GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.946 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(408 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5360 produtos de "GPCR/Proteína-G"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
CCR4 antagonist 3-1
CAS:<p>CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.</p>Fórmula:C14H12N2SPureza:99.53%Cor e Forma:SolidPeso molecular:240.32Calhex 231 hydrochloride
CAS:<p>Calhex 231 hydrochloride a potent CaSR negative-conversion modulator that blocks the increase in [3H]inositol phosphate, inhibits mir-208a-mediated .</p>Fórmula:C25H28Cl2N2OPureza:99.36%Cor e Forma:SolidPeso molecular:443.41SMANT hydrochloride
CAS:<p>SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.</p>Fórmula:C16H24BrClN2OPureza:99.81%Cor e Forma:SolidPeso molecular:375.73Monatepil maleate
CAS:<p>Monatepil maleate (AJ-2615 maleate) is a Ca2+-channel and α1-adrenergic receptor antagonist, and ACAT inhibitor with antihypertensive activity.</p>Fórmula:C32H34FN3O5SPureza:97.90%Cor e Forma:SolidPeso molecular:591.69CCR1 antagonist 7
CAS:<p>CCR1 antagonist 7 (compound 16r) is an antagonist of chemokine receptor 1 (CCR1) with an IC 50 of 4 nM [1].</p>Fórmula:C21H24ClN5O3SPureza:98%Cor e Forma:SolidPeso molecular:461.96PNU-177864
CAS:<p>PNU-177864 is a selective dopamine D3 receptor antagonist.</p>Fórmula:C18H21F3N2O3SPureza:99.92%Cor e Forma:SolidPeso molecular:402.43S 14506 hydrochloride
CAS:<p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>Fórmula:C24H27ClFN3O2Pureza:99.92%Cor e Forma:SolidPeso molecular:443.94Iodophenpropit dihydrobromide
CAS:<p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>Fórmula:C15H20BrIN4SPureza:98%Cor e Forma:SolidPeso molecular:495.22PF-03654746 Tosylate
CAS:<p>PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.</p>Fórmula:C25H32F2N2O4SPureza:98%Cor e Forma:SolidPeso molecular:494.6SB-277011 dihydrochloride
CAS:<p>SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.</p>Fórmula:C28H32Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:511.49Taprenepag isopropyl
CAS:<p>Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.</p>Fórmula:C27H28N4O5SPureza:99.44%Cor e Forma:SolidPeso molecular:520.6Zatosetron maleate
CAS:<p>Zatosetron maleate（LY 277359 maleate） is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.</p>Fórmula:C23H29ClN2O6Pureza:98.07%Cor e Forma:SolidPeso molecular:464.94PPTN
CAS:<p>PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.</p>Fórmula:C29H24F3NO2Pureza:99.86%Cor e Forma:SolidPeso molecular:475.5KLS-13019
CAS:<p>KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).</p>Fórmula:C22H29NO3Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:355.47LRH-1 Inhibitor-3
CAS:<p>LRH-1 Inhibitor-3 is an antagonist that inhibits LRH-1 transcriptional activity, reducing SHP, cyclin E1 (CCNE1), and G0S2,antiproliferation anticancer.</p>Fórmula:C23H25N3O2Pureza:98%Cor e Forma:SolidPeso molecular:375.46GALNON
CAS:<p>Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties</p>Fórmula:C40H46N4O6Pureza:98%Cor e Forma:SolidPeso molecular:678.82L-365260
CAS:<p>L-365260 is a nonpeptide gastrin and cerebral cholecystokinin receptor (CCK-B) antagonist used in the study of neurologic ojibwa and endocrine diseases.</p>Fórmula:C24H22N4O2Pureza:99.75%Cor e Forma:SolidPeso molecular:398.46Lusaperidone
CAS:<p>Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against liver cell damage and fibrosis in rats.</p>Fórmula:C22H21N3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:359.42Tecalcet Hydrochloride
CAS:<p>Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.</p>Fórmula:C18H23Cl2NOPureza:99.97%Cor e Forma:SolidPeso molecular:340.29Lavoltidine
CAS:<p>Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.</p>Fórmula:C19H29N5O2Pureza:98.30% - 98.36%Cor e Forma:SolidPeso molecular:359.47SARS-CoV-2-IN-57
