Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
Show 6 more subcategories
Found 3180 products of "Endocrinology/Hormones"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Azilsartan Medoxomil Potassium
CAS:<p>Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.</p>Formula:C30H23N4O8·KPurity:98.72%Color and Shape:SolidMolecular weight:606.62Neuropeptide AF (human)
CAS:<p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>Formula:C90H132N26O25Purity:98%Color and Shape:SolidMolecular weight:1978.17Saralasin
CAS:<p>Competitive non-selective angiotensin II antagonist.</p>Formula:C42H65N13O10Purity:98%Color and Shape:PowderMolecular weight:912Ac-RYYRWK-NH2
CAS:<p>Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.</p>Formula:C49H69N15O9Purity:98%Color and Shape:SolidMolecular weight:1012.17[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Formula:C63H101F3N22O17Color and Shape:SolidMolecular weight:1495.61hFSH-β-(33-53) (TFA)
<p>hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist.</p>Formula:C115H183N31O32SxC2HF3O2Color and Shape:SolidMolecular weight:2657.96Boc-ypgflt(O-tbu)
CAS:<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Formula:C44H64N6O11Color and Shape:SolidMolecular weight:853.01Faznolutamide
CAS:<p>Faznolutamide is an antiandrogen agent [1] [2] .</p>Formula:C19H17FN4O2SColor and Shape:SolidMolecular weight:384.43RLA-5331
<p>RLA-5331: iron activator with anti-androgen properties; inhibits mCRPC cell proliferation.</p>Formula:C40H43F3N6O7SColor and Shape:SolidMolecular weight:808.871-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone
CAS:<p>Methyl-2-quinolone from Evodia rutaecarpa blocks angiotensin II receptor with 48.2 μM IC50.</p>Formula:C25H35NOColor and Shape:SolidMolecular weight:365.55Deacylcortivazol
CAS:<p>Deacylcortivazol is a potent glucocorticoid that inhibits growth in glucocorticoid-resistant leukemia cells without receptor mediation.</p>Formula:C30H36N2O4Color and Shape:SolidMolecular weight:488.62PD 132002
CAS:<p>PD 132002 is a renin inhibitor.</p>Formula:C31H50N4O9SColor and Shape:SolidMolecular weight:654.82PROTAC ERα Y537S degrader-1
CAS:<p>PROTAC ERα Y537S degrader-1 comprises a ubiquitin E3 ligase binding group, a linker and a protein binding group.</p>Formula:C46H49N5O6Color and Shape:SolidMolecular weight:767.91PROTAC ERα Degrader-7
CAS:<p>PROTAC ERα Degrader-7 (Compound i-320) is a powerful PROTAC degrader targeting the estrogen receptor alpha (ERα), exhibiting a DC50 of 0.000006 µM. This compound consists of a cereblon-binding segment, LBM, connected to ERBM, an ERα-binding ligand that includes a benzofused partially saturated 6-membered carbocyclic or heterocyclic ring [1].</p>Formula:C46H49F2N5O4Color and Shape:SolidMolecular weight:773.91Angiotensin II (1-4), human
CAS:<p>Angiotensin II constricts blood vessels and boosts blood pressure by escalating norepinephrine release.</p>Formula:C24H37N7O8Purity:98%Color and Shape:SolidMolecular weight:551.59Glucocorticoids receptor agonist 2
CAS:<p>Arylpyrazole-based glucocorticoid agonist with potent anti-inflammatory effects; doesn't affect insulin secretion.</p>Formula:C25H25FN2OColor and Shape:SolidMolecular weight:388.48SNIPER(ER)-110
<p>SNIPER(ER)-110 links cIAP1 and estrogen ligands. SNIPER(ER)-51 degrades ER protein; DC50 <3 nM at 4h, 7.7 nM at 48h.</p>Formula:C66H83N5O11Purity:98%Color and Shape:SolidMolecular weight:1122.39Retosiban
CAS:<p>Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).</p>Formula:C27H34N4O5Purity:98%Color and Shape:SolidMolecular weight:494.58Olmesartan impurity
CAS:<p>Olmesartan impurity, related to parent RNH-6270, is an AT1R antagonist used for hypertension research.</p>Formula:C33H26N4OColor and Shape:SolidMolecular weight:494.598Cgp 44099
CAS:<p>Cgp 44099 is a potent plasma renin inhibitor from all subprimate species.</p>Formula:C69H104N14O13Purity:98%Color and Shape:SolidMolecular weight:1337.676PD 125967
