GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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PF-04628935
CAS:<p>PF-04628935: potent GHS-R1a antagonist/inverse agonist, IC50=4.6 nM, orally bioavailable, brain penetrant.</p>Fórmula:C24H26ClN7OSPureza:98%Cor e Forma:SolidPeso molecular:496.03Pitolisant oxalate
CAS:<p>Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Fórmula:C19H28ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:385.88WAY 161503 hydrochloride
CAS:<p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>Fórmula:C11H12Cl3N3OPureza:98%Cor e Forma:SolidPeso molecular:308.59SKF-83822
CAS:<p>SKF-83822 is an agonist of dopamine D1-like receptor.</p>Fórmula:C20H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:343.85Ro 19-1400
CAS:<p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>Fórmula:C31H56N2O8SPureza:98%Cor e Forma:SolidPeso molecular:616.85OUP-186
CAS:<p>OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.</p>Fórmula:C19H30ClN3SCor e Forma:SolidPeso molecular:367.98(Rac)-E1R
CAS:<p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>Fórmula:C13H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:232.28GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Fórmula:C21H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:387.9Abanoquil
CAS:Abanoquil is an antagonist of alpha-1 adrenoceptor.Fórmula:C22H25N3O4Cor e Forma:SolidPeso molecular:395.45Oxyfedrine
CAS:<p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>Fórmula:C19H23NO3Cor e Forma:SolidPeso molecular:313.39Tiamenidine
CAS:<p>Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.</p>Fórmula:C8H10ClN3SPureza:98%Cor e Forma:SolidPeso molecular:215.7AM6545
CAS:<p>AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.</p>Fórmula:C26H23Cl2N5O3SPureza:97.03%Cor e Forma:SolidPeso molecular:556.46Ipsapirone
CAS:<p>Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.</p>Fórmula:C19H23N5O3SPureza:99.51%Cor e Forma:SolidPeso molecular:401.48GRK5-IN-3
CAS:<p>GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5).GRK5-IN-3 significantly inhibits GRK5 (IC50: 0.22 μM) and GRK6 (IC50: 0.41 μM).</p>Fórmula:C23H21N7O3Cor e Forma:SolidPeso molecular:443.46JMV3002
CAS:<p>JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.</p>Fórmula:C35H34N6O3Cor e Forma:SolidPeso molecular:586.68IMTPPE
CAS:<p>IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.</p>Fórmula:C20H27N3O2SCor e Forma:SolidPeso molecular:373.51SSTR4 agonist 2
CAS:<p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Fórmula:C23H30N6O6Pureza:98%Cor e Forma:SolidPeso molecular:486.52Bag-1
CAS:<p>Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.</p>Fórmula:C22H27N3Cor e Forma:SolidPeso molecular:333.47LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Fórmula:C27H38ClN3OSPureza:98.06%Cor e Forma:SolidPeso molecular:488.13JNJ-17156516
CAS:<p>JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.</p>Fórmula:C26H22Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:481.37Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Fórmula:C23H21FN8OCor e Forma:SolidPeso molecular:444.46DMP 696
CAS:<p>DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.</p>Fórmula:C18H21Cl2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:410.3Rp-cAMPS sodium
CAS:<p>Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.</p>Fórmula:C10H11N5NaO5PSPureza:99.71%Cor e Forma:SolidPeso molecular:367.25GB-110
CAS:<p>GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.</p>Fórmula:C33H48N6O5Pureza:98%Cor e Forma:SolidPeso molecular:608.77GSK334429