CAS:<p>SARS-CoV-2-IN-57 (compound (+)-R-26) is a potent inhibitor of SARS-CoV-2 with an IC50 of 80 nM and demonstrates high affinity for the Sigma Receptor, exhibiting</p>Fórmula:C23H37N3OPureza:98%Cor e Forma:SolidPeso molecular:371.56A2AR-antagonist-1
CAS:<p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>Fórmula:C27H25N5O2Pureza:98%Cor e Forma:SolidPeso molecular:451.52Moprolol
CAS:<p>Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].</p>Fórmula:C13H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:239.31ML230
CAS:<p>ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor.</p>Fórmula:C25H21N5O3Pureza:98%Cor e Forma:SolidPeso molecular:439.47A-77636
CAS:<p>A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50</p>Fórmula:C20H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:329.43D4R agonist-1
CAS:<p>D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.</p>Fórmula:C19H22N4SPureza:98.44%Cor e Forma:SolidPeso molecular:338.47SORT-PGRN interaction inhibitor 3
CAS:<p>SORT-PGRN Interaction Inhibitor 3 (Compound 13), with an IC50 value of 0.17 μM, acts as an inhibitor of the SORT-PGRN interaction, and is utilized in the study</p>Fórmula:C15H19Cl2NO3Pureza:98%Cor e Forma:SolidPeso molecular:332.22AMX12006
CAS:<p>AMX12006, a potent and selective EP4 antagonist, exhibits cytotoxic and antitumor activity, demonstrating oral activity with an IC50 of 4.3 nM [1].</p>Fórmula:C26H22F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:481.47Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Fórmula:C19H24N2OPureza:98%Cor e Forma:SolidPeso molecular:296.41NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Fórmula:C25H27Cl2N3O2SPureza:98%Cor e Forma:SolidPeso molecular:504.47WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Fórmula:C14H18N2Pureza:98%Cor e Forma:SolidPeso molecular:214.31PF2562
CAS:<p>PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).</p>Fórmula:C19H17N5OPureza:98%Cor e Forma:SolidPeso molecular:331.37ROS 234 dioxalate
CAS:<p>ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)</p>Fórmula:C17H19N5O8Pureza:98%Cor e Forma:SolidPeso molecular:421.37VUF 5574
CAS:<p>VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.</p>Fórmula:C21H17N5O2Pureza:99.53%Cor e Forma:SolidPeso molecular:371.39N-Methyldopamine hydrochloride
CAS:<p>N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.</p>Fórmula:C9H14ClNO2Cor e Forma:SolidPeso molecular:203.67SR 2640 hydrochloride
CAS:<p>SR 2640 hydrochloride is a competitive antagonist of leukotriene D4 and E4 and can be used in studies about leukotrienes in human asthma.</p>Fórmula:C23H19ClN2O3Pureza:98.36%Cor e Forma:SolidPeso molecular:406.86BW 245C
CAS:<p>BW 245C is a DP1 agonist with an inhibitory effect on the aggregation response of collagen and can be used to study diseases such as stroke.</p>Fórmula:C19H32N2O5Pureza:≥99%Cor e Forma:SolidPeso molecular:368.47Glemanserin
CAS:<p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>Fórmula:C20H25NOPureza:99.93%Cor e Forma:SolidPeso molecular:295.42OMDM-6
CAS:<p>OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.</p>Fórmula:C28H42N2O3Pureza:99.66%Cor e Forma:SolidPeso molecular:454.64N-Arachidonyldopamine
CAS:<p>N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1</p>Fórmula:C28H41NO3Pureza:97.65%Cor e Forma:SolidPeso molecular:439.63VPC 23019
CAS:<p>VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively).</p>Fórmula:C17H29N2O5PPureza:98%Cor e Forma:SolidPeso molecular:372.4Ancarolol
CAS:Ancarolol is a blocking agent of beta-adrenergic.Fórmula:C18H24N2O4Pureza:98%Cor e Forma:SolidPeso molecular:332.39Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Fórmula:C18H20N2Pureza:99.85%Cor e Forma:SolidPeso molecular:264.36Wy 49051
CAS:<p>Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).</p>Fórmula:C28H33N5O3Pureza:99.89%Cor e Forma:SolidPeso molecular:487.59PF-03654746
CAS:<p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>Fórmula:C18H24F2N2OPureza:98.85% - 99.57%Cor e Forma:SolidPeso molecular:322.39Rolapitant
