Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(207 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(296 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3178 products of "Endocrinology/Hormones"
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Commendamide
CAS:<p>Commendamide, natural, mimics N-acyl-amides, activates GPR132 with EC50 of 11.8 μM, made by Cbeg12 gene in commensal bacteria.</p>Formula:C18H35NO4Color and Shape:SolidMolecular weight:329.47RG 13647
CAS:<p>RG 13647 is an agonist of angiotensin II peptide.</p>Formula:C30H27N3O5Purity:98%Color and Shape:SolidMolecular weight:509.55Valorphin
CAS:<p>Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.</p>Formula:C44H61N9O11Purity:98%Color and Shape:SolidMolecular weight:892.01Diisononyl phthalate
CAS:<p>Diisononyl phthalate (DINP), known as a plasticizer, is a phthalate. DINP is specifically a mixture of various isononyl esters of phthalic acid.</p>Formula:C26H42O4Color and Shape:Colorless Liquid In Water (Uscg 1999)Molecular weight:418.61PROTAC ER Degrader-3
CAS:<p>PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.</p>Formula:C71H77N7O12Purity:98%Color and Shape:SolidMolecular weight:1220.434Prednisolone farnesylate
CAS:<p>Prednisolone farnesylate is a novel transdermal corticosteroid with anti-inflammatory activity.</p>Formula:C36H50O6Purity:98%Color and Shape:SolidMolecular weight:578.78Dynorphin B (1-13)
CAS:<p>Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.</p>Formula:C74H115N21O17Purity:98%Color and Shape:SolidMolecular weight:1570.84ERRγ agonist-2
CAS:<p>ERRγ agonist-2 is a potent and selective ERRγ inverse agonist with a K d value of 6.5 μM.</p>Formula:C27H21N5O2Color and Shape:SolidMolecular weight:447.49Herkinorin
CAS:<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Formula:C28H30O8Color and Shape:SolidMolecular weight:494.539,10-Dihydrophenanthrene
CAS:<p>9,10-Dihydrophenanthrene has inhibitory activity against the androgen receptor and can be used in related research in the field of life sciences.</p>Formula:C14H12Purity:98.76%Color and Shape:SolidMolecular weight:180.25UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Formula:C82H138N32O21Purity:98%Color and Shape:SolidMolecular weight:1908.19Imidaprilate
CAS:<p>Imidaprilate, an active TA-6366 metabolite, is a potent ACE inhibitor with an IC50 of 2.6 nM, researched for hypertension.</p>Formula:C18H23N3O6Purity:98%Color and Shape:SolidMolecular weight:377.39T4-ATA (S-isomer)
<p>T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.</p>Formula:C19H15I4NO6SPurity:98%Color and Shape:SolidMolecular weight:893.01Antihypertensive agent 3
<p>Antihypertensive agent 3 (compound 4a), an angiotensin II receptor 1 antagonist, demonstrates antihypertensive activity in spontaneously hypertensive rats (SHRs</p>Formula:C16H13NO4SColor and Shape:SolidMolecular weight:315.34TrxR1 prodrug-1
<p>TrxR1 prodrug-1 (compound 5u) is a potent inhibitor of TrxR1, demonstrating significant antitumor activity in nude mice and NSCLC organoids.</p>Formula:C22H30N2O6S2Color and Shape:SolidMolecular weight:482.613DDHF20
<p>DDHF20 is an inhibitor of Staphylococcus aureus, specifically targeting and inhibiting its thioredoxin reductase (TrxR) by acting as a competitive inhibitor at the NADPH binding site. DDHF20 shows potential for research in combating infections related to Staphylococcus aureus.</p>Formula:C34H28O4Color and Shape:SolidMolecular weight:500.58Teriparatide