CAS:<p>GSK334429 is an antagonist of histamine H3 receptor.</p>Fórmula:C20H29F3N4OCor e Forma:SolidPeso molecular:398.47Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Fórmula:C22H26ClNPureza:98%Cor e Forma:SolidPeso molecular:339.9Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Fórmula:C20H25BrN4OCor e Forma:SolidPeso molecular:417.34S-5751
CAS:<p>S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.</p>Fórmula:C25H31NO4SCor e Forma:SolidPeso molecular:441.58Imiloxan hydrochloride
CAS:<p>Imiloxan hydrochloride is an α2-adrenoceptor antagonist.</p>Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75Gastrazole disodium
CAS:<p>Gastrazole, a CCK2 receptor antagonist, is used potentially for the treatment of pancreatic cancer.</p>Fórmula:C34H34FN5Na2O7Cor e Forma:SolidPeso molecular:689.652Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Fórmula:C18H29NO2Pureza:98%Cor e Forma:SolidPeso molecular:291.43Orexin receptor antagonist 2
CAS:<p>Compound 30, potent orexin antagonist with pKis of 7.69/9.78, potential for insomnia research.</p>Fórmula:C25H31N5O2Cor e Forma:SolidPeso molecular:433.55Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Fórmula:C25H27N3O5SPureza:98%Cor e Forma:SolidPeso molecular:481.56A 68930 hydrochloride
CAS:<p>A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].</p>Fórmula:C16H18ClNO3Cor e Forma:Off-White SolidPeso molecular:307.77PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Fórmula:C17H21N3Pureza:98%Cor e Forma:SolidPeso molecular:267.37AK-IN-1
CAS:<p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>Fórmula:C22H21N3O4Cor e Forma:SolidPeso molecular:391.42BI-L 239
CAS:BI-L 239 is an inhibition of 5-lipoxygenase products that cause bronchoconstriction.Fórmula:C16H15FOCor e Forma:SolidPeso molecular:242.29Sequifenadine
CAS:<p>Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].</p>Fórmula:C22H27NOCor e Forma:SolidPeso molecular:321.46NPC 17731
CAS:<p>NPC 17731 is a bradykinin receptor antagonist.</p>Fórmula:C59H95N19O14Cor e Forma:SolidPeso molecular:1294.5MK761
CAS:<p>MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.</p>Fórmula:C13H19N3O2Cor e Forma:SolidPeso molecular:249.31LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.41PD 119819
CAS:PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.Fórmula:C21H25Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:438.35Guanoxabenz hydrochloride
CAS:<p>Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.</p>Fórmula:C8H9Cl3N4OCor e Forma:SolidPeso molecular:283.54Foscarbidopa
CAS:<p>Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.</p>Fórmula:C10H15N2O7PPureza:96.17% - 97.27%Cor e Forma:SolidPeso molecular:306.21Zinterol hydrochloride
CAS:<p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>Fórmula:C19H27ClN2O4SCor e Forma:SolidPeso molecular:414.952-ThioUTP tetrasodium salt
CAS:<p>2-ThioUTP tetrasodium salt is a P2Y2 agonist.</p>Fórmula:C9H15N2O14P3SPureza:98%Cor e Forma:SolidPeso molecular:500.21Alprenolol tartrate, (S)-
CAS:<p>Alprenolol tartrate, (S)- is an 5-HT1A antagonist.</p>Fórmula:C19H29NO8Pureza:98%Cor e Forma:SolidPeso molecular:399.44Sultopride
CAS:<p>Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.</p>Fórmula:C17H26N2O4SCor e Forma:SolidPeso molecular:354.46CCG-224406
CAS:<p>CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.</p>Fórmula:C29H27FN6O5Cor e Forma:SolidPeso molecular:558.565-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45(Rac)-WAY-161503