CAS:<p>PD 125967 is a renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.</p>Formula:C51H67N5O4Color and Shape:SolidMolecular weight:814.11TF-505
CAS:<p>TF-505, a steroid 5α-reductase inhibitor, is used potentially for the treatment of benign prostatic hyperplasia.</p>Formula:C33H37NO4Purity:98%Color and Shape:SolidMolecular weight:511.65D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Formula:C25H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:410.98RS 21314
CAS:<p>RS 21314 is a thiol ester corticosteroid that is topical.</p>Formula:C24H30F2O5SColor and Shape:SolidMolecular weight:468.55PROTAC ERRα Degrader-3
CAS:<p>PROTAC ERRα Degrader-3 is a highly effective and selective von Hippel-Lindau-based ligand that efficiently degrades the ERRα protein.</p>Formula:C47H50F6N6O7SColor and Shape:SolidMolecular weight:957.0ARD-2585
CAS:<p>ARD-2585 is an orally active and selective androgen receptor PROTAC degrader with anticancer activity for the study of prostate cancer.</p>Formula:C41H43ClN8O5Color and Shape:SolidMolecular weight:763.28Urotensin II, mouse
CAS:<p>UTS2 is a human gene, alias U-II, on chromosome 1p36.23, codes for Urotensin-II, a potent vasoconstrictor. Formula: C64H85N13O18S2, Molar mass: 1388.6 g/mol.</p>Formula:C76H100N18O19S2Purity:98%Color and Shape:SolidMolecular weight:1633.86Estrone-N-O-C1-amido
CAS:<p>Estrone-N-O-C1-amido (ERα ligand 1) is an estrogen ligand derived from Estrone that specifically binds to estrogen receptor α (ERα).</p>Formula:C20H26N2O3Purity:98%Color and Shape:SolidMolecular weight:342.439PROTAC ERα Degrader-1
<p>PROTAC ERα Degrader-1 is a chemical compound.</p>Formula:C66H69N7O10Purity:98%Color and Shape:SolidMolecular weight:1120.29Arzoxifene
CAS:<p>Arzoxifene (LY353381), an oral SERM, combats breast cancer, supports bone health, and improves lipids, with few side effects.</p>Formula:C28H29NO4SColor and Shape:SolidMolecular weight:475.6OT-R antagonist 1
CAS:<p>OT-R antagonist 1: Nonpeptide, selective, low-weight blocker of oxytocin; IC50 = 8 nM for Ca2+ disruption.</p>Formula:C28H29N3O4Purity:98%Color and Shape:SolidMolecular weight:471.55Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formula:C49H75N15O14Purity:98%Color and Shape:SolidMolecular weight:1098.2ARD-2051
CAS:<p>ARD-2051 is a potent, orally active proteolysis-targeting chimera degrader of the androgen receptor (AR), exhibiting DC50 values of 0.6 nM in degrading AR</p>Formula:C43H45ClN8O5Purity:98%Color and Shape:SolidMolecular weight:789.32Raloxifene 6-Monomethyl Ether
CAS:<p>Compound 7, Raloxifene 6-Monomethyl Ether, blocks estrogen receptor α, inhibits MCF-7 cells; IC50=250 nM, pIC50=6.6.</p>Formula:C29H29NO4SColor and Shape:SolidMolecular weight:487.61PROTAC ER Degrader-15
<p>PROTAC ER Degrader-15 (Compound 40) is an orally active estrogen receptor (ER) degrader with anticancer properties, suitable for breast cancer research.</p>Formula:C47H47F4N5O5Color and Shape:SolidMolecular weight:837.9Dynorphin A (1-8)
CAS:<p>Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.</p>Formula:C46H72N14O10Purity:98%Color and Shape:SolidMolecular weight:981.15Raloxifene 4'-glucuronide
CAS:<p>Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.</p>Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71BWA-6047
<p>BWA-6047 is a dual AR/AR-V7 and GSPT1 PROTAC-type degrader (AR: DC50= 3.7 nM; AR-V7: DC50= 3.0 nM; GSPT1: DC50= 1.2 nM). It facilitates the ubiquitination and degradation of AR/AR-V7 and, through molecular glue properties, induces a PPI between GSPT1 and CRBN, leading to GSPT1 degradation. BWA-6047 is applicable in prostate cancer research.</p>Formula:C42H46ClN5O7Color and Shape:SolidMolecular weight:767.30858Bufrolin
CAS:<p>Bufrolin is a potent GPR35 agonist, mast cell stabilizer, and anti-inflammatory research agent.</p>Formula:C18H16N2O6Color and Shape:SolidMolecular weight:356.33ERα degrader 10