CAS:<p>Teriparatide is an agonist of PHT(IC50 of 2 nM in HEK293 cells).</p>Formula:C181H291N55O51S2Purity:98%Color and Shape:SolidMolecular weight:4117.72[Arg8]-Vasotocin
CAS:<p>[Arg8]-Vasotocin is a hormone present in the neurohypophysis of nonmammalian vertebrates that is related to vasopressin and oxytocin.</p>Formula:C43H67N15O12S2Purity:98%Color and Shape:SolidMolecular weight:1050.22PTP1B/AKR1B1-IN-2
<p>PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0</p>Formula:C23H23NO4S2Purity:98%Color and Shape:SolidMolecular weight:441.56ST-CY14
<p>ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.</p>Formula:C139H237N57O31S2Color and Shape:SolidMolecular weight:3266.86Eprosartan
CAS:<p>Eprosartan is a selective AT1 receptor blocker with IC50s of 9.2 nM (rat) and 3.9 nM (human), used for hypertension.</p>Formula:C23H24N2O4SPurity:>99.99%Color and Shape:SolidMolecular weight:424.51Hydrocortisone sodium succinate
CAS:<p>Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.</p>Formula:C25H34NaO8Color and Shape:SolidMolecular weight:485.529Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Color and Shape:Odour SolidL 363564
CAS:<p>L 363564 is a kidney renin inhibitor.</p>Formula:C54H76N12O10Color and Shape:SolidMolecular weight:1053.276AZ 1729
CAS:<p>FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.</p>Formula:C18H16FN5OSColor and Shape:SolidMolecular weight:369.42AKR1C3-IN-10
<p>AKR1C3-IN-10 (compound 5r), a selective inhibitor of AKR1C3 with an IC50 of 51 nM, demonstrates efficacy in a prostate cancer xenograft model [1].</p>Formula:C24H20N4O3Color and Shape:SolidMolecular weight:412.44Olmesartan medoxomil impurity C
CAS:<p>Impurity C of Olmesartan medoxomil is a selective AT1 inhibitor with an IC50 of 66.2 μM.</p>Formula:C29H28N6O5Color and Shape:SolidMolecular weight:540.57OBHSA
CAS:<p>OBHSA（Oxabicycloheptane sulfonamide） is a novel selective estrogen receptor depressant (SERD) that can be used to study breast cancer.</p>Formula:C27H24F3NO6SPurity:98%Color and Shape:SolidMolecular weight:547.54Neuropeptide EI, rat
CAS:<p>Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.</p>Formula:C63H98N16O23Purity:98%Color and Shape:SolidMolecular weight:1447.55Potassium Channel Targeted Library
<p>A unique collection of xnum potassium channel blockers and agonists for high throughput and high content screening;</p>Color and Shape:Odour SolidYp537
CAS:<p>Yp537 acts as an estrogen receptor (ER) inhibitor, specifically preventing the dimerization of the human estrogen receptor [1].</p>Formula:C64H104N13O22PSColor and Shape:SolidMolecular weight:1470.62hFSH-β-(33-53) (TFA)
<p>hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist.</p>Formula:C115H183N31O32SxC2HF3O2Color and Shape:SolidMolecular weight:2657.96(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin
CAS:<p>'(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin blocks oxytocin receptors, stopping oxytocin effects on CA1 neuron currents.'</p>Formula:C45H69N9O12S2Color and Shape:SolidMolecular weight:992.21Azilsartan Medoxomil Potassium
CAS:<p>Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.</p>Formula:C30H23N4O8·KPurity:98.72%Color and Shape:SolidMolecular weight:606.62Ro 64-6198
CAS:<p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.</p>Formula:C26H31N3OPurity:98%Color and Shape:SolidMolecular weight:401.54ERα degrader 10