CAS:<p>(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.</p>Fórmula:C11H11Cl2N3OPureza:99.51%Cor e Forma:SolidPeso molecular:272.13A-940894
CAS:<p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>Fórmula:C17H21N5Cor e Forma:SolidPeso molecular:295.38Bufetolol
CAS:Bufetolol is an antagonist of beta-adrenoceptor.Fórmula:C18H29NO4Pureza:98%Cor e Forma:SolidPeso molecular:323.43Kadsurenone
CAS:<p>Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.</p>Fórmula:C21H24O5Cor e Forma:SolidPeso molecular:356.41GRK5-IN-4
CAS:<p>GRK5-IN-4: potent, selective covalent inhibitor of GRK5 (IC50=1.1 μM), 90x more specific than GRK2, useful for heart failure research.</p>Fórmula:C26H25N7O3Cor e Forma:SolidPeso molecular:483.52MRS2603
CAS:<p>MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.</p>Fórmula:C14H12ClN4O8PPureza:98%Cor e Forma:SolidPeso molecular:430.69CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Fórmula:C18H20N6Cor e Forma:SolidPeso molecular:320.39Hexoprenaline
CAS:<p>Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.</p>Fórmula:C22H32N2O6Cor e Forma:SolidPeso molecular:420.5KW-8232
CAS:<p>KW-8232, an orally active anti-osteoporotic agent, reduces the biosynthesis of PGE2[1].</p>Fórmula:C37H41ClN4O6SCor e Forma:SolidPeso molecular:705.27Mosapramine
CAS:<p>Mosapramine is a dopamine D2-receptor antagonist.</p>Fórmula:C28H35ClN4OPureza:98%Cor e Forma:SolidPeso molecular:479.06SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Cor e Forma:SolidPeso molecular:376.29(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Fórmula:C16H26BrNOPureza:98%Cor e Forma:SolidPeso molecular:328.29SNT-207858 free base
CAS:<p>SNT-207858: selective MC-4 receptor antagonist, passes blood-brain barrier, orally active, IC50: 22 nM (binding), 11 nM (function).</p>Fórmula:C32H43Cl2N5O3Pureza:98%Cor e Forma:SolidPeso molecular:616.62VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Fórmula:C21H15N3OCor e Forma:SolidPeso molecular:325.36AZD-1678
CAS:<p>AZD-1678 is a potent CCR4 receptor antagonist.</p>Fórmula:C11H8Cl2FN3O3SCor e Forma:SolidPeso molecular:352.17CP 96345
CAS:<p>CP 96345 is a NK1 receptor antagonist.</p>Fórmula:C28H32N2OPureza:98%Cor e Forma:SolidPeso molecular:412.573-epi-Vitamin D3
CAS:<p>3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM in</p>Fórmula:C27H44OCor e Forma:SolidPeso molecular:384.64Fenmetozole Tosylate
CAS:<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Fórmula:C17H18Cl2N2O4SPureza:98%Cor e Forma:SolidPeso molecular:417.31S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Fórmula:C22H29Cl2N3O2SCor e Forma:SolidPeso molecular:470.45GSK-345931A
CAS:<p>GSK-345931A is an EP(1) antagonist with CNS uptake in mice/rats, offering strong pain relief in acute and prolonged inflammation.</p>Fórmula:C22H20ClNNaO3Cor e Forma:SolidPeso molecular:404.85Agroclavine
CAS:<p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>Fórmula:C16H18N2Cor e Forma:SolidPeso molecular:238.33RUSKI-201
CAS:<p>RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.</p>Fórmula:C20H27N3OSCor e Forma:SolidPeso molecular:357.51BMS-665053
CAS:<p>BMS-665053: CRF1 receptor antagonist, IC50 = 1.0 nM; inhibits cAMP in Y-79 cells, IC50 = 4.9 nM; anti-anxiety in rats, Cl = 17 mL/min/kg, t½ = 7.8 h.</p>Fórmula:C16H14Cl3F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:424.66Levobunolol
CAS:<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Fórmula:C17H25NO3Cor e Forma:White To Pink PowderPeso molecular:291.39MRS2179
CAS:<p>MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.</p>Fórmula:C11H17N5O9P2Cor e Forma:SolidPeso molecular:425.23CI 1020
