GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.943 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(196 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(69 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(164 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5337 produtos de "GPCR/Proteína-G"
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A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Fórmula:C23H25IN4Cor e Forma:SolidPeso molecular:484.38Baloncibart
CAS:<p>Baloncibart is a human IgG4K monoclonal antibody that targets NPR1.</p>Cor e Forma:LiquidLeukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Fórmula:C22H37NO4Cor e Forma:SolidPeso molecular:379.541Amylin (1-37), human acetate
<p>Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.</p>Pureza:96.21%Cor e Forma:Odour SolidCCR6 antagonist 2
<p>CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.</p>Fórmula:C19H24N4O4Cor e Forma:SolidPeso molecular:372.42Neuropeptide S(Rat)
CAS:<p>Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).</p>Fórmula:C95H160N34O27Pureza:98%Cor e Forma:SolidPeso molecular:2210.52Cortistatin-8
CAS:<p>ghrelin receptor antagonist</p>Fórmula:C47H68N12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1009.25K-(D-1-Nal)-FwLL-NH2 TFA
<p>K-(D-1-Nal)-FwLL-NH2 TFA: potent ghrelin inverse agonist; Ki=4.9 nM (COS7), 31 nM (HEK293T); blocks Gq/G13 signaling.</p>Fórmula:C53H68F3N9O8Cor e Forma:SolidPeso molecular:1016.16GLP-1R agonist 14
CAS:<p>GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].</p>Fórmula:C45H42F2N10O5Cor e Forma:SolidPeso molecular:840.88Sulamserod
CAS:<p>Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular related</p>Fórmula:C19H28ClN3O5SPureza:98.76%Cor e Forma:SolidPeso molecular:445.96APJ receptor agonist 1
CAS:<p>Potent APJ-R agonist 1, biphenyl acid, EC50: 0.093 nM (human), 0.12 nM (rat), targets apelin-13, promising for heart failure study.</p>Fórmula:C31H26ClN3O3Cor e Forma:SolidPeso molecular:524.02(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)
CAS:<p>(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14), a bombesin (BBN) antagonist, holds potential for cancer research applications [1].</p>Fórmula:C49H69N13O9Cor e Forma:SolidPeso molecular:984.15Ebiratide
CAS:<p>Ebiratide is an analog of ACTH 4-9.</p>Fórmula:C48H73N11O10SPureza:98%Cor e Forma:SolidPeso molecular:996.23Luseogliflozin hydrate
CAS:<p>Luseogliflozin hydrate: SGLT2 inhibitor, IC50 2.26 nM, oral, for type 2 diabetes research.</p>Fórmula:C23H32O7SCor e Forma:SolidPeso molecular:452.56GB-6
CAS:<p>GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to</p>Fórmula:C32H45N11O8Pureza:98%Cor e Forma:SolidPeso molecular:711.77GR231118
CAS:<p>Potent NPY Y1 antagonist & Y4 agonist; inhibits rat appetite; binds to NPFF receptors (Ki: 43-73 nM).</p>Fórmula:C110H170N34O24Pureza:98%Cor e Forma:Lyophilized PowderPeso molecular:2352.77(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat)
CAS:<p>(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat) is a corticotropin-releasing factor (CRF) antagonist known to counteract the inhibitory effects of IL-1a</p>Fórmula:C159H267N49O43Cor e Forma:SolidPeso molecular:3553.12SB234551
CAS:<p>SB234551 is a selective antagonist of endothelin ETA receptor.</p>Fórmula:C34H34N2O9Cor e Forma:SolidPeso molecular:614.64Femoxetine
CAS:<p>Femoxetine: antidepressant, enhances morphine, inhibits MAO-A/B, boosts mice's exercise capacity.</p>Fórmula:C20H25NO2Pureza:99.1% - 99.35%Cor e Forma:SolidPeso molecular:311.42Bucindolol Formate
<p>Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.</p>Fórmula:C23H27N3O4Pureza:99.76% - 99.88%Cor e Forma:SolidPeso molecular:409.48BAY-747
CAS:<p>BAY-747: oral, brain-penetrant sGC stimulator; improves rat memory, cognition, lowers blood pressure, aids Duchenne muscular dystrophy.</p>Fórmula:C22H26F2N4O2Cor e Forma:SolidPeso molecular:416.46Cenderitide
CAS:<p>Cenderitide fuses CNP with DNP, stimulates pGC-A/B, ups cGMP, curbs aldosterone, and aids GFR, not affecting BP—used in heart failure studies.</p>Fórmula:C158H263N49O50S3Cor e Forma:SolidPeso molecular:3745.27Cortistatin 14, human, rat
CAS:<p>Cortistatin 14: a neuropeptide similar to somatostatin; induces sleep, depresses neuronal activity; found in cortex, hippocampus.</p>Fórmula:C81H113N19O19S2Pureza:98%Cor e Forma:SolidPeso molecular:1721.01ELA-11(human)