CAS:<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Fórmula:C25H26F6N2O2Pureza:99.86%Cor e Forma:SolidPeso molecular:500.48Arbutamine
CAS:<p>Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.</p>Fórmula:C18H23NO4Pureza:95.06%Cor e Forma:SolidPeso molecular:317.38PD 144418
CAS:<p>PD 144418 displays potential antipsychotic activity.</p>Fórmula:C18H22N2OPureza:98%Cor e Forma:SolidPeso molecular:282.38Methiothepin maleate
CAS:<p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>Fórmula:C24H28N2O4S2Pureza:98%Cor e Forma:SolidPeso molecular:472.62Amitifadine hydrochloride
CAS:<p>Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).</p>Fórmula:C11H12Cl3NPureza:98%Cor e Forma:SolidPeso molecular:264.58F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Fórmula:C25H29ClF2N4O5Pureza:98.86%Cor e Forma:SolidPeso molecular:538.97Radioprotectin-1
CAS:<p>Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.</p>Fórmula:C23H19ClN2O6SPureza:98.63% - 99.27%Cor e Forma:SolidPeso molecular:486.92Rec 15/2615 dihydrochloride
CAS:<p>Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.</p>Fórmula:C26H35Cl2N5O5Pureza:97.04% - 99.76%Cor e Forma:SolidPeso molecular:568.49Donitriptan
CAS:<p>Donitriptan 是一种 5-HT 受体激动剂，对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>Fórmula:C23H25N5O2Pureza:98.76%Cor e Forma:SolidPeso molecular:403.48PGD2-IN-1
CAS:<p>PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.</p>Fórmula:C23H23Cl2N3O3Pureza:98.21%Cor e Forma:SolidPeso molecular:460.35Felypressin acetate
CAS:<p>Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.</p>Fórmula:C48H69N13O13S2Pureza:97.06%Cor e Forma:SolidPeso molecular:1100.27CGP 35949
CAS:<p>CGP 35949 is an LTD4 antagonist with phospholipase inhibitory activity.</p>Fórmula:C23H25ClN5NaO5Pureza:99.62%Cor e Forma:SolidPeso molecular:509.92RG-12915
CAS:<p>RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).</p>Fórmula:C20H25ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:360.88Nelonicline
CAS:<p>Nelonicline is a selective agonist of neuronal nicotinic receptors.</p>Fórmula:C17H19N3OSPureza:98%Cor e Forma:SolidPeso molecular:313.42CB2 modulator 1
CAS:<p>CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.</p>Fórmula:C18H19F3N4O2Pureza:99.6%Cor e Forma:SolidPeso molecular:380.36Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Fórmula:C17H20N4O2Pureza:99.97%Cor e Forma:SolidPeso molecular:312.37Niperotidine
CAS:<p>Niperotidine is an antagonist of histamine H2-receptor.</p>Fórmula:C20H26N4O5SPureza:98%Cor e Forma:SolidPeso molecular:434.51Ampreloxetine
CAS:<p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>Fórmula:C18H18F3NOPureza:98%Cor e Forma:SolidPeso molecular:321.34EP1-antagonist-1
CAS:<p>EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).</p>Fórmula:C19H15BrCl2N2O3Pureza:97.06%Cor e Forma:SolidPeso molecular:470.14EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Fórmula:C24H31N3O2Pureza:95.64% - 99.39%Cor e Forma:SolidPeso molecular:393.522(S)-(-)-Propranolol hydrochloride
CAS:<p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。</p>Fórmula:C16H22ClNO2Pureza:99.02% - 99.91%Cor e Forma:SolidPeso molecular:295.8Befetupitant
CAS:<p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>Fórmula:C29H29F6N3O2Pureza:98.72%Cor e Forma:SolidPeso molecular:565.55Aminaftone
CAS:<p>Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.</p>Fórmula:C18H15NO4Pureza:96.31% - 99.39%Cor e Forma:SolidPeso molecular:309.32AP521
CAS:<p>AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).</p>Fórmula:C20H19ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:402.89PG 01037 dihydrochloride
CAS:<p>PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.</p>Fórmula:C26H28Cl4N4OPureza:99.89%Cor e Forma:SolidPeso molecular:554.34WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Fórmula:C17H20Cl2FN3O2SPureza:98.43%Cor e Forma:SolidPeso molecular:420.33AM6545