CAS:<p>endothelin-A receptor (ETA) antagonist</p>Fórmula:C28H26O9Pureza:98%Cor e Forma:SolidPeso molecular:506.5MRS2768 tetrasodium salt
CAS:<p>MRS2768 tetrasodium: a P2Y2 agonist; offers cardioprotection against ischemia.</p>Fórmula:C15H16N2Na4O18P4Cor e Forma:SolidPeso molecular:728.14Idremcinal
CAS:<p>Idremcinal is a motilin receptor agonist.</p>Fórmula:C39H69NO12Cor e Forma:SolidPeso molecular:743.96CCG-273463
CAS:<p>CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.</p>Fórmula:C26H25BrN4O3Cor e Forma:SolidPeso molecular:521.41B-HT 933 dihydrochloride
CAS:<p>Azepexole (B-HT 933) dihydrochloride is an α2-adrenoceptor agonist, pKi: 8.3/α2A, 7.6/α2B, 7.5/α2C; IC50: 78.72 nM for peristalsis inhibition.</p>Fórmula:C9H17Cl2N3OCor e Forma:SolidPeso molecular:254.16Broxaterol
CAS:<p>Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.</p>Fórmula:C9H15BrN2O2Pureza:98%Cor e Forma:SolidPeso molecular:263.13(E)-Guanabenz
CAS:<p>(E)-Guanabenz is an oral α2-adrenoceptor agonist, antihypertensive, GADD34 inhibitor, and has neuroprotective properties.</p>Fórmula:C8H8Cl2N4Cor e Forma:SolidPeso molecular:231.08CFM 1571 hydrochloride
CAS:<p>CFM 1571 hydrochloride stimulates sGC with EC50 of 5.49 μM; potential for cardiovascular research.</p>Fórmula:C23H29ClN4O3Cor e Forma:SolidPeso molecular:444.96JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Fórmula:C20H28N2OPureza:98%Cor e Forma:SolidPeso molecular:312.45Atigliflozin
CAS:<p>Atigliflozin is an antihyperglycaemic drug candidate.</p>Fórmula:C18H22O7SCor e Forma:SolidPeso molecular:382.43Ro 363 hydrochloride
CAS:<p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>Fórmula:C19H26ClNO6Cor e Forma:SolidPeso molecular:399.87Substance P Receptor Antagonist 1
CAS:<p>Substance P Receptor Antagonist 1 may aid in treating GI, inflammatory, respiratory, and CNS disorders.</p>Fórmula:C24H29F3N2O2Pureza:98%Cor e Forma:SolidPeso molecular:434.49FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Fórmula:C27H29F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:465.53Pargolol hydrochloride
CAS:<p>Pargolol hydrochloride is an antagonist of β adrenergic receptor.</p>Fórmula:C16H24ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:313.82Octoclothepin maleate salt
CAS:<p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>Fórmula:C23H25ClN2O4SCor e Forma:SolidPeso molecular:460.97DW-1350
CAS:DW-1350 is an antagonist of LTB4 receptor.Fórmula:C25H31N3O3SPureza:98%Cor e Forma:SolidPeso molecular:453.6RTI 336
CAS:<p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>Fórmula:C24H26Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:429.38L-826266
CAS:<p>L-826266 is an antagonist of EP(1) receptor.</p>Fórmula:C27H21BrClNO4SCor e Forma:SolidPeso molecular:570.88LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Fórmula:C20H24N4O3Cor e Forma:SolidPeso molecular:368.43PQ-69
CAS:<p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>Fórmula:C20H19FN4OCor e Forma:SolidPeso molecular:350.39Autotaxin-IN-6
CAS:<p>Autotaxin-IN-6 is a strong ATX inhibitor with a 30 nM IC50, potentially aiding anticancer research by hindering cell migration.</p>Fórmula:C35H54BNO6Cor e Forma:SolidPeso molecular:595.62Izuforant
CAS:<p>Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).</p>Fórmula:C12H12BrN7Cor e Forma:SolidPeso molecular:334.17MK-8133
CAS:<p>MK-8133 is an antagonist of orexin-2 selective receptor with favorable development properties.</p>Fórmula:C23H21N5O2Cor e Forma:SolidPeso molecular:399.45Fluprostenol methyl ester
