fórmula:C19H27N5Pureza:98%Cor e Forma:SolidPeso molecular:325.45A-65186
CAS:<p>A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.</p>Fórmula:C25H35N3O4Pureza:98.85% - 99.94%Cor e Forma:SolidPeso molecular:441.56SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Fórmula:C18H20ClNO2Pureza:98.68%Cor e Forma:SolidPeso molecular:317.81Isothipendyl
CAS:Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.Fórmula:C16H19N3SCor e Forma:SolidPeso molecular:285.41S-15535
CAS:<p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>Fórmula:C21H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:336.43ER819762
CAS:<p>ER819762, an antagonist of the prostaglandin E2 EP4 receptor, inhibits Th1 differentiation and Th17 expansion.</p>Fórmula:C30H39N3O3Cor e Forma:SolidPeso molecular:489.65OSU 6162 hydrochloride
CAS:Dopamine stabilizerFórmula:C15H24ClNO2SPureza:98%Cor e Forma:SolidPeso molecular:317.88SCH-202676 HBr
CAS:<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Fórmula:C15H13N3SPureza:98%Cor e Forma:SolidPeso molecular:267.35JNJ-40255293
CAS:<p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>Fórmula:C23H22N4O3Pureza:98%Cor e Forma:SolidPeso molecular:402.455-HT6/5-HT2A receptor ligand-2
CAS:<p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>Fórmula:C20H18FN3O2Cor e Forma:SolidPeso molecular:351.37Hedgehog IN-3
CAS:<p>Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].</p>Fórmula:C18H13ClF3N5OCor e Forma:SolidPeso molecular:407.78RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Fórmula:C16H24Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:363.28NSC12404
CAS:<p>NSC-12404 is a selective non-lipid LPA2/3 agonist.</p>Fórmula:C21H13NO4Cor e Forma:SolidPeso molecular:343.33VUF-10497
CAS:<p>VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).</p>Fórmula:C18H20ClN5SPureza:98%Cor e Forma:SolidPeso molecular:373.9(R)-V-0219
<p>(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.</p>Fórmula:C20H25F3N4O2Cor e Forma:SolidPeso molecular:410.43SC-41930
CAS:<p>SC-41930 is a potent and selective antagonist of leukotriene B4 receptor.</p>Fórmula:C28H36O7Cor e Forma:SolidPeso molecular:484.58MJ 15
CAS:<p>MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.</p>Fórmula:C23H17Cl3N4OPureza:99.63%Cor e Forma:SolidPeso molecular:471.77OPC-14523 hydrochloride
CAS:<p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>Fórmula:C23H29Cl2N3O2Pureza:99.60%Cor e Forma:SolidPeso molecular:450.4ADRA1D receptor antagonist 1 HCl
CAS:<p>ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.</p>Fórmula:C15H14Cl2N4OPureza:98.13%Cor e Forma:SolidPeso molecular:337.2Hedgehog Antagonist VIII
CAS:<p>Hh antagonist VIII is a quinazolinyl-urea that inhibits Gli transcription in the Hh pathway, linked to cancer, with an IC50 of 70 nM.</p>Fórmula:C23H15ClF4N4O2Cor e Forma:SolidPeso molecular:490.84RS 79948 hydrochloride
CAS:<p>α2-adrenoreceptor antagonist</p>Fórmula:C19H29ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:400.96Romifidine
CAS:Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Fórmula:C9H9BrFN3Cor e Forma:SolidPeso molecular:258.09(Iso)-FK-480
CAS:(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.Fórmula:C26H19FN4O2Pureza:98.36% - 99.41%Cor e Forma:SolidPeso molecular:438.45L-749372
CAS:L-749372 is the beta 3 adrenergic receptor 3-Pyridyloxypropanolamine agonist.Fórmula:C22H24IN3O4SPureza:98%Cor e Forma:SolidPeso molecular:553.41SB-221284
CAS:5-HT2C/2B receptor antagonistFórmula:C16H14F3N3OSPureza:98%Cor e Forma:SolidPeso molecular:353.36BAY-27-9955
CAS:<p>BAY-27-9955 is a glucagon receptor antagonist.</p>Fórmula:C23H31FOCor e Forma:SolidPeso molecular:342.49mPGES-1 Inhibitor-1
