GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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Urocortin II, human TFA
<p>hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.</p>Fórmula:C196H340F3N63O56SPureza:98%Cor e Forma:SolidPeso molecular:4564.3Terazosin dimer impurity dihydrochloride
CAS:<p>Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.</p>Fórmula:C24H30Cl2N8O4Cor e Forma:SolidPeso molecular:565.46Azaline
CAS:<p>Azaline is a gonadorelin antagonist.</p>Fórmula:C74H106ClN23O12Pureza:98%Cor e Forma:SolidPeso molecular:1545.26SphK1&2-IN-1
CAS:<p>SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.</p>Fórmula:C14H14N2O3SPureza:99.59%Cor e Forma:SolidPeso molecular:290.34GRK2i
CAS:GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.Fórmula:C153H256N50O41SPureza:98%Cor e Forma:SolidPeso molecular:3484.08ACTH (34-39)
CAS:ACTH (34-39) is an adrenocorticotropic hormone fragment.Fórmula:C37H50N6O9Pureza:98%Cor e Forma:SolidPeso molecular:722.83Samelisant
CAS:<p>Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.</p>Fórmula:C21H31N3O3Pureza:99.59%Cor e Forma:SolidPeso molecular:373.49AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Fórmula:C21H25N5Cor e Forma:SolidPeso molecular:347.211Motilin, canine
CAS:<p>Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.</p>Fórmula:C120H194N36O34Pureza:98%Cor e Forma:SolidPeso molecular:2685.05human GALP (3-32)
<p>Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), as</p>Fórmula:C137H213N43O38SPureza:98%Cor e Forma:SolidPeso molecular:3102.49Tocrifluor T1117
CAS:<p>Fluorescent form of AM 251, CB1 receptor antagonist</p>Fórmula:C56H53Cl2N7O5Pureza:98%Cor e Forma:SolidPeso molecular:974.975-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFórmula:C17H22Cl2N6SPureza:98%Cor e Forma:SolidPeso molecular:413.37Teprotumumab
CAS:<p>Teprotumumab: human antibody, inhibits IGF-1R, used for thyroid eye diseases.</p>Pureza:SDS-PAGE:95.2%;SEC-HPLC:99.6%Cor e Forma:LiquidPeso molecular:145.62 kDa(Hyp³)-Bradykinin acetate
<p>(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.</p>Fórmula:C52H77N15O14Pureza:99.46%Cor e Forma:SolidPeso molecular:1136.26Prolactin-Releasing Peptide (12-31), rat
CAS:Prolactin-Releasing Peptide (12-31), rat, a fragment of PrRP, exhibits high affinity for GPR10 receptors and stimulates calcium mobilization in CHOK1 cellsFórmula:C104H158N32O26Peso molecular:2272.57AC-264613
CAS:<p>AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5.</p>Fórmula:C19H18BrN3O2Pureza:98%Cor e Forma:SolidPeso molecular:400.28Israpafant
CAS:<p>Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.</p>Fórmula:C28H29ClN4SCor e Forma:SolidPeso molecular:489.07Neuropeptide Y (1-24) (human)
CAS:Neuropeptide Y (1-24) inhibits rat vas deferens twitch and activates NMDA-induced neurons in rat hippocampus.Fórmula:C116H170N30O40SPeso molecular:2656.83PF-4363467
CAS:<p>PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.</p>Fórmula:C22H30N2O3SCor e Forma:SolidPeso molecular:402.55CB2R/FAAH modulator-3
CAS:<p>CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.</p>Fórmula:C22H31NO2Pureza:99.81%Cor e Forma:SoildPeso molecular:341.49Litoxetine HCl
<p>Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.</p>Fórmula:C16H20ClNOPureza:99.56% - 99.75%Cor e Forma:SoildPeso molecular:277.79(D-Ala2)-GRF (1-29) amide (human)
CAS:(D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-Fórmula:C149H246N44O42SPeso molecular:3357.88Maridebart
CAS:<p>Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].</p>Cor e Forma:Liquid[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Fórmula:C54H71N15O14Pureza:98%Cor e Forma:SolidPeso molecular:1154.23Sarafotoxin S6c
CAS:<p>Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).</p>Fórmula:C103H147N27O37S5Pureza:98%Cor e Forma:SolidPeso molecular:2516Setmelanotide Acetate(920014-72-8 free base)
CAS:<p>Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM</p>Fórmula:C51H72N18O11S2Pureza:99.71%Cor e Forma:SolidPeso molecular:1177.35Tezusomant
CAS:Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Fórmula:C120H171N23O32SCor e Forma:SolidPeso molecular:2479.84Cetirizine Impurity C
