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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3180 products of "Endocrinology/Hormones"

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  • GPR81 agonist 1

    CAS:
    <p>GPR81 agonist 1 is a GPR81 agonist that improves glycaemic control in insulin-resistant mouse models for the study of diabetes and obesity.</p>
    Formula:C22H30N4O2S2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:446.63
  • EM-800

    CAS:
    <p>EM-800, an ERα ligand &amp; prodrug of EM-652, inhibits E1-stimulated ZR-75-1 tumor growth in mice.</p>
    Formula:C39H47NO6
    Color and Shape:Solid
    Molecular weight:625.79
  • JTC-801 free base

    CAS:
    <p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>
    Formula:C26H25N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.5
  • ML138

    CAS:
    <p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>
    Formula:C19H14Cl2N4OS
    Color and Shape:Solid
    Molecular weight:417.31
  • Estrogen receptor antagonist 2

    CAS:
    <p>ER antagonist 2 selectively suppresses ERα, a key breast cancer driver, with research potential in the disease.</p>
    Formula:C26H31F4N5
    Color and Shape:Solid
    Molecular weight:489.55
  • LY88074 Methyl ether

    CAS:
    <p>LY88074 Methyl ether combats estrogen deficit, targeting osteoporosis and hyperlipidemia.</p>
    Formula:C22H16O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.42
  • (R)-Bicalutamide

    CAS:
    <p>(R)-Bicalutamide, an AR antagonist with antitumor properties, is crucial in prostate cancer research.</p>
    Formula:C18H14F4N2O4S
    Color and Shape:Solid
    Molecular weight:430.37
  • Cancer-Targeting Compound 1

    CAS:
    <p>Cancer-Targeting Compound 1 can be used in the study of hormone-related cancers, including the treatment or prevention of fibroids, uterine leiomyomas,</p>
    Formula:C15H13N3O2S
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:299.35
  • Xelaglifam

    CAS:
    <p>Xelaglifam is a potent agonist of G protein-coupled receptor 40 (GPR40) and exhibits hypoglycemic effects.</p>
    Formula:C30H28FNO5
    Color and Shape:Solid
    Molecular weight:501.55
  • GSK1521498 free base

    CAS:
    <p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>
    Formula:C24H20F2N4
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:402.44
  • Norethisterone enanthate

    CAS:
    <p>Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.</p>
    Formula:C27H38O3
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:410.59
  • BMS 183920

    CAS:
    <p>BMS 183920 is a potent Angiotensin II Receptor antagonist that improves improves Caco-2 cell permeability in vivo.</p>
    Formula:C26H19N5O3
    Purity:98.92%
    Color and Shape:Solid
    Molecular weight:449.46
  • GSK1521498 free base (hydrochloride)

    CAS:
    <p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>
    Formula:C24H21ClF2N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.9
  • TAK-875 Hemihydrate

    CAS:
    <p>TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than oleic acid.</p>
    Formula:C29H32O7SH2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:533.63
  • OT antagonist 3

    CAS:
    <p>OT antagonist 3 is an antagonist of oxytocin (OT).</p>
    Formula:C21H20N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.42
  • LY191704

    CAS:
    <p>LY 191704 is a 5α-reductase type 1 inhibitor.</p>
    Formula:C14H16ClNO
    Color and Shape:Solid
    Molecular weight:249.74
  • TUG-905

    CAS:
    <p>TUG-905 is an agonist for free fatty acid receptor 4 (FFA4/GPR120), and TUG-905 has the potential to treat agitation.</p>
    Formula:C27H30FNO5S
    Color and Shape:Solid
    Molecular weight:499.59
  • AT2R antagonist 1

    CAS:
    <p>AT2R antagonist 1: potent, selective ligand, Ki 29 nM, inhibits CYP enzymes, stable in liver microsomes.</p>
    Formula:C23H30N4O4S2
    Color and Shape:Solid
    Molecular weight:490.64
  • GSK1521498