CAS:<p>mPGES-1 Inhibitor-1 is an mPGES-1 inhibitor with anti-inflammatory and analgesic activity, which can be used to study acute liver injury.</p>Fórmula:C16H19ClN4O2Pureza:96.84% - 98.75%Cor e Forma:SolidPeso molecular:334.82-Acetylbenzoic acid
CAS:<p>2-Acetylbenzoic acid outperforms 2-propionyloxybenzoic in hindering platelet function and PG synthesis; both similar in blocking PGI2 creation.</p>Fórmula:C9H8O3Pureza:99.62%Cor e Forma:Off-White SolidPeso molecular:164.165-HT4 antagonist 1
CAS:<p>5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).</p>Fórmula:C23H36N4O5SPureza:99.75%Cor e Forma:SolidPeso molecular:480.62Mabuterol, (S)-
CAS:Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.Fórmula:C13H18ClF3N2OCor e Forma:SolidPeso molecular:310.74VL-0395
CAS:VL-0395 is an antagonist of CCK1 receptor.Fórmula:C25H21N3O4Pureza:98%Cor e Forma:SolidPeso molecular:427.45Bamirastine
CAS:<p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>Fórmula:C31H37N5O3Pureza:96.68%Cor e Forma:SolidPeso molecular:527.66Cicloprolol hydrochloride
CAS:<p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>Fórmula:C18H30ClNO4Pureza:97.26%Cor e Forma:SolidPeso molecular:359.89NVP-QAV-680
CAS:<p>NVP-QAV-680: Powerful, selective CRTh2 antagonist with nM potency inhibiting eosinophil/Th2 activation.</p>Fórmula:C18H18N2O4SPureza:98%Cor e Forma:SolidPeso molecular:358.41Levoprotiline hydrochloride
CAS:<p>Levoprotiline hydrochloride is an antidepressant.</p>Fórmula:C20H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:329.86Butaclamol free base
CAS:<p>Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.</p>Fórmula:C25H31NOPureza:98%Cor e Forma:SolidPeso molecular:361.52Argiprestocin
CAS:Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.Fórmula:C43H67N15O12S2Pureza:99.34%Cor e Forma:SolidPeso molecular:1050.22Quininib
CAS:<p>Quininib inhibits ocular angiogenesis, blocks HMEC-1 tubules, aortic sprouts, and retinal revascularization in OIR mice.</p>Fórmula:C17H13NOPureza:99.81%Cor e Forma:SolidPeso molecular:247.29(+/-)-PPCC oxalate
CAS:<p>Sigma receptor ligand with high sigma-1 affinity; binds sigma-2 as well (Ki = 1.5 & 50.8 nM). Selective over dopaminergic, muscarinic receptors, DAT, SERT.</p>Fórmula:C50H60N2O10Cor e Forma:SolidPeso molecular:849.034Sipagladenant
CAS:<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Fórmula:C20H19N3O4SCor e Forma:SolidPeso molecular:397.45AZ-GHS-22
CAS:<p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>Fórmula:C27H33ClN6O5S2Cor e Forma:SolidPeso molecular:621.17MLN3126
CAS:<p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>Fórmula:C21H19ClN2O5SCor e Forma:SolidPeso molecular:446.9KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Fórmula:C26H32N2O4Cor e Forma:SolidPeso molecular:436.54GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Cor e Forma:SolidPeso molecular:282.81(Rac)-SEP-363856
CAS:<p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>Fórmula:C9H13NOSPureza:98%Cor e Forma:SolidPeso molecular:183.27Ro 19-1400
CAS:<p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>Fórmula:C31H56N2O8SPureza:98%Cor e Forma:SolidPeso molecular:616.85L-902688
CAS:<p>L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).</p>Fórmula:C21H27F2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:419.47ALK4290
CAS:<p>ALK4290 (AKST4290), a potent oral CCR3 inhibitor with a Ki of 3.2 nM, may treat macular degeneration and Parkinsonism.</p>Fórmula:C27H34ClN5O3Cor e Forma:SolidPeso molecular:512.04SV-156
CAS:<p>SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).</p>Fórmula:C21H23BrN2O2Cor e Forma:SolidPeso molecular:415.32RPT193
CAS:RPT193 is an oral CCR4 inhibitor reducing Th2 cell migration in atopic dermatitis, asthma, and allergies.Fórmula:C27H34Cl3N5O2Cor e Forma:SolidPeso molecular:566.95SSTR4 agonist 2