CAS:<p>Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.</p>Fórmula:C58H90N16O13S2Pureza:98%Cor e Forma:SolidPeso molecular:1283.57CHS-114
<p>CHS-114 (SRF-114) is a fully human IgG1 antibody targeting the (CCR8) receptor. It shows potential for research in head and neck squamous cell carcinoma (HNSCC). The isotype control for CHS-114 can be referred to as HumanIgG1kappa, Isotype Control.</p>Cor e Forma:Odour LiquidGlucagon-like peptide 1 (1-37), human
CAS:<p>Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.</p>Fórmula:C186H275N51O59Pureza:98%Cor e Forma:SolidPeso molecular:4169.48Petrelintide acetate
<p>Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.</p>Fórmula:C185H305N49O61·xC2H4O2Cor e Forma:SolidPeso molecular:4191.69 (free base)PG 931 acetate
<p>PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.</p>Fórmula:C61H89N15O13Pureza:98.74%Cor e Forma:SolidPeso molecular:1240.45Piperulin A
CAS:<p>Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,</p>Fórmula:C23H28O6Cor e Forma:SolidPeso molecular:400.46HTR2A antagonist 1
<p>HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.</p>Fórmula:C35H43Cl2F2N5O4Cor e Forma:SolidPeso molecular:706.65Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide
<p>Biotin-labeled GLP-1-(7-36) amide; a gut peptide that enhances insulin release.</p>Fórmula:C165H252N44O48SCor e Forma:SolidPeso molecular:3652.1Cetirizine Impurity C
CAS:<p>Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.</p>Fórmula:C21H25ClN2O3Cor e Forma:SolidPeso molecular:388.89Prostaglandin F2α 1,11-lactone
CAS:<p>Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be used in studies about treating glaucoma.</p>Fórmula:C20H32O4Pureza:98%Cor e Forma:SolidPeso molecular:336.47TAK-683 acetate
<p>TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.</p>Fórmula:C66H87N17O15Cor e Forma:SolidPeso molecular:1358.5(Ala13)-Apelin-13 acetate
<p>(Ala13)-Apelin-13 acetate, an APJ antagonist, modulates CRF-induced enhanced colonic motility, visceral sensation, and gut barrier.</p>Fórmula:C65H111N23O18SPureza:98%Cor e Forma:SolidPeso molecular:1534.79HAEGTFTSD acetate(926018-45-3 free base)
<p>HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from</p>Fórmula:C42H61N11O19Pureza:98%Cor e Forma:SolidPeso molecular:1024.01Selepressin acetate
<p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>Fórmula:C48H77N13O13S2Cor e Forma:SolidPeso molecular:1108.33Peptide YY (pig)
CAS:<p>Peptide YY (pig), a 36 amino acid gut peptide from porcine duodenum, reduces appetite via Y2 receptor, affecting digestion and the heart.</p>Fórmula:C190H288N54O57Cor e Forma:SolidPeso molecular:4240.72Dotanoc
CAS:<p>Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.</p>Fórmula:C69H94N14O17S2Cor e Forma:SolidPeso molecular:1455.71JNJ-5207787
CAS:<p>JNJ-5207787, a blood-brain barrier-crossing Y2 receptor antagonist, is >100x selective against Y1/Y4/Y5 and inhibits human/rat Y2 with pIC50s of 7.0/7.1.</p>Fórmula:C32H38N4O2Pureza:98%Cor e Forma:SolidPeso molecular:510.67[Des-His1,Glu9]-Glucagon amide
CAS:<p>Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.</p>Fórmula:C148H221N41O47SPureza:98%Cor e Forma:SolidPeso molecular:3358.68PAR-4 Agonist Peptide, amide
CAS:<p>PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).</p>Fórmula:C34H48N8O7Pureza:98%Cor e Forma:SolidPeso molecular:680.79Kinetensin
CAS:<p>Kinetensin is a neurotensin-like peptide.</p>Fórmula:C56H85N17O11Pureza:98%Cor e Forma:White Lyophilised SolidPeso molecular:1172.38Pancreatic Polypeptide, bovine
CAS:<p>Agonist at Y4 neuropeptide Y receptors.</p>Fórmula:C186H287N53O56S2Pureza:98%Cor e Forma:SolidPeso molecular:4225.78PG-931 TFA
<p>PG-931 TFA, a potent MC4 receptor agonist (IC50 0.58 nM), excels in selectivity and helps reverse hemorrhagic shock in vivo.</p>Fórmula:C61H86F3N15O13Cor e Forma:SolidPeso molecular:1294.42Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Fórmula:C45H47N7O9S3Cor e Forma:SolidPeso molecular:926.09AC-263093
CAS:<p>AC-263093 is an NPFFR2 agonist with anxiolytic activity that increases c-Fos protein expression in the paraventricular nucleus of the hypothalamus.</p>Fórmula:C8H8Br2N4Pureza:99.78%Cor e Forma:SoildPeso molecular:319.98Tryptamine hydrochloride
CAS:<p>Tryptamine hydrochloride is a monoamine alkaloid, metabolite of tryptophan and CNS active substance, agonist of 5-HT4 receptor, TAAR1, AHR.</p>Fórmula:C10H13ClN2Pureza:99.89%Cor e Forma:SolidPeso molecular:196.68I-BOP
