Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(164 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(34 products)
- Vasopressin Receptor(48 products)
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Found 3419 products of "Endocrinology/Hormones"
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2-Ethylhexyl trans-4-methoxycinnamate
CAS:2-Ethylhexyl trans-4-methoxycinnamate is a sunscreen agent.Formula:C18H26O3Purity:98.92%Color and Shape:Pale Yellow LiquidMolecular weight:290.4Angiotensin amide
CAS:Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.Formula:C49H70N14O11Purity:98%Color and Shape:SolidMolecular weight:1031.174'-hydroxy Tamoxifen
CAS:It is a metabolite of tamoxifen and an estrogen receptor modulator.Formula:C26H29NO2Purity:98%Color and Shape:SolidMolecular weight:387.511α-Hydroxy-3-epi-vitamin D3
CAS:1α-Hydroxy-3-epi-vitamin D3, a natural metabolite derived from 1alpha,25-dihydroxyvitamin D3, effectively suppresses parathyroid hormone (PTH) secretion[1].Formula:C27H44O2Color and Shape:SolidMolecular weight:400.647Ac-RYYRIK-NH2
CAS:NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.Formula:C44H70N14O9Purity:98%Color and Shape:SolidMolecular weight:939.12Antitumor agent-195
Antitumor agent-195 (compound 16c) is a dual-targeting agent that simultaneously targets STAT3 and NQO1. At a concentration of 1 μM, it significantly inhibits the phosphorylation of STAT3 at the Tyr705 site and effectively induces apoptosis in MDA-MB-231 and MDA-MB-468 breast cancer cells. As a substrate of NQO1, Antitumor agent-195 markedly increases ROS production, causing severe DNA damage in a dose-dependent manner. It also demonstrates strong antitumor properties in MDA-MB-231 xenograft models.Formula:C22H22N2O4Color and Shape:SolidMolecular weight:378.42BigLEN(mouse)
CAS:GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.Formula:C78H130N24O22Purity:98%Color and Shape:SolidMolecular weight:1756.03(rel)-PROTAC ERRα Degrader-1
(rel)-PROTAC ERRα Degrader-1 is a relative configuration of PROTAC ERRα Degrader-1, which is an estrogen-related receptor alpha (ERRa) degrader.Formula:C54H49Cl2F6N7O8Purity:98%Color and Shape:SolidMolecular weight:1108.91PROTAC ER Degrader-4
CAS:PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).Formula:C53H67F3N6O8SPurity:98%Color and Shape:SolidMolecular weight:1005.2DAMGO (TFA)
CAS:DAMGO is a selective peptide agonist of the µ-opioid receptor .Formula:C28H36F3N5O8Purity:98%Color and Shape:SolidMolecular weight:627.61OT-R antagonist 2
CAS:OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .Formula:C28H29N3O4Purity:98%Color and Shape:SolidMolecular weight:471.55BI 653048
CAS:BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.Formula:C23H25F4N3O4SPurity:98%Color and Shape:SolidMolecular weight:515.523-epi-25-hydroxy Vitamin D3
CAS:3-epi-25-hydroxy Vitamin D3 lowers serum PTH in male weanling rats at 0.5 and 1 IU/g doses; doesn't affect females.Formula:C27H44O2Color and Shape:SolidMolecular weight:400.64GNE-274
CAS:GNE-274, akin to GDC-0927 but non-degrading, is a partial ER agonist in breast cancer, enhancing chromatin at ER sites, inhibiting ER-LBD.Formula:C29H31NO4Color and Shape:SolidMolecular weight:457.57Cgp 38560
CAS:CGP 38560 is a potent renin inhibitor.Formula:C40H67N5O9S2Color and Shape:SolidMolecular weight:826.12Nurr1 agonist 2
CAS:Nurr1 agonist 2 with EC50 of 0.07 μM, boosts TH & VMAT2 mRNA, binds Nurr1 LBD at Kd 0.14 μM, for parkinsonism study.Formula:C18H14O3SPurity:98.78%Color and Shape:SoildMolecular weight:310.37Methylprednisolone Acetate
Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.Formula:C24H32O6Purity:99.74%Color and Shape:Off-White SolidMolecular weight:416.51Axelopran