CAS:<p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41GCGR antagonist 2
CAS:<p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>Fórmula:C28H26N4O2Cor e Forma:SolidPeso molecular:450.53Ko-3290
CAS:<p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>Fórmula:C19H25N3O3Pureza:98%Cor e Forma:SolidPeso molecular:343.42SC 51089 free base
CAS:<p>SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.</p>Fórmula:C22H19ClN4O3Cor e Forma:SolidPeso molecular:422.86Metrenperone
CAS:<p>Metrenperone is used as a S(2)-receptor blocker.</p>Fórmula:C24H26FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:407.48O-2093
CAS:<p>anandamide uptake inhibitor</p>Fórmula:C34H43Cl2NO3Pureza:98%Cor e Forma:SolidPeso molecular:584.62Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.53TH-162
CAS:<p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>Fórmula:C19H23N5O4Cor e Forma:SolidPeso molecular:385.42Idremcinal
CAS:<p>Idremcinal is a motilin receptor agonist.</p>Fórmula:C39H69NO12Cor e Forma:SolidPeso molecular:743.96CCG-273463
CAS:<p>CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.</p>Fórmula:C26H25BrN4O3Cor e Forma:SolidPeso molecular:521.41ASP7657
CAS:<p>ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.</p>Fórmula:C28H26F3N3O3Cor e Forma:SolidPeso molecular:509.52RTI 336
CAS:<p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>Fórmula:C24H26Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:429.38L-826266
CAS:<p>L-826266 is an antagonist of EP(1) receptor.</p>Fórmula:C27H21BrClNO4SCor e Forma:SolidPeso molecular:570.88LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Fórmula:C20H24N4O3Cor e Forma:SolidPeso molecular:368.43CP-195543
CAS:<p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>Fórmula:C24H19F3O4Cor e Forma:SolidPeso molecular:428.4SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Fórmula:C17H20BrNO2Cor e Forma:SolidPeso molecular:350.25Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Fórmula:C22H27ClN2Cor e Forma:SolidPeso molecular:354.92NAEPA
CAS:<p>NAEPA, an LPA mimetic, is a selective agonist of the lysophosphatidic acid-1 (LPA1) receptor.</p>Fórmula:C20H40NO5PPureza:98%Cor e Forma:SolidPeso molecular:405.51EP2 receptor antagonist-1
CAS:<p>EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.</p>Fórmula:C24H22N4O5Cor e Forma:SolidPeso molecular:446.46S-777469
CAS:<p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>Fórmula:C23H27FN2O4Cor e Forma:SolidPeso molecular:414.47CB2 receptor agonist 3
CAS:<p>GP 2A is a selective agonist of CB2 receptor.</p>Fórmula:C24H23Cl2N3OCor e Forma:SolidPeso molecular:440.36DuP 734
CAS:<p>DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].</p>Fórmula:C17H23BrFNOCor e Forma:SolidPeso molecular:356.279GPR183 antagonist-2
CAS:<p>GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].</p>Fórmula:C20H18F2N4O5Cor e Forma:SolidPeso molecular:432.38CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Fórmula:C19H28ClN5OPureza:99.72%Cor e Forma:SolidPeso molecular:377.91Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Fórmula:C19H17NO7Pureza:95% - 97.34%Cor e Forma:SolidPeso molecular:371.34H3R-IN-1 Hydrochloride
CAS:<p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>Fórmula:C19H24ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:377.865-Carboxamidotryptamine maleate
CAS:<p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>Fórmula:C15H17N3O5Pureza:99.88%Cor e Forma:SolidPeso molecular:319.31Mirisetron
CAS:<p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>Fórmula:C24H31N3O2Pureza:99.88%Cor e Forma:SolidPeso molecular:393.52Iprindole
CAS:<p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>Fórmula:C19H28N2Pureza:99.54%Cor e Forma:SolidPeso molecular:284.44LPA2 antagonist 2