CAS:<p>I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).</p>Fórmula:C23H29IO5Cor e Forma:SolidPeso molecular:512.384[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS:<p>'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.</p>Fórmula:C39H64N8O10Cor e Forma:SolidPeso molecular:804.9712(S)-HpEPE
CAS:<p>12(S)-HpEPE, a fatty acid created by 12-lipoxygenase on EPA, has unclear biological activities but may resemble 12(S)-HpETE.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Fórmula:C47H67N11O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1026.2PACAP (1-27), human, ovine, rat
CAS:<p>PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.</p>Fórmula:C142H224N40O39SPureza:98%Cor e Forma:SolidPeso molecular:3147.66RFRP-1(human)
CAS:<p>Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.</p>Fórmula:C67H101N19O14SPureza:98%Cor e Forma:SolidPeso molecular:1428.72Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Fórmula:C18H20ClNO4Cor e Forma:SolidPeso molecular:349.81Guanylin TFA (mouse,rat)
<p>Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.</p>Fórmula:C60H90N16O22S4·xC2HF3O2Cor e Forma:SolidPeso molecular:1515.71 (free base)Methicillin sodium hydrate
CAS:<p>Methicillin sodium hydrate, a narrow-spectrum antibiotic, combats methicillin-resistant Staphylococcus strains and treats various infections.</p>Fórmula:C17H21N2NaO7SCor e Forma:SolidPeso molecular:420.41CB2R probe 1
CAS:<p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>Fórmula:C36H42N4O4Cor e Forma:SolidPeso molecular:594.746α-Prostaglandin I1
CAS:<p>6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.</p>Fórmula:C20H34O5Cor e Forma:SolidPeso molecular:354.48717-phenoxy trinor Prostaglandin F2α ethyl amide
CAS:<p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>Fórmula:C25H37NO5Cor e Forma:SolidPeso molecular:431.573Adrenomedullin (16-31), human TFA
<p>Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.</p>Fórmula:C84H130F3N25O23S2Cor e Forma:SolidPeso molecular:1979.21GHRF, bovine
CAS:<p>bGRF(1-44)-NH2 is a bovine GH-releasing factor that stimulates GH release and synergizes with Hydrocortisone.</p>Fórmula:C220H366N72O66SCor e Forma:SolidPeso molecular:5104.72Nolomirole
CAS:<p>Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.</p>Fórmula:C19H27NO4Cor e Forma:SolidPeso molecular:333.42Tafluprost acid
CAS:<p>Tafluprost acid is a selective agonist at the prostaglandin F receptor.</p>Fórmula:C22H28F2O5Cor e Forma:SolidPeso molecular:410.46[bAla8]-Neurokinin A(4-10)
CAS:<p>[bAla8]-Neurokinin A(4-10) is a neurokinin 2 (NK2) receptor agonist.</p>Fórmula:C35H56N8O10SPureza:98%Cor e Forma:SolidPeso molecular:780.94B-Raf IN 14
CAS:<p>B-Raf IN 14 is a BRAF inhibitor.</p>Fórmula:C15H14BrN5O3SPureza:98.32%Cor e Forma:SolidPeso molecular:424.27Urocortin III (human)
CAS:<p>Urocortin III, a human peptide, binds CRF-R2, affecting insulin via somatostatin feedback with K i values 13.5-100+ nM.</p>Fórmula:C185H307N53O50S2Cor e Forma:SolidPeso molecular:4137.93Thiothixene
CAS:<p>Thiothixene has a wide range of applications in life science related research.</p>Fórmula:C23H29N3O2S2Cor e Forma:SolidPeso molecular:443.62PG106 TFA
<p>PG106 TFA is a potent hMC3 antagonist (IC50=210 nM), inactive at hMC4 (EC50=9900 nM) and hMC5 receptors.</p>Fórmula:C53H70F3N13O11Cor e Forma:SolidPeso molecular:1122.2Mosapride citrate dihydrate
CAS:<p>Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.</p>Fórmula:C27H35ClFN3O11Pureza:98%Cor e Forma:SolidPeso molecular:632.04Ro 25-1553
CAS:<p>Ro 25-1553 is a 31-amino acid analog of vasoactive intestinal peptide (VIP) that functions as an agonist for the VIP2 receptor (VPAC2 receptor). In guinea pig models, Ro 25-1553 exhibits bronchodilator effects on tracheal smooth muscle contraction induced by neural stimuli or Carbachol.</p>Fórmula:C160H258N46O46Cor e Forma:SolidPeso molecular:3562.04Teprotumumab
CAS:<p>Teprotumumab: human antibody, inhibits IGF-1R, used for thyroid eye diseases.</p>Pureza:SDS-PAGE:95.2%;SEC-HPLC:99.6%Cor e Forma:LiquidPeso molecular:145.62 kDaKhusimol
CAS:<p>Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.</p>Fórmula:C15H24OPureza:98%Cor e Forma:SolidPeso molecular:220.35NTRC-824
CAS:<p>NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.</p>Fórmula:C25H26F3N3O6SPureza:98%Cor e Forma:SolidPeso molecular:553.55DETQ