CAS:<p>Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.</p>Fórmula:C21H25ClN2O3Cor e Forma:SolidPeso molecular:388.89GRK2-IN-1 hydrochloride (2055990-90-2 free base)
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).Fórmula:C24H26ClFN4O4Pureza:98%Cor e Forma:SolidPeso molecular:488.94Eloralintide
CAS:<p>Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.</p>Fórmula:C201H319N49O65S2Cor e Forma:SolidPeso molecular:4526.1GLP-1 receptor agonist 8
CAS:<p>GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.</p>Fórmula:C34H36ClFN6O4Cor e Forma:SolidPeso molecular:647.14AB21 oxalate
<p>AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM and 102 nM for S1R and S2R, respectively.</p>Fórmula:C25H30N2O5Pureza:98%Cor e Forma:SolidPeso molecular:438.52Fenoldopam
CAS:<p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>Fórmula:C16H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:305.76Seglitide acetate
CAS:<p>Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.</p>Fórmula:C46H60N8O9Pureza:98.87%Cor e Forma:SolidPeso molecular:869.02Noladin ether
CAS:<p>Noladin ether (2-AG ether) is a cannabinoid CB1 receptor agonist.</p>Fórmula:C23H40O3Cor e Forma:SolidPeso molecular:364.56Muscarinic toxin 3
CAS:<p>Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57</p>Fórmula:C319H489N89O97S8Pureza:98%Cor e Forma:SolidPeso molecular:7379.35S1R agonist 1
CAS:<p>Compound 6b: Selective S1R agonist, K i = 0.93 nM (S1R), 72 nM (S2R); neuroprotective against ROS, NMDA toxicity.</p>Fórmula:C20H25NOCor e Forma:SolidPeso molecular:295.42Lintitript
CAS:<p>Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and 200 nM for CCK1 and CCK2. The Ki value is 0.2 nM for CCK1.</p>Fórmula:C20H14ClN3O3SPureza:99.28%Cor e Forma:SolidPeso molecular:411.86(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Fórmula:C14H22N2O3Pureza:98.72%Cor e Forma:SolidPeso molecular:266.34Spns2-IN-1
<p>Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value of 1.4±0.3 μM, crucial for modulating the immune</p>Pureza:98%Cor e Forma:Odour Solid5-OMe-UDP trisodium salt
CAS:<p>Potent P2Y6 agonist</p>Fórmula:C10H16N2O13P2Pureza:98%Cor e Forma:SolidPeso molecular:434.19W140 HBr
CAS:<p>[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.</p>Fórmula:C16H28BrN2O4PPureza:99.85%Cor e Forma:SoildPeso molecular:423.28[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:<p>[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).</p>Fórmula:C48H69N13O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1068.27Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Fórmula:C74H92ClN17O13Pureza:98%Cor e Forma:SolidPeso molecular:1463.08Adenosine receptor antagonist 1
CAS:<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Fórmula:C22H15ClFN7OCor e Forma:SolidPeso molecular:447.86(D-Arg8)-Inotocin
CAS:<p>'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.</p>Fórmula:C39H68N14O11S2Pureza:98%Cor e Forma:SolidPeso molecular:973.17Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Fórmula:C161H274N48O46SPureza:98%Cor e Forma:SolidPeso molecular:3650.29Syk Inhibitor II hydrochloride
CAS:<p>Syk signaling is key in lupus. Syk inhibitors reduce inflammation and sepsis severity in FcgRIIb-/- mice, lowering cytokines and organ damage.</p>Fórmula:C14H16ClF3N6OPureza:99.05%Cor e Forma:SolidPeso molecular:376.77FXR/TGR5 agonist 1
CAS:<p>FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.</p>Fórmula:C31H32ClN3O3Cor e Forma:SolidPeso molecular:530.07Oxmetidine FA
<p>Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.</p>Fórmula:C20H23N5O5SPureza:97.34%Cor e Forma:SoildPeso molecular:445.49Bz-Dab(nbd)-awfpp-nle-NH2
CAS:<p>Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.</p>Fórmula:C56H65N13O11Cor e Forma:SolidPeso molecular:1096.2Gulgafafusp alfa
CAS:<p>Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].</p>Cor e Forma:LiquidNSC380324
<p>NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.</p>Fórmula:C31H24N4O4Cor e Forma:SolidPeso molecular:516.55Sulamserod
CAS:<p>Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular related</p>Fórmula:C19H28ClN3O5SPureza:98.76%Cor e Forma:SolidPeso molecular:445.96Pafenolol