CAS:LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.Fórmula:C20H16N2O6Pureza:96.13%Cor e Forma:SolidPeso molecular:380.35SDZ 205-557 hydrochloride
CAS:<p>5-HT3/5-HT4 receptor antagonist</p>Fórmula:C14H22Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:337.24RS 15385-197
CAS:<p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>Fórmula:C18H26N2O3SCor e Forma:SolidPeso molecular:350.48LBP-1
CAS:<p>LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.</p>Fórmula:C23H29ClN6O3Cor e Forma:SolidPeso molecular:472.97Seproxetine HCl
CAS:<p>Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.</p>Fórmula:C16H17ClF3NOPureza:98%Cor e Forma:SolidPeso molecular:331.76Amitifadine free base
CAS:<p>Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.</p>Fórmula:C11H11Cl2NCor e Forma:SolidPeso molecular:228.12BE 2254
CAS:<p>BE 2254 is an antagonist of central noradrenergic receptor.</p>Fórmula:C19H21NO2Cor e Forma:SolidPeso molecular:295.38LUF5831
CAS:<p>LUF5831 is an agonist of adenosine A1 receptor.</p>Fórmula:C15H12N4O2SCor e Forma:SolidPeso molecular:312.35Opiranserin
CAS:<p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>Fórmula:C21H34N2O5Pureza:98%Cor e Forma:SolidPeso molecular:394.51Ro 04-6790 dihydrochloride
CAS:<p>Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.</p>Fórmula:C12H18Cl2N6O2SPureza:98%Cor e Forma:SolidPeso molecular:381.28HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Fórmula:C21H21FN2O3Pureza:98%Cor e Forma:SolidPeso molecular:368.4(E)-Alprenoxime
CAS:(E)-Alprenoxime is the isomer of the Alprenoxime which is a site-activated ocular β-blocker.Fórmula:C15H22N2O2Pureza:98%Cor e Forma:SolidPeso molecular:262.35Caprospinol
CAS:Caprospinol inhibits β-Amyloid (Aβ) protein neurotoxicity.Fórmula:C33H52O4Pureza:98%Cor e Forma:SolidPeso molecular:512.76Draflazine
CAS:<p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>Fórmula:C30H33Cl2F2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:604.52Lergotrile mesylate
CAS:Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.Fórmula:C18H22ClN3O3SCor e Forma:SolidPeso molecular:395.9RGH 1756
CAS:<p>RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.</p>Fórmula:C26H30N4O2SPureza:98%Cor e Forma:SolidPeso molecular:462.61S 12024-2
CAS:<p>S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.</p>Fórmula:C16H26N2O5SPureza:98%Cor e Forma:SolidPeso molecular:358.45ML 10375
CAS:<p>ML 10375 is an antagonist of 5-HT4 receptor.</p>Fórmula:C17H25ClN2O3Cor e Forma:SolidPeso molecular:340.85L 659,877
CAS:<p>L 659,877 is an antagonist of the Tachykinin and neurokinin-2 receptor.</p>Fórmula:C38H50N8O7SPureza:98%Cor e Forma:SolidPeso molecular:762.92KSCM-11
CAS:<p>KSCM-11 is a sigma receptor ligand.</p>Fórmula:C25H30N2O3Pureza:98%Cor e Forma:SolidPeso molecular:406.52YM 114
CAS:<p>YM 114 is an anatagonist of 5-HT(3) receptor.</p>Fórmula:C16H18ClN3OPureza:98%Cor e Forma:SolidPeso molecular:303.79Mequitamium iodide
CAS:<p>Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.</p>Fórmula:C21H25IN2SCor e Forma:SolidPeso molecular:464.41Virodhamine trifluoroacetate
CAS:<p>Virodhamine trifluoroacetate: full GPR55 & CB2 agonist, partial CB1 antagonist, cannabinoid receptor mixed antagonist.</p>Fórmula:C24H38F3NO4Pureza:98%Cor e Forma:SolidPeso molecular:461.56ADX-10061
CAS:<p>ADX-10061 is a dopamine D1 receptor antagonist.</p>Fórmula:C19H20N2O4Cor e Forma:SolidPeso molecular:340.37Mepixanox
CAS:Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.Fórmula:C20H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:323.39Diftalone
CAS:<p>Diftalone is an anti-Inflammatory agent.</p>Fórmula:C16H12N2O2Pureza:98%Cor e Forma:SolidPeso molecular:264.28