<p>ERα degrader10 is a potent, selective, orally active estrogen receptor α (ERα) degrader. It demonstrates strong ERα binding affinity (IC50 of 24.0 nM) and degradation capability (EC50 of 5.3 nM). This compound degrades ERα through a proteasome-mediated pathway and is utilized in breast cancer research.</p>Color and Shape:Odour SolidPROTAC ER Degrader-14
CAS:<p>PROTAC ER Degrader-14 (compound 86) is a PROTAC-type estrogen receptor/ERR degrader. It comprises an E3 ubiquitin ligase ligand (blue part) (S)-Deoxy-thalidomide, a PROTAC linker (black part) N-Boc-piperazine, and a target protein ligand (red part) ER ligand-6. The combination of the E3 ligase and linker forms tert-Butyl (S)-4-(2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)piperazine-1-carboxylate.</p>Formula:C44H46FN5O5Color and Shape:SolidMolecular weight:743.865U-54494A hydrochloride
CAS:<p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>Formula:C18H25Cl3N2OColor and Shape:SolidMolecular weight:391.76Estrogen receptor modulator 6
CAS:<p>ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.</p>Formula:C18H16F2O3Color and Shape:SolidMolecular weight:318.32[Sar1, Ile8]-Angiotensin II
CAS:<p>[Sar1, Ile8]-Angiotensin II(3TFA) is a peptide that has multiple effects on vascular smooth muscle.</p>Formula:C46H73N13O10Purity:98%Color and Shape:SolidMolecular weight:968.15AKR1B10-IN-1
CAS:<p>AKR1B10-IN-1: potent AKR1B10 inhibitor, IC50 3.5 nM; hinders lung cancer cell growth, spread, and Cisplatin resistance.</p>Formula:C19H16FNO4Color and Shape:SolidMolecular weight:341.338ERD-308
CAS:<p>ERD-308, potent at 5nM, achieves >95% ER degradation in ER+ breast cancer, with DC50 of 0.17-0.43 nM.</p>Formula:C55H65N5O9S2Purity:98%Color and Shape:SolidMolecular weight:1004.26PROTAC ERα Degrader-2
CAS:<p>PROTAC ERα Degrader-2 is composed of a cIAP1 ligand binding group, a linker, and an estrogen receptor α (ERα) binding group, serving as an ERα degrader.</p>Formula:C42H61N5O8Purity:98%Color and Shape:SolidMolecular weight:763.96Ocedurenone
CAS:<p>Ocedurenone, a corticosteroid receptor antagonist, is a compound utilized in the investigation of kidney disease (WO2018054357, compound I).</p>Formula:C28H30ClN5O2Color and Shape:SolidMolecular weight:504.032-sec-Butylphenol
CAS:<p>2-sec-Butylphenol is an inhibitor of the androgen receptor and P450 aromatase, and can be used in research and experiments in the field of life sciences.</p>Formula:C10H14OColor and Shape:SolidMolecular weight:150.22[Sar1, Ile8]-Angiotensin II TFA
<p>[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.</p>Formula:C48H74F3N13O12Purity:98%Color and Shape:SolidMolecular weight:1082.18Dagrocorat hydrochloride
CAS:<p>PF-0251802 HCl is a bio-active chemical.</p>Formula:C29H30ClF3N2O2Color and Shape:SolidMolecular weight:531.01BAY 1003803
CAS:<p>BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.</p>Formula:C21H18ClF5N2O4Color and Shape:SolidMolecular weight:492.83Urotensin II (114-124), human
CAS:<p>Human Urotensin II (114-124) is an 11-amino acid peptide with vasoconstrictor properties and agonizes GPR14.</p>Formula:C64H85N13O18S2Purity:98%Color and Shape:SolidMolecular weight:1388.57Alclometasone
CAS:<p>Alclometasone is a glucocorticoid that reduces inflammation and treats various skin conditions like eczema and psoriasis.</p>Formula:C22H29ClO5Purity:98%Color and Shape:SolidMolecular weight:408.92Angiotensin II 5-valine