CAS:<p>Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.</p>Fórmula:C18H31N3O3Pureza:98.33%Cor e Forma:SolidPeso molecular:337.46A-286501
CAS:<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Fórmula:C11H14BrN5O2Pureza:98%Cor e Forma:SolidPeso molecular:328.17p-MPPF
CAS:<p>p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.</p>Fórmula:C25H27FN4O2Pureza:99.92%Cor e Forma:SolidPeso molecular:434.51LU AA33810
CAS:<p>LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Fórmula:C19H25N3O2S3Pureza:98%Cor e Forma:SolidPeso molecular:423.62IRL-1038 TFA
<p>IRL-1038 TFA is an ETB receptor antagonist used in the study of cardiovascular disease.</p>Fórmula:C70H93F3N14O17S2Pureza:98.79%Cor e Forma:SolidPeso molecular:1523.7CAP-100
<p>CAP-100 is a monoclonal antibody targeting CCR7. It neutralizes the ligand binding site and signaling of CCR7. This compound effectively inhibits migration, extravasation, homing, and survival in chronic lymphocytic leukemia (CLL) samples induced by CCR7. CAP-100 can mediate potent tumor cell killing through host immune mechanisms and exhibits favorable toxicity profiles in related hematopoietic cell subsets. It is involved in research on antitumor activity and diseases like chronic lymphocytic leukemia (CLL).</p>Cor e Forma:Odour LiquidGalanin-Like Peptide (porcine)
CAS:<p>Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.</p>Fórmula:C281H443N81O78Pureza:98%Cor e Forma:SolidPeso molecular:6204.021-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid
CAS:1-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid (Compound 31) is a metabolite of AB-FUBINACA. It acts as an MRGPRX4 antagonist with an IC50 greater than 2.5 μM.Fórmula:C15H11FN2O2Cor e Forma:SolidPeso molecular:270.26U 67827E
CAS:<p>U 67827E is a long-lasting cholecystokinin agonist. It acts by decreases food intake.</p>Fórmula:C53H68N10O17SPureza:98%Cor e Forma:SolidPeso molecular:1149.24Vazegepant
CAS:<p>Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.</p>Fórmula:C36H46N8O3Pureza:98.61%Cor e Forma:SolidPeso molecular:638.80Methicillin sodium hydrate
CAS:<p>Methicillin sodium hydrate, a narrow-spectrum antibiotic, combats methicillin-resistant Staphylococcus strains and treats various infections.</p>Fórmula:C17H21N2NaO7SCor e Forma:SolidPeso molecular:420.41LysoPalloT-NH-amide-C3-ph-m-O-C11
CAS:<p>LysoPalloT-NH-amide-C3-ph-m-O-C11 is an agonist of the GPR174 receptor with an EC50 value of 34 nM.</p>Fórmula:C27H47N2O9PCor e Forma:SolidPeso molecular:574.64GI-560192
CAS:<p>GI-560192 (RL-0070933), a potent smo modulator, EC50: 0.02µM; affects smoothened in cilia via hedgehog signaling.</p>Fórmula:C20H16N2O2Pureza:99.53%Cor e Forma:SoildPeso molecular:316.35AA 497 HCl
CAS:<p>AA 497, a beta-2 agonist, suppresses Ca spikes.</p>Fórmula:C14H22ClNO3Cor e Forma:SolidPeso molecular:287.78tetranor-PGJM
CAS:<p>Tetranor-PGJM is a metabolite of prostaglandin D2 and is associated with the anti-inflammatory effects of curcumin.</p>Fórmula:C16H22O6Cor e Forma:SolidPeso molecular:310.346Propranolol hydrochloride
CAS:<p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>Fórmula:C16H22ClNO2Pureza:99.94% - >99.99%Cor e Forma:White Or Almost White Powder White PowderPeso molecular:295.80N-Nitroso Atenolol
CAS:<p>N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.</p>Fórmula:C14H21N3O4Cor e Forma:SolidPeso molecular:295.33Survodutide TFA
<p>Survodutide TFA (BI 456906 TFA) is a GCGR/GLP-1R dual agonist, a peptide compound used in obesity research.</p>Fórmula:C192H289N47O61·xC2HF3OC2Pureza:99.29% - 99.96%Cor e Forma:SolidPeso molecular:4231.62 (free base)AD186
<p>AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for S1R and 27 nM for S2R.</p>Fórmula:C22H28N2Pureza:98%Cor e Forma:SolidPeso molecular:320.47Ala5-Galanin (2-11)
CAS:<p>Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1].</p>Fórmula:C54H81N13O13Pureza:98%Cor e Forma:SolidPeso molecular:1120.3Nocistatin(human)
CAS:<p>Blocker of nociceptin-induced allodynia and hyperalgesia</p>Fórmula:C149H238N42O53S3Pureza:98%Cor e Forma:SolidPeso molecular:3561.936α-Prostaglandin I1