    CAS:
    <p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>
    Formula:C24H23F2N4O4P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.43
  • Org30958

    CAS:
    <p>Org30958 is a potent inhibitor of aromatase in vivo.</p>
    Formula:C21H30O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.59
  • Estrogen receptor antagonist 1

    CAS:
    <p>"Potent estrogen receptor blocker with promise for breast cancer treatment per WO2021249533A1."</p>
    Formula:C28H33F4N5
    Color and Shape:Solid
    Molecular weight:515.59
  • (R)-DPN

    CAS:
    <p>estrogen receptor (ER) β agonist</p>
    Formula:C15H13NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.27
  • MK181

    CAS:
    <p>MK181 is an inhibitor of AKR1B10, a tumor marker and promising antineoplastic target.</p>
    Formula:C16H13BrClNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.64
  • GSK1104252A

    CAS:
    <p>GSK1104252A is a potent and selective agonist of GPR119.</p>
    Formula:C22H27FN4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:478.54
  • DIPPA hydrochloride

    CAS:
    <p>κ receptor antagonist</p>
    Formula:C22H24Cl3N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:484.87
  • Gumelutamide

    CAS:
    <p>Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.</p>
    Formula:C22H21ClN6O
    Color and Shape:Solid
    Molecular weight:420.89
  • Methylprednisolone Aceponate

    CAS:
    <p>Methylprednisolone Aceponate (SH 440), a non-halogenated corticosteroid, is a potent anti-inflammatory agent.</p>
    Formula:C27H36O7
    Purity:99.00% - 99.61%
    Color and Shape:Solid
    Molecular weight:472.57
  • DDD028

    CAS:
    <p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>
    Formula:C20H20N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.39
  • MK-3984

    CAS:
    <p>MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.</p>
    Formula:C17H12F7NO2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:395.27
  • LY117018

    CAS:
    <p>LY117018 shows antiproliferative effects on breast cancer cell lines. LY117018 is a Raloxifene analog and is a selective estrogen receptor modulator.</p>
    Formula:C27H25NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.56
  • Aldose reductase-IN-5

    CAS:
    <p>Aldose reductase-IN-5 inhibits ALR2, boosts inhibitory response and antioxidants, slowing diabetes complications.</p>
    Formula:C18H15NO5
    Color and Shape:Solid
    Molecular weight:325.32
  • ALR2-IN-2


    <p>ALR2-IN-2 inhibits ALR2 (27 nM IC50) &amp; ALR1 (228 nM IC50), used in diabetes complication research.</p>
    Formula:C17H11FN2O2S2
    Color and Shape:Solid
    Molecular weight:358.41
  • AT1R antagonist 1

    CAS:
    <p>AT1R Antagonist 1 (compound 10) serves as a potent, selective ligand for AT1R with considerable affinity, demonstrated by a K i value of 8.5 nM [1].</p>
    Formula:C28H32F3N5O4S2
    Color and Shape:Solid
    Molecular weight:623.71
  • SB 611812

    CAS:
    <p>SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.</p>
    Formula:C17H16Cl3F3N2O3S
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:491.74
  • Glucocorticoid receptor-IN-2

    CAS:
    <p>Glucocorticoid receptor-IN-2 selectively targets GR with anti-inflammatory effects (IC50: 0.171 nM) and activates MMTV (EC50: 0.94 nM).</p>
    Formula:C25H20F4N6O2
    Color and Shape:Solid
    Molecular weight:512.46
  • D-Methionine sulfoxide

    CAS:
    <p>D-Methionine sulfoxide inhibits peptide methionine sulfoxide reductase and can be used to inhibit ochre mites.D-Methionine sulfoxide can be added to chicken</p>
    Formula:C5H11NO3S
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:165.21
  • OP-1074

    CAS:
    <p>OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.</p>
    Formula:C29H31NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.56
  • Levormeloxifene

