GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Cor e Forma:SolidPeso molecular:381.44GW-493838
CAS:<p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>Fórmula:C21H21ClFN7O4Pureza:99.11% - 99.58%Cor e Forma:SolidPeso molecular:489.89CP 316311
CAS:<p>CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.</p>Fórmula:C21H29NO2Pureza:99.71% - >99.99%Cor e Forma:SolidPeso molecular:327.46(S)-(+)-Niguldipine hydrochloride
CAS:<p>(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.</p>Fórmula:C36H40ClN3O6Pureza:98.27%Cor e Forma:SolidPeso molecular:646.17Eclazolast
CAS:<p>Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.</p>Fórmula:C12H12ClNO4Pureza:98.36% - 98.58%Cor e Forma:SolidPeso molecular:269.68Safotibant
CAS:<p>Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema</p>Fórmula:C25H34N4O5SPureza:99.62% - 99.67%Cor e Forma:SolidPeso molecular:502.63Clemastine
CAS:<p>Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.</p>Fórmula:C21H26ClNOPureza:99.21%Cor e Forma:SolidPeso molecular:343.89Enerisant hydrochloride
CAS:<p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>Fórmula:C22H31ClN4O3Pureza:99.95%Cor e Forma:SolidPeso molecular:434.96LAS38096
CAS:<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Fórmula:C17H12N6OPureza:99.18% - 99.95%Cor e Forma:SolidPeso molecular:316.32LY 272015 hydrochloride
CAS:<p>LY 272015 hydrochloride is a 5-HT2B receptor antagonist.</p>Fórmula:C21H25ClN2O2Pureza:99.47%Cor e Forma:SolidPeso molecular:372.89JP1302
CAS:<p>JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.</p>Fórmula:C24H24N4Pureza:99.96%Cor e Forma:SolidPeso molecular:368.47SCH-336
CAS:<p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>Fórmula:C23H25NO8S3Pureza:95.01%Cor e Forma:SolidPeso molecular:539.64Seridopidine
CAS:<p>Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.</p>Fórmula:C14H20FNO2SPureza:99.65%Cor e Forma:SolidPeso molecular:285.387-Hydroxy-DPAT hydrobromide
CAS:<p>7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.</p>Fórmula:C16H26BrNOPureza:99.73%Cor e Forma:SolidPeso molecular:328.29JTE-907
CAS:<p>JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。</p>Fórmula:C24H26N2O6Pureza:99.93%Cor e Forma:SolidPeso molecular:438.47CB1 agonist 1
CAS:<p>CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.</p>Fórmula:C24H24N2O5SPureza:98.56%Cor e Forma:SolidPeso molecular:452.52CMF019
CAS:<p>CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).</p>Fórmula:C25H33N3O3SPureza:99.5%Cor e Forma:SolidPeso molecular:455.61SB-209670
CAS:<p>SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in rat vascular endothelium and vascular smooth muscle.</p>Fórmula:C29H28O9Pureza:97.80% - 99.40%Cor e Forma:SolidPeso molecular:520.53U 99194 maleate
CAS:<p>U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.</p>Fórmula:C21H31NO6Pureza:99.45%Cor e Forma:SolidPeso molecular:393.47A-437203
CAS:<p>A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.</p>Fórmula:C20H27F3N6OSPureza:98.80%Cor e Forma:SolidPeso molecular:456.53Adenosine antagonist-1
CAS:<p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>Fórmula:C18H13N7SPureza:99.28% - 99.95%Cor e Forma:SolidPeso molecular:359.41TC LPA5 4
CAS:<p>TC LPA5 4 is a LPA5 receptor antagonist.</p>Fórmula:C23H23ClN2O3Pureza:99.93%Cor e Forma:SolidPeso molecular:410.89RS 67333 hydrochloride
CAS:<p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>Fórmula:C19H30Cl2N2O2Pureza:98.78%Cor e Forma:SolidPeso molecular:389.36Butofilolol
CAS:<p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>Fórmula:C17H26FNO3Pureza:98.96% - >99.99%Cor e Forma:SolidPeso molecular:311.392Oxyfedrine L-form HCl
CAS:<p>Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.</p>Fórmula:C19H24ClNO3Pureza:99.5% - 99.57%Cor e Forma:SolidPeso molecular:349.85CGRP antagonist 1