<p>ERα degrader10 is a potent, selective, orally active estrogen receptor α (ERα) degrader. It demonstrates strong ERα binding affinity (IC50 of 24.0 nM) and degradation capability (EC50 of 5.3 nM). This compound degrades ERα through a proteasome-mediated pathway and is utilized in breast cancer research.</p>Color and Shape:Odour SolidHydrocortisone sodium succinate
CAS:<p>Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.</p>Formula:C25H34NaO8Color and Shape:SolidMolecular weight:485.529L 363564
CAS:<p>L 363564 is a kidney renin inhibitor.</p>Formula:C54H76N12O10Color and Shape:SolidMolecular weight:1053.276PTP1B/AKR1B1-IN-2
<p>PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0</p>Formula:C23H23NO4S2Purity:98%Color and Shape:SolidMolecular weight:441.56Ro 64-6198
CAS:<p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.</p>Formula:C26H31N3OPurity:98%Color and Shape:SolidMolecular weight:401.54AZ 1729
CAS:<p>FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.</p>Formula:C18H16FN5OSColor and Shape:SolidMolecular weight:369.42Estrogen receptor modulator 6
CAS:<p>ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.</p>Formula:C18H16F2O3Color and Shape:SolidMolecular weight:318.32[Sar1, Ile8]-Angiotensin II TFA
<p>[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.</p>Formula:C48H74F3N13O12Purity:98%Color and Shape:SolidMolecular weight:1082.18ZINC05925939
<p>ZINC05925939 is an estrogen receptor β (ESR2) inhibitor used in breast cancer research.</p>Formula:C17H17NO2Color and Shape:SolidMolecular weight:267.32UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Formula:C82H138N32O21Purity:98%Color and Shape:SolidMolecular weight:1908.19T4-ATA (S-isomer)
<p>T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.</p>Formula:C19H15I4NO6SPurity:98%Color and Shape:SolidMolecular weight:893.01Norleual
CAS:<p>Angiotensin IV analog, potent HGF/c-MET inhibitor (IC50=3 pM), halts MDCK cell growth and invasion, AT4 antagonist, impairs LTP, antiangiogenic.</p>Formula:C41H58N8O7Purity:98%Color and Shape:SolidMolecular weight:774.95Herkinorin
CAS:<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Formula:C28H30O8Color and Shape:SolidMolecular weight:494.53PROTAC ER Degrader-3
CAS:<p>PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.</p>Formula:C71H77N7O12Purity:98%Color and Shape:SolidMolecular weight:1220.434Methylpiperidino pyrazole
CAS:<p>Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.</p>Formula:C29H31N3O3Purity:98.84%Color and Shape:SolidMolecular weight:469.57[Orn5]-URP
CAS:<p>Urotensin-II receptor antagonist, no agonist effect, pEC50 7.24, blocks U-II in rat aorta assay.</p>Formula:C48H62N10O10S2Purity:98%Color and Shape:SolidMolecular weight:1003.2PL-017
CAS:<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Formula:C29H37N5O5Purity:98%Color and Shape:SolidMolecular weight:535.64[Met5]-Enkephalin, amide
CAS:<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Formula:C27H36N6O6SPurity:98%Color and Shape:SolidMolecular weight:572.68(Rac)-SNC80
CAS:<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Formula:C28H39N3O2Color and Shape:SolidMolecular weight:449.63Melanin Concentrating Hormone, salmon TFA
<p>MCH (salmon) TFA is a 19-amino-acid neuropeptide affecting appetite, energy, sleep, and heart health via GPCR SLC-1/GPR24 and MCHR2.</p>Formula:C91H140F3N27O26S4Color and Shape:SolidMolecular weight:2213.5(Rac)-Finerenone
CAS:<p>Rac-Finerenone, or (Rac)-BAY 94-8862, is an oral nonsteroidal MR antagonist with high selectivity and an IC50 of 18 nM.</p>Formula:C21H22N4O3Color and Shape:SolidMolecular weight:378.432Montirelin
CAS:<p>Montirelin is an analog of thyrotropin-releasing hormone.</p>Formula:C17H24N6O4SColor and Shape:SolidMolecular weight:408.483-Cl-Pyridine-amide-acrylaldehyde-piperazine
