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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • DMP-543

    CAS:
    <p>DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.</p>
    Formula:C26H18F2N2O
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:412.43
  • Nisoxetine hydrochloride

    CAS:
    Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor
    Formula:C17H21NO2·HCl
    Purity:99.21%
    Color and Shape:White Solid
    Molecular weight:307.82
  • 8-Bromo-cGMP sodium

    CAS:
    <p>8-Bromo-cGMP sodium: PKG activator, eases pain, dilates vessels, reduces Ca2+ currents &amp; insulin release.</p>
    Formula:C10H10BrN5NaO7P
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:446.09
  • YM758

    CAS:
    <p>YM758 is an inhibitor of If current channel.</p>
    Formula:C26H32FN3O4
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:469.55
  • Ralitoline

    CAS:
    <p>Ralitoline (Ralitolinum) is an anticonvulsant with anticancer activity and sodium channel blocking activity.</p>
    Formula:C13H13ClN2O2S
    Purity:98.45%
    Color and Shape:Solid
    Molecular weight:296.77
  • ABT 102

    CAS:
    <p>ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.</p>
    Formula:C21H24N4O
    Purity:98.38% - 99.86%
    Color and Shape:Solid
    Molecular weight:348.44
  • JNJ-26489112

    CAS:
    <p>JNJ-26489112 is a CNS-active agent and an inhibitor of voltage-gated Na+ channels and N-type Ca2+ channels.</p>
    Formula:C9H11ClN2O4S
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:278.71
  • NHE3-IN-1

    CAS:
    <p>NHE3-IN-1 是钠/质子交换剂 3 (NHE-3) 的抑制剂。</p>
    Formula:C12H10ClN3S
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:263.75
  • Silperisone HCl

    CAS:
    <p>Silperisone HCl is a muscle relaxant and vasodilator, treating myoclonus, hypertonia, dystonia, and myospasm by blocking Na+ and Ca2+ channels.</p>
    Formula:C15H25ClFNSi
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:301.9
  • GW 542573X

    CAS:
    <p>GW 542573X is a potent and selective small molecule Ca2+-activated K+ 2 (SK2) channel activator.GW 542573X induces a leftward shift in the Ca2+ response curve</p>
    Formula:C19H28N2O5
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:364.44
  • Divaplon

    CAS:
    <p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>
    Formula:C17H17N3O2
    Purity:97.44% - 98.25%
    Color and Shape:Solid
    Molecular weight:295.34
  • Stepronin

    CAS:
    <p>Stepronin (TTPG) shows expectorant activities and inhibits airway secretion.</p>
    Formula:C10H11NO4S2
    Purity:99.59%
    Color and Shape:White Or Off White Crystalline
    Molecular weight:273.33
  • Quinacainol

    CAS:
    <p>Quinacainol (RP 54272) is a new antiarrhythmic compound with class I antiarrhythmic effects in rats.</p>
    Formula:C21H30N2O
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:326.48
  • L-838417

    CAS:
    <p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>
    Formula:C19H19F2N7O
    Purity:98.12% - 99.70%
    Color and Shape:Solid
    Molecular weight:399.4
  • Indecainide

    CAS:
    <p>Indecainide (Ricainid) is an antiarrhythmic compound that is carcinogenic and may be used in studies secondary to coronary artery disease.</p>
    Formula:C20H24N2O
    Purity:98.01% - 98.96%
    Color and Shape:Solid
    Molecular weight:308.42
  • DMT1 blocker 1

    CAS:
    <p>DMT1 blocker 1 inhibits DMT1; IC50=0.64μM; may prevent intestinal iron absorption.</p>
    Formula:C16H14N4O2
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:294.31
  • Trombodipine

    CAS:
    <p>Trombodipine (PCA-4230) is a platelet aggregation inhibitor with antithrombotic activity and protection against Listeria monocytogenes.</p>
    Formula:C21H24N2O7S
    Purity:98.73% - 99.14%
    Color and Shape:Solid
    Molecular weight:448.49
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Formula:C14H12FNO
    Purity:99.51% - 99.56%
    Color and Shape:Solid
    Molecular weight:229.25
  • Tiludronate disodium

    CAS:
    Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.
    Formula:C7H7ClNa2O6P2S
    Purity:>99.99% - >99.99%
    Color and Shape:Fine White To Off-White Crystalline Powder
    Molecular weight:362.57
  • Progabide

    CAS:
    <p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>
    Formula:C17H16ClFN2O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:334.77
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Formula:C18H17N5O2
    Purity:98.30% - 98.94%
    Color and Shape:Solid
    Molecular weight:335.36
  • Gallopamil

    CAS:
    Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.
    Formula:C28H40N2O5
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:484.63
  • CP-060