CAS:<p>CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the</p>Fórmula:C29H26N4O4Pureza:99.55%Cor e Forma:SolidPeso molecular:494.54O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Fórmula:C17H22O2Pureza:99.85%Cor e Forma:SolidPeso molecular:258.36Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Fórmula:C22H22N2O7Pureza:>99.99%Cor e Forma:SolidPeso molecular:426.42Torbafylline
CAS:<p>Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, cancer, or sepsis.</p>Fórmula:C16H26N4O4Pureza:98.66% - 99.13%Cor e Forma:SoildPeso molecular:338.4Milveterol HCl
CAS:<p>Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).</p>Fórmula:C25H30ClN3O4Pureza:98.2%Cor e Forma:SolidPeso molecular:471.98Proxyfan
CAS:<p>Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.</p>Fórmula:C13H16N2OPureza:99.68%Cor e Forma:SolidPeso molecular:216.28Impromidine hydrochloride
CAS:<p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>Fórmula:C14H26Cl3N7SPureza:99.82%Cor e Forma:SolidPeso molecular:430.83ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Fórmula:C12H16N8Pureza:99.64% - 99.69%Cor e Forma:SolidPeso molecular:272.31AM-1235
CAS:<p>AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.</p>Fórmula:C24H21FN2O3Pureza:97.77%Cor e Forma:SolidPeso molecular:404.43K6PC-5
CAS:<p>K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels.</p>Fórmula:C19H37NO4Pureza:99.9%Cor e Forma:SolidPeso molecular:343.5Ticolubant
CAS:<p>Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.</p>Fórmula:C23H19Cl2NO3SPureza:99.59%Cor e Forma:SolidPeso molecular:460.37N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Fórmula:C18H21N5O4Pureza:99.83%Cor e Forma:SolidPeso molecular:371.39L-693,403 maleate
CAS:<p>L-693,403 maleate has analgesic activity.</p>Fórmula:C24H27NO4Pureza:99.88%Cor e Forma:SolidPeso molecular:393.48ANR 94
CAS:<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Fórmula:C9H13N5OPureza:98.9%Cor e Forma:SolidPeso molecular:207.23Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Fórmula:C24H27FN4O2Pureza:98.04%Cor e Forma:SolidPeso molecular:422.5BMS 182874
CAS:<p>BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.</p>Fórmula:C17H19N3O3SPureza:98.38%Cor e Forma:SolidPeso molecular:345.42Neldazosin
CAS:<p>Neldazosin is used as a potent α1-adrenoceptor antagonist.</p>Fórmula:C18H25N5O4Pureza:99.74% - 99.76%Cor e Forma:SolidPeso molecular:375.42N 0861
CAS:<p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>Fórmula:C13H17N5Pureza:98.78%Cor e Forma:SolidPeso molecular:243.31L 674573
CAS:<p>L 674573 is an inhibitor of leukotriene biosynthesis.</p>Fórmula:C28H27NO3SPureza:99.51%Cor e Forma:SolidPeso molecular:457.58SLF1081851
CAS:<p>SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.</p>Fórmula:C21H33N3OPureza:99.26%Cor e Forma:SolidPeso molecular:343.51SF-22
CAS:<p>SF-22 is a Y2R antagonist with potential anti-inflammatory activity that can be used to study diseases associated with neurological disorders.</p>Fórmula:C28H26N2O3SPureza:99.09%Cor e Forma:SolidPeso molecular:470.58Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Fórmula:C28H30ClN5O3Pureza:99.04%Cor e Forma:SolidPeso molecular:520.028-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Fórmula:C16H25NOPureza:98%Cor e Forma:SolidPeso molecular:247.38Runcaciguat
CAS:<p>Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.</p>Fórmula:C23H22Cl2F3NO3Pureza:99.17%Cor e Forma:SolidPeso molecular:488.33GS-9667
CAS:<p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>Fórmula:C21H24FN5O4SPureza:99.76% - 99.77%Cor e Forma:SolidPeso molecular:461.51Crinecerfont
CAS:<p>Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.</p>Fórmula:C27H28ClFN2OSPureza:98.01% - 98.55%Cor e Forma:SolidPeso molecular:483.04Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Fórmula:C14H20ClN3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:313.78Pimethixene maleate