CAS:<p>Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.</p>Fórmula:C24H31F3O6Cor e Forma:SolidPeso molecular:472.49SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Fórmula:C19H27IN2O4Cor e Forma:SolidPeso molecular:474.33QCC-374
CAS:<p>QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.</p>Fórmula:C28H33N3O2Pureza:98%Cor e Forma:SolidPeso molecular:443.58UK 1745
CAS:<p>UK 1745 is a novel drug of cardiotonic.</p>Fórmula:C16H23ClN2O2Cor e Forma:SolidPeso molecular:310.82CP-195543
CAS:<p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>Fórmula:C24H19F3O4Cor e Forma:SolidPeso molecular:428.4SM-130686
CAS:<p>SM-130,686: orally-active GHSR agonist, 50% as potent as ghrelin in stimulating growth hormone.</p>Fórmula:C22H24Cl2F3N3O3Cor e Forma:SolidPeso molecular:506.35ZK-90055 hydrochloride
CAS:ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.Fórmula:C16H23ClN2O4Pureza:99.26%Cor e Forma:SolidPeso molecular:342.82Guanethidine
CAS:<p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>Fórmula:C10H22N4Cor e Forma:SolidPeso molecular:198.31EP4 receptor antagonist 4
CAS:<p>EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].</p>Fórmula:C19H14N2OSCor e Forma:SolidPeso molecular:318.39SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Fórmula:C17H20BrNO2Cor e Forma:SolidPeso molecular:350.25Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Fórmula:C22H27ClN2Cor e Forma:SolidPeso molecular:354.92A 55453
CAS:<p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>Fórmula:C25H32N6O3Cor e Forma:SolidPeso molecular:464.565'-(N-Cyclopropyl)carboxamidoadenosine
CAS:<p>adenosine A2 receptor agonist</p>Fórmula:C13H16N6O4Pureza:98%Cor e Forma:SolidPeso molecular:320.3FRG8701
CAS:<p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>Fórmula:C22H30N2O4SPureza:98%Cor e Forma:SolidPeso molecular:418.55NAEPA
CAS:<p>NAEPA, an LPA mimetic, is a selective agonist of the lysophosphatidic acid-1 (LPA1) receptor.</p>Fórmula:C20H40NO5PPureza:98%Cor e Forma:SolidPeso molecular:405.51EP2 receptor antagonist-1
CAS:<p>EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.</p>Fórmula:C24H22N4O5Cor e Forma:SolidPeso molecular:446.46ROS 234
CAS:<p>ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.</p>Fórmula:C13H15N5Cor e Forma:SolidPeso molecular:241.29SDZ 21009
CAS:β-adrenoceptor and 5-HT1A/1B receptor antagonistFórmula:C19H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:348.44Adrenaline sulfate
CAS:<p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>Fórmula:C9H15NO7SCor e Forma:SolidPeso molecular:281.279PD-135666
CAS:<p>PD-135666 is an antagonist of CCK receptor.</p>Fórmula:C33H39N3O5Pureza:98%Cor e Forma:SolidPeso molecular:557.68PROTAC(H-PGDS)-7
CAS:<p>PROTAC(H-PGDS)-7, a potent H-PGDS degrader, inhibits PGD2 in KU812 cells; DC50 is 17.3 pM. Potential DMD treatment.</p>Fórmula:C40H38N8O7Cor e Forma:SolidPeso molecular:742.78Anatibant
CAS:<p>Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.</p>Fórmula:C34H36Cl2N6O5SPureza:98%Cor e Forma:SolidPeso molecular:711.66LUF 5834
CAS:A2A and A2B adenosine receptor partial agonistFórmula:C17H12N6OSPureza:98%Cor e Forma:SolidPeso molecular:348.38CB1R Allosteric modulator 1
CAS:<p>CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.</p>Fórmula:C24H24ClN3OCor e Forma:SolidPeso molecular:405.92SANT-2
CAS:<p>SANT-2 is a potent inhibitor of Shh signaling pathway.</p>Fórmula:C23H20ClN3O4Cor e Forma:SolidPeso molecular:437.88Nivasorexant
CAS:<p>Nivasorexant is a potent antagonist of the orexin receptor.</p>Fórmula:C23H23N7O2Cor e Forma:SolidPeso molecular:429.47SF 11