    CAS:
    <p>CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.</p>
    Formula:C30H42N2O5S
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:542.73
  • IKs124

    CAS:
    <p>IKs124 is a KCNE2/KCNQ1 potassium channel blocker, for hKCNE1 and hKCNE3, and can be used to study peptic ulcers.</p>
    Formula:C18H26N2O3S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:350.48
  • Hepcidin antagonist-1

    CAS:
    Heparin Antagonist-1 is an iron-regulating antagonist that can be used to study metabolic disorders such as iron deficiency diseases.
    Formula:C16H13Cl2N5
    Purity:99.53% - 99.76%
    Color and Shape:Solid
    Molecular weight:346.21
  • Sipatrigine

    CAS:
    Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, and calcium channels.
    Formula:C15H16Cl3N5
    Purity:98.64% - 99.77%
    Color and Shape:Solid
    Molecular weight:372.68
  • KR-32568

    CAS:
    <p>KR-32568 is a sodium/hydrogen exchanger 1 (NHE-1) inhibitor (IC50: 230 nM).</p>
    Formula:C13H12FN3O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:261.25
  • MK-0448

    CAS:
    <p>MK-0448 is a novel and selective blocker of the Kv1.5 (KCNA5) channel, a key channel involved in cardiac repolarization current I Kur.</p>
    Formula:C24H21FN4O2S
    Purity:99.25% - 99.79%
    Color and Shape:Solid
    Molecular weight:448.51
  • Rilmakalim

    CAS:
    <p>Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.</p>
    Formula:C21H23NO5S
    Purity:99.8% - 99.9%
    Color and Shape:Solid
    Molecular weight:401.48
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Formula:C17H14O6
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:314.29
  • Sulcardine sulfate

    CAS:
    <p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>
    Formula:C24H35N3O8S2
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:557.68
  • Pyr3

    CAS:
    <p>Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.</p>
    Formula:C16H11Cl3F3N3O3
    Purity:98.04%
    Color and Shape:Solid
    Molecular weight:456.63
  • PG01

    CAS:
    <p>PG01 is a potent CFTR Cl-channel potentiator, effective against ΔF508 (Ka 0.3 μM), and also against E193K, G970R and G551D (CFTR mutants), with Kd values of 0.</p>
    Formula:C28H29N3O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:439.55
  • RWJ-51204

    CAS:
    <p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>
    Formula:C21H19F2N3O3
    Purity:99.57% - 99.95%
    Color and Shape:Solid
    Molecular weight:399.39
  • SET 2

    CAS:
    <p>SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 of 0.46 μM. SET 2 shows selectivity over TRPV1, TRPV3 and TRPV4.</p>
    Formula:C17H21F3N4O2S
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:402.43
  • Saviprazole

    CAS:
    <p>Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.</p>
    Formula:C15H10F7N3O2S2
    Purity:97.07% - 97.17%
    Color and Shape:Solid
    Molecular weight:461.38
  • SKA-111

    CAS:
    SKA-111 activates KCa3.1 potassium channels, modulates membrane potential in endothelial cells, and dilates rat coronary arteries.
    Formula:C12H10N2S
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:214.29
  • SCH28080

    CAS:
    <p>SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of 20 nM (rabbit microsomal membrane).SCH28080 is a potent</p>
    Formula:C17H15N3O
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:277.32
  • (+)-KCC2 blocker 1

    CAS:
    <p>(+)-KCC2 blocker 1 is a selective blocker of KCC2 (IC50 = 0.4 μM).</p>
    Formula:C22H25NO5S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:415.5
  • TAK-653

    CAS:
    <p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>
    Formula:C19H23N3O3S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:373.47
  • AZD-1305

    CAS:
    <p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>
    Formula:C22H31FN4O4
    Purity:99.31% - 99.86%
    Color and Shape:Solid
    Molecular weight:434.5
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Formula:C21H23Cl2N3O
    Purity:99.56% - 99.97%
    Color and Shape:White To Off-White Solid
    Molecular weight:404.33
  • Elpetrigine

    CAS:
    <p>Elpetrigine (GW273293) is a potential sodium channel blocker with antiepileptic activity that can be used to study epilepsy.</p>
    Formula:C10H7Cl3N4
    Purity:99.04% - 99.43%
    Color and Shape:Solid
    Molecular weight:289.55
  • ZTZ240

    CAS:
    <p>ZTZ240 is a KCNQ2 channel activator used in the study of epilepsy.</p>
    Formula:C12H8ClFN2O
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:250.66
  • CNS-5161 hydrochloride

    CAS:
    <p>CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.</p>
    Formula:C16H19Cl2N3S2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:388.38
  • Temiverine hydrochloride

    CAS:
    Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.
    Formula:C24H36ClNO3
    Purity:99.26% - 99.43%
    Color and Shape:Solid
    Molecular weight:422
  • L-Cysteine S-sulfate