CAS:<p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>Fórmula:C23H23NO4SPureza:99.55%Cor e Forma:SolidPeso molecular:409.5NNC 92-1687
CAS:<p>NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.</p>Fórmula:C15H12N2O3SPureza:98.70% - 99.70%Cor e Forma:SolidPeso molecular:300.33Cianopramine
CAS:<p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>Fórmula:C20H23N3Pureza:99.92% - 99.92%Cor e Forma:SolidPeso molecular:305.42Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Fórmula:C15H23NOPureza:98.09% - 98.77%Cor e Forma:SolidPeso molecular:233.35AZD1940
CAS:<p>AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.</p>Fórmula:C20H29F2N3O2SPureza:98.68%Cor e Forma:SolidPeso molecular:413.52Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Fórmula:C26H32N2O5Pureza:99.17% - 99.67%Cor e Forma:SolidPeso molecular:452.54L-168049
CAS:<p>L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.</p>Fórmula:C24H20BrClN2OPureza:>99.99%Cor e Forma:SolidPeso molecular:467.79NF-56-EJ40
CAS:<p>NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM.</p>Fórmula:C27H29N3O3Pureza:99.65%Cor e Forma:SolidPeso molecular:443.54Lorglumide sodium salt
CAS:<p>Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).</p>Fórmula:C22H31Cl2N2NaO4Pureza:99.32%Cor e Forma:SolidPeso molecular:481.39Parogrelil Free Base
CAS:<p>Parogrelil Free Base is a phosphodiesterase inhibitor, improves claudication-limited exercise performance in patients with peripheral arterial disease.</p>Fórmula:C19H18BrClN4O2Pureza:99.16% - 99.17%Cor e Forma:SolidPeso molecular:449.73Remogliflozin etabonate
CAS:<p>Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.</p>Fórmula:C26H38N2O9Pureza:98.98%Cor e Forma:SolidPeso molecular:522.59APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Fórmula:C18H22N6O4Pureza:99.88%Cor e Forma:SolidPeso molecular:386.41Octimibate
CAS:<p>Octimibate: non-prostaglandin antiplatelet, treats cardiovascular disease, aids atherosclerosis/thrombosis research.</p>Fórmula:C29H30N2O3Pureza:99.51%Cor e Forma:SolidPeso molecular:454.56Sitaxsentan
CAS:<p>Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.</p>Fórmula:C18H15ClN2O6S2Pureza:97.99% - 98.71%Cor e Forma:SolidPeso molecular:454.9Agomelatine hydrochloride
CAS:<p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>Fórmula:C15H18ClNO2Pureza:99.57%Cor e Forma:SolidPeso molecular:279.76CYM50374
CAS:<p>CYM50374 inhibits Sphingosine-1-phosphate receptor 4 (S1P4 ) with an IC50 of µM.</p>Fórmula:C19H19NO3SPureza:98.35% - 98.4%Cor e Forma:SolidPeso molecular:341.42Pipoxazole
CAS:<p>Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.</p>Fórmula:C14H20N4OPureza:98.58% - 99.53%Cor e Forma:SolidPeso molecular:260.33SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Fórmula:C23H31Cl2NO8SPureza:99.37%Cor e Forma:SolidPeso molecular:552.47Taprizosin
CAS:<p>Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.</p>Fórmula:C25H26N6O4SPureza:96.34% - 99.11%Cor e Forma:SolidPeso molecular:506.58RG 7152
CAS:<p>RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.</p>Fórmula:C20H19N5O2Pureza:98.45%Cor e Forma:SolidPeso molecular:361.4ABT-080
CAS:<p>ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.</p>Fórmula:C37H31N2NaO4Pureza:98.42%Cor e Forma:SolidPeso molecular:590.64Antihistamine-1
CAS:<p>Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。</p>Fórmula:C23H24FN5Pureza:99.69%Cor e Forma:SolidPeso molecular:389.47FPL 55712
CAS:<p>FPL 55712 is a leukotriene receptor and SRS-A antagonist that inhibits bronchoconstriction and can be used in studies of asthma and coronary artery thrombosis.</p>Fórmula:C27H30O9Pureza:98.15% - 99.8%Cor e Forma:SolidPeso molecular:498.52ReN-1869
CAS:<p>ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases</p>Fórmula:C24H27NO2Pureza:99.83% - 99.98%Cor e Forma:SolidPeso molecular:361.48Nemazoline Free Base