CAS:<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Fórmula:C22H25Cl2NO3Cor e Forma:SolidPeso molecular:422.34Adrenomedullin (16-31), human
CAS:<p>Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).</p>Fórmula:C82H129N25O21S2Pureza:98%Cor e Forma:SolidPeso molecular:1865.19Ecnoglutide
CAS:<p>Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .</p>Fórmula:C194H304N48O61Cor e Forma:SolidPeso molecular:4284.76Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Fórmula:C25H31F3N6O8Pureza:98.08%Cor e Forma:SoildPeso molecular:600.55Ono 3708
CAS:<p>Ono-3708 is a potent antagonist of the thromboxane A2/prostaglandin endoperoxide receptor in vitro and in vivo.</p>Fórmula:C23H37NO4Pureza:98%Cor e Forma:SolidPeso molecular:391.54Brexpiprazole S-oxide
CAS:<p>Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).</p>Fórmula:C25H27N3O3SPureza:98%Cor e Forma:SolidPeso molecular:449.57Cetirizine methyl ester
CAS:<p>Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.</p>Fórmula:C22H27ClN2O3Cor e Forma:SolidPeso molecular:402.91TT-OAD2 free base
CAS:<p>TT-OAD2 free base, a non-peptide GLP-1 receptor agonist, can treat diabetes; has an EC50 of 5 nM.</p>Fórmula:C50H47Cl2N3O6Pureza:98%Cor e Forma:SolidPeso molecular:856.83Guanylate cyclase-IN-1
CAS:<p>Guanylate cyclase-IN-1 (Example 46) is a specific inhibitor of guanylate cyclase, employed in research related to cardiovascular diseases.</p>Fórmula:C20H17FN8OCor e Forma:SolidPeso molecular:404.409Neuropeptide Y 13-36 (porcine)
CAS:<p>Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.</p>Fórmula:C135H209N41O36Cor e Forma:SolidPeso molecular:2982.408Hemopressin (human, mouse)
CAS:<p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>Fórmula:C50H79N13O12Pureza:98%Cor e Forma:SolidPeso molecular:1054.26Clomipramine D3
CAS:<p>Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).</p>Fórmula:C19H23ClN2Pureza:98%Cor e Forma:SolidPeso molecular:317.87Alcaftadine carboxylic acid
CAS:<p>Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.</p>Fórmula:C19H21N3O2Cor e Forma:SolidPeso molecular:323.39Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Fórmula:C86H115FN16O21Cor e Forma:SolidPeso molecular:1727.93(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:<p>V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.</p>Fórmula:C52H74N14O12S2Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:1151.38LUF6096
CAS:<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Fórmula:C22H21Cl2N3OPureza:99.5%Cor e Forma:SolidPeso molecular:414.33Cholecystokinin Octapeptide, desulfated
CAS:<p>Cholecystokinin Octapeptide, desulfated (CCK Octapeptide, non-sulfated) is an octapeptide composed of 8 amino acids from cholecystokinin-8.</p>Fórmula:C49H62N10O13S2Pureza:97.12%Cor e Forma:SolidPeso molecular:1063.21Men 10208
CAS:<p>Men 10208 is an antagonist of the neurokinin A receptor.</p>Fórmula:C61H75N15O12Pureza:98%Cor e Forma:SolidPeso molecular:1210.36Pobilukast
CAS:<p>Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.</p>Fórmula:C26H34O5SPureza:99.65% - 99.84%Cor e Forma:SolidPeso molecular:458.61Dulaglutide
CAS:<p>Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).</p>Cor e Forma:SolidGW-328267
CAS:<p>GW-328267 is an agonist of the adenosine A2 receptor.</p>Fórmula:C21H26N10O4Cor e Forma:SolidPeso molecular:482.5Benzomalvin B
CAS:<p>Benzomalvin B, a metabolite from Penicillium, blocks 24% NK1 receptor binding at 100 μg/ml.</p>Fórmula:C24H17N3O2Cor e Forma:SolidPeso molecular:379.41917-trifluoromethylphenyl trinor Prostaglandin F2α ethyl amide
CAS:<p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>Fórmula:C26H36F3NO4Cor e Forma:SolidPeso molecular:483.572GLP-1R Antagonist 1
CAS:<p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>Fórmula:C16H11ClF6N4O2Pureza:99.84%Cor e Forma:SolidPeso molecular:440.73Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:<p>CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.</p>Fórmula:C163H267N51O50S2Pureza:98%Cor e Forma:SolidPeso molecular:3805.31Metaterol
CAS:<p>Metaterol is a bioactive chemical.</p>Fórmula:C11H17NO2Cor e Forma:SolidPeso molecular:195.2582Carazolol-d7
CAS:<p>Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.</p>Fórmula:C18H22N2O2Cor e Forma:SolidPeso molecular:305.42Nocistatin(human)
CAS:<p>Blocker of nociceptin-induced allodynia and hyperalgesia</p>Fórmula:C149H238N42O53S3Pureza:98%Cor e Forma:SolidPeso molecular:3561.93LY 293284