    CAS:
    <p>Levormeloxifene is a selective modulator of the estrogen receptor. It inhibits the production of vaginal tropoelastin and transforming growth factor-beta 1.</p>
    Formula:C30H35NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.6
  • L 158809

    CAS:
    <p>L 158809 is an antagonist of the angiotensin II type 1 receptor.</p>
    Formula:C24H23N7
    Color and Shape:Solid
    Molecular weight:409.49
  • OBHS

    CAS:
    <p>OBHS is an inhibitor of estrogen receptor alpha (ERα).</p>
    Formula:C24H20O6S
    Color and Shape:Solid
    Molecular weight:436.48
  • Nitromifene

    CAS:
    <p>Nitromifene is the estrogen receptor antagonist.</p>
    Formula:C27H28N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.52
  • A 81282

    CAS:
    <p>A 81282 is a selective antagonist of angiotensin receptors. It has the activity of lowering blood pressure.</p>
    Formula:C23H23N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.47
  • (±)-AC 7954 hydrochloride

    CAS:
    <p>(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.</p>
    Formula:C19H21Cl2NO2
    Purity:99.42%
    Color and Shape:White Solid
    Molecular weight:366.28
  • DK3

    CAS:
    <p>DK3 is a potent and selective agonist of estrogen-related receptor alpha (ERRα). ERRα is a potential drug target for cancer and metabolic diseases [1].</p>
    Formula:C16H14N2O2
    Color and Shape:Solid
    Molecular weight:266.29
  • SHR1653

    CAS:
    <p>SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR).</p>
    Formula:C21H21ClFN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.88
  • Capesaris

    CAS:
    <p>Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.</p>
    Formula:C19H13F2NO3
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:341.31
  • Androgen receptor antagonist 1

    CAS:
    <p>Androgen receptor antagonist 1, an oral full AR antagonist (IC50 59 nM), for PROTAC synthesis, reducing AR protein by 24–47% in LNCaP cells at 1–10 μM.</p>
    Formula:C21H25ClN4O3
    Purity:99.054%
    Color and Shape:Solid
    Molecular weight:416.9
  • PF-4455242 HCl

    CAS:
    <p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>
    Formula:C21H29ClN2O2S
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:408.99
  • SB-568849

    CAS:
    <p>SB-568849 is a melanin-concentrating hormone receptor 1 antagonist (pKi: 7.7).</p>
    Formula:C28H31F3N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.55
  • Dimethomorph

    CAS:
    <p>Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .</p>
    Formula:C21H22ClNO4
    Purity:99.2%
    Color and Shape:Solid Crystalline
    Molecular weight:387.86
  • FSHR agonist 1

    CAS:
    <p>FSHR agonist 1: high-affinity, allosteric FSHR activator, pEC50 of 7.72, interacts with TMD.</p>
    Formula:C26H33N3O3S
    Color and Shape:Solid
    Molecular weight:467.62
  • MCH-1 antagonist 1

    CAS:
    <p>MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).</p>
    Formula:C25H26N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.5
  • CP-866087

    CAS:
    <p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>
    Formula:C24H28N2O2
    Purity:99.56% - >99.99%
    Color and Shape:Soild
    Molecular weight:376.49
  • SB 706375

    CAS:
    <p>urotensin-II (UT) receptor antagonist</p>
    Formula:C20H22BrF3N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:539.36
  • ATC0065 HCl

    CAS:
    <p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>
    Formula:C25H31BrCl2F3N5O
    Color and Shape:Solid
    Molecular weight:625.35
  • GPR84 antagonist 8

    CAS:
    <p>GPR84 antagonist 8 is a selective GPR84 antagonist applicable for investigating inflammatory and fibrotic diseases.</p>
    Formula:C23H23N3O5
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:421.45
  • J9

    CAS:
    <p>J9 is an inhibitor of Glucocorticoid resistance. J9 reverses Dexamethasone Resistance in T-cell Acute Lymphoblastic Leukemia.</p>
    Formula:C12H12N4
    Color and Shape:Solid
    Molecular weight:212.25
  • Camizestrant