CAS:<p>Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.</p>Fórmula:C10H11Cl2N3Pureza:98.06% - 98.83%Cor e Forma:SolidPeso molecular:244.12A2A receptor antagonist 1
CAS:<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Fórmula:C16H12FN5OPureza:99.52% - 99.93%Cor e Forma:SolidPeso molecular:309.3Bavisant
CAS:<p>Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.</p>Fórmula:C19H27N3O2Pureza:99.21% - 99.65%Cor e Forma:SolidPeso molecular:329.44Quinupramine
CAS:<p>Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.</p>Fórmula:C21H24N2Pureza:99.77%Cor e Forma:SolidPeso molecular:304.43CL 316243
CAS:<p>CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.</p>Fórmula:C20H18ClNNa2O7Pureza:98.00% - 99.68%Cor e Forma:SolidPeso molecular:465.79Amosulalol
CAS:<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Fórmula:C18H24N2O5SPureza:99.5%Cor e Forma:SolidPeso molecular:380.46LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Fórmula:C21H24Cl2N2O2Pureza:98.58%Cor e Forma:SolidPeso molecular:407.33ML 10302 hydrochloride
CAS:<p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>Fórmula:C15H22Cl2N2O3Pureza:99.99%Cor e Forma:SolidPeso molecular:349.2548740 RP
CAS:<p>48740 RP (RP 55779) is an antagonist of platelet-activating factor.</p>Fórmula:C12H11N3OSPureza:99.79%Cor e Forma:SolidPeso molecular:245.3Remoxipride hydrochloride
CAS:<p>Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-</p>Fórmula:C16H24BrClN2O3Pureza:99.88%Cor e Forma:SolidPeso molecular:407.73SK609 HCl
CAS:<p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>Fórmula:C10H15Cl2NPureza:99.02%Cor e Forma:SolidPeso molecular:220.14PNU-282987 free base
CAS:<p>PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.</p>Fórmula:C14H17ClN2OPureza:99.64%Cor e Forma:SolidPeso molecular:264.75Bedoradrine sulfate
CAS:<p>Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Fórmula:C24H32N2O5H2O4SPureza:99.31%Cor e Forma:SolidPeso molecular:477.56Immethridine dihydrobromide
CAS:<p>Immethridine dihydrobromide is a histamine H3 receptor agonist.</p>Fórmula:C9H11Br2N3Pureza:97.61% - 98.14%Cor e Forma:SolidPeso molecular:321.01KSK94
CAS:<p>KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.</p>Fórmula:C25H26N4OPureza:99.60%Cor e Forma:SolidPeso molecular:398.5L-161982
CAS:<p>L-161982 is a selective EP4 receptor antagonist that inhibits PGE2-induced ERK phosphorylation and cell proliferation in HCA-7 cells.Cost-effective and quality-assured.</p>Fórmula:C32H29F3N4O4S2Pureza:99.58% - 99.6%Cor e Forma:SolidPeso molecular:654.72CV-6209
CAS:<p>CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.</p>Fórmula:C34H60ClN3O6Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:642.31Egis-11150
CAS:<p>Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.</p>Fórmula:C19H21ClFN5O2Pureza:97.49% - >99.99%Cor e Forma:SolidPeso molecular:405.85Landipirdine
CAS:<p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>Fórmula:C18H19FN2O3SPureza:97.61% - 99.37%Cor e Forma:SolidPeso molecular:362.42KP136
CAS:<p>KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).</p>Fórmula:C16H18N4O3Pureza:98.3% - 98.61%Cor e Forma:SolidPeso molecular:314.34Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Fórmula:C24H32N4O2SPureza:99.74%Cor e Forma:SolidPeso molecular:440.6Medifoxamine
CAS:<p>Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine</p>Fórmula:C16H19NO2Pureza:97.14%Cor e Forma:SolidPeso molecular:257.33Evodenoson
CAS:<p>Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.</p>Fórmula:C23H29N7O6Pureza:99.75% - 99.83%Cor e Forma:SolidPeso molecular:499.52Pirodomast
CAS:<p>Pirodomast is a thromboxane A (TXA2) synthase inhibitor.</p>Fórmula:C18H17N3O2Pureza:99.64%Cor e Forma:SolidPeso molecular:307.35SB 218795
CAS:<p>SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.</p>Fórmula:C25H20N2O3Pureza:99.70%Cor e Forma:SolidPeso molecular:396.44UNC0006