CAS:<p>LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.</p>Fórmula:C19H26N2OCor e Forma:SolidPeso molecular:298.4217-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:<p>Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.</p>Fórmula:C27H39NO4Cor e Forma:SolidPeso molecular:441.612Prosaptide TX14(A)
CAS:<p>GPR37L1/GPR37 agonist with EC50 of 5/7 nM, activates G proteins, enhances ERK, myelin synthesis, neuro/glioprotection.</p>Fórmula:C69H110N16O26Pureza:98%Cor e Forma:SolidPeso molecular:1579.72Orexin B, rat, mouse TFA
<p>Orexin B, rat/mouse TFA, activates OX1-R & OX2-R receptors, influencing food intake, energy, and sleep regulation.</p>Fórmula:C128H216F3N45O36SCor e Forma:SolidPeso molecular:3050.42Fpl 14294
CAS:<p>Fpl 14294 is a novel CCK-8 agonist with effective intranasal anorectic activity in the rat.</p>Fórmula:C45H56N8O13S3Pureza:98%Cor e Forma:SolidPeso molecular:1013.17Naratriptan D3 Hydrochloride
CAS:<p>Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.</p>Fórmula:C17H26ClN3O2SPureza:98%Cor e Forma:SolidPeso molecular:374.94Ularitide
CAS:<p>Ularitide is a 32-amino acid peptide from ANP prohormone, resistant to dog kidney cortex peptidase.</p>Fórmula:C145H234N52O44S3Pureza:98%Cor e Forma:SolidPeso molecular:3505.97LY 344864 racemate
CAS:<p>LY 344864 racemate is a 5-HT1F receptor agonist.</p>Fórmula:C21H22FN3OPureza:99.75%Cor e Forma:SoildPeso molecular:351.42Mirtazapine N-oxide
CAS:<p>Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.</p>Fórmula:C17H19N3OCor e Forma:SolidPeso molecular:281.359Brain Natriuretic Peptide-45, rat
CAS:<p>BNP-45 (rat) is a circulating form of rat brain natriuretic peptide isolated from rat heart with potent hypotensive and natriuretic potency.</p>Fórmula:C213H349N71O65S3Pureza:98%Cor e Forma:SolidPeso molecular:5040.67(+)-5-trans Cloprostenol
CAS:<p>Cloprostenol, a synthetic PGF2α derivative, induces estrus and treats reproductive issues in livestock; its minor impurity, (+)-5-trans, is less effective.</p>Fórmula:C22H29ClO6Cor e Forma:SolidPeso molecular:424.92Neuropeptide Y(29-64)
CAS:<p>Neuropeptide Y(29-64) is a 36 amino acid peptide, a fragment of Neuropeptide Y.</p>Fórmula:C189H284N54O58SPureza:98%Cor e Forma:SolidPeso molecular:4272.7Orforglipron hemicalcium hydrate
CAS:<p>Orforglipron hemicalcium hydrate (LY3502970 hemicalcium hydrate; GLP-1 receptor agonist 1 hemicalcium hydrate) represents the hemicalcium hydrate form of the calcium salt of Orforglipron, an orally active agonist targeting the Glucagon-like peptide-1 receptor (GLP-1R). This compound has demonstrated efficacy in mitigating type 2 diabetes [1].</p>Fórmula:C48H48F2N10O5Ca·H2OCor e Forma:SolidPeso molecular:921.02Mitemcinal fumarate
CAS:<p>Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.</p>Fórmula:C84H142N2O28Cor e Forma:SolidPeso molecular:1628.02Sorbinicate
CAS:<p>Sorbinicate is an antihypercholesterolaemic and vasodilating nicotinic acid ester.</p>Fórmula:C42H32N6O12Pureza:98%Cor e Forma:SolidPeso molecular:812.74Pellotine
CAS:<p>Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.</p>Fórmula:C13H19NO3Cor e Forma:SolidPeso molecular:237.295Suntinorexton
CAS:<p>Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.</p>Fórmula:C23H28F2N2O4SPureza:99.89%Cor e Forma:SolidPeso molecular:466.54CRL-42872 free base
CAS:<p>CRL-42872 free base is a bioactive chemical.</p>Fórmula:C22H26N6O6SCor e Forma:SolidPeso molecular:502.54ACTH (34-39)
CAS:ACTH (34-39) is an adrenocorticotropic hormone fragment.Fórmula:C37H50N6O9Pureza:98%Cor e Forma:SolidPeso molecular:722.83Elabela(19-32)
CAS:<p>APJ receptor agonist with Ki of 0.93 nM, derived from ELA-32, activates Gαi1, β-arrestin-2, lowers rat heart arterial pressure, effective in vivo.</p>Fórmula:C75H119N25O17S2Pureza:98%Cor e Forma:SolidPeso molecular:1707.03Firazorexton
CAS:<p>Firazorexton is a potent orexin type 2 receptor (OX2R) agonist.</p>Fórmula:C22H25F3N2O4SCor e Forma:SolidPeso molecular:470.51Mapenterol hydrochloride
CAS:<p>Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.</p>Fórmula:C14H21Cl2F3N2OPureza:98.11% - 99.98%Cor e Forma:SolidPeso molecular:361.23Luseogliflozin
CAS:<p>Luseogliflozin inhibits SGLT2 for glucose uptake with 1.10 nM potency.</p>Fórmula:C23H30O6SCor e Forma:SolidPeso molecular:434.55Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Fórmula:C161H274N48O46SPureza:98%Cor e Forma:SolidPeso molecular:3650.29ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate
