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Pim
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Uzansertib phosphate
CAS:2088852-47-3
Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, …
Formula:
C26H29F3N5O7P
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
611.51
Ref: TM-T12477
1mg | 94.00 € | ||
5mg | 275.00 € | ||
10mg | 410.00 € | ||
25mg | 677.00 € | ||
50mg | 922.00 € | ||
100mg | 1,290.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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FD1024
CAS:1422456-47-0
FD1024 is a potent PIM inhibitor, displaying inhibitory concentrations (IC50s) of 1.96 nM, 38.9 nM, …
Formula:
C21H20F2N4O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.47
Ref: TM-T79456
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pim-1 kinase inhibitor 5
CAS:2928606-67-9
Pim-1 kinase inhibitor 5 (Compound 4c), with an IC50 of 0.61 μM, exhibits cytotoxicity against …
Formula:
C22H13Cl2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
406.26
Ref: TM-T78980
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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HS94
CAS:1892594-93-2
HS94 (DAPK3 inhibitor HS94) is a selective and potent DAPK3 inhibitor with a Ki value …
Formula:
C15H15N5O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.38
Ref: TM-T77777
1mg | 40.00 € | ||
5mg | 85.00 € | ||
10mg | 116.00 € | ||
25mg | 224.00 € | ||
50mg | 333.00 € | ||
100mg | 494.00 € | ||
500mg | 1,058.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pim-1 kinase inhibitor 8
CAS:916038-47-6
Pim-1 kinase inhibitor 8 is a Pim-1 kinase inhibitor with anticancer activity that inhibits cell …
Formula:
C14H17N3O3
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
275.3
Ref: TM-T83627
1mg | 61.00 € | ||
5mg | 133.00 € | ||
10mg | 206.00 € | ||
25mg | 414.00 € | ||
50mg | 664.00 € | ||
100mg | 1,045.00 € | ||
500mg | 2,116.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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PIM-IN-2
CAS:1006699-45-1
PIM-IN-2 (Pim-2) is a potent inhibitor of Pim kinases, demonstrating an inhibition concentration half-maximal (IC50) …
Formula:
C19H22N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
338.4
Ref: TM-T81460
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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(2R)-Octyl-α-hydroxyglutarate
CAS:1391194-67-4
(2R)-Octyl-α-hydroxyglutarate ((2R)-Octyl-2-HG) is a D-isomer 2-Hydroxyglutarate modified form.
Formula:
C13H24O5
Color and Shape:
Solid
Molecular weight:
260.33
Ref: TM-T19611
1ml | 130.00 € | ||
2mg | 91.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pim-1/2 kinase inhibitor 1
CAS:6320-51-0
Orally active Pim-1/2 inhibitor blocks kinase phosphorylation; used in prostate cancer research.
Formula:
C11H9NO3S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
235.26
Ref: TM-T9229
1mg | 40.00 € | ||
2mg | 95.00 € | ||
5mg | 83.00 € | ||
10mg | 122.00 € | ||
25mg | 237.00 € | ||
50mg | 369.00 € | ||
100mg | 553.00 € | ||
500mg | 1,160.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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CX-6258 hydrochloride
CAS:1353859-00-3
CX-6258 hydrochloride (Pim-Kinase Inhibitor X) is an effective, orally efficacious Pim1/2/3 kinase inhibitor (IC50: 5/25/16 …
Formula:
C26H24ClN3O3·HCl
Purity:
97.98%
Color and Shape:
Solid
Molecular weight:
498.4
Ref: TM-T6148
1mg | 42.00 € | ||
1ml | 87.00 € | ||
2mg | 55.00 € | ||
5mg | 87.00 € | ||
10mg | 142.00 € | ||
25mg | 249.00 € | ||
50mg | 415.00 € | ||
100mg | 601.00 € | ||
500mg | 1,236.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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Hispidulin
CAS:1447-88-7
Hispidulin, a natural flavone with a broad spectrum of biological activities, is a Pim-1 inhibitor …
Formula:
C16H12O6
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
300.26
Ref: TM-TQ0201
1ml | 69.00 € | ||
10mg | 88.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
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(Z)-SMI-4a
CAS:438190-29-5
(Z)-SMI-4a (TCS PIM-1 4a) is a selective ATP-competitive Pim-1 kinase inhibitor with an IC50 of …
Formula:
C11H6F3NO2S
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
273.23
Ref: TM-T3058
1ml | 52.00 € | ||
5mg | 51.00 € | ||
10mg | 71.00 € | ||
25mg | 142.00 € | ||
50mg | 212.00 € | ||
100mg | 318.00 € | ||
200mg | 479.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
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Quercetagetin
CAS:90-18-6
Quercetagetin, a flavonoid from Citrus unshiu, inhibits pim-1 kinase (IC50: 0.34 μM), cell-permeable.