CAS:<p>6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.</p>Fórmula:C20H34O5Cor e Forma:SolidPeso molecular:354.487(+)-ORM-10921
CAS:<p>(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.</p>Fórmula:C18H23NO2Pureza:99.85%Cor e Forma:SoildPeso molecular:285.38Sibenadet hydrochloride
CAS:<p>Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.</p>Fórmula:C22H29ClN2O5S2Cor e Forma:SolidPeso molecular:501.06Ularitide
CAS:<p>Ularitide is a 32-amino acid peptide from ANP prohormone, resistant to dog kidney cortex peptidase.</p>Fórmula:C145H234N52O44S3Pureza:98%Cor e Forma:SolidPeso molecular:3505.97Anticancer agent 258
CAS:<p>Anticanceragent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates nuclear receptor activity. It exhibits an EC50 of 63 nM for Nurr in N2A cells and an IC50 of 0.1 pM for Nur77 in HEK293 cells. Anticanceragent 258 is applicable in studies related to cancer, metabolic disorders, and neurological diseases.</p>Fórmula:C17H12F2N4Cor e Forma:SolidPeso molecular:310.3PSA1 (141-150)
CAS:<p>This Prostate Specific Antigen 1 peptide was used in the immunotherapy of cancer experiments.</p>Fórmula:C55H93N13O13SPureza:98%Cor e Forma:SolidPeso molecular:1176.47Galanin (1-19), human
CAS:<p>Galanin (1-19), human: a fragment of GAL neuropeptide influencing hormone release, pain response, and eating behavior.</p>Fórmula:C89H130N26O25Pureza:98%Cor e Forma:SolidPeso molecular:1964.145-HT1AR agonist 2
<p>5-HT1AR Agonist 2 (Compound 4f) is a potent agonist of the 5-HT1A receptor with a Ki value of 10.0 nM. It also binds to SERT, D2, and 5-HT6 receptors with Ki values of 2.8 nM, 23 nM, and 192 nM, respectively. Furthermore, this compound demonstrates stability in microsomes and induces hypothermia in mice.</p>Fórmula:C31H31N5O3Cor e Forma:SolidPeso molecular:521.61Pancreatic Polypeptide, rat
CAS:<p>Rat Pancreatic Polypeptide: 36-amino acid peptide, NPYR4 agonist, secreted by islet PP cells.</p>Fórmula:C195H298N58O57SPureza:98%Cor e Forma:SolidPeso molecular:4398.87Bremelanotide
CAS:<p>Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.</p>Fórmula:C50H68N14O10Pureza:98%Cor e Forma:White PowderPeso molecular:1025.16Boc-Phe-Leu-Phe-Leu-Phe
CAS:<p>Boc-Phe-Leu-Phe-Leu-Phe is a chemotactic peptide antagonist that inhibits the release of peptide leukotrienes induced by FMLP.</p>Fórmula:C44H59N5O8Cor e Forma:SolidPeso molecular:785.97Pentagastrin meglumine
CAS:<p>Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.</p>Fórmula:C44H66N8O14SCor e Forma:SolidPeso molecular:963.11isomer-Cilansetron
CAS:<p>isomer-Cilansetron is an isomer of Cilansetron.</p>Fórmula:C20H21N3OPureza:99.92% - 99.96%Cor e Forma:SoildPeso molecular:319.4Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Fórmula:C25H31F3N6O8Pureza:98.08%Cor e Forma:SoildPeso molecular:600.55Val9-Oxytocin
CAS:<p>Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.</p>Fórmula:C46H72N12O12S2Pureza:98%Cor e Forma:SolidPeso molecular:1049.27CCR2 antagonist 1
CAS:CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).Fórmula:C28H32BrF3N2OCor e Forma:SolidPeso molecular:549.4716,16-dimethyl Prostaglandin F2α
CAS:<p>16,16-dimethyl Prostaglandin F2α can be used in related research in the field of life sciences. Its product number is T37993 and CAS number is 39746-23-1.</p>Fórmula:C22H38O5Cor e Forma:SolidPeso molecular:382.541Glucagon (19-29), human
CAS:Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.Fórmula:C61H89N15O18SPureza:98%Cor e Forma:SolidPeso molecular:1352.53Isoprenaline
CAS:<p>Isoprenaline is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.</p>Fórmula:C11H17NO3Pureza:99.31%Cor e Forma:SolidPeso molecular:211.26Des His1, Glu8 Exendin-4
<p>Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose and is used in the study of diabetes and obesity.</p>Fórmula:C179H277N47O59SPureza:99.92%Cor e Forma:SolidPeso molecular:4063.46YM 09538
CAS:<p>YM 09538 is a biochemical.</p>Fórmula:C18H25ClN2O5SCor e Forma:SolidPeso molecular:416.92GR 94800