CAS:<p>SF 11 is a potent and brain penetrant neuropeptide Y Y2 receptor antagonist with IC50 of 199 nM. Antidepressant-like activity</p>Fórmula:C27H30N2O2SPureza:99.51%Cor e Forma:SolidPeso molecular:446.6INCB38579
CAS:<p>INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.</p>Fórmula:C25H34N6OCor e Forma:SolidPeso molecular:434.58LY 393558
CAS:<p>Dual 5-HT1B/1D receptor antagonist</p>Fórmula:C26H31FN4O4S2Pureza:98%Cor e Forma:SolidPeso molecular:546.68AGI-41998
CAS:<p>AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.</p>Fórmula:C22H16BrF3N4O2Cor e Forma:SolidPeso molecular:505.29Latanoprost ethyl amide
CAS:<p>Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.</p>Fórmula:C25H39NO4Cor e Forma:SolidPeso molecular:417.58Remogliflozin
CAS:<p>Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).</p>Fórmula:C23H34N2O7Cor e Forma:SolidPeso molecular:450.53Orexin receptor antagonist 3
CAS:<p>Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist.</p>Fórmula:C21H22N8O3Cor e Forma:SolidPeso molecular:434.45Palmitoyl serinol
CAS:<p>Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.</p>Fórmula:C19H39NO3Cor e Forma:SolidPeso molecular:329.52Repinotan HCl
CAS:<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Fórmula:C21H25ClN2O4SPureza:99.57%Cor e Forma:SolidPeso molecular:436.95Aligeron
CAS:<p>Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibit</p>Fórmula:C20H24N2Pureza:99.09% - >99.99%Cor e Forma:SolidPeso molecular:292.42SNT-207858
CAS:<p>SNT-207858: selective, BBB-penetrating, oral MC-4 receptor antagonist with 22 nM IC50 (binding), 11 nM (function).</p>Fórmula:C32H45Cl4N5O3Pureza:98%Cor e Forma:SolidPeso molecular:689.54AP-521 (Free base)
CAS:<p>AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.</p>Fórmula:C20H18N2O3SCor e Forma:SolidPeso molecular:366.43BRD5814
CAS:<p>BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.</p>Fórmula:C21H23ClF3NO2Cor e Forma:SolidPeso molecular:413.86Adriforant
CAS:<p>Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.</p>Fórmula:C13H22N6Pureza:99.84%Cor e Forma:SolidPeso molecular:262.35LY 306669
CAS:LY 306669 is an antagonist of leukotriene B4 receptor.Fórmula:C23H29FN4NaO2Cor e Forma:SolidPeso molecular:435.499Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Fórmula:C26H32N2O7Cor e Forma:SolidPeso molecular:484.549Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Cor e Forma:SolidPeso molecular:369.29GPR55 agonist 3
CAS:<p>Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.</p>Fórmula:C19H16F4N4Cor e Forma:SolidPeso molecular:376.35GPR183-IN-2
CAS:<p>GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.</p>Fórmula:C19H23BrN2O3Cor e Forma:SolidPeso molecular:407.3A2A/A1 AR antagonist-1
CAS:<p>A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).</p>Fórmula:C15H12N6O2Cor e Forma:SolidPeso molecular:308.29Epanolol
CAS:<p>Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.</p>Fórmula:C20H23N3O4Pureza:98%Cor e Forma:SolidPeso molecular:369.41Proglumide sodium
CAS:Non-selective cholecystokinin (CCK) antagonistFórmula:C18H26N2NaO4Pureza:98%Cor e Forma:SolidPeso molecular:357.4Fosnetupitant
CAS:Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.Fórmula:C31H35F6N4O5PPureza:98%Cor e Forma:SolidPeso molecular:688.6MAT2A-IN-2
CAS:<p>MAT2A-IN-2 is a potent inhibitor of MAT2A. MAT2A-IN-2 has potential for cancer disease research.</p>Fórmula:C23H17F3N6O2Cor e Forma:SolidPeso molecular:466.42Melatonin receptor agonist 1