CAS:<p>AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.</p>Fórmula:C26H23Cl2N5O3SPureza:97.03%Cor e Forma:SolidPeso molecular:556.46LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Fórmula:C27H38ClN3OSPureza:98.06%Cor e Forma:SolidPeso molecular:488.13Rp-cAMPS sodium
CAS:<p>Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.</p>Fórmula:C10H11N5NaO5PSPureza:99.71%Cor e Forma:SolidPeso molecular:367.25Aligeron
CAS:<p>Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibit</p>Fórmula:C20H24N2Pureza:99.09% - >99.99%Cor e Forma:SolidPeso molecular:292.42Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Cor e Forma:SolidPeso molecular:369.292-Iodomelatonin
CAS:<p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.</p>Fórmula:C13H15IN2O2Pureza:99.7%Cor e Forma:SolidPeso molecular:358.17TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Cor e Forma:SolidPeso molecular:377.48GR 113808
CAS:<p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>Fórmula:C19H27N3O4SPureza:98.16%Cor e Forma:SolidPeso molecular:393.5ST3932
CAS:<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Fórmula:C12H16N8OPureza:98%Cor e Forma:SolidPeso molecular:288.31PRX933 hydrochloride
CAS:<p>PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.</p>Fórmula:C16H22ClN5O2Pureza:99.51% - 99.89%Cor e Forma:SolidPeso molecular:351.84H4R antagonist 1
CAS:<p>H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.</p>Fórmula:C11H11BrN8Cor e Forma:SolidPeso molecular:335.16Iferanserin
CAS:<p>Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.</p>Fórmula:C23H28N2OCor e Forma:SolidPeso molecular:348.48Deramciclane
CAS:<p>Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.</p>Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47(±)-Tazifylline
CAS:<p>(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.</p>Fórmula:C23H32N6O3SPureza:99.54%Cor e Forma:SolidPeso molecular:472.6SK1-IN-1
CAS:<p>SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be used to study cancer and neurodegenerative diseases.</p>Fórmula:C22H30N4O3Pureza:98.72%Cor e Forma:SolidPeso molecular:398.5Tedatioxetine hydrobromide
CAS:<p>Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.</p>Fórmula:C18H22BrNSPureza:99.65%Cor e Forma:SolidPeso molecular:364.34BAY-1316957
CAS:<p>BAY-1316957 is a highly potent and selective EP4 receptor antagonist. With an IC50 of 15.3 nM. Good oral bioavailability[1].</p>Fórmula:C27H27N3O3Cor e Forma:SolidPeso molecular:441.52(S)-Terazosin
CAS:<p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>Fórmula:C19H25N5O4Cor e Forma:SolidPeso molecular:387.43Licogliflozin
CAS:<p>Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).</p>Fórmula:C23H28O7Pureza:98%Cor e Forma:SolidPeso molecular:416.46L-692429
CAS:<p>L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can be used to study acromegaly and obesity.</p>Fórmula:C29H31N7O2Pureza:98.64% - 99.90%Cor e Forma:SolidPeso molecular:509.614T-0509
CAS:<p>T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-</p>Fórmula:C18H23NO5Pureza:97.52% - 98.43%Cor e Forma:SolidPeso molecular:333.38SLM6031434 HCl
CAS:<p>SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.</p>Fórmula:C22H31ClF3N5O2Pureza:98%Cor e Forma:SolidPeso molecular:489.96p-MPPF dihydrochloride
CAS:<p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>Fórmula:C25H29Cl2FN4O2Pureza:99.55%Cor e Forma:SolidPeso molecular:507.43Arvanil
CAS:<p>Arvanil (N-Vanillylarachidonamide) is a synthetic capsaicin-amphetamine hybrid that acts as a ligand for VR1 and CB1, offering neuroprotective effects.</p>Fórmula:C28H41NO3Pureza:99.49%Cor e Forma:SolidPeso molecular:439.63PGN-9856
CAS:PGN-9856 is an EP2 receptor ligand and EP2 receptor agonist with anti-inflammatory and intraocular pressure-lowering properties, useful for glaucoma research.Fórmula:C21H15F2NO4Pureza:99.27%Cor e Forma:SolidPeso molecular:383.35LPA2 antagonist 1