    CAS:
    <p>L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.</p>
    Formula:C3H7NO5S2
    Purity:99.90% - 99.92%
    Color and Shape:Solid
    Molecular weight:201.22
  • N106

    CAS:
    <p>N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.</p>
    Formula:C17H14N4O3S
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:354.38
  • DFP00173

    CAS:
    <p>DFP00173: Potent, selective AQP3 inhibitor; IC50 ~0.1-0.4 μM; less effective on AQP7, AQP9.</p>
    Formula:C11H7Cl2N3O3S
    Purity:99.53% - 99.53%
    Color and Shape:Solid
    Molecular weight:332.16
  • Ru-32514

    CAS:
    Ru-32514 is a benzodiazepine receptor agonist.
    Formula:C18H17N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:307.35
  • XE991

    CAS:
    <p>XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and can be used in the study of neurological disorders.</p>
    Formula:C26H20N2O
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:376.45
  • Golexanolone

    CAS:
    Golexanolone can be used to study neurological diseases.
    Formula:C21H31NO2
    Purity:99.90% - 99.99%
    Color and Shape:Solid
    Molecular weight:329.48
  • TWIK-1/TREK-1-IN-3

    CAS:
    <p>TWIK-1/TREK-1-IN-3 is a potassium channel TREK-1 inhibitor TWIK-1/TREK-1-IN-3 has antidepressant activity and can be used to study depression.</p>
    Formula:C19H27F3N2O2
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:372.43
  • WY-47766

    CAS:
    <p>WY-47766, a proton pump inhibitor, is used potentially for the treatment of postmenopausal osteoporosis.</p>
    Formula:C14H13N3O2S
    Purity:97.63% - 99.83%
    Color and Shape:Solid
    Molecular weight:287.34
  • VU 0240551

    CAS:
    VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.
    Formula:C16H14N4OS2
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:342.44
  • DMCM hydrochloride

    CAS:
    <p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>
    Formula:C17H19ClN2O4
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:350.8
  • UCCF-853

    CAS:
    <p>UCCF-853 是一种小分子 CFTR 调节剂,可用于研究囊性纤维化。</p>
    Formula:C14H8ClF3N2O
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:312.67
  • FR183998 free base

    CAS:
    <p>FR183998 free base is an inhibitor of Na+/Ca2+ Exchanger.</p>
    Formula:C17H19Cl2N5O2S
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:428.34
  • NS-2710

    CAS:
    <p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Formula:C22H20N4O
    Purity:99.7% - 99.82%
    Color and Shape:Solid
    Molecular weight:356.42
  • Sarmazenil

    CAS:
    <p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>
    Formula:C15H14ClN3O3
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:319.74
  • R(+)-IAA-94

    CAS:
    <p>R(+)-IAA-94 (Methylindazone) blocks epithelial chloride channels; inhibits Nef-sdAb19 binding.</p>
    Formula:C17H18Cl2O4
    Purity:98.95% - 99.17%
    Color and Shape:Solid
    Molecular weight:357.23
  • TC-N 1752

    CAS:
    TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. TC-N 1752 shows analgesic activities.
    Formula:C25H27F3N6O3
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:516.52
  • Olvanil

    CAS:
    <p>Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.</p>
    Formula:C26H43NO3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:417.62
  • Ro 25-6981

    CAS:
    <p>Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.</p>
    Formula:C22H29NO2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:339.47
  • VRT-532

    CAS:
    <p>VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.</p>
    Formula:C16H14N2O
    Purity:99.88% - 99.93%
    Color and Shape:Solid
    Molecular weight:250.3
  • CFTR corrector 8

    CAS:
    <p>CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.</p>
    Formula:C29H27F2NO7
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:539.52
  • Mavatrep

    CAS:
    <p>Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can be used for studies about inflammatory pain.</p>
    Formula:C25H21F3N2O
    Purity:98.51% - 99.31%
    Color and Shape:Solid
    Molecular weight:422.44
  • Dasolampanel

    CAS:
    Dasolampanel (NGX-426) is an ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study of chronic pain disorders.
    Formula:C17H20ClN5O3
    Purity:98.70%
    Color and Shape:Solid
    Molecular weight:377.83
  • Saripidem

    CAS:
    <p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>
    Formula:C19H20ClN3O
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:341.83
  • Butibufen

    CAS:
    Butibufen (FF-106) is a non-steroidal anti-inflammatory compound and LOX inhibitor with analgesic and antipyretic activity for the study of rheumatic diseases.
    Formula:C14H20O2
    Purity:98.11% - 98.91%
    Color and Shape:Solid
    Molecular weight:220.31
  • UCL 2077