CAS:<p>Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].</p>Fórmula:C15H19N3O2Cor e Forma:SolidPeso molecular:273.33Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Fórmula:C18H20ClNPureza:98%Cor e Forma:SolidPeso molecular:285.81LUF6000
CAS:LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).Fórmula:C22H20Cl2N4Cor e Forma:SolidPeso molecular:411.33WIN 62,577
CAS:<p>WIN 62,577 is a allosteric antagonist of mAChR.</p>Fórmula:C29H31N3OPureza:98%Cor e Forma:SolidPeso molecular:437.58GPR183 antagonist-2
CAS:<p>GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].</p>Fórmula:C20H18F2N4O5Cor e Forma:SolidPeso molecular:432.38YQA14
CAS:<p>YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.</p>Fórmula:C23H27ClN4O3Pureza:99.52%Cor e Forma:SolidPeso molecular:442.94AChE-IN-14
CAS:<p>AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.</p>Fórmula:C28H35NO3Cor e Forma:SolidPeso molecular:433.58SB357134
CAS:<p>SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.</p>Fórmula:C17H18Br2FN3O3SPureza:98%Cor e Forma:SolidPeso molecular:523.21MRS 1334
CAS:<p>antagonist for the human adenosine A3 receptor</p>Fórmula:C31H26N2O6Pureza:98%Cor e Forma:SolidPeso molecular:522.55PF-06256142
CAS:PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).Fórmula:C21H16N4O2Pureza:98%Cor e Forma:SolidPeso molecular:356.38AZD5213
CAS:<p>AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.</p>Fórmula:C19H25N3O2Cor e Forma:SolidPeso molecular:327.42(R,R)-Reboxetine mesylate
CAS:<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Fórmula:C20H27NO6SCor e Forma:SolidPeso molecular:409.5TCS-OX2-29 HCl
CAS:TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.Fórmula:C23H32ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:433.97A331440
CAS:<p>A331440 is an modulator of L-histidine and histamine H3 receptor.</p>Fórmula:C22H27N3OCor e Forma:SolidPeso molecular:349.47UP202-56
CAS:UP202-56 is an adenosinergic agonist and is an adenosine analog.Fórmula:C33H37N7O4Pureza:98%Cor e Forma:SolidPeso molecular:595.69Spirendolol
CAS:Spirendolol is an antagonist of β adrenergic receptor.Fórmula:C21H31NO3Pureza:98%Cor e Forma:SolidPeso molecular:345.48S(-)-Bisoprolol
CAS:<p>S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.</p>Fórmula:C18H31NO4Cor e Forma:SolidPeso molecular:325.44UCSF678
CAS:<p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>Fórmula:C15H18N2O2SCor e Forma:SolidPeso molecular:290.38Centanafadine
CAS:<p>Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).</p>Fórmula:C15H15NPureza:98%Cor e Forma:SolidPeso molecular:209.29PF-592379
CAS:PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).Fórmula:C13H21N3OPureza:98%Cor e Forma:SolidPeso molecular:235.33HEMADO
CAS:<p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>Fórmula:C17H23N5O4Pureza:98%Cor e Forma:SolidPeso molecular:361.4GR-203040 HCl
CAS:<p>GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.</p>Fórmula:C20H26Cl2N6OCor e Forma:SolidPeso molecular:437.37EGIS-7625
CAS:<p>EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.</p>Fórmula:C18H24Cl2N4O2Pureza:98%Cor e Forma:SolidPeso molecular:399.32Carbinoxamine
CAS:<p>Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.</p>Fórmula:C16H19ClN2OPureza:98%Cor e Forma:LiquidPeso molecular:290.79hA2A/hCA XII modulator 1
CAS:<p>Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>Fórmula:C24H19N7O4SCor e Forma:SolidPeso molecular:501.52DV 7028 hydrochloride
CAS:<p>DV 7028 hydrochloride is a 5-HT2A receptor antagonist.</p>Fórmula:C21H26ClFN4O3Pureza:98%Cor e Forma:SolidPeso molecular:436.91S20928
