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Glucocorticoid Receptor

Glucocorticoid Receptor

The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.

Found 153 products of "Glucocorticoid Receptor"

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  • Org-34517
    Targetmol
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    Org-34517

    CAS:
    <p>Org-34517, a glucocorticoid receptor (GR) antagonist, is used potentially for the treatment of depression.</p>
    Formula:C28H30O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.54

    Ref: TM-T28265

  • AZD2906
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    AZD2906

    CAS:
    <p>AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.</p>
    Formula:C26H25FN4O3
    Color and Shape:Solid
    Molecular weight:460.5

    Ref: TM-T14374

  • Prednisolone Tebutate
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    Prednisolone Tebutate

    CAS:
    <p>Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.</p>
    Formula:C27H38O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.59

    Ref: TM-T12535

  • AZD9567
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    AZD9567

    CAS:
    <p>AZD9567: potent, selective SGRM, oral, IC50=3.8nM, effective in SCW joint inflammation.</p>
    Formula:C27H28F2N4O3
    Purity:98.4%
    Color and Shape:Solid
    Molecular weight:494.53

    Ref: TM-T14386

  • Lorundrostat
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    Lorundrostat

    CAS:
    <p>Lorundrostat is an aldosterone synthase inhibitor.</p>
    Formula:C24H33N7O2
    Purity:95.47%
    Color and Shape:Solid
    Molecular weight:451.56

    Ref: TM-T62747

  • Glucocorticoid receptor agonist-1
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    Glucocorticoid receptor agonist-1

    CAS:
    <p>Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].</p>
    Formula:C35H39NO6
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:569.69

    Ref: TM-T37908

  • Dagrocorat
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    Dagrocorat

    CAS:
    <p>Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor.</p>
    Formula:C29H29F3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:494.55

    Ref: TM-T15048

  • HP210
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    HP210

    CAS:
    <p>HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-</p>
    Formula:C22H19N3O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.54

    Ref: TM-T78073

  • Spirorenone
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    Spirorenone

    CAS:
    <p>Spirorenone (INN) is a novel aldosterone antagonist with anti-salt corticosteroid activity, used in metabolic disease research.</p>
    Formula:C24H28O3
    Purity:98.28% - 99.84%
    Color and Shape:Solid
    Molecular weight:364.48

    Ref: TM-T68765

  • Halobetasol
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    Halobetasol

    CAS:
    <p>Halobetasol (Ulobetasol), a corticosteroid, is utilized in the research of severe localized psoriasis [1].</p>
    Formula:C22H27ClF2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:428.9

    Ref: TM-T78512

  • Dexamethasone palmitate
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    Dexamethasone palmitate

    CAS:
    <p>DXP, a lipophilic prodrug of Dexamethasone, has 47x less glucocorticoid receptor affinity; it's an agonist &amp; anti-inflammatory.</p>
    Formula:C38H59FO6
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:630.87

    Ref: TM-T15102

  • Amebucort
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    Amebucort

    CAS:
    <p>Amebucort is a synthetic glucocorticoid corticosteroid. It may used for the research of inflammatory disorders.</p>
    Formula:C28H40O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.61

    Ref: TM-T14209

  • RU28362
    Targetmol
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    RU28362

    CAS:
    <p>RU28362 is an agonist of glucocorticoid receptor.</p>
    Formula:C23H28O3
    Color and Shape:Solid
    Molecular weight:352.47

    Ref: TM-T28623

  • Glucocorticoid receptor agonist
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    Glucocorticoid receptor agonist

    CAS:
    <p>Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.</p>
    Formula:C20H20F4N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.38

    Ref: TM-T11417

  • Glucocorticoid receptor-IN-1
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    Glucocorticoid receptor-IN-1

    CAS:
    <p>Glucocorticoid receptor-IN-1 selectively modulates GR with anti-inflammatory effects, represses hMMP1 (IC50: 2.11 nM), and activates MMTV (EC50: 5.59 nM).</p>
    Formula:C24H19F4N7O2
    Color and Shape:Solid
    Molecular weight:513.45

    Ref: TM-T63551

  • Fosdagrocorat
    Targetmol
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    Fosdagrocorat

    CAS:
    <p>Fosdagrocorat is an agonist of the dissociated glucocorticoid receptor.</p>
    Formula:C29H30F3N2O5P
    Color and Shape:Solid
    Molecular weight:574.53

    Ref: TM-T15340

  • Baxdrostat
    Targetmol
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    Baxdrostat

    CAS:
    <p>Baxdrostat is an aldosterone synthase inhibitor.</p>
    Formula:C22H25N3O2
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:363.45

    Ref: TM-T61373

  • Dazucorilant
    Targetmol
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    Dazucorilant

    CAS:
    <p>Dazucorilant (CORT113176), a selective non-steroidal GR modulator, has high affinity with a K i &lt;1 nM, useful for neurological research.</p>
    Formula:C29H22F4N4O3S
    Color and Shape:Solid
    Molecular weight:582.57

    Ref: TM-T38983

  • ORIC-101
    Targetmol
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    ORIC-101

    CAS:
    <p>ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.</p>
    Formula:C34H47NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.74

    Ref: TM-T16404

  • C108297
    Targetmol
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    C108297

    CAS:
    <p>C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.</p>
    Formula:C30H36FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.69

    Ref: TM-T26935