CAS:<p>UNC0006 is a β-arrestin-biased dopamine D2 ligand.</p>Fórmula:C24H29Cl2N3O2Pureza:99.35% - 99.97%Cor e Forma:SolidPeso molecular:462.41Rezatomidine
CAS:<p>Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.</p>Fórmula:C13H16N2SPureza:98.34%Cor e Forma:SolidPeso molecular:232.34PSB-16133 sodium
CAS:<p>PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.</p>Fórmula:C28H21N2NaO5S2Pureza:98.03% - 98.93%Cor e Forma:SolidPeso molecular:552.60Upacicalcet
CAS:<p>Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.</p>Fórmula:C11H14ClN3O6SPureza:99.83%Cor e Forma:SolidPeso molecular:351.76Tildacerfont
CAS:<p>Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.</p>Fórmula:C20H26ClN5OSPureza:>99.99%Cor e Forma:SolidPeso molecular:419.97KI-7
CAS:<p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>Fórmula:C23H18N2O2Pureza:98.33%Cor e Forma:SolidPeso molecular:354.4CP 96021
CAS:<p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>Fórmula:C29H21FN4OSPureza:97.81% - 99.62%Cor e Forma:SoildPeso molecular:492.57Ricasetron
CAS:<p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>Fórmula:C19H27N3OPureza:99.52%Cor e Forma:SolidPeso molecular:313.44Imiloxan
CAS:<p>Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.</p>Fórmula:C14H16N2O2Pureza:98.13% - 99.8%Cor e Forma:SolidPeso molecular:244.29RLX-33
CAS:<p>RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.</p>Fórmula:C24H19ClN4O4Pureza:99.89%Cor e Forma:SolidPeso molecular:462.89AZD8542
CAS:<p>AZD8542 is an antagonist of Smoothened (SMO) with potential as an oncology therapeutic.</p>Fórmula:C25H24N4O2Pureza:99.96%Cor e Forma:SolidPeso molecular:412.48ASP-4058
CAS:<p>ASP-4058: Safe, oral S1P1/S1P5 agonist; improves autoimmune encephalomyelitis in mice.</p>Fórmula:C19H12F6N4O2Pureza:99.30% - 99.53%Cor e Forma:SolidPeso molecular:442.31Sonedenoson
CAS:<p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>Fórmula:C18H20ClN5O5Pureza:99.79%Cor e Forma:SolidPeso molecular:421.84Nonabine
CAS:<p>Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.</p>Fórmula:C25H33NO2Pureza:99.46% - 99.95%Cor e Forma:SolidPeso molecular:379.54Edonentan
CAS:<p>Edonentan is A potent endothelin A (ETA) receptor antagonist that can be used to study heart failure.</p>Fórmula:C28H32N4O5SPureza:98.07% - 99.6%Cor e Forma:SolidPeso molecular:536.64Linetastine
CAS:<p>Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.</p>Fórmula:C35H40N2O6Pureza:99.76%Cor e Forma:SolidPeso molecular:584.7Rocepafant
CAS:<p>Rocepafant (LAU8080), a PAF antagonist, reduces neonatal rat brain damage and inhibits TNF-α toxicity in L929 cells.</p>Fórmula:C26H23ClN6OS2Pureza:97.31% - 98.95%Cor e Forma:SolidPeso molecular:535.08SDZ-62-434
CAS:<p>SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.</p>Fórmula:C23H27Cl2N3Pureza:98.38%Cor e Forma:SolidPeso molecular:416.395-HT2 antagonist 1
CAS:<p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>Fórmula:C22H29FN4O2Pureza:99.76%Cor e Forma:SolidPeso molecular:400.49CCR2 antagonist 5
CAS:<p>JNJ-41443532: oral hCCR2 antagonist, IC50=37 nM, anti-chemotaxis, treats inflammation & diabetes.</p>Fórmula:C22H25F3N4O3SPureza:99.09%Cor e Forma:SolidPeso molecular:482.52SR144528
CAS:<p>SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).</p>Fórmula:C29H34ClN3OPureza:99.63%Cor e Forma:SolidPeso molecular:476.05GSK2239633A
CAS:<p>GSK2239633A is an allosteric antagonist of CC-chemokine receptor 4 (CCR4) with a pIC50 of 7.96 for the binding of [125I]-TARC to human CCR4.</p>Fórmula:C24H25ClN4O5S2Pureza:99.82%Cor e Forma:SolidPeso molecular:549.06Rafabegron
CAS:<p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>Fórmula:C21H23ClN2O4Pureza:99.21%Cor e Forma:SolidPeso molecular:402.87SMO-IN-2
CAS:<p>SMO-IN-2 is a SMO inhibitor with antiproliferative activity and anticancer activity and inhibits Hh signaling.SMO-IN-2 can be used in the study of cancer.</p>Fórmula:C25H25F4N5O2Pureza:98.64%Cor e Forma:SolidPeso molecular:503.49CCR1 antagonist 6