CAS:<p>ngiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors.</p>Formula:C49H69N13O12Purity:98%Color and Shape:SolidMolecular weight:N/AAdrenocorticotropic hormone
CAS:<p>ACTH, a polypeptide, is secreted by the pituitary gland and regulates cortisol and androgen.</p>Color and Shape:SolidNeuropeptide AF (human)
CAS:<p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>Formula:C90H132N26O25Purity:98%Color and Shape:SolidMolecular weight:1978.17DPC-AJ1951 TFA
<p>DPC-AJ1951 TFA is a 14 amino acid peptide, potent PTH/PPR agonist, tested in bone resorption assays.</p>Formula:C78H128F3N23O21Color and Shape:SolidMolecular weight:1781.02PROTAC ERα Degrader-8
CAS:<p>PROTAC ERα Degrader-8 (compound ii-56), a highly potent degrader of Erα, achieves a DC50 of just 0.000006 μM in MCF7 cells [1].</p>Formula:C47H51N5O4Color and Shape:SolidMolecular weight:749.94Handle region peptide, rat
CAS:<p>Rat handle region peptide acts as prorenin receptor blocker, curbs diabetic kidney disease, and reduces eye inflammation.</p>Formula:C54H101N15O12SPurity:98%Color and Shape:SolidMolecular weight:1184.54PROTAC AR Degrader-9
<p>PROTAC AR Degrader-9 (Compound c6) is a PROTAC-based degrader specifically targeting the androgen receptor. It effectively degrades the androgen receptor in human dermal papilla cells (HDPC) with a DC50 of 262.38 nM. Additionally, this compound enhances the expression of paracrine factors, such as TGF-β1 and β-catenin, thereby promoting hair regeneration in mouse models. [Pink: ligand for target protein AR ligand-38; Black: linker; Blue: ligand for E3 ligase Cereblon]</p>Formula:C43H49ClN6O5Color and Shape:SolidMolecular weight:765.339Cl-4AS-1
CAS:<p>steroidal androgen receptor agonist</p>Formula:C26H33ClN2O2Purity:98%Color and Shape:SolidMolecular weight:441.01[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Formula:C63H101F3N22O17Color and Shape:SolidMolecular weight:1495.61Melanin Concentrating Hormone, salmon TFA
<p>MCH (salmon) TFA is a 19-amino-acid neuropeptide affecting appetite, energy, sleep, and heart health via GPCR SLC-1/GPR24 and MCHR2.</p>Formula:C91H140F3N27O26S4Color and Shape:SolidMolecular weight:2213.5PROTAC ER Degrader-15
<p>PROTAC ER Degrader-15 (Compound 40) is an orally active estrogen receptor (ER) degrader with anticancer properties, suitable for breast cancer research.</p>Formula:C47H47F4N5O5Color and Shape:SolidMolecular weight:837.9Aclerastide
CAS:<p>Aclerastide, an angiotensin receptor agonist, decreases fibrosis in wounds; effect increases with use duration, blocked by AT antagonist.</p>Formula:C42H64N12O11Color and Shape:SolidMolecular weight:913.03Floramanoside C
CAS:<p>Floramanoside C exhibits 2,2-diphenyl-1-picrylhydrazyl scavenging and aldose reductase inhibitory activities [1].</p>Formula:C21H18O15Color and Shape:SolidMolecular weight:510.36TRV-120027
CAS:<p>TRV120027: β-arrestin-1-biased agonist, angiotensin II type 1 receptor, reduces vasoconstriction, boosts heart muscle contraction.</p>Formula:C43H67N13O10Purity:98%Color and Shape:SolidMolecular weight:926.09ARD-2051
CAS:<p>ARD-2051 is a potent, orally active proteolysis-targeting chimera degrader of the androgen receptor (AR), exhibiting DC50 values of 0.6 nM in degrading AR</p>Formula:C43H45ClN8O5Purity:98%Color and Shape:SolidMolecular weight:789.32TAN67
