Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3180 products of "Endocrinology/Hormones"
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G15
CAS:<p>G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)</p>Formula:C19H16BrNO2Purity:98.46% - 98.59%Color and Shape:SolidMolecular weight:370.24DY131
CAS:<p>DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.</p>Formula:C18H21N3O2Purity:98.65% - 99.66%Color and Shape:SolidMolecular weight:311.38Nandrolone phenylpropionate
CAS:<p>Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis</p>Formula:C27H34O3Purity:99.2% - 99.46%Color and Shape:White Or Milky Crystalline PowderMolecular weight:406.56panomifene
CAS:<p>Panomiphene (Gyki-13504, EGIS-5650) is an anti-estrogen drug that is a tamoxifen (TMX) analogue.</p>Formula:C25H24F3NO2Color and Shape:SolidMolecular weight:427.46AMG 837 hemicalcium
CAS:<p>AMG 837 hemicalcium: oral GPR40 agonist, binds human FFA1 (pIC50: 8.13), boosts insulin, lowers glucose in rodents.</p>Formula:C52H40CaF6O6Color and Shape:SolidMolecular weight:914.954VPC-13163
CAS:<p>VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.</p>Formula:C16H14N2Purity:98.02%Color and Shape:SolidMolecular weight:234.3Pipendoxifene
CAS:<p>Pipendoxifene (ERA-923) is an antiestrogen that blocks ER-alpha and inhibits MCF-7 breast cancer cell growth, effective even when tamoxifen-resistant.</p>Formula:C29H32N2O3Color and Shape:SolidMolecular weight:456.58α-Zearalenol
CAS:<p>α-Zearalenol is one of the major metabolites of Zearalenone.</p>Formula:C18H24O5Purity:90% - 99.72%Color and Shape:SolidMolecular weight:320.38Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Formula:C38H54N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:782.88Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formula:C30H39N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:597.66MCOPPB
CAS:<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Formula:C26H40N4Color and Shape:SolidMolecular weight:408.62MS21570
CAS:<p>MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.</p>Formula:C10H11N3S2Purity:97.79%Color and Shape:SolidMolecular weight:237.34Palosuran hydrochloride 540769-28-6(free base)
<p>Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.</p>Formula:C25H31ClN4O2Purity:99.75%Color and Shape:SolidMolecular weight:454.99b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Antide acetate
<p>Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. </p>Formula:C84H112ClN17O16Purity:99.57%Color and Shape:SolidMolecular weight:1651.34Bisphenol B
CAS:<p>Bisphenol B has a binding affinity for estrogen receptors.</p>Formula:C16H18O2Purity:97.35% - 99.62%Color and Shape:Crystal Or Tan Granules Odorless Slightly Brown SolidMolecular weight:242.31H-Val-Pro-Pro-OH
CAS:<p>H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).</p>Formula:C15H25N3O4Purity:98.23%Color and Shape:SolidMolecular weight:311.38DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59Urotensin II (114-124), human acetate
<p>Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor and agonist for the orphan receptor GPR14.</p>Formula:C66H89N13O20S2Purity:>99.99%Color and Shape:SolidMolecular weight:1448.63Apalutamide
CAS:<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Formula:C21H15F4N5O2SPurity:99.03% - 99.91%Color and Shape:SolidMolecular weight:477.43AZD1981
CAS:<p>AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma and other trials.</p>Formula:C19H17ClN2O3SPurity:98.87% - 99.67%Color and Shape:SolidMolecular weight:388.87TC-O 9311
CAS:<p>TC-O 9311 (TCO-9311) is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).</p>Formula:C20H19N3O4Purity:99.24% - 99.84%Color and Shape:SolidMolecular weight:365.38Timapiprant
CAS:<p>Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).</p>Formula:C21H17FN2O2Purity:97.44% - 99.51%Color and Shape:SolidMolecular weight:348.374-CMTB
CAS:<p>4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).</p>Formula:C14H15ClN2OSPurity:99.59%Color and Shape:SolidMolecular weight:294.8AS1269574
CAS:<p>AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.</p>Formula:C13H14BrN3OPurity:99.99%Color and Shape:SolidMolecular weight:308.17(Sar¹)-Angiotensin II acetate