<p>3-Cl-Pyridine-amide-acrylaldehyde-piperazine serves as a synthetic intermediate for LO-4-25. LO-4-25 is a ligand for the androgen receptor (AR) DNA binding domain and is linked to a truncated fumaramide handle via a connector. In 22Rv1 cells, LO-4-25 demonstrates potent degradation of both AR and AR-V7.</p>Color and Shape:Odour SolidAkuammicine
CAS:<p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>Formula:C20H22N2O2Color and Shape:SolidMolecular weight:322.408Glucocorticoids receptor agonist 1
CAS:<p>GRA-1, an arylpyrazole, is a potent glucocorticoid receptor agonist with robust anti-inflammatory effects and preserves insulin secretion.</p>Formula:C20H23FN2OColor and Shape:SolidMolecular weight:326.41CP 85339
CAS:<p>CP 85339 is an aspartic acid protease inhibitor for X-ray analysis of peptide-renin complexes.</p>Formula:C31H49ClN4O6SColor and Shape:SolidMolecular weight:641.26Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formula:C31H41N7O9Purity:98%Color and Shape:SolidMolecular weight:655.709Brain Natriuretic Peptide (1-32), rat
CAS:<p>Rat Brain Natriuretic Peptide (1-32) is a 32-amino-acid peptide from heart, released when ventricles stretch excessively.</p>Formula:C146H239N47O44S3Purity:98%Color and Shape:SolidMolecular weight:3452.944',2-Dihydroxy-4,6-dimethoxydihydrochalcone
CAS:<p>4',2-Dihydroxy-4,6-dimethoxydihydrochalcone, an estrogen-like compound, binds to bovine estrogen receptors, IC50 15 μM.</p>Formula:C17H18O5Color and Shape:SolidMolecular weight:302.32Lyciumin A
CAS:<p>Lyciumin A, a cyclic octapeptide, inhibits proteases and could aid in hypertension studies.</p>Formula:C42H51N9O12Color and Shape:SolidMolecular weight:873.921[(pF)Phe4]Nociceptin(1-13)NH2
CAS:<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Formula:C61H99FN22O15Purity:98%Color and Shape:SolidMolecular weight:1399.6PSDalpha
<p>PSDalpha, a conjugate of PS, TB, and 17β-estradiol, degrades ERα with peak absorption at 465 nm, effectively inhibiting MCF-7 cell growth.</p>Formula:C44H39N3O2SColor and Shape:SolidMolecular weight:673.86PROTAC ERRα Degrader-2
CAS:<p>PROTAC ERRα Degrader-2 is a compound consisting of an MDM2 ligand binding group, a linker, and an estrogen-related receptor alpha (ERRα) binding group.</p>Formula:C57H55Cl2F6N7O8Purity:98%Color and Shape:SolidMolecular weight:1150.99Aliskiren D6 Hydrochloride
CAS:<p>Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).</p>Formula:C30H54ClN3O6Purity:98%Color and Shape:SolidMolecular weight:594.26Rofleponide
CAS:<p>Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.</p>Formula:C25H34F2O6Purity:99.32%Color and Shape:SolidMolecular weight:468.53Dermorphin Analog
<p>Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.</p>Formula:C44H59N11O10Purity:98%Color and Shape:SolidMolecular weight:901.43Imidaprilate
CAS:<p>Imidaprilate, an active TA-6366 metabolite, is a potent ACE inhibitor with an IC50 of 2.6 nM, researched for hypertension.</p>Formula:C18H23N3O6Purity:98%Color and Shape:SolidMolecular weight:377.39Potassium Channel Targeted Library
<p>A unique collection of xnum potassium channel blockers and agonists for high throughput and high content screening;</p>Color and Shape:Odour SolidAngiotensin II (5-8), human
CAS:<p>Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II</p>Formula:C26H36N6O5Purity:98%Color and Shape:SolidMolecular weight:512.6Dipropyl phthalate
CAS:<p>Dipropyl phthalate is a weak androgen receptor inhibitor, and can be used in biochemical experiments and drug synthesis.</p>Formula:C14H18O4Purity:98.62%Color and Shape:SolidMolecular weight:250.29UFP-803
CAS:<p>UT receptor ligand acts mainly as silent antagonist with slight agonist effects; blocks U-II in rat aorta, pIC50 = 7.46, & inhibits plasma leakage in mice.</p>Formula:C50H64N10O12S2Purity:98%Color and Shape:SolidMolecular weight:1061.24[Ala17]-MCH
