EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
Read more
Selatinib
CAS:1275595-86-2
Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer …
Formula:
C29H26ClFN4O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
565.06
Ref: TM-T34602
| 1mg | 96.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 345.00 € | ||
| 25mg | 637.00 € | ||
| 50mg | 926.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
LY 456236 hydrochloride
CAS:338736-46-2
LY 456236 hydrochloride (MPMQ hydrochloride) is an mGlu1 receptor antagonist with an ic50 value of …
Formula:
C16H16ClN3O2
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
317.77
Ref: TM-T22954
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 608.00 € | ||
| 500mg | 1,262.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Cloperastine fendizoate
CAS:85187-37-7
Cloperastine fendizoate (Hustazol) inhibits the hERG K+ currents in a concentration-dependent manner (IC50: 27 nM).
Formula:
C40H38ClNO5
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
648.19
Ref: TM-T13619
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EMI1
CAS:35773-42-3
EMI1 targets mutated EGFR in drug-resistant NSCLC research.
Formula:
C20H18N2O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
334.37
Ref: TM-T61016
| 5mg | 39.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 293.00 € | ||
| 200mg | 414.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
CGP52411
CAS:145915-58-8
CGP52411 is an orally active, and ATP-competitive inhibitor of EGFR (IC50: 0.3 μM).
Formula:
C20H15N3O2
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
329.35
Ref: TM-T10782
| 1mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 294.00 € | ||
| 50mg | 429.00 € | ||
| 100mg | 603.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EGFR-IN-16
CAS:133550-22-8
EGFR-IN-16 (AG473) is an inhibitor of EGFR in human A431 cells.
Formula:
C16H11NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
265.26
Ref: TM-T8525
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 346.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EGFR-IN-88
CAS:2944452-34-8
EGFR-IN-88 (Compound 4i), an EGFR inhibitor with an IC50 of 87 nM, exhibits cytotoxic effects …
Formula:
C22H18Cl2N4O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
473.37
Ref: TM-T79694
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EGFR-IN-89
CAS:2413029-40-8
EGFR-IN-89 (compound 13k) is a fourth-generation inhibitor selectively targeting EGFR mutations, exhibiting potent activity with …
Formula:
C26H31FN8O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
538.64
Ref: TM-T79775
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Antiproliferative agent-34
CAS:2910858-34-1
Antiproliferative Agent-34 (Compound A14), a multitarget kinase inhibitor, demonstrates IC50 values of 177 nM for …
Formula:
C27H27N7O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
529.55
Ref: TM-T79368
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EGFR-IN-73
CAS:2857033-34-0
EGFR-IN-73 (Compound 3f) effectively inhibits the prevalent EGFR mutation, EGFR Del19, exhibiting an IC50 value …
Formula:
C19H17ClFN3O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
405.81
Ref: TM-T73165
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EGFR-IN-82
CAS:2568086-81-5
EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of …
Formula:
C32H41BrN9O2P
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
694.6
Ref: TM-T78788
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
PD 174265
CAS:216163-53-0
PD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) …
Formula:
C17H15BrN4O
Purity:
98.88%
Color and Shape:
Solid
Molecular weight:
371.23
Ref: TM-T28339
| 5mg | 35.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 61.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 111.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Tarlox-TKI
CAS:2135696-72-7
Tarlox-TKI (Kinase inhibitor-1) is a pan-ErbB inhibitor, the active ingredient of Tarloxotinib, which has antitumor …
Formula:
C19H18BrClN6O
Purity:
97.03%
Color and Shape:
Solid
Molecular weight:
461.74
Ref: TM-T11761
| 1mg | 142.00 € | ||
| 1mL*10mM (DMSO) | 253.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
(E/Z)-CP-724714
CAS:537705-08-1
(E/Z)-CP-724714, comprising racemic mixtures of (E)-CP-724714 and (Z)-CP-724714 isomers, is a potent, selective, and orally …
Formula:
C27H27N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
469.54
Ref: TM-T6046
| 25mg | 1,410.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EAI001
CAS:892772-75-7
EAI001 is a potent and selective mutant epidermal growth factor receptor (EGFR) variant inhibitor that …
Formula:
C19H15N3O2S
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
349.41
Ref: TM-T61191
| 5mg | 55.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 446.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Mutated EGFR-IN-2
CAS:2050906-97-1
Mutated EGFR-IN-2 is an inhibitor of mutant-selective EGFR.
Formula:
C29H35FN8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
562.64
Ref: TM-T12130
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
EGFR-IN-5
CAS:2225887-26-1
EGFR-IN-5 inhibits EGFR & mutants; IC50: EGFR 10.4nM, L858R 1.1nM, L858R/T790M 34nM, L858R/T790M/C797S 7.2nM.
Formula:
C31H38FN9O
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
571.69
Ref: TM-T11160
| 1mg | 106.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 442.00 € | ||
| 25mg | 887.00 € | ||
| 50mg | 1,346.00 € | ||
| 100mg | 2,349.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Sunvozertinib
CAS:2370013-12-8
Sunvozertinib (DZD9008) is a potent ErbBs and BTK inhibitor, with inhibitory effects on EGFR, Her2.Cost-effective …
Formula:
C29H35ClFN7O3
Purity:
98.11% - 99.71%
Color and Shape:
Liquid
Molecular weight:
584.08
Ref: TM-T64124
| 1mg | 36.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 370.00 € | ||
| 500mg | 1,375.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
A-935142
CAS:1031335-85-9
A-935142 enhances hERG (Kv 11.1) channels, slows inactivation, promotes activation, and shortens repolarization.
Formula:
C18H19F3N2O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
352.35
Ref: TM-T14077
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Tyrphostin AG 112
CAS:144978-82-5
Tyrphostin AG 112 is an inhibitor of EGFR phosphorylation.
Formula:
C13H8N4O
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
236.23
Ref: TM-T8534
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 267.00 € | ||
| 500mg | 649.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