CAS:<p>LPA2 antagonist 1 is a potent LPA2 antagonist.</p>Fórmula:C20H23Cl2N5O2S2Pureza:99.85%Cor e Forma:SolidPeso molecular:500.47Cyclazosin HCl
CAS:<p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>Fórmula:C23H28ClN5O4Pureza:99.10%Cor e Forma:SolidPeso molecular:473.95L-694,247
CAS:<p>L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.</p>Fórmula:C20H21N5O3SPureza:98.36%Cor e Forma:White SolidPeso molecular:411.486-Chloromelatonin
CAS:<p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>Fórmula:C13H15ClN2O2Pureza:98.01% - 99.25%Cor e Forma:SolidPeso molecular:266.72Usmarapride free base
CAS:<p>Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.</p>Fórmula:C21H29N5O2Pureza:99.91% - 99.91%Cor e Forma:SolidPeso molecular:383.49S 32212 hydrochloride
CAS:<p>S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .</p>Fórmula:C25H29ClN4O2Pureza:97.11% - 99.57%Cor e Forma:SolidPeso molecular:452.98SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Fórmula:C18H20ClNO2Pureza:98.68%Cor e Forma:SolidPeso molecular:317.81CCX777
CAS:<p>CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer research.</p>Fórmula:C31H43N7O3SPureza:98.73%Cor e Forma:SolidPeso molecular:593.78Levobunolol hydrochloride
CAS:<p>Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂，可用于治疗青光眼和上斜肌肌障碍的研究。</p>Fórmula:C17H26ClNO3Pureza:98.49% - >99.99%Cor e Forma:SolidPeso molecular:327.85Org41841
CAS:<p>Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.</p>Fórmula:C19H22N4O2S2Pureza:99.46% - 99.92%Cor e Forma:SolidPeso molecular:402.53MRE3008F20
CAS:<p>MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.</p>Fórmula:C21H20N8O3Pureza:97.29%Cor e Forma:SolidPeso molecular:432.44MJ 15
CAS:<p>MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.</p>Fórmula:C23H17Cl3N4OPureza:99.63%Cor e Forma:SolidPeso molecular:471.77L748337
CAS:<p>L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.</p>Fórmula:C26H31N3O5SPureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:497.61Pridefine
CAS:<p>Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.</p>Fórmula:C19H21NPureza:99.15% - 99.66%Cor e Forma:SolidPeso molecular:263.38JNJ-39220675
CAS:<p>JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.</p>Fórmula:C21H24FN3O2Pureza:98.13% - 99.89%Cor e Forma:SolidPeso molecular:369.43OPC-14523 hydrochloride
CAS:<p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>Fórmula:C23H29Cl2N3O2Pureza:99.60%Cor e Forma:SolidPeso molecular:450.4E-3620
CAS:<p>E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.</p>Fórmula:C20H27Cl2N3O2Pureza:98.88% - 98.88%Cor e Forma:SolidPeso molecular:412.35PF 03654746 FA
<p>PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.</p>Fórmula:C19H26F2N2O3Pureza:99.44%Cor e Forma:SoildPeso molecular:368.42ADRA1D receptor antagonist 1 HCl
CAS:<p>ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.</p>Fórmula:C15H14Cl2N4OPureza:98.13%Cor e Forma:SolidPeso molecular:337.2AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Fórmula:C17H20ClN5O2SPureza:>99.99%Cor e Forma:SolidPeso molecular:393.89Romifidine
CAS:<p>Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.</p>Fórmula:C9H9BrFN3Cor e Forma:SolidPeso molecular:258.09SLV-310
CAS:<p>SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.</p>Fórmula:C25H24FN3O2Pureza:99.39%Cor e Forma:SolidPeso molecular:417.48SC 51089
CAS:<p>SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.</p>Fórmula:C22H20Cl2N4O3Pureza:98%Cor e Forma:SolidPeso molecular:459.33(Iso)-FK-480
CAS:<p>(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.</p>Fórmula:C26H19FN4O2Pureza:98.36% - 99.41%Cor e Forma:SolidPeso molecular:438.45LY377604
CAS:<p>LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.</p>Fórmula:C31H32N4O4Pureza:99.72% - >99.99%Cor e Forma:SolidPeso molecular:524.61ST1936
CAS:<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Fórmula:C13H17ClN2Pureza:98%Cor e Forma:SolidPeso molecular:236.74SM-2470