CAS:<p>CCR1 antagonist 6 is a CCR1 antagonist (IC50: 3 nM).</p>Fórmula:C21H23ClN4O3SPureza:99.02% - 99.15%Cor e Forma:SolidPeso molecular:446.952'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Fórmula:C16H22ClN5O4Pureza:99.93%Cor e Forma:SolidPeso molecular:383.83Cyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Fórmula:C19H21N3SPureza:97.01%Cor e Forma:SolidPeso molecular:323.46Tiopinac
CAS:<p>Tiopinac: tricyclic with anti-inflammatory, analgesic, antipyretic properties; inhibits prostaglandin synthesis; mild anti-platelet effects in humans.</p>Fórmula:C16H12O3SPureza:>99.99%Cor e Forma:SolidPeso molecular:284.33SC 19220
CAS:<p>SC 19220 is a prostaglandin E2 receptor EP1 antagonist that inhibits RANKL-induced osteoclastogenesis.</p>Fórmula:C16H14ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:331.755-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Fórmula:C22H20FN3O3Pureza:98.78% - 99.26%Cor e Forma:SolidPeso molecular:393.41Fipamezole
CAS:<p>Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.</p>Fórmula:C14H15FN2Pureza:99.32% - >99.99%Cor e Forma:SolidPeso molecular:230.28Sergliflozin etabonate
CAS:<p>Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.</p>Fórmula:C23H28O9Pureza:97.88%Cor e Forma:SolidPeso molecular:448.46Noberastine
CAS:<p>Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.</p>Fórmula:C17H21N5OPureza:99.72% - >99.99%Cor e Forma:SolidPeso molecular:311.38Fananserin
CAS:<p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>Fórmula:C23H24FN3O2SPureza:99.88%Cor e Forma:SolidPeso molecular:425.52Halopemide
CAS:<p>Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).</p>Fórmula:C21H22ClFN4O2Pureza:96.57%Cor e Forma:SolidPeso molecular:416.88BMS CCR2 22
CAS:BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Fórmula:C28H34F3N5O4SPureza:99.65%Cor e Forma:SolidPeso molecular:593.66Bedoradrine
CAS:<p>Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Fórmula:C24H32N2O5Pureza:>99.99%Cor e Forma:SolidPeso molecular:428.52Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Fórmula:C14H20FNO2SPureza:99.39%Cor e Forma:SolidPeso molecular:285.38Isbogrel
CAS:<p>Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.</p>Fórmula:C18H19NO2Pureza:99.58%Cor e Forma:SolidPeso molecular:281.35NGD 94-1
CAS:<p>NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.</p>Fórmula:C18H20N6Pureza:99.61%Cor e Forma:SolidPeso molecular:320.39Spizofurone
CAS:<p>Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.</p>Fórmula:C12H10O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:202.21CyPPA
CAS:<p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>Fórmula:C16H23N5Pureza:99.88%Cor e Forma:SolidPeso molecular:285.39PF-00217830
CAS:<p>PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.</p>Fórmula:C26H30N4O2Pureza:98.72%Cor e Forma:SolidPeso molecular:430.54DA-6886
CAS:<p>DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.</p>Fórmula:C19H28Cl2N6O2Pureza:99.28% - 99.91%Cor e Forma:SolidPeso molecular:443.37MK-0686
CAS:<p>MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.</p>Fórmula:C22H19ClF4N2O4Pureza:99.88%Cor e Forma:SolidPeso molecular:486.84PD 168568 dihydrochloride
CAS:<p>PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).</p>Fórmula:C22H29Cl2N3OPureza:99.71%Cor e Forma:SolidPeso molecular:422.39(Z)-Thiothixene
CAS:<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Fórmula:C23H29N3O2S2Pureza:99.21%Cor e Forma:Yellow To Yellow With A Tan Cast PowderPeso molecular:443.63ML-354
CAS:<p>ML354 is a selective antagonist of PAR4 with an IC 50 of 140 nM [1].</p>Fórmula:C16H14N2O3Pureza:99.44%Cor e Forma:SolidPeso molecular:282.29R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Fórmula:C27H27ClFN3OSPureza:97.7%Cor e Forma:SolidPeso molecular:496.04JZP-361