CAS:<p>Potent and selective tachykinin NK2 receptor antagonist</p>Fórmula:C49H61N9O8Pureza:98%Cor e Forma:SolidPeso molecular:904.082Adrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Fórmula:C194H304N58O59S4Pureza:98%Cor e Forma:SolidPeso molecular:4521.17Setmelanotide
CAS:<p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>Fórmula:C49H68N18O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1117.31WS 9326A
CAS:<p>WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger.</p>Fórmula:C54H68N8O13Pureza:98%Cor e Forma:SolidPeso molecular:1037.181TGR5 agonist 1
<p>Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].</p>Fórmula:C28H48NNaO6SCor e Forma:SolidPeso molecular:549.74CGRP 8-37 (rat)
CAS:<p>CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.</p>Fórmula:C138H224N42O41Pureza:99.28%Cor e Forma:SolidPeso molecular:3127.51Cortistatin-8
CAS:<p>ghrelin receptor antagonist</p>Fórmula:C47H68N12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1009.25RC-3095
CAS:<p>RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.</p>Fórmula:C56H79N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1106.32GRK-IN-1
CAS:<p>4-Amino-5-(bromomethyl)-2-methylpyrimidine used in vitamin B1 analogs and esters synthesis.</p>Fórmula:C6H10Br3N3Cor e Forma:SolidPeso molecular:363.879Vapreotide diacetate
CAS:<p>Vapreotide diacetate, a synthetic somatostatin analog, blocks NK1R to provide analgesic effects.</p>Fórmula:C61H78N12O13S2Pureza:98%Cor e Forma:SolidPeso molecular:1251.47Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Fórmula:C10H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:233.69GLP-1R/GIPR agonist-1
<p>GLP-1R/GIPR agonist-1 is a dual receptor agonist for GLP-1 (glucagon-like peptide-1) and GIP (glucose-dependent insulinotropic polypeptide). It mimics the action of endogenous hormones GLP-1 and GIP, enhancing insulin secretion while suppressing glucagon release, thus lowering blood sugar. This compound is used in research related to metabolic disorders such as diabetes, obesity, and non-alcoholic steatohepatitis (NASH).</p>Fórmula:C220H342N55O69Peso molecular:4858.49434MCL0129
CAS:<p>MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.</p>Fórmula:C34H47FN4OPureza:98%Cor e Forma:SolidPeso molecular:546.7611-deoxy Prostaglandin E1
CAS:<p>11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and cause</p>Fórmula:C20H34O4Cor e Forma:SolidPeso molecular:338.48RFRP-1(human)
CAS:<p>Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.</p>Fórmula:C67H101N19O14SPureza:98%Cor e Forma:SolidPeso molecular:1428.72[D-Trp34]-Neuropeptide Y Acetate
<p>[D-Trp34]-Neuropeptide Y Acetate is a potent Y5 receptor agonist that increases rat food intake; less potent at Y1, Y2, Y4, Y6.</p>Fórmula:C198H293N55O58Pureza:99.73%Cor e Forma:SoildPeso molecular:4371.78Sch 202596
CAS:<p>Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.</p>Fórmula:C25H22Cl2O12Cor e Forma:SolidPeso molecular:585.34Torososide B
CAS:<p>Torososide B is an anti-allergic compound that inhibits leukotriene release from calcium ionophore A-stimulated rat peritoneal mast cells.</p>Fórmula:C40H52O25Cor e Forma:SolidPeso molecular:932.83Human growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Fórmula:C215H358N72O66SPureza:98%Cor e Forma:SolidPeso molecular:5039.65Albenatide
CAS:<p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>Fórmula:C26H47N7O9SPureza:98%Cor e Forma:SolidPeso molecular:633.76Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:<p>Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.</p>Fórmula:C161H240N46O41S2Cor e Forma:SolidPeso molecular:3540.09LY-53857 free base
CAS:<p>LY-53857 free base is a bioactive chemical.</p>Fórmula:C23H32N2O3Cor e Forma:SolidPeso molecular:384.51Esprolol
CAS:<p>Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.</p>Fórmula:C17H27NO4Pureza:71.58% - 99.16%Cor e Forma:SoildPeso molecular:309.4Cholecystokinin Octapeptide, desulfated
CAS:<p>Cholecystokinin Octapeptide, desulfated (CCK Octapeptide, non-sulfated) is an octapeptide composed of 8 amino acids from cholecystokinin-8.</p>Fórmula:C49H62N10O13S2Pureza:97.12%Cor e Forma:SolidPeso molecular:1063.21Apelin-17(human, bovine)
