EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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Gefitinib
CAS:184475-35-2
Gefitinib (ZD1839) is an EGFR first-generation inhibitor with oral activity that inhibits the EGFR 19 …
Formula:
C22H24ClFN4O3
Purity:
100% - 99.92%
Color and Shape:
Light-Yellow Crystalline Powder
Molecular weight:
446.9
Ref: TM-T1181
| 1g | 80.00 € | ||
| 5g | 144.00 € | ||
| 100mg | 54.00 € | ||
| 500mg | 62.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
O-Desmethyl gefitinib
CAS:847949-49-9
O-Desmethyl gefitinib is an active EGFR inhibitor (IC50: 36 nM), a metabolite of Gefitinib, formed …
Formula:
C21H22ClFN4O3
Purity:
99.6%
Color and Shape:
Solid
Molecular weight:
432.88
Ref: TM-T16369
| 1mg | 56.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 342.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 783.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
4-Quinazolinamine, N-(3-chlorophenyl)-6,7-dimethoxy-
CAS:153436-53-4
Formula:
C16H14ClN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
315.7543
Ref: IN-DA0020DN
| 50mg | 113.00 € | ||
| 100mg | 186.00 € | ||
| 250mg | 291.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Erlotinib
CAS:183321-74-6
Erlotinib (NSC-718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment …
Formula:
C22H23N3O4
Purity:
98.19% - 99.98%
Color and Shape:
White To Off-White Powder
Molecular weight:
393.44
Ref: TM-T0373
| 50mg | 47.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Mubritinib
CAS:366017-09-6
Formula:
C25H23F3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
468.4709
Ref: IN-DA0078T8
| 5mg | 81.00 € | ||
| 10mg | 111.00 € | ||
| 50mg | 328.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lapatinib ditosylate monohydrate
CAS:388082-78-8
Lapatinib ditosylate monohydrate: a drug for advanced breast cancer; may cause liver issues.
Formula:
C29H26ClFN4O4S·2(C7H8O3S)·H2O
Purity:
100% - 98%
Color and Shape:
Colourless To Light-Yellow Crystal
Molecular weight:
943.47
Ref: TM-T0078L
| 50mg | 52.00 € | ||
| 100mg | 69.00 € | ||
| 200mg | 92.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![(2E)-2-Cyano-3-(3,4-Dihydroxyphenyl)-N-[(1S)-1-Phenylethyl]-2-Propenamide](https://static.cymitquimica.com/products/IN/thumb/DA003988.jpg)
(2E)-2-Cyano-3-(3,4-Dihydroxyphenyl)-N-[(1S)-1-Phenylethyl]-2-Propenamide
CAS:133550-37-5
Formula:
C18H16N2O3
Purity:
97%
Color and Shape:
Solid
Molecular weight:
308.3312
Ref: IN-DA003988
| 1g | To inquire | ||
| 1mg | 197.00 € | ||
| 100mg | 233.00 € | ||
| 250mg | 527.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Norcantharidin
CAS:5442-12-6
Norcantharidin (Norcantharadine) is a synthetic anticancer compound which is a dual inhibitor for c-Met and …
Formula:
C8H8O4
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
168.15
Ref: TM-T2894
| 20mg | 54.00 € | ||
| 50mg | 84.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AV-412
CAS:451493-31-5
AV-412 (MP412) is an EGFR inhibitor (EGFR, EGFR T790M, EGFR L858R, EGFR L858R/T790M and ErbB2 …
Formula:
C41H44ClFN6O7S2
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
851.41
Ref: TM-T10419
| 1mg | 43.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 415.00 € | ||
| 100mg | 604.00 € | ||
| 1mL*10mM (DMSO) | 135.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TYRPHOSTIN B48
CAS:133550-35-3
Formula:
C16H12N2O3
Purity:
95%
Color and Shape:
Solid
Molecular weight:
280.2781
Ref: IN-DA009ARY
| 10mg | 66.00 € | ||
| 20mg | 72.00 € | ||
| 50mg | 102.00 € | ||