CAS:<p>JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.</p>Fórmula:C22H20ClN5OPureza:99.82%Cor e Forma:SolidPeso molecular:405.88Ancriviroc
CAS:<p>Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.</p>Fórmula:C28H37BrN4O3Pureza:99.76% - 99.82%Cor e Forma:SolidPeso molecular:557.52Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Fórmula:C21H24BrN3O3SPureza:98.36% - 99.65%Cor e Forma:SolidPeso molecular:478.4Soquinolol
CAS:<p>Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long</p>Fórmula:C17H26N2O3Pureza:97.48% - 98.63%Cor e Forma:SolidPeso molecular:306.4Dabelotine
CAS:<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Fórmula:C15H22N2O2Pureza:98.55%Cor e Forma:SolidPeso molecular:262.35GR 46611
CAS:<p>GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.</p>Fórmula:C23H27N3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:377.48Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Fórmula:C20H26ClNO2Pureza:99.63%Cor e Forma:SolidPeso molecular:347.88Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Fórmula:C16H19NOPureza:99.47%Cor e Forma:SolidPeso molecular:241.33Ex26
CAS:<p>Ex26 (S1P1-IN-Ex26) is an S1P1 antagonist used in experimental autoimmune encephalomyelitis, atherosclerosis, and gastric cancer.</p>Fórmula:C28H28ClFN2O3Pureza:99.62%Cor e Forma:SolidPeso molecular:494.99Elinogrel
CAS:<p>Elinogrel (PRT060128) is a competitive and reversible antagonist of platelet P2Y12 with IC50 of 20 nM and exhibits potent antiplatelet effects.</p>Fórmula:C20H15ClFN5O5S2Pureza:98.78%Cor e Forma:SolidPeso molecular:523.95Xamoterol hemifumarate
CAS:<p>Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationship</p>Fórmula:C36H54N6O14Pureza:99.79%Cor e Forma:White SolidPeso molecular:794.37FK-453
CAS:<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Fórmula:C23H25N3O2Pureza:99.44%Cor e Forma:SolidPeso molecular:375.46SLP9101555
<p>SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of 90 nM.SLP9101555 has a high affinity for SphK2, which is 200-fold</p>Fórmula:C16H22BrClN2Pureza:99.45%Cor e Forma:SolidPeso molecular:357.72MLS1547
CAS:<p>MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).</p>Fórmula:C19H19ClN4OPureza:99.64%Cor e Forma:SolidPeso molecular:354.83CYM5181
CAS:<p>CYM5181 is related to the body's immune system and can be used to study multiple sclerosis, transplant rejection, and adult respiratory distress syndrome.</p>Fórmula:C17H17N3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:311.34AZ-1355
CAS:<p>AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.</p>Fórmula:C17H17NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:299.32NP10679
CAS:<p>NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.</p>Fórmula:C23H26F3N3O3Pureza:99.43%Cor e Forma:SolidPeso molecular:449.47Sinitrodil
CAS:<p>Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.</p>Fórmula:C10H10N2O5Pureza:98.98%Cor e Forma:SolidPeso molecular:238.2CB2R PAM
CAS:<p>CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in neuropathic pain relief.</p>Fórmula:C21H24BrFN2O2Pureza:99.09%Cor e Forma:SolidPeso molecular:435.33Molindone
CAS:<p>Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.</p>Fórmula:C16H24N2O2Pureza:99.37% - 99.46%Cor e Forma:Off-White SolidPeso molecular:276.37Dimethindene
CAS:<p>Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.</p>Fórmula:C20H24N2Pureza:98.3% - 98.99%Cor e Forma:SolidPeso molecular:292.42Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Fórmula:C24H22N4Pureza:99.91%Cor e Forma:SolidPeso molecular:366.46LTB4-IN-1
CAS:<p>LTB4-IN-1 (Anti-inflammatory agent 2) with IC50 of 70 nM is an inhibitor of leukotriene synthesis (LTB4).</p>Fórmula:C26H30N2O4SPureza:99.93%Cor e Forma:SolidPeso molecular:466.59Selodenoson
CAS:<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Fórmula:C17H24N6O4Pureza:99.52%Cor e Forma:SolidPeso molecular:376.41Midaglizole hydrochloride