CAS:<p>Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).</p>Fórmula:C96H156N34O20SPureza:98%Cor e Forma:SolidPeso molecular:2138.56Men 10208
CAS:<p>Men 10208 is an antagonist of the neurokinin A receptor.</p>Fórmula:C61H75N15O12Pureza:98%Cor e Forma:SolidPeso molecular:1210.36Apelin-36(rat, mouse)
CAS:Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.Fórmula:C185H304N68O43SPureza:98%Cor e Forma:SolidPeso molecular:4200.93NI-203
<p>NI-203 is a monoclonal antibody inhibitor that targets amylin and shows potential for research in type 2 diabetes.</p>Cor e Forma:Odour LiquidPHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44Kinetensin
CAS:Kinetensin is a neurotensin-like peptide.Fórmula:C56H85N17O11Pureza:98%Cor e Forma:White Lyophilised SolidPeso molecular:1172.38Amylin, amide, rat
CAS:<p>Amylin: peptide, 50% similar to CGRP, found with somatostatin in stomach cells, reduces acid secretion in mice.</p>Fórmula:C167H272N52O53S2Pureza:99.92%Cor e Forma:SolidPeso molecular:3920.44Thromboxane B1
CAS:<p>Thromboxane B1 (TXB1) is a lipid eicosanoid, part of the TXB family, involved in blood clotting.</p>Fórmula:C20H36O6Cor e Forma:SolidPeso molecular:372.5YM 16638
CAS:<p>YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.</p>Fórmula:C18H22N2O5S3Pureza:99.18%Cor e Forma:SolidPeso molecular:442.57Corynanthine
CAS:<p>Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.</p>Fórmula:C21H26N2O3Pureza:98%Cor e Forma:SolidPeso molecular:354.44Sphingosine-1-phosphate (d16:1)
CAS:<p>C16 S1P binds S1P1/EDG-1 (115%), S1P3/EDG-3 (83%), S1P2/EDG-5 (103%) receptors; elevated in glaucoma.</p>Fórmula:C16H34NO5PCor e Forma:SolidPeso molecular:351.424HHS-0701
CAS:HHS-0701: SuTEx ligand, strong PTGR2 inhibitor, blocks 15-Keto-PGE2 metabolism.Fórmula:C20H20N4O3SPureza:97.24%Cor e Forma:SoildPeso molecular:396.46ent-Prostaglandin E2
CAS:<p>Enzymatic PGE2 is optically pure; radical peroxidation makes it racemic. In oxidative stress, rac-PGE2 forms via 15-E2t-isoprostane.</p>Fórmula:C20H32O5Cor e Forma:SolidPeso molecular:352.471SHU 9119
CAS:<p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>Fórmula:C54H71N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1074.2585-methoxy-α-Ethyltryptamine
CAS:<p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>Fórmula:C13H18N2OPureza:98.25%Cor e Forma:SolidPeso molecular:218.29Antibacterial agent 189
Antibacterialagent 189 (compound 3a) is a potent antibacterial agent with high binding affinity to the target proteins OMPA/exo-1,3-β-glucanase. It demonstrates effective antibacterial activity against Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Candida albicans, and Aspergillus flavus. Additionally, Antibacterialagent 189 exhibits strong binding affinity to the target proteins SMO and SUFU/GLI-1.Fórmula:C37H28N4OPeso molecular:544.22631(±)-9-Nor-9α-hydroxy Hexahydrocannabinol
CAS:<p>(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.</p>Fórmula:C20H30O3Cor e Forma:SolidPeso molecular:318.45Nadolol
CAS:<p>Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.</p>Fórmula:C17H27NO4Pureza:99.87% - 99.92%Cor e Forma:White To Off-White Crystalline Powder SolidPeso molecular:309.40N,N′-Diferuloylputrescine
CAS:<p>N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.</p>Fórmula:C24H28N2O6Pureza:98%Cor e Forma:SolidPeso molecular:440.4915(R)-17-phenyl trinor Prostaglandin F2α
CAS:<p>17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocular</p>Fórmula:C23H32O5Cor e Forma:SolidPeso molecular:388.5Vapitadine
CAS:<p>Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.</p>Fórmula:C17H20N4OPureza:99.77% - 99.86%Cor e Forma:SoildPeso molecular:296.37TGR5 agonist 4
<p>TGR5 agonist 4 (compound 19), a derivative of cholic acid, selectively activates the TGR5 receptor with an effective concentration (EC50) of 4 μM [1].</p>Fórmula:C24H38F2O5Cor e Forma:SolidPeso molecular:444.555-trans Latanoprost (free acid)
CAS:<p>Latanoprost, a prodrug eye drop, turns into active acid inside the body and treats high eye pressure. Its trans isomer also likely reduces eye pressure.</p>Fórmula:C23H34O5Cor e Forma:SolidPeso molecular:390.52hNTS1R agonist-1