CAS:Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.Formula:C26H39N3O4Color and Shape:SolidMolecular weight:457.61Raloxifene 6-glucuronide
CAS:Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8.Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71PTP1B/AKR1B1-IN-1
PTP1B/AKR1B1-IN-1 is a dual inhibitor targeting protein tyrosine phosphatase 1B (PTP1B) and aldose reductase (AKR1B1), exhibiting inhibitory potency with IC50sFormula:C22H21NO4S2Purity:98%Color and Shape:SolidMolecular weight:427.54Dipropyl phthalate
CAS:Dipropyl phthalate is a weak androgen receptor inhibitor, and can be used in biochemical experiments and drug synthesis.Formula:C14H18O4Purity:98.62%Color and Shape:SolidMolecular weight:250.29PROTAC ERRα Degrader-2
CAS:PROTAC ERRα Degrader-2 is a compound consisting of an MDM2 ligand binding group, a linker, and an estrogen-related receptor alpha (ERRα) binding group.Formula:C57H55Cl2F6N7O8Purity:98%Color and Shape:SolidMolecular weight:1150.99Aliskiren D6 Hydrochloride
CAS:Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).Formula:C30H54ClN3O6Purity:98%Color and Shape:SolidMolecular weight:594.26UFP-803
CAS:UT receptor ligand acts mainly as silent antagonist with slight agonist effects; blocks U-II in rat aorta, pIC50 = 7.46, & inhibits plasma leakage in mice.Formula:C50H64N10O12S2Purity:98%Color and Shape:SolidMolecular weight:1061.24Brain Natriuretic Peptide (1-32), rat
CAS:Rat Brain Natriuretic Peptide (1-32) is a 32-amino-acid peptide from heart, released when ventricles stretch excessively.Formula:C146H239N47O44S3Purity:98%Color and Shape:SolidMolecular weight:3452.94Lyciumin A
CAS:Lyciumin A, a cyclic octapeptide, inhibits proteases and could aid in hypertension studies.
Formula:C42H51N9O12Color and Shape:SolidMolecular weight:873.921Akuammicine
CAS:Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.Formula:C20H22N2O2Color and Shape:SolidMolecular weight:322.408Glucocorticoids receptor agonist 1
CAS:GRA-1, an arylpyrazole, is a potent glucocorticoid receptor agonist with robust anti-inflammatory effects and preserves insulin secretion.Formula:C20H23FN2OColor and Shape:SolidMolecular weight:326.41(Rac)-Finerenone
CAS:Rac-Finerenone, or (Rac)-BAY 94-8862, is an oral nonsteroidal MR antagonist with high selectivity and an IC50 of 18 nM.Formula:C21H22N4O3Color and Shape:SolidMolecular weight:378.432Montirelin
CAS:Montirelin is an analog of thyrotropin-releasing hormone.Formula:C17H24N6O4SColor and Shape:SolidMolecular weight:408.48[(pF)Phe4]Nociceptin(1-13)NH2
CAS:Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.Formula:C61H99FN22O15Purity:98%Color and Shape:SolidMolecular weight:1399.6Dermorphin Analog
Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.Formula:C44H59N11O10Purity:98%Color and Shape:SolidMolecular weight:901.43OT-R antagonist 1
CAS:OT-R antagonist 1: Nonpeptide, selective, low-weight blocker of oxytocin; IC50 = 8 nM for Ca2+ disruption.Formula:C28H29N3O4Purity:98%Color and Shape:SolidMolecular weight:471.55[Orn5]-URP
CAS:Urotensin-II receptor antagonist, no agonist effect, pEC50 7.24, blocks U-II in rat aorta assay.Formula:C48H62N10O10S2Purity:98%Color and Shape:SolidMolecular weight:1003.2Olmesartan impurity
CAS:Olmesartan impurity, related to parent RNH-6270, is an AT1R antagonist used for hypertension research.Formula:C33H26N4OColor and Shape:SolidMolecular weight:494.598Cgp 44099
CAS:Cgp 44099 is a potent plasma renin inhibitor from all subprimate species.Formula:C69H104N14O13Purity:98%Color and Shape:SolidMolecular weight:1337.676Norleual
CAS:Angiotensin IV analog, potent HGF/c-MET inhibitor (IC50=3 pM), halts MDCK cell growth and invasion, AT4 antagonist, impairs LTP, antiangiogenic.