| 100mg | 147.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
LCH-7749944
CAS:796888-12-5
LCH-7749944 suppresses human gastric cancer cell growth, induces apoptosis, and inhibits PAK4 with IC50 of …
Formula:
C20H22N4O2
Purity:
99.28%
Color and Shape:
Solid
Molecular weight:
350.41
Ref: TM-T11826
| 1mg | 82.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 261.00 € | ||
| 25mg | 466.00 € | ||
| 50mg | 699.00 € | ||
| 100mg | 1,013.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
WHI-P154
CAS:211555-04-3
Formula:
C16H14BrN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
376.2047
Ref: IN-DA00BF57
| 1g | 611.00 € | ||
| 10mg | 55.00 € | ||
| 50mg | 121.00 € | ||
| 100mg | 184.00 € | ||
| 250mg | 233.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![2-Propenethioamide, 3-[3,5-bis(1,1-dimethylethyl)-4-hydroxyphenyl]-2-cyano-, (2E)-](https://static.cymitquimica.com/products/IN/thumb/DA001L5Z.jpg)
2-Propenethioamide, 3-[3,5-bis(1,1-dimethylethyl)-4-hydroxyphenyl]-2-cyano-, (2E)-
CAS:148741-30-4
Formula:
C18H24N2OS
Purity:
95%
Color and Shape:
Solid
Molecular weight:
316.4610
Ref: IN-DA001L5Z
| 25mg | 64.00 € | ||
| 100mg | 167.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
4-Quinazolinamine, N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)-, hydrochloride (1:1)
CAS:183319-69-9
Formula:
C22H24ClN3O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
429.8967
Ref: IN-DA0027I4
| 1g | 24.00 € | ||
| 5g | 41.00 € | ||
| 10g | 62.00 € | ||
| 25g | 118.00 € | ||
| 100g | 258.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-fur…](https://static.cymitquimica.com/products/IN/thumb/DA0039KT.jpg)
N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine
CAS:231277-92-2
Formula:
C29H26ClFN4O4S
Purity:
99%
Color and Shape:
Solid
Molecular weight:
581.0575
Ref: IN-DA0039KT
| 1g | 59.00 € | ||
| 5g | 135.00 € | ||
| 25g | 276.00 € | ||
| 25mg | 23.00 € | ||
| 250mg | 54.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
1,5-Dihydroxyxanthone
CAS:14686-65-8
1,5-Dihydroxyxanthone inhibits EGFR-tyrosine kinase (IC50: 90.34 nM) and may block AChE/BChE.
Formula:
C13H8O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
228.203
Ref: TM-TN2504
| 5mg | 1,707.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
JH-XI-10-02
CAS:2209085-22-1
JH-XI-10-02 selectively degrades CDK8 (IC50: 159 nM) through proteasome, sparing CDK8 mRNA and CDK19.
Formula:
C53H69N5O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
920.161
Ref: TM-T13743
| 2mg | 1,366.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Petosemtamab
CAS:2213450-26-9
Petosemtamab (MCLA 158), a dual-action monoclonal antibody targets EGFR & LGR5, used in solid tumor …
Purity:
> 95% - > 95%
Color and Shape:
Liquid
Molecular weight:
145.97 kDa
Ref: TM-T76890
| 1mg | 332.00 € | ||
| 5mg | 862.00 € | ||
| 10mg | 1,392.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Pertuzumab
CAS:380610-27-5
Pertuzumab (anti-HER2) a humanized monoclonal antibody and the first in the class of agents called …
Purity:
98.00%
Color and Shape:
Liquid
Molecular weight:
148 kDa
Ref: TM-T9909
| 1mg | 177.00 € | ||
| 5mg | 537.00 € | ||
| 10mg | 773.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Mutated EGFR-IN-3
CAS:2375107-27-8
Mutated EGFR-IN-3: ATP-competitive, selective dibenzodiazepinone inhibitor for EGFR mutations, IC50 12-13 nM.
Formula:
C31H29FN4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
508.59
Ref: TM-T12131
| 25mg | 1,435.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