<p>Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (</p>Fórmula:C37H62N10O9Pureza:98%Cor e Forma:SolidPeso molecular:790.95APJ receptor agonist 1
CAS:<p>Potent APJ-R agonist 1, biphenyl acid, EC50: 0.093 nM (human), 0.12 nM (rat), targets apelin-13, promising for heart failure study.</p>Fórmula:C31H26ClN3O3Cor e Forma:SolidPeso molecular:524.02Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Fórmula:C20H22Cl2N2O4Cor e Forma:SolidPeso molecular:425.31Thiethylperazine
CAS:<p>Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.</p>Fórmula:C22H29N3S2Pureza:98.72%Cor e Forma:SolidPeso molecular:399.62Flibanserin-d4
CAS:<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Fórmula:C20H21F3N4OPureza:98%Cor e Forma:SolidPeso molecular:394.43Fexofenadine-d6
CAS:<p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>Fórmula:C32H39NO4Pureza:98%Cor e Forma:SolidPeso molecular:507.69SYL-4
CAS:SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Fórmula:C20H15N3O5SPureza:95.76%Cor e Forma:SoildPeso molecular:409.42Alosetron D3 Hydrochloride
CAS:<p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Fórmula:C17H19ClN4OPureza:98%Cor e Forma:SolidPeso molecular:333.83Bombesin
CAS:<p>Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.</p>Fórmula:C71H110N24O18SCor e Forma:While Lyophilized PowderPeso molecular:1619.85MK-761 TFA
<p>MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.</p>Fórmula:C15H20F3N3O4Cor e Forma:SolidPeso molecular:363.332Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Fórmula:C21H26D6Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:433.45Argipressin
CAS:<p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>Fórmula:C46H65N15O12S2Pureza:98%Cor e Forma:White PowderPeso molecular:1084.23Substance P TFA
CAS:<p>Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.</p>Fórmula:C65H99F3N18O15SPureza:98%Cor e Forma:SolidPeso molecular:1461.673-O-Methyldopa-d3
CAS:3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Fórmula:C10H10D3NO4Peso molecular:214.23Mozavaptan hydrochloride
CAS:<p>Mozavaptan is a vasopressin receptor antagonist.</p>Fórmula:C27H30ClN3O2Cor e Forma:SolidPeso molecular:464Hydroxyzine D8
CAS:Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Fórmula:C21H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:382.95Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Fórmula:C27H40N8O6Cor e Forma:SolidPeso molecular:572.66Cetirizine D4
CAS:<p>Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:392.91Dapagliflozin impurity
CAS:Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Fórmula:C21H25ClO7Cor e Forma:SolidPeso molecular:424.87Calcitonin (salmon)
CAS:<p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>Fórmula:C145H240N44O48S2Pureza:99.41% - 99.80%Cor e Forma:PowderPeso molecular:3431.85Aripiprazole (D8)
CAS:<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Fórmula:C23H27Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:456.44Asenapine hydrochloride
CAS:<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Fórmula:C17H17Cl2NOCor e Forma:SolidPeso molecular:322.23L-798106
CAS:L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Fórmula:C27H22BrNO4SPureza:98.97%Cor e Forma:SolidPeso molecular:536.44Sumanirole maleate
CAS:<p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>Fórmula:C15H17N3O5Pureza:98%Cor e Forma:SolidPeso molecular:319.31(Rac)-Mirabegron-d5
CAS:<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Fórmula:C21H24N4O2SPureza:98%Cor e Forma:SolidPeso molecular:401.54ML 00253764
CAS:melanocortin MC4 receptor antagonistFórmula:C18H18BrFN2OCor e Forma:SolidPeso molecular:377.25BMS-986020 sodium
CAS:<p>BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.</p>Fórmula:C29H25N2NaO5Cor e Forma:SolidPeso molecular:504.51Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Fórmula:C19H24N2OSPureza:99.15%Cor e Forma:SolidPeso molecular:328.474-Hydroxyatomoxetine D3
CAS:<p>4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.</p>Fórmula:C17H21NO2Pureza:98%Cor e Forma:SolidPeso molecular:274.37Ipragliflozin (L-Proline)
CAS:Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.Fórmula:C26H30FNO7SCor e Forma:SolidPeso molecular:519.58(S)-ZINC-3573