CAS:<p>S20928 is an antagonist of melatonin receptor.</p>Fórmula:C17H19NOCor e Forma:SolidPeso molecular:253.34Ibodutant
CAS:Ibodutant is an effective and selective tachykinin NK2 receptor antagonist (pKi: 10.1).Fórmula:C37H48N4O4SPureza:98%Cor e Forma:SolidPeso molecular:644.87Vicagrel
CAS:Vicagrel, an oral antiplatelet, boosts aspirin's effect, targeting P2Y12 and fights clots in heart and vessel diseases.Fórmula:C18H18ClNO4SPureza:98%Cor e Forma:SolidPeso molecular:379.86MRS1177
CAS:<p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>Fórmula:C20H12ClN5O2Pureza:98%Cor e Forma:SolidPeso molecular:389.79PA-9
CAS:<p>PA-9 is the first small-molecule PAC1 receptor antagonist.</p>Fórmula:C17H18N6O2Pureza:98%Cor e Forma:SolidPeso molecular:338.36Vasopressin V2 receptor antagonist 1
CAS:<p>Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).</p>Fórmula:C33H37ClN4O4Cor e Forma:SolidPeso molecular:589.12threo Ifenprodil hemitartrate
CAS:σ receptor agonist and NR2B subunit-selective NMDA receptor antagonistFórmula:C21H27NO2C4H6O6Pureza:98%Cor e Forma:SolidPeso molecular:400.49MG 1
CAS:<p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>Fórmula:C17H25N3O2Pureza:98.98% - >99.99%Cor e Forma:SolidPeso molecular:303.4I942
CAS:<p>I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to regulate inflammatory gene expression in human umbilical</p>Fórmula:C20H19NO4SPureza:99.75%Cor e Forma:SolidPeso molecular:369.43SM-2470
CAS:<p>SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.</p>Fórmula:C23H30ClN5O3Pureza:98.91%Cor e Forma:SolidPeso molecular:459.97TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75Iso-SLR 080811
CAS:<p>Iso-SLR 080811 is an isomer of SLR 080811, suitable for relevant research in the life sciences. SLR080811 is a selective SphK2 inhibitor (Ki=1.3 μM).</p>Fórmula:C21H32ClN5OPureza:98.34%Cor e Forma:SolidPeso molecular:405.97L-817,818
CAS:somatostatin sst5 receptor agonistFórmula:C33H36N4O3Pureza:98%Cor e Forma:SolidPeso molecular:536.66TSI-01
CAS:<p>TSI-01,Pro-inflammatory phospholipid mediator. Inhibits LPCAT2 (IC50=0.47 μM). Suppresses PAF biosynthesis in macrophages.</p>Fórmula:C14H11Cl2NO4Pureza:99.87%Cor e Forma:SolidPeso molecular:328.15CB1R Allosteric modulator 3
CAS:<p>CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.</p>Fórmula:C22H17ClN2O2Pureza:98.18%Cor e Forma:SolidPeso molecular:376.84RXFP3/4 agonist 2
CAS:RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.Fórmula:C22H22N6O2Pureza:99.82%Cor e Forma:SolidPeso molecular:402.455-HT7 agonist 1
CAS:<p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>Fórmula:C19H20ClN3Pureza:98.61%Cor e Forma:SolidPeso molecular:325.84PM226
CAS:<p>CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.</p>Fórmula:C22H31NO3Cor e Forma:SolidPeso molecular:357.49Alniditan
CAS:<p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>Fórmula:C17H26N4OPureza:98%Cor e Forma:SolidPeso molecular:302.41GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Cor e Forma:SolidPeso molecular:377.48GR 113808
CAS:<p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>Fórmula:C19H27N3O4SPureza:98.16%Cor e Forma:SolidPeso molecular:393.5Amgen-23
CAS:<p>Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.</p>Fórmula:C23H25Cl2N3O2SPureza:97.31%Cor e Forma:SolidPeso molecular:478.44Setastine HCl
CAS:<p>Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.</p>Fórmula:C22H29Cl2NOCor e Forma:SolidPeso molecular:394.38CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Fórmula:C24H23N3O4S2Pureza:98%Cor e Forma:SolidPeso molecular:481.59
