CymitQuimica logo
Glucocorticoid Receptor

Glucocorticoid Receptor

The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.

Found 153 products of "Glucocorticoid Receptor"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • AL-438

    CAS:
    <p>AL-438 is a non-steroidal selective glucocorticoid receptor modulator.</p>
    Formula:C23H25NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:347.45
  • BAY 1003803

    CAS:
    <p>BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.</p>
    Formula:C21H18ClF5N2O4
    Color and Shape:Solid
    Molecular weight:492.83
  • OP-3633

    CAS:
    <p>OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.</p>
    Formula:C30H39NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.64
  • CP-472555

    CAS:
    <p>CP-472555 is a selective nonsteroidal glucocorticoid receptor antagonist with anti-GR and anti-obesity activity in animal models.</p>
    Formula:C31H32N2O2
    Color and Shape:Solid
    Molecular weight:464.60
  • PPARγ/GR modulator 1


    <p>PPARγ/GR Modulator 1, an orally active dual agonist for the Peroxisome Proliferator-Activated Receptor Gamma (PPARγ) and Glucocorticoid Receptor (GR), exhibits</p>
    Formula:C14H10FNO4
    Color and Shape:Solid
    Molecular weight:275.23
  • EX-A5386

    CAS:
    <p>EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50&lt;100nM.</p>
    Formula:C29H27FN4O2
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:482.55
  • Triamcinolone Benetonide

    CAS:
    <p>Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid exhibiting potent anti-inflammatory properties.</p>
    Formula:C35H42FNO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:623.71
  • Glucocorticoids receptor agonist 2

    CAS:
    <p>Arylpyrazole-based glucocorticoid agonist with potent anti-inflammatory effects; doesn't affect insulin secretion.</p>
    Formula:C25H25FN2O
    Color and Shape:Solid
    Molecular weight:388.48
  • Prednisolone farnesylate

    CAS:
    <p>Prednisolone farnesylate is a novel transdermal corticosteroid with anti-inflammatory activity.</p>
    Formula:C36H50O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:578.78
  • Betamethasone 17-benzoate

    CAS:
    <p>Betamethasone 17-benzoate is a representative steroid. It also can be used in the treatment of recurrent aphothous ulcers (RAU).</p>
    Formula:C29H33FO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:496.57
  • Dexamethasone cipecilate

    CAS:
    <p>Dexamethasone cipecilate is a long-acting intranasal corticosteroid and a highly lipophilic anti-inflammatory corticosteroid.</p>
    Formula:C33H43FO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:570.69
  • Rofleponide

    CAS:
    <p>Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.</p>
    Formula:C25H34F2O6
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:468.53
  • Flucloronide

    CAS:
    <p>Flucloronide is a corticosteroid for topical use on the skin. It has anti-inflammatory properties.</p>
    Formula:C24H29Cl2FO5
    Color and Shape:Solid
    Molecular weight:487.39
  • NR3C1 Protein, Human, Recombinant (His)


    <p>NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene.</p>
    Color and Shape:Lyophilized Powder
    Molecular weight:10.95 kDa (predicted)
  • Prednisolone valerate acetate

    CAS:
    <p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>
    Formula:C28H38O7
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:486.6
  • Diflorasone Diacetate

    CAS:
    <p>Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.</p>
    Formula:C26H32F2O7
    Color and Shape:Crystals
    Molecular weight:494.53
  • Hydrocortisone buteprate

    CAS:
    <p>Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.</p>
    Formula:C28H40O7
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:488.61
  • Hydrocortisone cypionate

    CAS:
    <p>Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid.</p>
    Formula:C29H42O6
    Color and Shape:Solid
    Molecular weight:486.64
  • Desoxycorticosterone pivalate

    CAS:
    <p>DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.</p>
    Formula:C26H38O4
    Color and Shape:Solid
    Molecular weight:414.58
  • Anti-NR3C1 Antibody (9X89)


    <p>Anti-NR3C1 Antibody (9X89) is an antibody targeting NR3C1. Anti-NR3C1 Antibody (9X89) can be used in ELISA, WB, FCM.</p>
    Color and Shape:Odour Liquid
  • Isoflupredone Acetate

    CAS:
    <p>Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.</p>
    Formula:C23H29FO6
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:420.47
  • (20S)-Protopanaxatriol

    CAS:
    <p>(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid</p>
    Formula:C30H52O4
    Purity:95% - 99%
    Color and Shape:Solid
    Molecular weight:476.73
  • Fluorometholone Acetate

    CAS:
    <p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>
    Formula:C24H31FO5
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:418.50
  • Mirodenafil dihydrochloride

    CAS:
    <p>Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>
    Formula:C26H39Cl2N5O5S
    Purity:99.64% - 99.78%
    Color and Shape:Solid
    Molecular weight:604.59
  • Canrenoate potassium

    CAS:
    <p>Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.</p>
    Formula:C22H29KO4
    Purity:99.04% - 99.18%
    Color and Shape:Light Yellow To Tan Powder
    Molecular weight:396.56
  • Apararenone

    CAS:
    <p>Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.</p>
    Formula:C17H17FN2O4S
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:364.39
  • Beclometasone

    CAS:
    <p>Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma.</p>
    Formula:C22H29ClO5
    Purity:99.41% - 99.68%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:408.92
  • Desoximetasone