    CAS:
    <p>Camizestrant (Estrogen receptor antagonist 2) is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].</p>
    Formula:C24H28F4N6
    Purity:97.25% - 99.57%
    Color and Shape:Solid
    Molecular weight:476.51
  • L 366682

    CAS:
    <p>L 366682 is an oxytocin antagonist.</p>
    Formula:C40H53N9O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:755.91
  • OT antagonist 1

    CAS:
    <p>OT antagonist 1 is a potent and selective antagonist of Oxytocin(Ki of 50 nM)</p>
    Formula:C22H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:390.44
  • VPC-13789

    CAS:
    <p>VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.</p>
    Formula:C21H16F3N3O
    Color and Shape:Solid
    Molecular weight:383.37
  • Axomadol

    CAS:
    <p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>
    Formula:C16H25NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.37
  • (R,R)-THC

    CAS:
    <p>agonist at ERα receptor and antagonist at ERβ receptor</p>
    Formula:C22H24O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.42
  • LY285434

    CAS:
    <p>LY285434 is a suitable angiotensin II receptor antagonist.</p>
    Formula:C23H25N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.48
  • Chlorothalonil

    CAS:
    <p>Chlorothalonil (DAC 2787): Broad-spectrum, efficient, low-toxicity fungicide for fruits, vegetables, rice, wheat, cotton.</p>
    Formula:C8Cl4N2
    Purity:98.01% - 98.71%
    Color and Shape:Colorless Crystals Solid
    Molecular weight:265.91
  • D36

    CAS:
    <p>D36 is an androgen receptor allosteric antagonist. It also has inverse agonist properties.</p>
    Formula:C21H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.43
  • FERb 033

    CAS:
    <p>ERβ receptor agonist</p>
    Formula:C13H9ClFNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:281.67
  • BTI-A-404

    CAS:
    <p>BTI-A-404 is a potent and selective competitive inverse agonist of human GPR43.</p>
    Formula:C22H26N4O2
    Color and Shape:Solid
    Molecular weight:378.47
  • CPSA

    CAS:
    <p>CPSA is an effective and selective AKR1C1 inhibitor.</p>
    Formula:C13H9ClO3
    Color and Shape:Solid
    Molecular weight:248.66
  • MK-4541

    CAS:
    <p>MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.</p>
    Formula:C22H31F3N2O3
    Color and Shape:Solid
    Molecular weight:428.49
  • SCH 221510

    CAS:
    <p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>
    Formula:C28H31NO
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:397.55
  • VPC-3033

    CAS:
    <p>VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.</p>
    Formula:C21H14O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:298.33
  • CR-665 Acetate

    CAS:
    <p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>
    Formula:C38H53N9O6
    Color and Shape:Solid
    Molecular weight:731.899
  • Dehydro Olmesartan

    CAS:
    <p>Dehydro Olmesartan, from Olmesartan, is an AT1R blocker for researching hypertension.</p>
    Formula:C24H24N6O2
    Color and Shape:Solid
    Molecular weight:428.49
  • KB-130015

    CAS:
    <p>KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.</p>
    Formula:C18H14I2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.11
  • RU 43044

    CAS:
    <p>RU 43044 is a selective glucocorticoid receptor antagonist that has exhibited an antidepressant-like effect.</p>
    Formula:C29H34O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58
  • LY 281217

    CAS:
    <p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>
    Formula:C32H42N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:578.7
  • Idoxifene

    CAS:
    <p>Idoxifene is a tissue-specific selective estrogen receptor modulator.</p>
    Formula:C28H30INO
    Color and Shape:Solid
    Molecular weight:523.45
  • L-366509

    CAS:
    <p>L-366,509 is an antagonist of oxytocin.</p>
    Formula:C25H33NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.6
  • Cyprodinil