Formula:C41H58N8O7Purity:98%Color and Shape:SolidMolecular weight:774.95Retosiban
CAS:Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).Formula:C27H34N4O5Purity:98%Color and Shape:SolidMolecular weight:494.58SNIPER(ER)-110
SNIPER(ER)-110 links cIAP1 and estrogen ligands. SNIPER(ER)-51 degrades ER protein; DC50 <3 nM at 4h, 7.7 nM at 48h.Formula:C66H83N5O11Purity:98%Color and Shape:SolidMolecular weight:1122.39TF-505
CAS:TF-505, a steroid 5α-reductase inhibitor, is used potentially for the treatment of benign prostatic hyperplasia.Formula:C33H37NO4Purity:98%Color and Shape:SolidMolecular weight:511.65Deacylcortivazol
CAS:Deacylcortivazol is a potent glucocorticoid that inhibits growth in glucocorticoid-resistant leukemia cells without receptor mediation.Formula:C30H36N2O4Color and Shape:SolidMolecular weight:488.62PL-017
CAS:μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.Formula:C29H37N5O5Purity:98%Color and Shape:SolidMolecular weight:535.64PROTAC ERRα Degrader-3
CAS:PROTAC ERRα Degrader-3 is a highly effective and selective von Hippel-Lindau-based ligand that efficiently degrades the ERRα protein.Formula:C47H50F6N6O7SColor and Shape:SolidMolecular weight:957.0Estrone-N-O-C1-amido
CAS:Estrone-N-O-C1-amido (ERα ligand 1) is an estrogen ligand derived from Estrone that specifically binds to estrogen receptor α (ERα).Formula:C20H26N2O3Purity:98%Color and Shape:SolidMolecular weight:342.439Urotensin II, mouse
CAS:UTS2 is a human gene, alias U-II, on chromosome 1p36.23, codes for Urotensin-II, a potent vasoconstrictor. Formula: C64H85N13O18S2, Molar mass: 1388.6 g/mol.Formula:C76H100N18O19S2Purity:98%Color and Shape:SolidMolecular weight:1633.86PROTAC ERα Degrader-1
PROTAC ERα Degrader-1 is a chemical compound.Formula:C66H69N7O10Purity:98%Color and Shape:SolidMolecular weight:1120.29Arzoxifene
CAS:Arzoxifene (LY353381), an oral SERM, combats breast cancer, supports bone health, and improves lipids, with few side effects.Formula:C28H29NO4SColor and Shape:SolidMolecular weight:475.6Imlunestrant tosylate
CAS:Imlunestrant (LY-3484356) tosylate, an oral SERD, targets ER+ aBC/EEC by blocking estrogen receptors and gene transcription.Formula:C36H32F4N2O6SColor and Shape:SolidMolecular weight:696.71Melanin Concentrating Hormone, salmon
CAS:Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.Formula:C89H139N27O24S4Purity:98%Color and Shape:White PowderMolecular weight:2099.48RS 21314
CAS:RS 21314 is a thiol ester corticosteroid that is topical.Formula:C24H30F2O5SColor and Shape:SolidMolecular weight:468.55Orphanin FQ(1-11)
CAS:Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.Formula:C49H75N15O14Purity:98%Color and Shape:SolidMolecular weight:1098.218-Oxocortisol
CAS:18-Oxocortisol, a naturally occurring mineralocorticoid and adrenal biomarker, is produced by CYP11B2.