Formula:
C15H10O8
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
318.24
Ref: TM-T8114
1mg | 87.00 € | ||
1ml | 213.00 € | ||
5mg | 198.00 € | ||
10mg | 297.00 € | ||
25mg | 498.00 € | ||
50mg | 719.00 € | ||
100mg | 975.00 € | ||
500mg | 1,941.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
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TCS PIM-1 1
CAS:491871-58-0
TCS PIM-1 1 (SC 204330) is a potent ATP-competitive inhibitor of Pim-1 kinase with an …
Formula:
C18H11BrN2O2
Purity:
97%
Color and Shape:
Solid
Molecular weight:
367.2
Ref: TM-T2253
1ml | 96.00 € | ||
2mg | 45.00 € | ||
5mg | 63.00 € | ||
10mg | 87.00 € | ||
25mg | 184.00 € | ||
50mg | 339.00 € | ||
100mg | 501.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SGI-1776
CAS:1025065-69-3
SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, …
Formula:
C20H22F3N5O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
405.42
Ref: TM-T3078
1ml | 98.00 € | ||
2mg | 52.00 € | ||
5mg | 95.00 € | ||
10mg | 169.00 € | ||
25mg | 299.00 € | ||
50mg | 428.00 € | ||
100mg | 549.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
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Pim1/AKK1-IN-1
CAS:1093222-27-5
Pim1/AKK1-IN-1: LKB1/AAK1 inhibitor with Kd 35/53/75/380 nM for Pim1/AKK1/MST2/LKB1, also targets MPSK1, TNIK.
Formula:
C20H13N5O
Purity:
97.84%
Color and Shape:
Solid
Molecular weight:
339.35
Ref: TM-T5093
1mg | 88.00 € | ||
1ml | 201.00 € | ||
2mg | 129.00 € | ||
5mg | 180.00 € | ||
10mg | 273.00 € | ||
25mg | 479.00 € | ||
50mg | 697.00 € | ||
100mg | 978.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TP-3654
CAS:1361951-15-6
TP-3654 is a second-generation Pim kinase inhibitor (Ki values against Pim-1/3: 5/42 nM).
Formula:
C22H25F3N4O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
418.46
Ref: TM-T4523
1ml | 57.00 € | ||
5mg | 56.00 € | ||
10mg | 83.00 € | ||
25mg | 148.00 € | ||
50mg | 231.00 € | ||
100mg | 345.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
HJ-PI01
CAS:6192-43-4
HJ-PI01 (HJ-PI01) is a Pim-2 inhibitor. HJ-PI01 (HJ-PI01) induces apoptosis and autophagic cell death in …
Formula:
C14H11NO2
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
225.24
Ref: TM-T9583
1mg | 52.00 € | ||
1ml | 114.00 € | ||
5mg | 118.00 € | ||
10mg | 184.00 € | ||
25mg | 424.00 € | ||
50mg | 626.00 € | ||
100mg | 891.00 € | ||
500mg | 1,789.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZD1208
CAS:1204144-28-4
AZD1208 is a novel, orally bioavailable, highly selective PIM kinase inhibitor with single nanomolar potency …
Formula:
C21H21N3O2S
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
379.48
Ref: TM-T2300
1ml | 57.00 € | ||
2mg | 38.00 € | ||
5mg | 51.00 € | ||
10mg | 74.00 € | ||
25mg | 117.00 € | ||
50mg | 210.00 € | ||
100mg | 370.00 € | ||
200mg | 487.00 € | ||
500mg | 778.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TCS-PIM-1-4a
CAS:327033-36-3
SMI-4a, a Pim inhibitor, activates AMPK, halts mTORC1, and kills various myeloid/lymphoid cells (IC50=0.8-40μM).
Formula:
C11H6F3NO2S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
273.23
Ref: TM-T4215
1ml | 55.00 € | ||
5mg | 51.00 € | ||
10mg | 75.00 € | ||
25mg | 122.00 € | ||
50mg | 210.00 € | ||
100mg | 315.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SMI-16a
CAS:587852-28-6
SMI-16a (PIM1/2 Kinase Inhibitor VI) , a cell-permeable thiazolidinedione compound, acts as an effective, ATP-competitive …
Formula:
C13H13NO3S
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
263.31
Ref: TM-T3989
1mg | 35.00 € | ||
1ml | 92.00 € | ||
2mg | 47.00 € | ||
5mg | 69.00 € | ||
10mg | 96.00 € | ||
25mg | 158.00 € | ||
50mg | 231.00 € | ||
100mg | 346.00 € |
Estimated delivery in United States, on Friday 16 Aug 2024