EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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Naluzotan
CAS:740873-06-7
Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of …
Formula:
C23H38N4O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
450.64
Ref: TM-T16265
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PP 3
CAS:5334-30-5
PP 3 is a Negative control for the Src kinase inhibitor PP 2
Formula:
C11H9N5
Purity:
98.92%
Color and Shape:
Whit To Off-White Solid
Molecular weight:
211.22
Ref: TM-T23176
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 139.00 € | ||
| 50mg | 200.00 € | ||
| 100mg | 302.00 € | ||
| 500mg | 719.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Osimertinib
CAS:1421373-65-0
Osimertinib (AZD-9291) is a small molecule tyrosine kinase receptor inhibitor and antineoplastic agent that is …
Formula:
C28H33N7O2
Purity:
100% - 99.83%
Color and Shape:
Solid
Molecular weight:
499.61
Ref: TM-T2490
| 1g | 153.00 € | ||
| 2mg | 38.00 € | ||
| 5mg | 53.00 € | ||
| 10mg | 61.00 € | ||
| 25mg | 75.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 103.00 € | ||
| 200mg | 115.00 € | ||
| 500mg | 126.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Butein
CAS:487-52-5
Butein is a cAMP-specific PDE inhibitor, protein tyrosine kinase inhibitor, and SIRT1 activator.Cost-effective and quality-assured.
Formula:
C15H12O5
Purity:
100% - 99.85%
Color and Shape:
Solid
Molecular weight:
272.25
Ref: TM-T6427
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 540.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PD158780
CAS:171179-06-9
PD 158780 blocks all ErbB receptors: EGFR, ErbB2-4, with IC50s: 8μM, 49-52 nM.
Formula:
C14H12BrN5
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
330.18
Ref: TM-T5410
| 1mg | 40.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 546.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
β-Hydroxyisovalerylshikonin
CAS:7415-78-3
Beta-Hydroxyisovalerylshikonin is an inhibitor of protein-tyrosine kinases such as v-Src and EGFR, and has been …
Formula:
C21H24O7
Purity:
98.16%
Color and Shape:
Solid
Molecular weight:
388.41
Ref: TM-TN1440
| 1mg | 134.00 € | ||
| 5mg | 395.00 € | ||
| 10mg | 575.00 € | ||
| 25mg | 894.00 € | ||
| 50mg | 1,199.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
TAS6417
CAS:1661854-97-2
Zipalertinib (TAS6417, CLN-081) is a novel, highly potent, orally active covalent EGFR tyrosine kinase inhibitor.Cost-effective …
Formula:
C23H20N6O
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
396.44
Ref: TM-T16996
| 1mg | 96.00 € | ||
| 2mg | 122.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,513.00 € | ||
| 500mg | 3,045.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PD153035 hydrochloride
CAS:183322-45-4
PD153035 hydrochloride (ZM 252868) is a effective and selective inhibitor of EGFR; few influence against …
Formula:
C16H15BrClN3O2
Purity:
100% - ≥95%
Color and Shape:
Solid
Molecular weight:
396.67
Ref: TM-T1761
| 5mg | 35.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 81.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 233.00 € | ||
| 500mg | 530.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
EAI045
CAS:1942114-09-1
EAI045, an allosteric inhibitor, targets towards drug-resistant EGFR mutants but avoids the wild-type receptor.
Formula:
C19H14FN3O3S
Purity:
99.36% - 99.73%
Color and Shape:
Solid
Molecular weight:
383.4
Ref: TM-T6824
| 5mg | 43.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 195.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
AZ7550
CAS:1421373-99-0
AZ7550, an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).
Formula:
C27H31N7O2
Purity:
97.07%
Color and Shape:
Solid
Molecular weight:
485.58
Ref: TM-T13564
| 1mg | 129.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 417.00 € | ||
| 25mg | 689.00 € | ||
| 50mg | 920.00 € | ||
| 100mg | 1,287.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
CP-380736
CAS:179688-29-0
CP-380736 (PF-00520893) inhibits EGFR, a kinase key in cancer-signaling pathways like MAPK, JNK, and Akt.