CAS:<p>Potent MCH receptor agonist with EC50 of 17 nM (MCH1) & 54 nM (MCH2); prefers MCH1 (Ki 0.16 nM) over MCH2 (Ki 34 nM).</p>Formula:C97H155N29O26S4Purity:98%Color and Shape:SolidMolecular weight:2271.71Aclerastide
CAS:<p>Aclerastide, an angiotensin receptor agonist, decreases fibrosis in wounds; effect increases with use duration, blocked by AT antagonist.</p>Formula:C42H64N12O11Color and Shape:SolidMolecular weight:913.03Yp537
CAS:<p>Yp537 acts as an estrogen receptor (ER) inhibitor, specifically preventing the dimerization of the human estrogen receptor [1].</p>Formula:C64H104N13O22PSColor and Shape:SolidMolecular weight:1470.62Methylprednisolone Acetate
<p>Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.</p>Formula:C24H32O6Purity:99.74%Color and Shape:Off-White SolidMolecular weight:416.51Nurr1 agonist 2
CAS:<p>Nurr1 agonist 2 with EC50 of 0.07 μM, boosts TH & VMAT2 mRNA, binds Nurr1 LBD at Kd 0.14 μM, for parkinsonism study.</p>Formula:C18H14O3SPurity:98.78%Color and Shape:SoildMolecular weight:310.37Axelopran
CAS:<p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>Formula:C26H39N3O4Color and Shape:SolidMolecular weight:457.61Cgp 38560
CAS:<p>CGP 38560 is a potent renin inhibitor.</p>Formula:C40H67N5O9S2Color and Shape:SolidMolecular weight:826.12Raloxifene 6-glucuronide
CAS:<p>Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8.</p>Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71GPR88 agonist 2
<p>GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].</p>Color and Shape:Odour SolidGLL 398
CAS:<p>GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.</p>Formula:C25H23BO4Purity:98%Color and Shape:SolidMolecular weight:398.26BI 653048
CAS:<p>BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.</p>Formula:C23H25F4N3O4SPurity:98%Color and Shape:SolidMolecular weight:515.523-epi-25-hydroxy Vitamin D3
CAS:<p>3-epi-25-hydroxy Vitamin D3 lowers serum PTH in male weanling rats at 0.5 and 1 IU/g doses; doesn't affect females.</p>Formula:C27H44O2Color and Shape:SolidMolecular weight:400.64DAMGO (TFA)
CAS:<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Formula:C28H36F3N5O8Purity:98%Color and Shape:SolidMolecular weight:627.61Linuron
CAS:<p>Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.</p>Formula:C9H10Cl2N2O2Purity:99.08%Color and Shape:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An HerbicideMolecular weight:249.09OT-R antagonist 2
CAS:<p>OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .</p>Formula:C28H29N3O4Purity:98%Color and Shape:SolidMolecular weight:471.55GNE-274
CAS:<p>GNE-274, akin to GDC-0927 but non-degrading, is a partial ER agonist in breast cancer, enhancing chromatin at ER sites, inhibiting ER-LBD.</p>Formula:C29H31NO4Color and Shape:SolidMolecular weight:457.57Galloylalbiflorin
CAS:<p>Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.</p>Formula:C30H32O15Color and Shape:SolidMolecular weight:632.57PTP1B/AKR1B1-IN-1
<p>PTP1B/AKR1B1-IN-1 is a dual inhibitor targeting protein tyrosine phosphatase 1B (PTP1B) and aldose reductase (AKR1B1), exhibiting inhibitory potency with IC50s</p>Formula:C22H21NO4S2Purity:98%Color and Shape:SolidMolecular weight:427.54BigLEN(mouse)
CAS:<p>GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.</p>Formula:C78H130N24O22Purity:98%Color and Shape:SolidMolecular weight:1756.03ODM-204
CAS:<p>ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).</p>Formula:C20H21F3N4Purity:98%Color and Shape:SolidMolecular weight:374.40
![1-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT38593.webp&w=3840&q=75)
![[Orn5]-URP](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1928.webp&w=3840&q=75)
![[Met5]-Enkephalin, amide](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1255.webp&w=3840&q=75)
![[(pF)Phe4]Nociceptin(1-13)NH2](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1885.webp&w=3840&q=75)
![[Ala17]-MCH](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1997.webp&w=3840&q=75)