    CAS:
    <p>Cyprodinil is a fungicide blocking methionine synthesis in fungi and hinders B. cinerea, P. herpotrichoides, H. oryzae growth; it's also an AR agonist.</p>
    Formula:C14H15N3
    Color and Shape:Solid
    Molecular weight:225.29
  • Dup 747

    CAS:
    <p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>
    Formula:C24H28Cl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.4
  • Androgen receptor antagonist 3

    CAS:
    <p>Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].</p>
    Formula:C22H18ClN
    Color and Shape:Solid
    Molecular weight:331.84
  • BMS-986124

    CAS:
    <p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>
    Formula:C16H15BrClNO3S2
    Color and Shape:Solid
    Molecular weight:448.78
  • Aldose reductase-IN-4

    CAS:
    <p>Aldose reductase-IN-4 (compund IIc) is an inhibitor of aldose reductase with IC50s of 11.70 μM and 0.98 μM for ALR1 and ALR2, respectively [1].</p>
    Formula:C14H10FNO3S
    Color and Shape:Solid
    Molecular weight:291.3
  • Aldose reductase-IN-6

    CAS:
    <p>AR inhibitor Aldose reductase-IN-6: IC50 3.164 μM, Ki 0.018 μM, non-toxic to normal cells.</p>
    Formula:C20H16N4O2S
    Color and Shape:Solid
    Molecular weight:376.43
  • BMS-819881

    CAS:
    <p>BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for</p>
    Formula:C24H21ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.95
  • Olmesartan methyl ester

    CAS:
    <p>Olmesartan methyl ester: an intermediate for synthesizing Olmesartan medoxomil, a strong AT1 receptor blocker.</p>
    Formula:C25H28N6O3
    Color and Shape:Solid
    Molecular weight:460.53
  • Fenhexamid

    CAS:
    <p>Fenhexamid (Elevate), a sterol biosynthesis inhibitor, shows antifungal activity against the plant pathogenic fungus.</p>
    Formula:C14H17Cl2NO2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:302.20
  • DK1

    CAS:
    <p>DK1: potent ERRα modulator, lowers blood glucose, promising for diabetes research.</p>
    Formula:C16H13ClN2O2
    Color and Shape:Solid
    Molecular weight:300.74
  • GPR40 agonist 1

    CAS:
    <p>GPR40 agonist 1 is an effective new GPR40 agonist (EC50s: 17 nM and 2 nM for rGPR40 and hGPR40).</p>
    Formula:C27H30FN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.54
  • Endomorphin 1 acetate

    CAS:
    <p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>
    Formula:C36H42N6O7
    Color and Shape:Solid
    Molecular weight:670.75
  • SIM-688

    CAS:
    <p>SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).</p>
    Formula:C34H31F3N2O2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:556.62
  • ORL1 antagonist 1

    CAS:
    <p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>
    Formula:C20H22ClN5
    Purity:98.92%
    Color and Shape:Solid
    Molecular weight:367.88
  • Opioid receptor modulator 1

    CAS:
    <p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>
    Formula:C18H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.38
  • L-159282

    CAS:
    <p>L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity.</p>
    Formula:C30H28N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:524.63
  • Estrogen receptor-IN-1

    CAS:
    <p>Estrogen receptor-IN-1 (compound 16) is an effective estrogen receptor (ER) inhibitor with IC 50 s of 13, 5μM for ERα and Erβ, respectively [1].</p>
    Formula:C14H16OSi
    Color and Shape:Solid
    Molecular weight:228.36
  • Tolonidine

    CAS:
    <p>Tolonidine is orally active and has been shown to possess hypotensive. Tolonidine is a derivative of imidazoline.</p>
    Formula:C10H12ClN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.68
  • LY2048978

    CAS:
    <p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>
    Formula:C19H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.41
  • RU 45144

    CAS:
    <p>RU 45144 is an estradiol derivative with antiestrogenic activity.</p>
    Formula:C28H37NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.6
  • AZD7268

    CAS:
    <p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>
    Formula:C29H30N4O2S
    Color and Shape:Solid
    Molecular weight:498.64