CAS:<p>ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate is a platelet aggregation inhibitor.</p>Fórmula:C22H18N4O3Pureza:99.86%Cor e Forma:SolidPeso molecular:386.4Mabuterol free base
CAS:<p>Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.</p>Fórmula:C13H18ClF3N2OPureza:98%Cor e Forma:SolidPeso molecular:310.74(Iso)-Landipirdine
CAS:<p>(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.</p>Fórmula:C18H19FN2O3SPureza:98.50%Cor e Forma:SoildPeso molecular:362.42Neuropeptide FF
CAS:<p>Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).</p>Fórmula:C54H76N14O10Pureza:98%Cor e Forma:SolidPeso molecular:1081.27AMTG-DA1
<p>AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.</p>Fórmula:C101H149IN22O25Cor e Forma:SolidPeso molecular:2197.0109β-MSH, human
CAS:<p>beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).</p>Fórmula:C118H174N34O35SPureza:98%Cor e Forma:SolidPeso molecular:2660.924-P-PDOT
CAS:<p>4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.</p>Fórmula:C19H21NOPureza:99.91%Cor e Forma:SolidPeso molecular:279.38PY-60
CAS:<p>PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.</p>Fórmula:C16H15N3O2SPureza:99.5% - 99.67%Cor e Forma:SolidPeso molecular:313.37Pasireotide
CAS:<p>Pasireotide (SOM 230) is a cyclohexapeptide, mimicking somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).</p>Fórmula:C58H66N10O9Pureza:98%Cor e Forma:SolidPeso molecular:1047.21M1145
CAS:<p>Potent GAL2 agonist with EC50 = 38 nM; Ki: 6.55 nM (GAL2), 497 nM (GAL3), 587 nM (GAL1); enhances galanin signaling.</p>Fórmula:C128H205N37O32Pureza:98%Cor e Forma:SolidPeso molecular:2774.26PD-149164
CAS:<p>PD-149164 is an agonist of the CCK-A receptor.</p>Fórmula:C33H38FN3O5Cor e Forma:SolidPeso molecular:575.67GHRF, porcine
CAS:<p>GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing the</p>Fórmula:C219H365N73O66SCor e Forma:SolidPeso molecular:5108.76CB1R antagonist 2
<p>CB1R antagonist 2 (Compound 11g) functions as an antagonist of the cannabinoid receptor 1 (CB1R), inhibiting the MAPK/NF-κB signaling pathway and exhibiting anti-inflammatory properties. In RAW264.7 cells, it suppresses LPS-induced expression of IL-6, IL-1β, and TNF-α. In murine models, it improves OVA-induced allergic rhinitis.</p>Fórmula:C24H26N4OCor e Forma:SolidPeso molecular:386.4915(R)-17-phenyl trinor Prostaglandin F2α
CAS:<p>17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocular</p>Fórmula:C23H32O5Cor e Forma:SolidPeso molecular:388.5MM 419447
CAS:<p>MM 419447, a linaclotide metabolite, is a guanylate cyclase-C agonist showing potential in IBS-C research.</p>Fórmula:C50H70N14O19S6Cor e Forma:SolidPeso molecular:1363.55Tebufelone
CAS:<p>Tebufelone is a potent NSAID, inhibits CO, has anti-inflammatory and analgesic properties, and blocks lipoxygenase products (IC50 ~20-22 microM).</p>Fórmula:C20H28O2Pureza:99.32%Cor e Forma:SolidPeso molecular:300.44dCNP
<p>dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.</p>Fórmula:C141H248N38O36S3Cor e Forma:SolidPeso molecular:3147.91Parstatin(mouse)
CAS:<p>Peptide inhibits endothelial migration/proliferation (IC50 ~20μM), induces cell cycle arrest, triggers apoptosis, and has cardioprotective effects.</p>Fórmula:C189H326N58O57S3Pureza:98%Cor e Forma:SolidPeso molecular:4419.19IRAK inhibitor 4 trans
<p>IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.</p>Fórmula:C33H35F3N6O3Pureza:98%Cor e Forma:SolidPeso molecular:620.66Urocortin, rat
CAS:<p>Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.</p>Fórmula:C206H338N62O64Pureza:98%Cor e Forma:SolidPeso molecular:4707.26Prostaglandin J2
CAS:<p>PGJ2, a PGD2 metabolite, is a DP agonist (Ki: 0.9 nM hDP, 6.6 nM hCRTH2), induces cAMP (EC50: 1.2 nM), oxidative stress, neuronal apoptosis, and neurotoxicity.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.45Vedaprofen
CAS:<p>Vedaprofen (PM 150) is a COX-1 inhibitor with anti-inflammatory effects, blocking E. coli clamp at IC50 222 μM, Ki 131 μM.</p>Fórmula:C19H22O2Pureza:99.24% - 99.70%Cor e Forma:SolidPeso molecular:282.3817-phenyl trinor Prostaglandin E2 ethyl amide
CAS:<p>17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.</p>Fórmula:C25H35NO4Cor e Forma:SolidPeso molecular:413.55Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:<p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>Fórmula:C47H66N12O11Pureza:98%Cor e Forma:SolidPeso molecular:975.11Acetyl-Amylin (8-37) (human)