Formula:
C14H18N2O5
Purity:
99.91%
Color and Shape:
White To Off-White Solid
Molecular weight:
294.3
Ref: TM-T19814
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 163.00 € | ||
| 200mg | 237.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Tyrphostin 23
CAS:118409-57-7
Tyrphostin 23 (AG18) inhibits EGFR with IC50 of 35 μM.
Formula:
C10H6N2O2
Purity:
99.19% - 99.7%
Color and Shape:
Yellow-Tan Solid
Molecular weight:
186.17
Ref: TM-T2063
| 10mg | 59.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 333.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
EGFR-IN-12
CAS:879127-07-8
EGFR-IN-12 (EGFR Inhibitor) is a cell permeable and selective inhibitor of EGFR kinase (IC50: 21 …
Formula:
C21H18F3N5O
Purity:
98.30% - 99.19%
Color and Shape:
Solid
Molecular weight:
413.4
Ref: TM-T5168
| 1mg | 81.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 255.00 € | ||
| 25mg | 511.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 985.00 € | ||
| 500mg | 1,977.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
ALK-IN-1
CAS:1197958-12-5
ALK-IN-1 (AP26113) is a potent ALK inhibitor, demonstrated ability overcome Crizotinib resistance mediated by a …
Formula:
C26H34ClN6O2P
Purity:
100% - 97.66%
Color and Shape:
Solid
Molecular weight:
529.01
Ref: TM-T3059
| 5mg | 48.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 143.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 345.00 € | ||
| 500mg | 561.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Zorifertinib
CAS:1626387-80-1
Zorifertinib (AZD3759) is an orally active, effective and central nervous system-penetrant EGFR inhibitor.
Formula:
C22H23ClFN5O3
Purity:
98.29% - 99.36%
Color and Shape:
White To Off-White Solid
Molecular weight:
459.9
Ref: TM-T3659
| 25mg | 43.00 € | ||
| 50mg | 56.00 € | ||
| 100mg | 88.00 € | ||
| 200mg | 116.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
MTX-211
CAS:1952236-05-3
MTX-211, an inhibitor of EGFR and PI3K, is used for the therapy of cancer and …
Formula:
C20H14Cl2FN5O2S
Purity:
100% - 97.28%
Color and Shape:
Solid
Molecular weight:
478.33
Ref: TM-T4296
| 1mg | 62.00 € | ||
| 5mg | 180.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 450.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 840.00 € | ||
| 200mg | 1,116.00 € | ||
| 1mL*10mM (DMSO) | 183.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Desmethyl Erlotinib hydrochloride
CAS:183320-51-6
Desmethyl Erlotinib hydrochloride (OSI 420) is an active metabolite of erlotinib which is an orally …
Formula:
C21H21N3O4·HCl
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
415.87
Ref: TM-T6619
| 1mg | 59.00 € | ||
| 2mg | 82.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 186.00 € | ||
| 25mg | 332.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 711.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
AG 555
CAS:133550-34-2
AG 555 (Tyrphostin B46) is an EGFR tyrosine kinase inhibitor.
Formula:
C19H18N2O3
Purity:
100% - 99.51%
Color and Shape:
Solid
Molecular weight:
322.36
Ref: TM-T4326
| 5mg | 46.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 243.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
WHI-P258
CAS:21561-09-1
WHI-P258, a weak JAK3 inhibitor, is used as a negative control in drug development.
Formula:
C16H15N3O2
Purity:
99.59% - 99.95%
Color and Shape:
Solid
Molecular weight:
281.31
Ref: TM-T2035
| 5mg | 34.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 140.00 € | ||
| 100mg | 230.00 € | ||
| 200mg | 336.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
AG-1478
CAS:153436-53-4
AG-1478 (NSC-693255) (Tyrphostin AG-1478) is a selective EGFR inhibitor.
Formula:
C16H14ClN3O2
Purity:
99.03% - 99.71%
Color and Shape:
Solid
Molecular weight:
315.75
Ref: TM-T2047
| 5mg | 54.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 355.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
