Glucocorticoid Receptor
The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.
Found 165 products of "Glucocorticoid Receptor"
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RU 43044
CAS:RU 43044 is a selective glucocorticoid receptor antagonist that has exhibited an antidepressant-like effect.Formula:C29H34O2Purity:98%Color and Shape:SolidMolecular weight:414.58J9
CAS:J9 is an inhibitor of Glucocorticoid resistance. J9 reverses Dexamethasone Resistance in T-cell Acute Lymphoblastic Leukemia.Formula:C12H12N4Color and Shape:SolidMolecular weight:212.25Isoflupredone
CAS:Isoflupredone, a synthetic corticosteroid, inhibits inflammation and immune response in animals.Formula:C21H27FO5Purity:97.62% - 99.85%Color and Shape:SolidMolecular weight:378.43Ref: TM-T41303
1mg63.00€2mg90.00€5mg137.00€10mg235.00€25mg512.00€50mg740.00€100mg1,035.00€1mL*10mM (DMSO)150.00€Paramethasone Acetate
CAS:Paramethasone Acetate is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive effects that can be used in the treatment of systemic lupusFormula:C24H31FO6Purity:99.73%Color and Shape:SolidMolecular weight:434.5Prednisolone sodium metazoate
CAS:Prednisolone sodium metazoate is used in the treatment of Inflammatory Bowel Disease, Ulcerative Colitis, and GI Disorders.Formula:C28H32NaO9SColor and Shape:SolidMolecular weight:567.6Mazipredone
CAS:Mazipredone is a water-soluble, long-acting prednisolone derivative used topically for skin conditions & parenterally as a glucocorticoid.Formula:C26H38N2O4Color and Shape:SolidMolecular weight:442.59Prednisolone hemisuccinate
CAS:Prednisolone hemisuccinate is a soluble glucocorticoid and cortisol exerts anti-inflammatory, immunosuppressive, and antiallergic by binding to GR receptor.Formula:C25H32O8Purity:99.96%Color and Shape:SolidMolecular weight:460.52GSK9027
CAS:GSK9027, a nonsteroidal GR agonist, is a partial 2×GRE reporter gene activator, less potent than dexamethasone.Formula:C27H19F4N3O2SPurity:99.31%Color and Shape:SolidMolecular weight:525.52Methylprednisolone Aceponate
CAS:Methylprednisolone Aceponate (SH 440), a non-halogenated corticosteroid, is a potent anti-inflammatory agent.Formula:C27H36O7Purity:99.00% - 99.61%Color and Shape:SolidMolecular weight:472.57Ref: TM-T1171L
2mg35.00€5mg52.00€10mg73.00€25mg105.00€50mg156.00€100mg224.00€200mg310.00€1mL*10mM (DMSO)54.00€Prednisolone Tebutate
CAS:Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.Formula:C27H38O6Purity:98%Color and Shape:SolidMolecular weight:458.59PF-3882845
CAS:PF-3882845, a high affinity MR antagonist (IC50=2.7 nM) for hypertension, also targets progesterone receptor (IC50: 310 nM).Formula:C24H22ClN3O2Purity:99.63%Color and Shape:SolidMolecular weight:419.9RU 25055
CAS:RU 25055 is a synthetic antiglucocorticoid.Formula:C24H26O2SPurity:98%Color and Shape:SolidMolecular weight:378.53(S)-Baxdrostat
CAS:(S)-Baxdrostat is an S-enantiomer of Baxdrostat, which functions as an inhibitor of aldosterone synthase [1].Formula:C22H25N3O2Color and Shape:SolidMolecular weight:363.45Fludrocortisone
CAS:Fludrocortisone （Florinef） is a synthetic corticosteroid with moderate glucocorticoid potency and greater mineralocorticoid potency.Cost-effective and quality-assured.Formula:C21H29FO5Purity:98.56% - 98.66%Color and Shape:White SolidMolecular weight:380.45RU 28318, potassium salt
CAS:mineralocorticoid receptor (MR) antagonistFormula:C25H38KO4Purity:98%Color and Shape:SolidMolecular weight:441.67Lorundrostat
CAS:Lorundrostat is an aldosterone synthase inhibitor.Formula:C24H33N7O2Purity:95.47%Color and Shape:SolidMolecular weight:451.56AZD9567
CAS:AZD9567: potent, selective SGRM, oral, IC50=3.8nM, effective in SCW joint inflammation.Formula:C27H28F2N4O3Purity:98.4%Color and Shape:SolidMolecular weight:494.53Ref: TM-T14386
1mg190.00€5mg485.00€10mg700.00€25mg1,063.00€50mg1,431.00€100mg1,918.00€1mL*10mM (DMSO)533.00€Glucocorticoid receptor agonist-1
CAS:Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].
Formula:C35H39NO6Purity:99.68%Color and Shape:SolidMolecular weight:569.69Glucocorticoid receptor-IN-1
CAS:Glucocorticoid receptor-IN-1 selectively modulates GR with anti-inflammatory effects, represses hMMP1 (IC50: 2.11 nM), and activates MMTV (EC50: 5.59 nM).Formula:C24H19F4N7O2Color and Shape:SolidMolecular weight:513.45Dexamethasone palmitate
CAS:DXP, a lipophilic prodrug of Dexamethasone, has 47x less glucocorticoid receptor affinity; it's an agonist & anti-inflammatory.Formula:C38H59FO6Purity:99.28%Color and Shape:SolidMolecular weight:630.87
