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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2290 products of "Membrane Transporter/Ion Channel"

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  • AMG-0347

    CAS:
    <p>AMG-0347 inhibits TRPA1 ion channels in sensory neurons, blocking pain perception.</p>
    Formula:C24H26F3N3O2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:445.48
  • Bupivacaine hydrochloride monohydrate

    CAS:
    Bupivacaine hydrochloride monohydrate is an NMDA receptor inhibitor that inhibits SCN5A channels and is commonly used in the study of chronic pain.
    Formula:C18H31ClN2O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:342.9
  • Soraprazan

    CAS:
    BS3 Crosslinker (Bis(sulfosuccinimidyl)suberate) is an ADC linker that can be used to synthesize antibody-coupled active molecules.
    Formula:C21H25N3O3
    Purity:97.69% - 99.84%
    Color and Shape:Solid
    Molecular weight:367.44
  • EMD57033

    CAS:
    <p>EMD57033 activates cardiac troponin C, enhances Ca2+ sensitivity to boost heart contraction.</p>
    Formula:C22H23N3O4S
    Purity:99.72% - >99.99%
    Color and Shape:Solid
    Molecular weight:425.5
  • C 101248

    CAS:
    <p>C 101248 (KCNK13-IN-1) is a selective and potent tandem pore halogen inhibitor of K+ channel 1 (THIK-1) inhibitor and a human and mouse KCNK13 inhibitor.</p>
    Formula:C15H12N6O
    Purity:99.14% - 99.31%
    Color and Shape:Solid
    Molecular weight:292.3
  • Funapide

    CAS:
    <p>Funapide (TV 45070) is a potent Nav1.7 inhibitor, potentially treating inflammation and various pains.</p>
    Formula:C22H14F3NO5
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:429.35
  • Aneratrigine hydrochloride

    CAS:
    <p>Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.</p>
    Formula:C19H21Cl2F2N5O2S2
    Purity:98.37% - 99.16%
    Color and Shape:Solid
    Molecular weight:524.43
  • Reldesemtiv

    CAS:
    <p>Reldesemtiv (CK-2127107) boosts exercise capacity, targeting fast muscle troponin, EC50 3.4 μM.</p>
    Formula:C19H18F2N6O
    Purity:97.27%
    Color and Shape:Solid
    Molecular weight:384.38
  • AMG2850

    CAS:
    <p>AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).</p>
    Formula:C19H17F6N3O
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:417.35
  • Metaphit methylsulfate

    CAS:
    <p>Metaphit methylsulfate is a specific PCP antagonist and an acylating agent for the [3H] phencyclidine binding site in rat brain homogenate. It inhibits PCP-induced motor activity through a presynaptic mechanism.</p>
    Formula:C19H28N2O3S2
    Color and Shape:Solid
    Molecular weight:396.567
  • 3-Bromoamphetamine hydrochloride

    CAS:
    <p>3-Bromoamphetamine hydrochloride is a para-substituted amphetamine that functions as a monoamine releaser.</p>
    Formula:C9H13BrClN
    Color and Shape:Solid
    Molecular weight:250.563
  • ML-SI1

    CAS:
    <p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>
    Formula:C23H26Cl2N2O3
    Color and Shape:Solid
    Molecular weight:449.37
  • URAT1 inhibitor 3


    <p>URAT1 inhibitor 3: potent oral URAT1 blocker, IC50=0.8 nM, for gout/hyperuricemia study.</p>
    Formula:C14H8Cl2N2O2
    Color and Shape:Solid
    Molecular weight:307.13
  • YY-23

    CAS:
    <p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>
    Formula:C33H54O8
    Color and Shape:Solid
    Molecular weight:578.777
  • PD-217014

    CAS:
    <p>PD-217014 is an α2δ ligand that exhibits visceral analgesic activity and can suppress visceral hypersensitivity. Its antihyperalgesic effects are dose-dependent.</p>
    Formula:C10H17NO2
    Color and Shape:Solid
    Molecular weight:183.25
  • MRS4738


    <p>MRS4738 is a potent antagonist with high affinity for the P2Y14R receptor. It demonstrates in vivo anti-hyperallodynic and antiasthmatic activity [1].</p>
    Formula:C30H24F3NO2
    Color and Shape:Solid
    Molecular weight:487.51
  • ABCA1 inducer 2

    CAS:
    <p>ABCA1 inducer 2 is a non-lipogenic inducer of ABCA1. It increases the expression of ABCA1 by targeting the LXR pathway, thereby reducing lipid accumulation induced by ox-LDL and inhibiting foam cell formation. ABCA1 inducer 2 holds potential as an anti-atherosclerotic agent.</p>
    Formula:C16H11BrN2O
    Color and Shape:Solid
    Molecular weight:327.175
  • pan-HCN-IN-1

    CAS:
    <p>Pan-HCN-IN-1 (Compound J&amp;J12e) is an inhibitor of the hyperpolarization-activated and cyclic-nucleotide-gated 1 (HCN1) ion channel, with an IC50 of 58 nM. Pan-HCN-IN-1 reduces the voltage sag response and enhances EPSP summation in ex vivo rat brain slices [1].</p>
    Formula:C23H37N3O2
    Color and Shape:Solid
    Molecular weight:387.56
  • Sesamodil

    CAS:
    <p>Sesamodil (SD 3211) is a novel calcium antagonist that can be used to study hypertension.</p>
    Formula:C29H32N2O6S
    Purity:98.58% - 99.01%
    Color and Shape:Solid
    Molecular weight:536.64
  • S 0960

    CAS:
    <p>S 0960 is a dimeric bile acid analogue, a specific inhibitor of the sodium-dependent bile salt transporter in the ileum, used in metabolic disease research.</p>
    Formula:C48H79NO8
    Purity:99.32% - >99.99%
    Color and Shape:Solid
    Molecular weight:798.14