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JAK/STAT signaling
Products of "JAK/STAT signaling"
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Ilginatinib
CAS:1239358-86-1
Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H20FN7
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
389.43
Ref: TM-T12266
1mg | 93.00 € | ||
1ml | 213.00 € | ||
2mg | 133.00 € | ||
5mg | 218.00 € | ||
10mg | 303.00 € | ||
25mg | 444.00 € | ||
50mg | 639.00 € | ||
100mg | 916.00 € | ||
500mg | 1,838.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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JAK2 Inhibitor V
CAS:195371-52-9
JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting …
Formula:
C23H24N2O
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
344.45
Ref: TM-T3042
1ml | 63.00 € | ||
2mg | 39.00 € | ||
5mg | 56.00 € | ||
10mg | 83.00 € | ||
25mg | 153.00 € | ||
50mg | 268.00 € | ||
100mg | 494.00 € | ||
500mg | 1,100.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Ilginatinib maleate
CAS:1354799-87-3
Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C25H24FN7O4
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
505.5
Ref: TM-T12266L
1mg | 93.00 € | ||
1ml | 245.00 € | ||
2mg | 134.00 € | ||
5mg | 217.00 € | ||
10mg | 303.00 € | ||
25mg | 444.00 € | ||
50mg | 642.00 € | ||
100mg | 917.00 € | ||
500mg | 1,839.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Uzansertib phosphate
CAS:2088852-47-3
Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, …
Formula:
C26H29F3N5O7P
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
611.51
Ref: TM-T12477
1mg | 94.00 € | ||
5mg | 275.00 € | ||
10mg | 410.00 € | ||
25mg | 677.00 € | ||
50mg | 922.00 € | ||
100mg | 1,290.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Ilginatinib hydrochloride
CAS:1239358-85-0
Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H21ClFN7
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
425.89
Ref: TM-T12266L2
1mg | 91.00 € | ||
1ml | 207.00 € | ||
5mg | 217.00 € | ||
10mg | 304.00 € | ||
25mg | 447.00 € | ||
50mg | 639.00 € | ||
100mg | 916.00 € | ||
500mg | 1,845.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Brepocitinib P-Tosylate
CAS:2140301-96-6
Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and …
Formula:
C25H29F2N7O4S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
561.6
Ref: TM-T12427
1mg | 35.00 € | ||
1ml | 87.00 € | ||
5mg | 69.00 € | ||
10mg | 102.00 € | ||
25mg | 212.00 € | ||
50mg | 384.00 € | ||
100mg | 616.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Delgocitinib
CAS:1263774-59-9
Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the …
Formula:
C16H18N6O
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
310.35
Ref: TM-T15096
1mg | 167.00 € | ||
1ml | 347.00 € | ||
5mg | 500.00 € | ||
10mg | 722.00 € | ||
25mg | 1,096.00 € | ||
50mg | 1,486.00 € | ||
100mg | 2,016.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Golidocitinib
CAS:2091134-68-6
Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: …
Formula:
C25H31N9O2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
489.57
Ref: TM-T10431
1ml | 168.00 € | ||
2mg | 94.00 € | ||
5mg | 160.00 € | ||
10mg | 262.00 € | ||
25mg | 457.00 € | ||
50mg | 605.00 € | ||
100mg | 861.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Gusacitinib
CAS:1425381-60-7
Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 …
Formula:
C24H28N8O2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
460.53
Ref: TM-T14331
1mg | 47.00 € | ||
1ml | 116.00 € | ||
5mg | 94.00 € | ||
10mg | 121.00 € | ||
25mg | 185.00 € | ||
50mg | 343.00 € | ||
100mg | 510.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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JAK1-IN-10
CAS:2416858-88-1
JAK1-IN-10 (compound 9), a cyano-substituted cyclic hydrazine derivative, functions as a potent and selective inhibitor …
Formula:
C15H17N7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T79078
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-34
CAS:2068766-90-3
JAK-IN-34 (compound 11n) is a potent inhibitor of Janus kinases (JAKs), demonstrating IC50 values of …
Formula:
C27H26N6O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
450.53
Ref: TM-T82017
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-29
JAK-IN-29 (Compound 3) is a potent inhibitor of Janus kinases (JAK) [1].
Formula:
C17H14ClN5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
355.78
Ref: TM-T79222
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-25
CAS:2127110-22-7
JAK-IN-25 (compound 19), a potent JAK inhibitor, exhibits IC50 values of 6 nM for TYK2, …
Formula:
C19H17N5O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
379.37
Ref: TM-T78175
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-33
JAK-IN-33 (Compound 3 (R)) is a selective inhibitor of the Janus kinase (JAK) family [1].
Purity:
98%
Ref: TM-T82018
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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WDR5-IN-6
CAS:326901-92-2
WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a …
Formula:
C13H8Cl2N2O2S
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
327.19
Ref: TM-T77495
1mg | 45.00 € | ||
5mg | 96.00 € | ||
10mg | 142.00 € | ||
25mg | 275.00 € | ||
50mg | 447.00 € | ||
100mg | 708.00 € | ||
500mg | 1,439.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK/HDAC-IN-2
JAK/HDAC-IN-2, a potent 2-amino-4-phenylaminopyrimidine dual-target inhibitor, effectively suppresses JAK1/2 and HDAC3/6 at nanomolar concentrations.
Formula:
C28H38N6O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
570.7
Ref: TM-T78708
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK kinase-IN-1
CAS:2698389-43-2
JAK kinase-IN-1 (Example 1) functions as a potent inhibitor targeting the JAK family, which includes …
Formula:
C17H19F2N7OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
407.44
Ref: TM-T79807
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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Pumecitinib
CAS:2401057-12-1
Pumecitinib is a Janus kinase (JAK) inhibitor. Pumecitinib exhibits anti-inflammatory activity.
Formula:
C17H20N8O2S
Purity:
99.89%
Color and Shape:
Soild
Molecular weight:
400.46
Ref: TM-T67758
1mg | 35.00 € | ||
1ml | 96.00 € | ||
5mg | 79.00 € | ||
10mg | 114.00 € | ||
25mg | 202.00 € | ||
50mg | 322.00 € | ||
100mg | 459.00 € | ||
500mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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FD1024
CAS:1422456-47-0
FD1024 is a potent PIM inhibitor, displaying inhibitory concentrations (IC50s) of 1.96 nM, 38.9 nM, …
Formula:
C21H20F2N4O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.47
Ref: TM-T79456
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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TAK-901
CAS:934541-31-8
TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid …
Formula:
C28H32N4O3S
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
504.64
Ref: TM-T2709
5mg | 76.00 € | ||
25mg | 209.00 € | ||
50mg | 363.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024