CAS:<p>SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.</p>Fórmula:C23H30ClN5O3Pureza:98.91%Cor e Forma:SolidPeso molecular:459.97RXFP3/4 agonist 2
CAS:<p>RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.</p>Fórmula:C22H22N6O2Pureza:99.82%Cor e Forma:SolidPeso molecular:402.45mPGES-1 Inhibitor-1
CAS:<p>mPGES-1 Inhibitor-1 is an mPGES-1 inhibitor with anti-inflammatory and analgesic activity, which can be used to study acute liver injury.</p>Fórmula:C16H19ClN4O2Pureza:96.84% - 98.75%Cor e Forma:SolidPeso molecular:334.8Org-13011 fumarate
CAS:<p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>Fórmula:C22H29F3N4O5Pureza:98.92%Cor e Forma:SolidPeso molecular:486.48Enciprazine
CAS:<p>Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.</p>Fórmula:C23H32N2O6Pureza:98.63%Cor e Forma:SolidPeso molecular:432.51Adatanserin
CAS:<p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>Fórmula:C21H31N5OPureza:99.33%Cor e Forma:SolidPeso molecular:369.5Amgen-23
CAS:<p>Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.</p>Fórmula:C23H25Cl2N3O2SPureza:97.31%Cor e Forma:SolidPeso molecular:478.44AM404
CAS:<p>AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.</p>Fórmula:C26H37NO2Cor e Forma:SolidPeso molecular:395.58RS 56812 hydrochloride
CAS:<p>5-HT3 partial agonist</p>Fórmula:C18H22ClN3O2Pureza:98.62%Cor e Forma:SolidPeso molecular:347.84PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Fórmula:C15H20Cl2N2OPureza:98.67%Cor e Forma:SolidPeso molecular:315.24MK-2894
CAS:<p>MK-2894 is a highly potent and selective antagonist of second generation EP4 .</p>Fórmula:C25H22F3NO3SPureza:99.22%Cor e Forma:SolidPeso molecular:473.51A-65186
CAS:<p>A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.</p>Fórmula:C25H35N3O4Pureza:98.85% - 99.94%Cor e Forma:SolidPeso molecular:441.56UCM-05194
CAS:<p>UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD 19.6 nM, inactive at LPA2-6/autotaxin).</p>Fórmula:C19H30BrO6PPureza:90% - 91.22%Cor e Forma:SolidPeso molecular:465.32UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Fórmula:C23H28Cl2N4O2Pureza:98.78% - 98.78%Cor e Forma:SolidPeso molecular:463.4Falintolol
CAS:<p>Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.</p>Fórmula:C12H24N2O2Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:228.33ML-354
CAS:<p>ML354 is a selective antagonist of PAR4 with an IC 50 of 140 nM [1].</p>Fórmula:C16H14N2O3Pureza:99.44%Cor e Forma:SolidPeso molecular:282.29Olorinab
CAS:<p>Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.</p>Fórmula:C18H23N5O3Pureza:97.67% - 98.47%Cor e Forma:SolidPeso molecular:357.41CGRP antagonist 1
CAS:<p>CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the</p>Fórmula:C29H26N4O4Pureza:99.55%Cor e Forma:SolidPeso molecular:494.54O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Fórmula:C17H22O2Pureza:99.85%Cor e Forma:SolidPeso molecular:258.36Pavinetant
CAS:<p>Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.</p>Fórmula:C26H25N3O3SPureza:99.8%Cor e Forma:SolidPeso molecular:459.56Midaglizole hydrochloride
CAS:<p>Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).</p>Fórmula:C16H19Cl2N3Pureza:99.39% - 99.82%Cor e Forma:SolidPeso molecular:324.25NF-56-EJ40
CAS:<p>NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM.</p>Fórmula:C27H29N3O3Pureza:99.65%Cor e Forma:SolidPeso molecular:443.54Proxyfan
CAS:<p>Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.</p>Fórmula:C13H16N2OPureza:99.68%Cor e Forma:SolidPeso molecular:216.28Impromidine hydrochloride
CAS:<p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>Fórmula:C14H26Cl3N7SPureza:99.82%Cor e Forma:SolidPeso molecular:430.83BMS 182874
CAS:<p>BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.</p>Fórmula:C17H19N3O3SPureza:98.38%Cor e Forma:SolidPeso molecular:345.42CB1R antagonist 1