CAS:<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Formula:C23H26Br2N2OColor and Shape:SolidMolecular weight:506.28218-Oxocortisol
CAS:<p>18-Oxocortisol, a naturally occurring mineralocorticoid and adrenal biomarker, is produced by CYP11B2.</p>Formula:C21H28O6Color and Shape:SolidMolecular weight:376.449AL-438
CAS:<p>AL-438 is a non-steroidal selective glucocorticoid receptor modulator.</p>Formula:C23H25NO2Purity:98%Color and Shape:SolidMolecular weight:347.45Dynorphin A (1-8)
CAS:<p>Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.</p>Formula:C46H72N14O10Purity:98%Color and Shape:SolidMolecular weight:981.15Prednicarbate
CAS:<p>Prednicarbate (Hoe 777), a corticosteroid, has antipruritic, anti-inflammatory effects, reduces lymphocytes, and inhibits vasodilators.</p>Formula:C27H36O8Purity:99.88%Color and Shape:SolidMolecular weight:488.57Ditekiren
CAS:<p>Ditekiren is a renin inhibitor with orally active.</p>Formula:C50H75N9O8Purity:98%Color and Shape:SolidMolecular weight:930.19Thyroxine sulfate
CAS:<p>Thyroxine sulfate is a sulfoconjugated derivative of Thyroxine and is also a metabolite of Thyroxine.</p>Formula:C15H11I4NO7SColor and Shape:SolidMolecular weight:856.93RTI-13951-33 hydrochloride
<p>RTI-13951-33 HCl: potent, selective GPR88 agonist; brain-penetrant; EC50 = 25nM; curbs rat alcohol behaviors.</p>Formula:C28H35Cl2N3O3Purity:98%Color and Shape:SolidMolecular weight:532.5GLL 398
CAS:<p>GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.</p>Formula:C25H23BO4Purity:98%Color and Shape:SolidMolecular weight:398.26Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formula:C31H41N7O9Purity:98%Color and Shape:SolidMolecular weight:655.709Koreanoside E
CAS:<p>Koreanoside E is a useful organic compound for research related to life sciences. The catalog number is T125538 and the CAS number is 1804014-67-2.</p>Formula:C27H30O11Color and Shape:SolidMolecular weight:530.526Vasopressin Dimer (parallel) (TFA)
<p>Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, and</p>Formula:C94H131F3N30O26S4Purity:98%Color and Shape:SolidMolecular weight:2282.49ARD-69
<p>ARD-69, a potent PROTAC, degrades AR in prostate cancer, with low DC50 values in AR+ cell lines, and suppresses AR gene expression.</p>Formula:C62H74ClFN8O7SColor and Shape:SolidMolecular weight:1129.8311-Ketodihydrotestosterone
CAS:<p>11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20.4 nM, EC50: 1.35 nM for human AR).</p>Formula:C19H28O3Color and Shape:SolidMolecular weight:304.427β-Hydroxy-epi-androsterone
CAS:<p>7β-Hydroxy-epi-androsterone (7β-Hydroxy-EpiA) is an endogenous androgenic derivative of dehydroepiandrosterone that possesses the ability to bind to ERβ,</p>Formula:C19H30O3Color and Shape:SolidMolecular weight:306.44Zankiren
CAS:<p>Zankiren is a renin inhibitor. Zankiren can reduce blood pressure, plasma renin activity, and angiotension II.</p>Formula:C35H55N5O6S2Color and Shape:SolidMolecular weight:705.97[Arg14,Lys15]Nociceptin
CAS:<p>Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>Formula:C82H137N31O22Purity:98%Color and Shape:SolidMolecular weight:1909.18Angiotensin II (5-8), human
CAS:<p>Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II</p>Formula:C26H36N6O5Purity:98%Color and Shape:SolidMolecular weight:512.6SNIPER(ER)-87
CAS:<p>SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (</p>Formula:C59H73N5O10SPurity:98%Color and Shape:SolidMolecular weight:1044.32Urotensin II (114-124), human TFA