CAS:<p>Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).</p>Fórmula:C16H19Cl2N3Pureza:99.39% - 99.82%Cor e Forma:SolidPeso molecular:324.25OPC-51803
CAS:<p>OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.</p>Fórmula:C26H32ClN3O2Pureza:98.93% - >99.99%Cor e Forma:SolidPeso molecular:454L 651896
CAS:<p>L 651896 is an inhibitor of 5-lipoxygenase.</p>Fórmula:C18H18O3Pureza:96.06% - 99.85%Cor e Forma:SolidPeso molecular:282.33D18024
CAS:<p>D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.</p>Fórmula:C29H31ClFN3OPureza:99.86%Cor e Forma:SolidPeso molecular:492.03GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Fórmula:C28H34Cl2N2OPureza:98.08%Cor e Forma:SolidPeso molecular:485.49E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Fórmula:C17H18ClN5O2S2Pureza:96.32% - 99.53%Cor e Forma:SolidPeso molecular:423.94ORM-10921
CAS:<p>ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.</p>Fórmula:C18H23NO2Pureza:99.46% - 99.85%Cor e Forma:SolidPeso molecular:285.38rel-(1R,2R)-Vesamicol Hydrochloride
CAS:<p>Vesamicol hydrochloride ((±)-AH5183 hydrochloride) is a acetylcholine transport inhibitor.</p>Fórmula:C17H26ClNOPureza:99.88%Cor e Forma:SolidPeso molecular:295.85Opigolix
CAS:<p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>Fórmula:C25H19F3N4O5SPureza:98.60% - 98.97%Cor e Forma:SolidPeso molecular:544.5Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Fórmula:C24H24FN3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:405.46Ronacaleret HCl
CAS:<p>Ronacaleret HCl (SB-751689) is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.</p>Fórmula:C25H32ClF2NO4Pureza:99.97%Cor e Forma:SolidPeso molecular:483.98GW438014A
CAS:<p>GW438014A 是一种有效且具有选择性的 NPY-Y5 受体拮抗剂。GW438014A 对食物摄入并减少肥胖啮齿动物的体重增加具有抑制作用。</p>Fórmula:C23H23N3O4SPureza:99.89%Cor e Forma:SolidPeso molecular:437.51VA-K-14 hydrochloride
CAS:<p>VA-K-14 hydrochloride（VAK14 HCl） is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonal</p>Fórmula:C18H16ClN3SPureza:97.15%Cor e Forma:SolidPeso molecular:341.86Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Fórmula:C20H21N3OPureza:99.82% - 99.98%Cor e Forma:SolidPeso molecular:319.4SB228357
CAS:<p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>Fórmula:C22H17F4N3O2Pureza:99.82%Cor e Forma:SolidPeso molecular:431.38Sarizotan HCl
CAS:<p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>Fórmula:C22H22ClFN2OPureza:96%Cor e Forma:SolidPeso molecular:384.87ISAM-140
CAS:<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Fórmula:C19H19N3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:337.37Teniloxazine
CAS:<p>Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.</p>Fórmula:C16H19NO2SPureza:99.23%Cor e Forma:SolidPeso molecular:289.39Abt-288
CAS:<p>ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.</p>Fórmula:C23H24N4OPureza:98.17% - 98.49%Cor e Forma:SolidPeso molecular:372.46RS 42358-197
CAS:<p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>Fórmula:C19H23ClN2OPureza:99.70%Cor e Forma:SolidPeso molecular:330.85Pirmagrel
CAS:<p>pirmagrel is a potent thromboxane synthase inhibitor.</p>Fórmula:C13H16N2O2Pureza:98.02%Cor e Forma:SolidPeso molecular:232.28Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Fórmula:C13H19NO3Pureza:99.67%Cor e Forma:SolidPeso molecular:237.29Uridine 5'-diphosphate
CAS:<p>Uridine 5'-diphosphate acts as a P2Y6 receptor agonist, exhibiting an EC50 value of 0.013 μM for the human P2Y6 receptor [1].</p>Fórmula:C9H14N2O12P2Pureza:98%Cor e Forma:SolidPeso molecular:404.16L 659837
CAS:<p>L 659837 is an antagonist of ANC-2, lactam, and tackykinin.</p>Fórmula:C40H52N8O7SCor e Forma:SolidPeso molecular:788.96PD 160170
CAS:<p>neuropeptide Y1 receptor antagonist</p>Fórmula:C18H17N3O4SPureza:98%Cor e Forma:SolidPeso molecular:371.41Pecavaptan
CAS:<p>Pecavaptan is a vasopressin receptor antagonist.</p>Fórmula:C22H19Cl2F3N6O3Cor e Forma:SolidPeso molecular:543.33