    CAS:
    <p>UCL 2077 blocks KCNQ channels, related to epilepsy, and selective slow-afterhyperpolarization channels, with 500 nM IC50, sparing Ca2+ channels.</p>
    Formula:C25H22N2
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:350.46
  • MSP3

    CAS:
    <p>MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective effects.</p>
    Formula:C16H19NO3S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:305.39
  • Nelonemdaz

    CAS:
    Nelonemdaz (Neu2000) is an NMDA receptor antagonist with antioxidant activity that can be used to study cerebral infarction reperfusion injury.
    Formula:C15H8F7NO3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:383.22
  • ELB-139

    CAS:
    <p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>
    Formula:C14H16ClN3O
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:277.75
  • GNE-8324

    CAS:
    <p>GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, but not excitatory, neurons.</p>
    Formula:C18H18FN3OS
    Purity:98.68% - 99.34%
    Color and Shape:Solid
    Molecular weight:343.42
  • Enecadin

    CAS:
    Enecadin is a neuroprotective agent.
    Formula:C21H28FN3O
    Purity:98.53%
    Color and Shape:Solid
    Molecular weight:357.46
  • UK 66914

    CAS:
    <p>UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.</p>
    Formula:C18H24N4O3S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:376.47
  • Protonstatin-1

    CAS:
    <p>Protonstatin-1: treats hypoglycemia &amp; Alzheimer's, inhibits IGFIR kinase, used in cancer studies.</p>
    Formula:C8H5NO2S2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:211.26
  • FEMA-4809

    CAS:
    <p>FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling agent.</p>
    Formula:C17H17N3O2S
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:327.4
  • Transcainide

    CAS:
    Transcainide (R 54718), an oral lidocaine-like antiarrhythmic, blocks BTX-activated Na+ channels in heart/muscle.
    Formula:C22H35N3O2
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:373.53
  • Cerebrocrast

    CAS:
    <p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>
    Formula:C26H35F2NO7
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:511.56
  • Delucemine Hydrochloride

    CAS:
    <p>Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.</p>
    Formula:C16H18ClF2N
    Purity:98.49% - 99.30%
    Color and Shape:Solid
    Molecular weight:297.77
  • Muscimol HBr

    CAS:
    Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
    Formula:C4H7BrN2O2
    Purity:98.13%
    Color and Shape:Off-White Powder
    Molecular weight:195.01
  • Neboglamine hydrochloride

    CAS:
    Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.
    Formula:C13H25ClN2O3
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:292.8
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Formula:C17H17Cl2NO
    Purity:99%
    Color and Shape:Solid
    Molecular weight:322.23
  • HC-070

    CAS:
    HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).
    Formula:C22H20Cl2N4O4
    Purity:98.48%
    Color and Shape:Solid
    Molecular weight:475.32
  • Abeprazan hydrochloride

    CAS:
    <p>Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting H+, K+ -atPase</p>
    Formula:C19H18ClF3N2O3S
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:446.87
  • RL648_81

    CAS:
    <p>RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.</p>
    Formula:C17H17F4N3O2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:371.33
  • NC-1300-B

    CAS:
    NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.
    Formula:C17H19N3OS
    Purity:99.50%
    Color and Shape:Solid
    Molecular weight:313.42
  • Nerisopam

    CAS:
    <p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>
    Formula:C18H19N3O2
    Purity:97.07%
    Color and Shape:Solid
    Molecular weight:309.36
  • FR-167356

    CAS:
    <p>FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone metastasis.</p>
    Formula:C19H17Cl2NO3
    Purity:98.44% - 99.74%
    Color and Shape:Solid
    Molecular weight:378.25
  • TASK-1-IN-1

    CAS:
    <p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>
    Formula:C22H20N2O2
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:344.41
  • Losigamone

    CAS:
    Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.
    Formula:C12H11ClO4
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:254.67
  • NNC 05-711

    CAS:
    <p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>
    Formula:C21H23ClN2O3
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:386.87
  • NaV1.2/1.6 channel blocker-1

    CAS:
    <p>NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.</p>
    Formula:C14H14N2OS
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:258.34
  • SKF96067

    CAS:
    <p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>
    Formula:C21H22N2O2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:334.41
  • Bamocaftor

    CAS:
    <p>Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF patients.</p>
    Formula:C28H32F3N5O4S
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:591.65
  • Lirequinil

    CAS:
    <p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>
    Formula:C26H25ClN2O3
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:448.94
  • Elismetrep

    CAS:
    <p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>
    Formula:C27H21F3N2O5S
    Purity:99.37% - 99.93%
    Color and Shape:Solid
    Molecular weight:542.53
  • Aptiganel

    CAS:
    <p>Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.</p>
    Formula:C20H21N3
    Purity:98.13% - 98.90%
    Color and Shape:Solid
    Molecular weight:303.4