    CAS:
    <p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>
    Formula:C22H29FO4
    Purity:99.06% - 99.89%
    Color and Shape:Solid
    Molecular weight:376.46
  • Osilodrostat

    CAS:
    <p>Osilodrostat (LCI699) is a potent inhibitor of human 11β-hydroxylase (CYP11B1) and aldosterone synthase (CYP11B2).Cost-effective and quality-assured.</p>
    Formula:C13H10FN3
    Purity:99.10% - 99.36%
    Color and Shape:Solid
    Molecular weight:227.24
  • Fludrocortisone acetate

    CAS:
    <p>Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and</p>
    Formula:C23H31FO6
    Purity:96.92% - 98.03%
    Color and Shape:Crystalline Solid
    Molecular weight:422.49
  • Fluorometholone

    CAS:
    <p>Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery.</p>
    Formula:C22H29FO4
    Purity:99% - 99.15%
    Color and Shape:Solid
    Molecular weight:376.46
  • Hydrocortisone hemisuccinate

    CAS:
    <p>Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.</p>
    Formula:C25H34O8
    Purity:98.01% - 98.7%
    Color and Shape:Solid
    Molecular weight:462.53
  • AZD9977

    CAS:
    <p>AZD9977 is a novel, selective modulator of mineralocorticoid receptor .</p>
    Formula:C20H18FN3O5
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:399.37
  • Halobetasol propionate

    CAS:
    <p>Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.</p>
    Formula:C25H31ClF2O5
    Purity:99.89%
    Color and Shape:Distributed As 0 05% Ointment
    Molecular weight:484.96
  • Fluocinonide

    CAS:
    <p>Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.</p>
    Formula:C26H32F2O7
    Purity:98.33% - 99.70%
    Color and Shape:Solid
    Molecular weight:494.52
  • Corticosterone

    CAS:
    <p>Corticosterone (Kendall's compound B) is an adrenocortical steroid with salocorticoid and glucocorticoid activity that is orally active.</p>
    Formula:C21H30O4
    Purity:98.44% - ≥95%
    Color and Shape:Solid
    Molecular weight:346.46
  • Velsecorat

    CAS:
    <p>Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).</p>
    Formula:C32H32F2N4O6
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:606.62
  • AL 082D06

    CAS:
    <p>AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.</p>
    Formula:C23H24ClN3O2
    Purity:99.05% - 99.06%
    Color and Shape:Solid
    Molecular weight:409.91
  • Methylprednisolone succinate

    CAS:
    <p>Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.</p>
    Formula:C26H34O8
    Purity:98.41% - 99.82%
    Color and Shape:White Or Almost-White Solid Powder
    Molecular weight:474.54
  • Ciclesonide

    CAS:
    <p>Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.</p>
    Formula:C32H44O7
    Purity:99.89% - >99.99%
    Color and Shape:Solid
    Molecular weight:540.69
  • Vamorolone

    CAS:
    <p>Vamorolone (VBP15) is a steroid-like drug that treats muscular dystrophy with fewer side effects and inhibits NF-κB.</p>
    Formula:C22H28O4
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:356.46
  • Diflorasone

    CAS:
    <p>Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene expression.</p>
    Formula:C22H28F2O5
    Purity:99.02% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.45
  • Beclometasone dipropionate monohydrate

    CAS:
    <p>Beclometasone dipropionate monohydrate, precursor to oral glucocorticoid for inflammation and asthma research.</p>
    Formula:C28H39ClO8
    Color and Shape:Solid
    Molecular weight:539.06
  • Cortodoxone

    CAS:
    <p>Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.</p>
    Formula:C21H30O4
    Purity:99.26% - 99.87%
    Color and Shape:Solid
    Molecular weight:346.46
  • Osilodrostat phosphate

    CAS:
    <p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>
    Formula:C13H13FN3O4P
    Color and Shape:Solid
    Molecular weight:325.23
  • LY404039

    CAS:
    <p>LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).</p>
    Formula:C7H9NO6S
    Purity:99% - 99.92%
    Color and Shape:Solid
    Molecular weight:235.22
  • Finerenone

    CAS:
    <p>Finerenone (BAY-948862) is a selective and orally nonsteroidal antagonist of the mineralocorticoid receptor (MR). Cost effective and quality assured.</p>
    Formula:C21H22N4O3
    Purity:99.45% - 99.91%
    Color and Shape:Solid
    Molecular weight:378.42
  • Betamethasone disodium phosphate

    CAS:
    <p>Betamethasone disodium phosphate (Betamethasone 21-phosphate disodium salt) has anti-inflammatory activity and may be used in the study of rheumatoid arthritis.</p>
    Formula:C22H28FNa2O8P
    Purity:99.37%
    Color and Shape:White Powder
    Molecular weight:516.41
  • Triamcinolone hexacetonide

    CAS:
    <p>Triamcinolone hexacetonide, an exogenous synthetic corticosteroid, is a GR agonist used in the study of auto-reactive pericarditis and diabetic macular edema.</p>
    Formula:C30H41FO7
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:532.64
  • Hydrocortisone aceponate

    CAS:
    <p>Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) is an effective topical glucocorticoid used in the form of a cream to treat various skin</p>
    Formula:C26H36O7
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:460.56