
Enzyme
Enzyme inhibitors are molecules that bind to enzymes and decrease their activity. These inhibitors are widely used in research to study enzyme kinetics, regulation, and the role of specific enzymes in metabolic pathways. Enzyme inhibitors are also crucial in drug development, as many therapeutic agents function by inhibiting enzymes involved in disease processes. By targeting enzymes, these inhibitors can modulate biochemical pathways and offer potential treatments for various diseases. At CymitQuimica, we provide a comprehensive selection of high-quality enzyme inhibitors to support your research in biochemistry, pharmacology, and drug discovery.
Subcategories of "Enzyme"
- Carbonic Anhydrase(198 products)
- Hydroxylase(36 products)
- MPO(2 products)
- Reductase(56 products)
- Tyrosinase(79 products)
Found 3709 products for "Enzyme".
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Tyrosinase-IN-43
Tyrosinase-IN-43 (Compound 12j) is a competitive tyrosinase inhibitor with an IC50 value of 10.49 μM for tyrosinase. It exhibits significant antioxidant activity and can be used in the study and treatment of pigmentation-related conditions such as melasma, freckles, age spots, and post-inflammatory hyperpigmentation.Acesulfame
CAS:Acesulfame inhibits CA9/12 and can be used to study inflammation-related diseases.Formula:C4H5NO4SColor and Shape:SolidMolecular weight:163.15hCAIX-IN-17
hCA IX-IN-1 inhibits hCA I/II/IX/XII with Ki of 331.4/28.4/9.4/17.8 nM, has anticancer properties.Formula:C19H18N2O3SColor and Shape:SolidMolecular weight:354.42VM4-037
CAS:VM4-037 is a PET imaging agent used for carbonic anhydrase IX.Formula:C26H29FN6O7S2Color and Shape:SolidMolecular weight:620.67β-Amylase, from soy
CAS:Purity:≥ 10.0units/mgColor and Shape:White to off-white powderMolecular weight:-Calmodulin-dependent Protein Kinase II fragment 290-309
CAS:Formula:C103H185N31O24SMolecular weight:2273.83hCA/VEGFR-2-IN-3
hCA/VEGFR-2-IN-3 (compound 8j) is an indolinonylbenzenesulfonamide with potential as a dual inhibitor of cancer-associated hCA IX/XII and VEGFR-2.Formula:C24H28N6O6SPurity:98%Color and Shape:SolidMolecular weight:528.58Xanthine Oxidase, ammonium sulfate suspension
CAS:Color and Shape:Faint brown to dark brown suspensionhCAII-IN-8
CAS:Compound CDy9 is a highly selective inhibitor of carbonic anhydrase (CA) with an IC50 value of 0.18 μM for hCA II.Formula:C15H16N2O5SPurity:99.73%Color and Shape:White SolidMolecular weight:336.36Ref: TM-T67774
5mg42.00€1mL*10mM (DMSO)52.00€10mg64.00€25mg116.00€50mg167.00€100mg241.00€200mg339.00€Tyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Color and Shape:Odour SolidhCA/VEGFR-2-IN-4
hCA/VEGFR-2-IN-4 (compound 15b), an indolinylbenzenesulfonamide, serves as a potential dual inhibitor targeting cancer-related human carbonic anhydrases hCA IX/Formula:C22H23FN6O5SPurity:98%Color and Shape:SolidMolecular weight:502.52CAIX-IN-4
CAIX-IN-4 (Compound 8b) is a selective inhibitor of carbonic anhydrase IX (CAIX) with an IC50 value of 0.32 μM. It holds potential for research in cancer, such as renal cell carcinoma.Color and Shape:Odour SolidLysozyme, from chicken egg white
CAS:Purity:≥ 20,000U/mgColor and Shape:White to off-white powderMolecular weight:-DOTA-XYIMSR-01