CAS:<p>CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.</p>Fórmula:C18H23F3N2O3SPureza:99.65%Cor e Forma:SolidPeso molecular:404.45CyPPA
CAS:<p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>Fórmula:C16H23N5Pureza:99.88%Cor e Forma:SolidPeso molecular:285.39SLF1081851
CAS:<p>SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.</p>Fórmula:C21H33N3OPureza:99.26%Cor e Forma:SolidPeso molecular:343.51ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Fórmula:C12H16N8Pureza:99.64% - 99.69%Cor e Forma:SolidPeso molecular:272.31K6PC-5
CAS:<p>K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels.</p>Fórmula:C19H37NO4Pureza:99.9%Cor e Forma:SolidPeso molecular:343.5Cianopramine
CAS:<p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>Fórmula:C20H23N3Pureza:99.92% - 99.92%Cor e Forma:SolidPeso molecular:305.42Rafabegron
CAS:<p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>Fórmula:C21H23ClN2O4Pureza:99.21%Cor e Forma:SolidPeso molecular:402.87N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Fórmula:C18H21N5O4Pureza:99.83%Cor e Forma:SolidPeso molecular:371.39LAS38096
CAS:<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Fórmula:C17H12N6OPureza:99.18% - 99.95%Cor e Forma:SolidPeso molecular:316.32SDZ-62-434
CAS:<p>SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.</p>Fórmula:C23H27Cl2N3Pureza:98.38%Cor e Forma:SolidPeso molecular:416.39BAY 60-6583
CAS:<p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>Fórmula:C19H17N5O2SPureza:98.46% - 99.8%Cor e Forma:SolidPeso molecular:379.44ISAM-140
CAS:<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Fórmula:C19H19N3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:337.37Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Fórmula:C15H23NOPureza:98.09% - 98.77%Cor e Forma:SolidPeso molecular:233.35Nonabine
CAS:<p>Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.</p>Fórmula:C25H33NO2Pureza:99.46% - 99.95%Cor e Forma:SolidPeso molecular:379.54(R)-ZINC-3573
CAS:<p>ZINC-3573: Potent, selective MRGPRX2 activator; triggers mast cell degranulation and calcium release.</p>Fórmula:C18H21N5Pureza:99.75%Cor e Forma:SolidPeso molecular:307.39Edonentan
CAS:<p>Edonentan is A potent endothelin A (ETA) receptor antagonist that can be used to study heart failure.</p>Fórmula:C28H32N4O5SPureza:98.07% - 99.6%Cor e Forma:SolidPeso molecular:536.64U 99194 maleate
CAS:<p>U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.</p>Fórmula:C21H31NO6Pureza:99.45%Cor e Forma:SolidPeso molecular:393.47Perphenazine dihydrochloride
CAS:<p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>Fórmula:C21H28Cl3N3OSPureza:99.67%Cor e Forma:SolidPeso molecular:476.89Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Cor e Forma:SolidPeso molecular:381.44ST 91
CAS:<p>ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.</p>Fórmula:C13H20ClN3Pureza:99.83%Cor e Forma:SolidPeso molecular:253.77Parogrelil Free Base
CAS:<p>Parogrelil Free Base is a phosphodiesterase inhibitor, improves claudication-limited exercise performance in patients with peripheral arterial disease.</p>Fórmula:C19H18BrClN4O2Pureza:99.16% - 99.17%Cor e Forma:SolidPeso molecular:449.73SB-209670
CAS:<p>SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in rat vascular endothelium and vascular smooth muscle.</p>Fórmula:C29H28O9Pureza:97.80% - 99.40%Cor e Forma:SolidPeso molecular:520.53NNC 92-1687
CAS:<p>NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.</p>Fórmula:C15H12N2O3SPureza:98.70% - 99.70%Cor e Forma:SolidPeso molecular:300.33FPL 55712
CAS:<p>FPL 55712 is a leukotriene receptor and SRS-A antagonist that inhibits bronchoconstriction and can be used in studies of asthma and coronary artery thrombosis.</p>Fórmula:C27H30O9Pureza:98.15% - 99.8%Cor e Forma:SolidPeso molecular:498.52BMS CCR2 22
CAS:BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Fórmula:C28H34F3N5O4SPureza:99.65%Cor e Forma:SolidPeso molecular:593.66Fipamezole