CAS:<p>(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.</p>Fórmula:C18H21N5Cor e Forma:SolidPeso molecular:307.401Zagociguat
CAS:<p>Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and can be used in the research of neurological diseases.</p>Fórmula:C16H10F4N6Pureza:99.37%Cor e Forma:SolidPeso molecular:362.28Lanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Fórmula:C54H69N11O10S2Cor e Forma:SolidPeso molecular:1096.32Revdofilimab
CAS:<p>Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.</p>Pureza:98.80% - 98.80%Cor e Forma:Liquidβ2AR/M-receptor agonist-2
CAS:<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Fórmula:C36H49ClN4O7SCor e Forma:SolidPeso molecular:717.315-HT3 antagonist 5
CAS:<p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>Fórmula:C16H13N3O2Pureza:99.84%Cor e Forma:SolidPeso molecular:279.29Ceralifimod
CAS:Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Fórmula:C27H33NO4Cor e Forma:SolidPeso molecular:435.56SANT 2
CAS:<p>SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.</p>Fórmula:C26H26ClN3O4Pureza:99.23%Cor e Forma:SolidPeso molecular:479.96Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Fórmula:C10H16N8S2Pureza:98%Cor e Forma:SolidPeso molecular:312.42Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Fórmula:C15H21D3N2O4SCor e Forma:SolidPeso molecular:331.454,4-Diphenylbutylamine hydrochloride
CAS:<p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>Fórmula:C16H20ClNCor e Forma:SolidPeso molecular:261.79(S)-(+)-Dimethindene maleate
CAS:<p>(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors</p>Fórmula:C24H28N2O4Pureza:99.94%Cor e Forma:SolidPeso molecular:408.49Etofylline clofibrate
CAS:<p>Etofylline clofibrate has a hypolipidemic and antithrombotic effect and it also has an agonistic interaction with intimal PGI2.</p>Fórmula:C19H21ClN4O5Cor e Forma:SolidPeso molecular:420.85Cetirizine D8
CAS:<p>Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:396.94Diacetolol D7
CAS:<p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>Fórmula:C16H24N2O4Pureza:98%Cor e Forma:SolidPeso molecular:315.42R121919
CAS:<p>R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.</p>Fórmula:C22H32N6Pureza:99.75%Cor e Forma:SolidPeso molecular:380.53Virodhamine
CAS:<p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>Fórmula:C22H37NO2Pureza:98%Cor e Forma:SoildPeso molecular:347.53Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Fórmula:C18H18ClN3SPureza:99.93%Cor e Forma:SolidPeso molecular:343.87MRGPRX4 modulator-2
CAS:MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value of less than 100 nM. Its notable applications include research on autoimmune diseases such as psoriasis, multiple sclerosis, Steven Johnson's Syndrome, and various chronic itch conditions [1].Fórmula:C15H9ClF4O3Pureza:99.24%Cor e Forma:SolidPeso molecular:348.68Bromperidol hydrochloride
CAS:<p>Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.</p>Fórmula:C21H24BrClFNO2Cor e Forma:SolidPeso molecular:456.78GB-88
CAS:GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.Fórmula:C32H42N4O4Cor e Forma:SolidPeso molecular:546.7Glucagon (1-29), bovine, human, porcine
CAS:Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.Fórmula:C153H225N43O49SPureza:99.56% - 99.56%Cor e Forma:SolidPeso molecular:3482.75LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Fórmula:C18H14FN5OPureza:99.03% - >99.99%Cor e Forma:SolidPeso molecular:335.34Quetiapine-d4 hemifumarate
CAS:<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Fórmula:C25H29N3O6SPureza:98%Cor e Forma:White SolidPeso molecular:503.61GLP-1 receptor agonist 7
CAS:<p>GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.</p>Fórmula:C31H30ClFN4O5Cor e Forma:SolidPeso molecular:593.05GLP-1R modulator C5
CAS:<p>GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.</p>Fórmula:C24H21NO3Pureza:99.59%Cor e Forma:SolidPeso molecular:371.43SAR247799
CAS:<p>SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.</p>Fórmula:C21H16ClN3O5Cor e Forma:SolidPeso molecular:425.82
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