CAS:<p>Acetyl-Amylin (8-37) (human) is a specific amylin antagonist [1] .</p>Fórmula:C140H218N42O46Cor e Forma:SolidPeso molecular:3225.48Hydroxybupropion
CAS:<p>Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).</p>Fórmula:C13H18ClNO2Pureza:99.73%Cor e Forma:Off-White SolidPeso molecular:255.74Neuropeptide Y (18-36) (porcine)
CAS:<p>"Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."</p>Fórmula:C112H174N36O27Cor e Forma:SolidPeso molecular:2456.8SR142948A
CAS:<p>SR142948A is a selective and reversible non-peptide neurotensin receptor antagonist blocking hypothermia and analgesic effects, NMDA-induced dopamine release.</p>Fórmula:C39H52ClN5O6Pureza:98%Cor e Forma:SolidPeso molecular:722.31Gastrin I, rat
CAS:<p>Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.</p>Fórmula:C94H128N22O31S2Cor e Forma:SolidPeso molecular:2126.3SHU 9119
CAS:<p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>Fórmula:C54H71N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1074.258TDI-10229
CAS:<p>TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.</p>Fórmula:C16H16ClN5Pureza:99.85% - 99.89%Cor e Forma:SoildPeso molecular:313.78Parstatin(human) TFA
<p>Parstatin(human) TFA, a cell-penetrating PAR-1 thrombin receptor agonist peptide, effectively inhibits angiogenesis, as indicated by studies [1] [2].</p>Fórmula:C193H331F3N64O55S3Cor e Forma:SolidPeso molecular:4581.28Parstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Fórmula:C191H330N64O53S3Pureza:98%Cor e Forma:SolidPeso molecular:4467.29MGV354
<p>MGV354 is a soluble activator of guanylate cyclase(sGC) with EC 50 s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively [1] [2].</p>Fórmula:C35H37N5O3Pureza:98%Cor e Forma:SolidPeso molecular:575.7Neuropeptide Y (3-36) (porcine)
CAS:<p>Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.</p>Fórmula:C176H271N53O54Cor e Forma:SolidPeso molecular:3993.36Senktide TFA
<p>Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.</p>Cor e Forma:Odour SolidLEK 8804
CAS:<p>LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.</p>Fórmula:C19H19N3OCor e Forma:SolidPeso molecular:305.37Dehydro Aripiprazole (hydrochloride)
CAS:<p>Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.</p>Fórmula:C23H26Cl3N3O2Cor e Forma:SolidPeso molecular:482.83Amylin, amide, rat
CAS:<p>Amylin: peptide, 50% similar to CGRP, found with somatostatin in stomach cells, reduces acid secretion in mice.</p>Fórmula:C167H272N52O53S2Pureza:99.92%Cor e Forma:SolidPeso molecular:3920.44Atilmotin
CAS:<p>Atilmotin is a gastrointestinal agent for treating motility disorders.</p>Fórmula:C86H135N20O19Cor e Forma:SolidPeso molecular:1753.146(R)-Preclamol hydrochloride
CAS:<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Fórmula:C14H22ClNOCor e Forma:SolidPeso molecular:255.78HL2-m5
CAS:<p>HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.</p>Fórmula:C70H101N15O24S3Cor e Forma:SolidPeso molecular:1632.83MRS2500 tetraammonium
CAS:<p>Highly potent and selective antagonist of the platelet P2Y1 receptor</p>Fórmula:C13H21IN6O8P2Pureza:98%Cor e Forma:SolidPeso molecular:578.19α-Helical CRF(9-41) TFA
<p>α-Helical CRF(9-41) TFA acts as a competitive antagonist for the CRF2 receptor, possessing a binding constant (K B) of approximately 100 nM.</p>Fórmula:C168H275F3N46O55S2Cor e Forma:SolidPeso molecular:3940.42Pramlintide TFA
<p>Pramlintide TFA, a polypeptide analogue of human amylin and an antidiabetic agent, exhibits antineoplastic properties in colorectal cancer [1].</p>Fórmula:C173H268N51F3O55S2Cor e Forma:SolidPeso molecular:4063.4Clopidogrel-related Compound B hydrochloride
CAS:<p>Clopidogrel Related Compound B is a useful organic compound for research related to life sciences.</p>Fórmula:C16H17Cl2NO2SCor e Forma:SolidPeso molecular:358.28RWJ 676070
CAS:<p>RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.</p>Fórmula:C30H26ClFN2O5Cor e Forma:SolidPeso molecular:548.99Neuropeptide Y (2-36) (porcine)
CAS:<p>Porcine Neuropeptide Y (2-36) is 97.14% similar to rat/human, an agonist for Y5, Y2, Y1 receptors, used in obesity research.</p>Fórmula:C181H278N54O55Cor e Forma:SolidPeso molecular:4090.47Substance P(1-7)
CAS:<p>Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.</p>Fórmula:C41H65N13O10Pureza:98%Cor e Forma:SolidPeso molecular:900.04Sphinganine 1-phosphate