CAS:<p>Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.</p>Fórmula:C14H15FN2Pureza:99.32% - >99.99%Cor e Forma:SolidPeso molecular:230.28SB 699551 dihydrochloride
CAS:<p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>Fórmula:C34H47Cl2N3OPureza:99.83%Cor e Forma:SolidPeso molecular:584.66Antihistamine-1
CAS:<p>Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。</p>Fórmula:C23H24FN5Pureza:99.69%Cor e Forma:SolidPeso molecular:389.47Halopemide
CAS:<p>Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).</p>Fórmula:C21H22ClFN4O2Pureza:96.57%Cor e Forma:SolidPeso molecular:416.88Isbogrel
CAS:<p>Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.</p>Fórmula:C18H19NO2Pureza:99.58%Cor e Forma:SolidPeso molecular:281.35DA-6886
CAS:<p>DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.</p>Fórmula:C19H28Cl2N6O2Pureza:99.28% - 99.91%Cor e Forma:SolidPeso molecular:443.37ANR 94
CAS:<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Fórmula:C9H13N5OPureza:98.9%Cor e Forma:SolidPeso molecular:207.23Pimethixene maleate
CAS:<p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>Fórmula:C23H23NO4SPureza:99.55%Cor e Forma:SolidPeso molecular:409.5Efletirizine
CAS:<p>Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.</p>Fórmula:C21H24F2N2O3Pureza:99.39%Cor e Forma:SolidPeso molecular:390.42Neldazosin
CAS:<p>Neldazosin is used as a potent α1-adrenoceptor antagonist.</p>Fórmula:C18H25N5O4Pureza:99.74% - 99.76%Cor e Forma:SolidPeso molecular:375.428-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Fórmula:C16H25NOPureza:98%Cor e Forma:SolidPeso molecular:247.38BMS-817399
CAS:<p>BMS-817399: oral CCR1 antagonist with binding and chemotaxis inhibition IC50s, potential for rheumatoid arthritis research.</p>Fórmula:C23H36ClN3O4Pureza:99.7%Cor e Forma:SolidPeso molecular:454Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Fórmula:C14H20ClN3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:313.78RG 7152
CAS:<p>RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.</p>Fórmula:C20H19N5O2Pureza:98.45%Cor e Forma:SolidPeso molecular:361.4Medifoxamine
CAS:<p>Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine</p>Fórmula:C16H19NO2Pureza:97.14%Cor e Forma:SolidPeso molecular:257.33R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Fórmula:C27H27ClFN3OSPureza:97.7%Cor e Forma:SolidPeso molecular:496.04RO3244794
CAS:<p>RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.</p>Fórmula:C25H19F2NO5Pureza:99.36%Cor e Forma:SolidPeso molecular:451.42PNU-282987 free base
CAS:<p>PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.</p>Fórmula:C14H17ClN2OPureza:99.64%Cor e Forma:SolidPeso molecular:264.75Dabelotine
CAS:<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Fórmula:C15H22N2O2Pureza:98.55%Cor e Forma:SolidPeso molecular:262.35AZ-1355
CAS:<p>AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.</p>Fórmula:C17H17NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:299.32RS 67333 hydrochloride
CAS:<p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>Fórmula:C19H30Cl2N2O2Pureza:98.78%Cor e Forma:SolidPeso molecular:389.36Itasetron
CAS:<p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>Fórmula:C16H20N4O2Pureza:98.58% - 99.33%Cor e Forma:SolidPeso molecular:300.36KSK68
CAS:<p>KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.</p>Fórmula:C23H28N2O2Pureza:99.11%Cor e Forma:SolidPeso molecular:364.48Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Fórmula:C20H26ClNO2Pureza:99.63%Cor e Forma:SolidPeso molecular:347.88FK-453
CAS:<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Fórmula:C23H25N3O2Pureza:99.44%Cor e Forma:SolidPeso molecular:375.46Selodenoson
CAS:<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Fórmula:C17H24N6O4Pureza:99.52%Cor e Forma:SolidPeso molecular:376.41Ecopipam
CAS:<p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>Fórmula:C19H20ClNOPureza:99.68%Cor e Forma:SolidPeso molecular:313.82