CAS:DOTA-XYIMSR-01 is a molecular probe targeting CAIX, capable of being labeled with 177Lu for the treatment and localization of malignant gliomas. The uptake of [177Lu]Lu-XYIMSR-01 in U87MG tumors is 6.19% injected dose per gram (% ID/g), with a tumor-to-muscle uptake ratio of 20.14. In an orthotopic glioma model, co-administration with temozolomide significantly enhances survival rates and inhibits tumor growth in mice. DOTA-XYIMSR-01 shows potential for research in the field of cancer treatment.Formula:C61H88N16O22S2Color and Shape:SolidMolecular weight:1461.57hCAIX/XII-IN-11
hCAIX/XII-IN-11 (Compound 6c) is an inhibitor of hCA IX and hCA XII, exhibiting Ki values of 0.7 μM for both isoforms. This compound is applicable in cancer research.Formula:C13H10FN3O4Color and Shape:SolidMolecular weight:291.065535,6-Dihydro-2H-pyran-2-one
CAS:5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.Formula:C5H6O2Color and Shape:SolidMolecular weight:98.1TPH1-IN-1
TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.Formula:C21H18N6O4SColor and Shape:SolidMolecular weight:450.47CAIX/CAXII-IN-4
CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.Formula:C23H21N5O3SColor and Shape:SolidMolecular weight:447.51hCAIX-IN-19
hCAIX-IN-19 is a sulfonamide inhibitor with an inhibition constant (KI) of 6.2 nM for hCAIX, exhibiting significant selectivity towards hCAIX over hCAI (hCA I/Color and Shape:Odour SolidhCAIX/XII-IN-14
hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.Formula:C16H14F3N3O4SColor and Shape:SolidMolecular weight:401.36Barbituric acid
CAS:Barbituric acid is a pyrimidine derivative and the basic skeleton of barbiturate drugs, barbiturate drugs and other heterocyclic compounds.Formula:C4H4N2O3Purity:99.83%Molecular weight:128.09hCAII-IN-6
"hCAII-IN-6 (S-13) inhibits hCA II (4.4 nM) and isoforms I, IV, IX (9.2, 480.2, 14.7 nM). For glaucoma research."Formula:C20H25N3O4SColor and Shape:SolidMolecular weight:403.5hCA/VEGFR-2-IN-2
Compound 8g (hCA/VEGFR-2-IN-2) is an indolinonylbenzenesulfonamide identified as a potential dual inhibitor targeting cancer-associated isozymes hCA IX/XII andFormula:C23H26N6O5SPurity:98%Color and Shape:SolidMolecular weight:498.55Peroxidase
CAS:Purity:≥ 85units/mg (dry basis)Color and Shape:Beige to light-brown, reddish brown or dark brown lyophilised powderMolecular weight:-DPP IV/hCA II-IN-1
CAS:DPP IV/hCA II-IN-1: strong DPP IV & CA inhibitor, IC50=0.049μM (DPP IV), Ki=0.0361-3.034μM (CA II-IV).Formula:C17H20N2O5SColor and Shape:SolidMolecular weight:364.42Chlorothiazide
CAS:Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.Formula:C7H6ClN3O4S2Purity:98.46% - 98.91%Color and Shape:White SolidMolecular weight:295.72P-Hydroxybenzoate Hydroxylase
CAS:Color and Shape:Yellowish lyophilised powderMolecular weight:55 ~ 60 kDaTrypsin, bovine origin
CAS:Purity:≥ 2000units/mg (USP)Color and Shape:White or almost white crystalline powderMolecular weight:-GZ22-4
GZ22-4 is a near-infrared (NIR) fluorescent probe with a high affinity for carbonic anhydrase IX (CAIX), exhibiting a dissociation constant (Kd) of 0.2 nM. It is applicable in studies for visualizing CAIX-positive tumors.Formula:C88H126F3N6NaO24S4Color and Shape:SolidMolecular weight:1858.75561