<p>Urotensin II (114-124), human TFA, is an 11-amino acid peptide and potent vasoconstrictor, acting as GPR14 agonist.</p>Formula:C66H86F3N13O20S2Purity:98%Color and Shape:SolidMolecular weight:1502.5915,26-Dihydroxylanosta-7,9(11),24-trien-3-one
CAS:<p>15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is a natural product that can be used as a reference standard. The CAS number of 15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is 420781-85-7.</p>Formula:C30H46O3Color and Shape:SolidMolecular weight:454.7Raloxifene 6-Monomethyl Ether
CAS:<p>Compound 7, Raloxifene 6-Monomethyl Ether, blocks estrogen receptor α, inhibits MCF-7 cells; IC50=250 nM, pIC50=6.6.</p>Formula:C29H29NO4SColor and Shape:SolidMolecular weight:487.61AKR1C3-IN-9
<p>AKR1C3-IN-9: Selective AKR1C3 inhibitor, IC50=8.92 nM; reverses DOX resistance in breast cancer.</p>Formula:C20H20N2O4Purity:99.98%Color and Shape:SoildMolecular weight:352.38MT-7716 free base
CAS:<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Formula:C27H28N4O2Purity:98%Color and Shape:SolidMolecular weight:440.54PROTAC ERα Degrader-7
CAS:<p>PROTAC ERα Degrader-7 (Compound i-320) is a powerful PROTAC degrader targeting the estrogen receptor alpha (ERα), exhibiting a DC50 of 0.000006 µM. This compound consists of a cereblon-binding segment, LBM, connected to ERBM, an ERα-binding ligand that includes a benzofused partially saturated 6-membered carbocyclic or heterocyclic ring [1].</p>Formula:C46H49F2N5O4Color and Shape:SolidMolecular weight:773.91CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formula:C34H35N5O4Color and Shape:SolidMolecular weight:577.67Imlunestrant tosylate
CAS:<p>Imlunestrant (LY-3484356) tosylate, an oral SERD, targets ER+ aBC/EEC by blocking estrogen receptors and gene transcription.</p>Formula:C36H32F4N2O6SColor and Shape:SolidMolecular weight:696.71Arzoxifene
CAS:<p>Arzoxifene (LY353381), an oral SERM, combats breast cancer, supports bone health, and improves lipids, with few side effects.</p>Formula:C28H29NO4SColor and Shape:SolidMolecular weight:475.6EX-A5386
CAS:<p>EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.</p>Formula:C29H27FN4O2Purity:99.89%Color and Shape:SoildMolecular weight:482.55KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Formula:C38H38N2O5Color and Shape:SolidMolecular weight:602.72Triphenylethylene
CAS:<p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formula:C20H16Color and Shape:White PowderMolecular weight:256.34Angiotensin II (1-4), human TFA
<p>Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure.</p>Formula:C26H38F3N7O10Purity:98%Color and Shape:SolidMolecular weight:665.62Ganoderic acid Df
CAS:<p>Ganoderic acid Df, a lanostane triterpenoid from Ganoderma lucidum, inhibits aldose reductase with IC50 of 22.8 μM.</p>Formula:C30H44O7Color and Shape:SolidMolecular weight:516.67Melanin Concentrating Hormone, salmon
CAS:<p>Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>Formula:C89H139N27O24S4Purity:98%Color and Shape:White PowderMolecular weight:2099.48Urotensin II, mouse
CAS:<p>UTS2 is a human gene, alias U-II, on chromosome 1p36.23, codes for Urotensin-II, a potent vasoconstrictor. Formula: C64H85N13O18S2, Molar mass: 1388.6 g/mol.</p>Formula:C76H100N18O19S2Purity:98%Color and Shape:SolidMolecular weight:1633.86
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