Formula:C21H28O6Color and Shape:SolidMolecular weight:376.449ARD-2051
CAS:ARD-2051 is a potent, orally active proteolysis-targeting chimera degrader of the androgen receptor (AR), exhibiting DC50 values of 0.6 nM in degrading ARFormula:C43H45ClN8O5Purity:98%Color and Shape:SolidMolecular weight:789.32Raloxifene 6-Monomethyl Ether
CAS:Compound 7, Raloxifene 6-Monomethyl Ether, blocks estrogen receptor α, inhibits MCF-7 cells; IC50=250 nM, pIC50=6.6.Formula:C29H29NO4SColor and Shape:SolidMolecular weight:487.61Handle region peptide, rat
CAS:Rat handle region peptide acts as prorenin receptor blocker, curbs diabetic kidney disease, and reduces eye inflammation.Formula:C54H101N15O12SPurity:98%Color and Shape:SolidMolecular weight:1184.54PROTAC ER Degrader-15
PROTAC ER Degrader-15 (Compound 40) is an orally active estrogen receptor (ER) degrader with anticancer properties, suitable for breast cancer research.Formula:C47H47F4N5O5Color and Shape:SolidMolecular weight:837.9Dynorphin A (1-8)
CAS:Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.Formula:C46H72N14O10Purity:98%Color and Shape:SolidMolecular weight:981.151-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
CAS:1-Methyl-quinolone alkaloid inhibits DAG acyltransferase, blocks angiotensin II receptor (IC50s: 20.1 & 34.1 μM), and fights H. pylori (MIC: 10 μg/mL).Formula:C23H31NOColor and Shape:SolidMolecular weight:337.5Raloxifene 4'-glucuronide
CAS:Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71[Nphe1]Nociceptin(1-13)NH2
CAS:Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.Formula:C61H100N22O15Purity:98%Color and Shape:SolidMolecular weight:1381.6Olmesartan medoxomil impurity C
CAS:Impurity C of Olmesartan medoxomil is a selective AT1 inhibitor with an IC50 of 66.2 μM.Formula:C29H28N6O5Color and Shape:SolidMolecular weight:540.57Azilsartan Medoxomil Potassium
CAS:Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.Formula:C30H23N4O8·KPurity:99.99%Color and Shape:SolidMolecular weight:606.62Hydrocortisone sodium succinate
CAS:Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.Formula:C25H34NaO8Color and Shape:SolidMolecular weight:485.529L 363564
CAS:L 363564 is a kidney renin inhibitor.Formula:C54H76N12O10Color and Shape:SolidMolecular weight:1053.276ST-CY14
ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.Formula:C139H237N57O31S2Color and Shape:SolidMolecular weight:3266.86PTP1B/AKR1B1-IN-2
PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0Formula:C23H23NO4S2Purity:98%Color and Shape:SolidMolecular weight:441.56AZ 1729
CAS:FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.Formula:C18H16FN5OSColor and Shape:SolidMolecular weight:369.42Estrogen receptor modulator 6
CAS:ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.
Formula:C18H16F2O3Color and Shape:SolidMolecular weight:318.32Ro 64-6198
CAS:Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.Formula:C26H31N3OPurity:98%Color and Shape:SolidMolecular weight:401.54AKR1B10-IN-1
CAS:AKR1B10-IN-1: potent AKR1B10 inhibitor, IC50 3.5 nM; hinders lung cancer cell growth, spread, and Cisplatin resistance.Formula:C19H16FNO4Color and Shape:SolidMolecular weight:341.338UFP-101
CAS:Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.
Formula:C82H138N32O21Purity:98%Color and Shape:SolidMolecular weight:1908.19T4-ATA (S-isomer)
T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.Formula:C19H15I4NO6SPurity:98%Color and Shape:SolidMolecular weight:893.01U-54494A hydrochloride
CAS:U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.Formula:C18H25Cl3N2OColor and Shape:SolidMolecular weight:391.76[Sar1, Ile8]-Angiotensin II TFA
[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.Formula:C48H74F3N13O12Purity:98%Color and Shape:SolidMolecular weight:1082.18Herkinorin
CAS:Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.Formula:C28H30O8Color and Shape:SolidMolecular weight:494.53PROTAC ER Degrader-3
CAS:PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.Formula:C71H77N7O12Purity:98%Color and Shape:SolidMolecular weight:1220.434Alclometasone
CAS:Alclometasone is a glucocorticoid that reduces inflammation and treats various skin conditions like eczema and psoriasis.Formula:C22H29ClO5Purity:98%Color and Shape:SolidMolecular weight:408.92Dynorphin B (1-13)
CAS:Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Formula:C74H115N21O17Purity:98%Color and Shape:SolidMolecular weight:1570.84Antihypertensive agent 3