<p>(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor.</p>Formula:C51H75N13O12Purity:99.89%Color and Shape:SoildMolecular weight:1062.222-(pentylsulfanyl)pyrimidine-4,6-diol
CAS:<p>2-(pentylsulfanyl)pyrimidine-4,6-diol 是一种新型 GRP84 激动剂。</p>Formula:C9H14N2O2SPurity:97.58%Color and Shape:SolidMolecular weight:214.28Norgestrel
CAS:<p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>Formula:C21H28O2Purity:99.71% - 99.72%Color and Shape:Crystals From Methanol White Crystalline PowderMolecular weight:312.45JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Formula:C26H25N3O2·HClPurity:99.27% - 99.59%Color and Shape:SolidMolecular weight:447.96Gluten Exorphin C
CAS:<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Formula:C29H45N5O8Purity:99.39%Color and Shape:SolidMolecular weight:591.7Leucylarginylproline
CAS:<p>Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).</p>Formula:C17H32N6O4Purity:99.58%Color and Shape:SolidMolecular weight:384.47Nafoxidine
CAS:<p>Nafoxidine is an estrogen antagonist that has been used in the treatment of breast cancer.</p>Formula:C29H31NO2Purity:99.93%Color and Shape:SolidMolecular weight:425.56CVN424
CAS:<p>CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.</p>Formula:C24H29F2N5O3Purity:99.02%Color and Shape:SolidMolecular weight:473.52Carbetocin acetate
CAS:<p>Carbetocin acetate is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.</p>Formula:C47H73N11O14SPurity:98.16% - 99.22%Color and Shape:SolidMolecular weight:1048.22GSK1292263
CAS:<p>GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.</p>Formula:C23H28N4O4SPurity:98.34% - 99.53%Color and Shape:SolidMolecular weight:456.56JNJ-63533054
CAS:<p>JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.</p>Formula:C17H17ClN2O2Purity:99.71% - 99.88%Color and Shape:SolidMolecular weight:316.78Zaprinast
CAS:<p>Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist.</p>Formula:C13H13N5O2Purity:99.73% - 99.77%Color and Shape:White To Off White PowderMolecular weight:271.27XCT790
CAS:<p>XCT790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα).</p>Formula:C23H13F9N4O3SPurity:99% - 99.61%Color and Shape:SolidMolecular weight:596.42Osilodrostat phosphate
CAS:<p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>Formula:C13H13FN3O4PColor and Shape:SolidMolecular weight:325.23Sparsentan
CAS:<p>Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM,</p>Formula:C32H40N4O5SPurity:97.94% - 98.69%Color and Shape:SolidMolecular weight:592.75PSN 375963
CAS:<p>PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.</p>Formula:C17H23N3OPurity:99.63%Color and Shape:SolidMolecular weight:285.38Kisspeptin-10, human (TFA)(374675-21-5,FREE)
<p>Kisspeptin-10 TFA: vasoconstrictor, inhibits angiogenesis & metastasis; key in kidney development & osteoblast differentiation via GPR54 & NFATc4/BMP2.</p>Formula:C63H83N17O14·C2HF3O2Purity:>99.99%Color and Shape:SolidMolecular weight:1416.46Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66MBX-2982
CAS:<p>MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.</p>Formula:C22H24N8OSPurity:98% - 99.96%Color and Shape:SolidMolecular weight:448.54Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formula:C25H34N2O5Purity:98%Color and Shape:SolidMolecular weight:442.55Delapril hydrochloride
CAS:<p>Delapril HCl (indalapril) is a prodrug forming two ACE inhibitors, blocking angiotensin I-II conversion.</p>Formula:C26H33ClN2O5Purity:97.18% - 97.45%Color and Shape:White Crystalline PowderMolecular weight:489.01Asimadoline hydrochloride
CAS:<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Formula:C27H31ClN2O2Purity:98.94% - 99.32%Color and Shape:SolidMolecular weight:451.01Trans-Tranilast
CAS:<p>Trans-Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. It has been used for the treatment of allergic disorders such as atopic dermatitis.</p>Formula:C18H17NO5Purity:99.41% - ≥95%Color and Shape:SolidMolecular weight:327.33Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Formula:C46H74N14O11Purity:99.84%Color and Shape:SolidMolecular weight:999.17