CAS:<p>Sphinganine 1-phosphate has protects kidney and liver through activation of the S1P1 receptor in mice and acts as an agonist for S1P4 in Homo sapien.</p>Fórmula:C18H40NO5PCor e Forma:SolidPeso molecular:381.49Misoprostol acid
CAS:<p>Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.</p>Fórmula:C21H36O5Pureza:98%Cor e Forma:SolidPeso molecular:368.51LY-53857 free base
CAS:<p>LY-53857 free base is a bioactive chemical.</p>Fórmula:C23H32N2O3Cor e Forma:SolidPeso molecular:384.51Wy 43657
CAS:<p>Wy 43657 is a gonadorelin antagonist.</p>Fórmula:C71H86N14O13Pureza:98%Cor e Forma:SolidPeso molecular:1343.554APTAA-LHRH
CAS:<p>APTAA-LHRH is a gonadorelin antagonist.</p>Fórmula:C69H91Cl2N17O14Pureza:98%Cor e Forma:SolidPeso molecular:1453.47Roxatidine
CAS:<p>Roxatidine, a metabolite of Roxatidine acetate, is a H2-receptor antagonist that prevents ulcers and has anti-inflammatory properties.</p>Fórmula:C17H26N2O3Cor e Forma:SolidPeso molecular:306.4Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:<p>Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.</p>Fórmula:C161H240N46O41S2Cor e Forma:SolidPeso molecular:3540.09Synephrine hemitartrate
CAS:<p>Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.</p>Fórmula:C9H13NO2C4H6O6Cor e Forma:SolidPeso molecular:242.26Lys-[Des-Arg9]Bradykinin
CAS:<p>Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.</p>Fórmula:C50H73N13O11Pureza:98%Cor e Forma:SolidPeso molecular:1032.21FXR/TGR5 agonist 1
CAS:<p>FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.</p>Fórmula:C31H32ClN3O3Cor e Forma:SolidPeso molecular:530.07Antibacterial agent 189
<p>Antibacterialagent 189 (compound 3a) is a potent antibacterial agent with high binding affinity to the target proteins OMPA/exo-1,3-β-glucanase. It demonstrates effective antibacterial activity against Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Candida albicans, and Aspergillus flavus. Additionally, Antibacterialagent 189 exhibits strong binding affinity to the target proteins SMO and SUFU/GLI-1.</p>Fórmula:C37H28N4OPeso molecular:544.22631tetranor-PGJM
CAS:<p>Tetranor-PGJM is a metabolite of prostaglandin D2 and is associated with the anti-inflammatory effects of curcumin.</p>Fórmula:C16H22O6Cor e Forma:SolidPeso molecular:310.346Prostaglandin F1α
CAS:<p>Prostaglandin F1α (PGF1α) is a lipid mediator and an endogenous metabolite of prostacyclin, regulate smooth muscle contraction.</p>Fórmula:C20H36O5Cor e Forma:SolidPeso molecular:356.5Adenosine 3'-monophosphate (sodium salt hydrate)
<p>Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.</p>Fórmula:C10H15N5NaO8PCor e Forma:SolidPeso molecular:387.22AGN 191976
CAS:<p>AGN 191976 is a novel thromboxane A2-mimetic.</p>Fórmula:C21H32O6Cor e Forma:SolidPeso molecular:380.481Galanin (1-30), human
CAS:<p>Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.</p>Fórmula:C139H210N42O43Pureza:98%Cor e Forma:SolidPeso molecular:3157.46Exendin-3/4 (59-86)
<p>Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.</p>Fórmula:NAPureza:98%Cor e Forma:SolidPeso molecular:3055.49SYD5115
<p>SYD5115 is an orally active TSH-R antagonist.</p>Fórmula:C22H32F2N4O3Peso molecular:438.244258-iso Prostaglandin E1
CAS:<p>8-iso Prostaglandin E1 causes spasm in the pulmonary veins of dogs and also acts as a vasodilator.</p>Fórmula:C20H34O5Cor e Forma:Light Yellow Crystalline SolidPeso molecular:354.48(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Fórmula:C22H24ClF4N5OSPureza:98.36%Cor e Forma:SoildPeso molecular:517.97Glucagon-like peptide 1 (1-37), human TFA
<p>Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.</p>Fórmula:C188H276N51F3O61Pureza:98%Cor e Forma:SolidPeso molecular:4283.5PACAP-Related Peptide (PRP), human
<p>PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.</p>Fórmula:C139H229N41O42Pureza:98%Cor e Forma:SolidPeso molecular:3146.57[Nle11]-Substance P
CAS:<p>'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'</p>Fórmula:C64H100N18O13Pureza:98%Cor e Forma:SolidPeso molecular:1329.5915(S)-15-methyl Prostaglandin E2
CAS:<p>15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.</p>Fórmula:C21H34O5Cor e Forma:SolidPeso molecular:366.49Somatostatin 1-28 acetate
<p>Somatostatin 1-28 acetate circulates in human plasma.</p>Pureza:99.22%Cor e Forma:Soild
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