Antihypertensive agent 3 (compound 4a), an angiotensin II receptor 1 antagonist, demonstrates antihypertensive activity in spontaneously hypertensive rats (SHRsFormula:C16H13NO4SColor and Shape:SolidMolecular weight:315.34Neuropeptide AF (human)
CAS:Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.Formula:C90H132N26O25Purity:98%Color and Shape:SolidMolecular weight:1978.173-Cl-Pyridine-amide-acrylaldehyde-piperazine
3-Cl-Pyridine-amide-acrylaldehyde-piperazine serves as a synthetic intermediate for LO-4-25. LO-4-25 is a ligand for the androgen receptor (AR) DNA binding domain and is linked to a truncated fumaramide handle via a connector. In 22Rv1 cells, LO-4-25 demonstrates potent degradation of both AR and AR-V7.Color and Shape:Odour SolidAntihypertensive agent 2
Antihypertensive agent 2 (Compound 4g) exhibits effective antagonistic activities against angiotensin II receptor 1 and reduces blood pressure with equal orFormula:C22H15NO3Color and Shape:SolidMolecular weight:341.36CTAP
CAS:Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.Formula:C51H69N13O11S2Purity:98%Color and Shape:White Solid/PowderMolecular weight:1104.32SL910102
CAS:SL910102 is a nonpeptide angiotensin antagonist of the AT1 receptor.Formula:C30H30N6OPurity:98%Color and Shape:SolidMolecular weight:490.60β-Naltrexamine dihydrochloride
CAS:β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.Formula:C20H28Cl2N2O3Purity:95.98%Color and Shape:SoildMolecular weight:415.35CTOP
CAS:Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.Formula:C50H67N11O11S2Purity:98%Color and Shape:SolidMolecular weight:1062.28Cebranopadol hemicitrate
CAS:Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.Color and Shape:SolidThyroxine sulfate
CAS:Thyroxine sulfate is a sulfoconjugated derivative of Thyroxine and is also a metabolite of Thyroxine.Formula:C15H11I4NO7SColor and Shape:SolidMolecular weight:856.93Gluten Exorphin B5
CAS:Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.Formula:C30H38N6O7Purity:98%Color and Shape:SolidMolecular weight:594.66Estrogen receptor modulator 13
Estrogen receptor modulator13 (Compound 5D) is an estrogen receptor antagonist with significant cytotoxic effects on MCF7 cells, exhibiting an IC50 value of 8.50 μM. Estrogen receptor modulator13 holds potential for breast cancer research.Formula:C25H19ClN2O2SColor and Shape:SolidMolecular weight:446.08558ARD-69
ARD-69, a potent PROTAC, degrades AR in prostate cancer, with low DC50 values in AR+ cell lines, and suppresses AR gene expression.Formula:C62H74ClFN8O7SColor and Shape:SolidMolecular weight:1129.83Lactandrate
CAS:Lactandrate is a homo-aza-steroidal ester of p-bis(2-chloroethyl) amino phenyl acetic acid.Formula:C31H44Cl2N2O3Color and Shape:SolidMolecular weight:563.67β-Hydroxy-epi-androsterone
CAS:7β-Hydroxy-epi-androsterone (7β-Hydroxy-EpiA) is an endogenous androgenic derivative of dehydroepiandrosterone that possesses the ability to bind to ERβ,Formula:C19H30O3Color and Shape:SolidMolecular weight:306.44CP-472555
CAS:CP-472555 is a selective nonsteroidal glucocorticoid receptor antagonist with anti-GR and anti-obesity activity in animal models.Formula:C31H32N2O2Color and Shape:SolidMolecular weight:464.60[Arg14,Lys15]Nociceptin
CAS:Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.Formula:C82H137N31O22Purity:98%Color and Shape:SolidMolecular weight:1909.18THR-β agonist 6
CAS:THR-β Agonist 6, a selective and orally active compound targeting the thyroid hormone receptor β (THR-β), demonstrates specificity with EC50 values of 0.03 μMFormula:C20H14Cl2N6O3Color and Shape:SolidMolecular weight:457.27β-Endorphin, equine
CAS:Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.Formula:C154H248N42O44SPurity:98%Color and Shape:SolidMolecular weight:3423.94DPP-4/GPR119 modulator 1
CAS:Orally active DPP-4 inhibitor/GPR119 agonist, Compound 22 lowers glucose, moderate hERG inhibition, IC50 4.9 µM, for diabetes research.Formula:C30H39ClN10O3Color and Shape:SolidMolecular weight:623.15Bexirestrant
CAS:Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.Formula:C29H26F3NO2Color and Shape:SolidMolecular weight:477.527Ganoderic acid Df
CAS:Ganoderic acid Df, a lanostane triterpenoid from Ganoderma lucidum, inhibits aldose reductase with IC50 of 22.8 μM.Formula:C30H44O7Color and Shape:SolidMolecular weight:516.67
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